公开(公告)号：US20110166162A1

公开(公告)日：2011-07-07

申请号：US12999349

申请日：2009-06-17

申请人： Wolfgang von Deyn ,  Michael Puhl ,  Matthias Pohlman ,  Michael Rack ,  Liliana Parra Rapado ,  Jürgen Langewald ,  Douglas D. Anspaugh ,  Hassan Oloumi-Sadeghi ,  Gale F. Matt Hews ,  Deborah L. Culbertson ,  Nancy B. Rankl ,  Hennicke Kamp ,  Bennard van Ravenzwaay

发明人： Wolfgang von Deyn ,  Michael Puhl ,  Matthias Pohlman ,  Michael Rack ,  Liliana Parra Rapado ,  Jürgen Langewald ,  Douglas D. Anspaugh ,  Hassan Oloumi-Sadeghi ,  Gale F. Matt Hews ,  Deborah L. Culbertson ,  Nancy B. Rankl ,  Hennicke Kamp ,  Bennard van Ravenzwaay

IPC分类号： A01N43/54 ,  C07D417/06 ,  C07D401/06 ,  A01N43/40 ,  A01P11/00 ,  A01P15/00 ,  A01P7/04 ,  A01P5/00 ,  A01P7/00

CPC分类号： C07D417/06 ,  A01N43/80 ,  C02F1/001 ,  C02F2209/03 ,  C02F2303/16 ,  C07D417/14

摘要： The present invention relates to sulfonamide compounds of formula (I) wherein R1 is H, halogen, CN, C1-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, C3-C7-cycloalkyl, C3-C7-cycloalkyl-C1-C4-alkyl, C1-C6-alkoxy, C2-C6-alkenyloxy, C2-C6-alkynyloxy, C1-C6-alkylthio, C2-C6-alkenylthio, C2-C6-alkynylthio, C1-C6-haloalkyl or C1-C6-haloalkoxy; R2 and R3 are H, halogen, CN, C1-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, C3-C7-cycloalkyl, C3-C7-cycloalkyl-C1-C4-alkyl, C1-C6-alkoxy, C2-C6-alkenyloxy, C2-C6-alkynyloxy, C1-C6-alkylthio, C2-C6-alkenylthio, C2-C6-alkynylthio, C1-C6-haloalkyl or C1-C6-haloalkoxy; or R2 together with R3 form a fused 5 or 6-membered carbocycle or heterocycle; R4 is halogen, CN, C1-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, C1-C6-alkoxy, C1-C6-alkylthio, C1-C6-alkylsulfinyl, C1-C6-alkylsulfonyl, C1-C6-haloalkyl, C1-C6-haloalkoxy, C1-C6-haloalkylthio, C1-C6-haloalkylsulfinyl or C1-C6-haloalksulfonyl; n is 0, 1, 2 or 3; R5 is phenyl or a 5- or 6-membered heterocycle; X is O or NRx, wherein Rx is H, C1-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, C3-C7-cycloalkyl, C1-C6-alkoxy, C2-C6-alkenyloxy, C2-C6-alkynyloxy, C1-C6-alkylcarbonyl or C1-C6-alkylcarbonyloxy; Y is N or C(Ry), wherein Ry is H, halogen, CN, C1-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, C3-C7-cycloalkyl, C3-7-cycloalkyl-C1-C4-alkyl, C1-C6-alkoxy, C2-C6-alkenyloxy, C2-C6-alkynyloxy, C1-C6-alkylthio, C2-C6-alkenylthio, C2-C6-alkynylthio, C1-C6-haloalkyl and C1-C6-haloalkoxy; and Z is a chemical bond, O or N(Rz), wherein Rz is C1-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, C3-C7-cycloalkyl, C1-C6-alkoxy, C2-C6-alkenyloxy, C1-C6-alkylcarbonyl or C1-C6-alkylcarbonyloxy; as well as to the N-oxides and salts thereof. These compounds are useful for combating animal pests. The invention also relates to a process for the preparation of these compounds and to intermediate compounds used in said process. The invention further relates to a method for controlling animal pests by using the compounds of formula (I), the N-oxides or the salts thereof, to plant propagation material and to an agricultural and veterinary composition comprising said compounds, the N-oxides or the salts thereof.

公开(公告)号：US07563921B2

公开(公告)日：2009-07-21

申请号：US12137624

申请日：2008-06-12

申请人： Wolfgang von Deyn ,  Henricus Maria Martinus Bastiaans ,  Matthias Pohlman ,  Michael Rack ,  Ernst Baumann ,  Michael Puhl ,  Michael Hofmann ,  Livio Tedeschi ,  Markus Kordes ,  Christopher Koradin ,  Douglas D. Anspaugh ,  Deborah L. Culbertson ,  Henry van Tuyl Cotter ,  Hassan Oloumi-Sadeghi

发明人： Wolfgang von Deyn ,  Henricus Maria Martinus Bastiaans ,  Matthias Pohlman ,  Michael Rack ,  Ernst Baumann ,  Michael Puhl ,  Michael Hofmann ,  Livio Tedeschi ,  Markus Kordes ,  Christopher Koradin ,  Douglas D. Anspaugh ,  Deborah L. Culbertson ,  Henry van Tuyl Cotter ,  Hassan Oloumi-Sadeghi

IPC分类号： C07C319/20 ,  C07C323/32 ,  C07C311/15 ,  A01N25/00 ,  A01N25/26 ,  A01P17/00 ,  A61K31/18

CPC分类号： C07C319/20 ,  A01N41/06 ,  C07C311/29 ,  C07C323/62

摘要： The invention relates to 2-cyano-3-(halo)alkoxy-benzenesulfonamide compounds I where the variables Alk and R1 to R5 are as defined in claim 1, and/or to their agriculturally useful salts. Moreover, the present invention relates to the use of compounds I and/or their salts for combating animal pests; agricultural compositions comprising such an amount of at least one compound of the general formula I and/or at least one agriculturally useful salt of I and at least one inert liquid and/or solid agronomically acceptable carrier that it has a pesticidal action and, if desired, at least one surfactant; and a method of combating animal pests which comprises contacting the animal pests, their habit, breeding ground, food supply, plant, seed, soil, area, material or environment in which the animal pests are growing or may grow, or the materials, plants, seeds, soils, surfaces or spaces to be protected from animal attack or infestation with a pesticidally effective amount of at least one 2-cyano-3-(halo)alkoxy-benzenesulfonamide compound of the formula I and/or at least one agriculturally acceptable salt thereof. a method for the for the protection of seeds from soil insects and of the resulting plant's roots and shoots from soil and foliar insects comprising contacting the seeds before sowing and/or after pregermination with a 2-cyano-3-(halo)alkoxy-benzenesulfonamide compound of the general formula I.

摘要翻译： 本发明涉及2-氰基-3-（卤代）烷氧基 - 苯磺酰胺化合物I，其中变量Alk和R1至R5如权利要求1所定义，和/或其农业上有用的盐。 此外，本发明涉及化合物I和/或其盐对抗动物害虫的用途; 包含至少一种式I化合物和/或至少一种农业上可用的I盐和至少一种惰性液体和/或其农业上可接受的载体的农药组合物，其具有杀虫作用，如果需要 ，至少一种表面活性剂; 以及一种对抗动物害虫的方法，包括使动物有害生物，其习惯，繁殖地，食物供应，植物，种子，土壤，区域，动物害虫生长或可能生长的区域，材料或环境，或材料，植物 ，防止动物攻击或侵染的种子，土壤，表面或空间，其中农药有效量的至少一种式I的2-氰基-3-（卤代）烷氧基 - 苯磺酰胺化合物和/或至少一种农业上可接受的 的盐。 包括从土壤和叶面昆虫中保护种子免受土壤昆虫和所得植物的根和芽的方法，包括在种子播种前和/或后发芽后将种子与2-氰基-3-（卤代）烷氧基 - 苯磺酰胺 通式Ⅰ的化合物

公开(公告)号：US20080306297A1

公开(公告)日：2008-12-11

申请号：US12137624

申请日：2008-06-12

申请人： Wolfgang von Deyn ,  Henricus Maria Martinus Bastiaans ,  Matthias Pohlman ,  Michael Rack ,  Ernst Baumann ,  Michael Puhl ,  Michael Hofmann ,  Livio Tedeschi ,  Markus Kordes ,  Christopher Koradin ,  Douglas D. Anspaugh ,  Deborah L. Culbertson ,  Henry van Tuyl Cotter ,  Hassan Oloumi-Sadeghi

发明人： Wolfgang von Deyn ,  Henricus Maria Martinus Bastiaans ,  Matthias Pohlman ,  Michael Rack ,  Ernst Baumann ,  Michael Puhl ,  Michael Hofmann ,  Livio Tedeschi ,  Markus Kordes ,  Christopher Koradin ,  Douglas D. Anspaugh ,  Deborah L. Culbertson ,  Henry van Tuyl Cotter ,  Hassan Oloumi-Sadeghi

IPC分类号： C07C255/53

CPC分类号： C07C319/20 ,  A01N41/06 ,  C07C311/29 ,  C07C323/62

摘要： Novel 2-cyano-3-(halo)alkoxy-benzenesulfonamide compounds for combating animal pestsThe invention relates to 2-cyano-3-(halo)alkoxy-benzenesulfonamide compounds I where the variables Alk and R1 to R5 are as defined in claim 1, and/or to their agriculturally useful salts.Moreover, the present invention relates to the use of compounds I and/or their salts for combating animal pests; agricultural compositions comprising such an amount of at least one compound of the general formula I and/or at least one agriculturally useful salt of I and at least one inert liquid and/or solid agronomically acceptable carrier that it has a pesticidal action and, if desired, at least one surfactant; and a method of combating animal pests which comprises contacting the animal pests, their habit, breeding ground, food supply, plant, seed, soil, area, material or environment in which the animal pests are growing or may grow, or the materials, plants, seeds, soils, surfaces or spaces to be protected from animal attack or infestation with a pesticidally effective amount of at least one 2-cyano-3-(halo)alkoxy-benzenesulfonamide compound of the formula I and/or at least one agriculturally acceptable salt thereof. a method for the for the protection of seeds from soil insects and of the resulting plant's roots and shoots from soil and foliar insects comprising contacting the seeds before sowing and/or after pregermination with a 2-cyano-3-(halo)alkoxybenzenesulfonamide compound of the general formula I

摘要翻译： 用于对抗动物害虫的新型2-氰基-3-（卤代）烷氧基 - 苯磺酰胺化合物本发明涉及2-氰基-3-（卤代）烷氧基 - 苯磺酰胺化合物I，其中变量Alk和R1至R5如权利要求1中所定义 ，和/或其农业上有用的盐。 此外，本发明涉及化合物I和/或其盐对抗动物害虫的用途; 包含至少一种式I化合物和/或至少一种农业上可用的I盐和至少一种惰性液体和/或其农业上可接受的载体的农药组合物，其具有杀虫作用，如果需要 ，至少一种表面活性剂; 以及一种对抗动物害虫的方法，包括使动物有害生物，其习惯，繁殖地，食物供应，植物，种子，土壤，区域，动物害虫生长或可能生长的区域，材料或环境，或材料，植物 ，防止动物攻击或侵染的种子，土壤，表面或空间，其中农药有效量的至少一种式I的2-氰基-3-（卤代）烷氧基 - 苯磺酰胺化合物和/或至少一种农业上可接受的 的盐。 包括从土壤和叶面昆虫中保护种子免受土壤昆虫和所得植物的根和芽的方法，包括在种子播种前和/或后发芽之前将种子与2-氰基-3-（卤代）烷氧基苯磺酰胺化合物接触 通式I

公开(公告)号：US07544637B2

公开(公告)日：2009-06-09

申请号：US11791398

申请日：2005-11-24

申请人： Wolfgang von Deyn ,  Henricus Maria Martinus Bastiaans ,  Matthias Pohlman ,  Michael Rack ,  Ernst Baumann ,  Michael Puhl ,  Michael Hofmann ,  Livio Tedeschi ,  Markus Kordes ,  Christopher Koradin ,  Douglas D. Anspaugh ,  Deborah L. Culbertson ,  Henry van Tuyl Cotter ,  Hassan Oloumi-Sadeghi

发明人： Wolfgang von Deyn ,  Henricus Maria Martinus Bastiaans ,  Matthias Pohlman ,  Michael Rack ,  Ernst Baumann ,  Michael Puhl ,  Michael Hofmann ,  Livio Tedeschi ,  Markus Kordes ,  Christopher Koradin ,  Douglas D. Anspaugh ,  Deborah L. Culbertson ,  Henry van Tuyl Cotter ,  Hassan Oloumi-Sadeghi

IPC分类号： C07C311/15 ,  A01N25/00 ,  A01N25/26 ,  A01P17/00 ,  A61K31/18

CPC分类号： C07C319/20 ,  A01N41/06 ,  C07C311/29 ,  C07C323/62

摘要： The invention relates to 2-cyano-3-(halo)alkoxy-benzenesulfonamide compounds I where the variables Alk and R1 to R5 are as defined in claim 1, and/or to their agriculturally useful salts. Moreover, the present invention relates to the use of compounds I and/or their salts for combating animal pests; agricultural compositions comprising such an amount of at least one compound of the general formula I and/or at least one agriculturally useful salt of I and at least one inert liquid and/or solid agronomically acceptable carrier that it has a pesticidal action and, if desired, at least one surfactant; and a method of combating animal pests which comprises contacting the animal pests, their habit, breeding ground, food supply, plant, seed, soil, area, material or environment in which the animal pests are growing or may grow, or the materials, plants, seeds, soils, surfaces or spaces to be protected from animal attack or infestation with a pesticidally effective amount of at least one2-cyano-3-(halo)alkoxy-benzenesulfonamide compound of the formula I and/or at least one agriculturally acceptable salt thereof. a method for the for the protection of seeds from soil insects and of the resulting plant's roots and shoots from soil and foliar insects comprising contacting the seeds before sowing and/or after pregermination with a 2-cyano-3-(halo)alkoxy-benzenesulfonamide compound of the general formula I

摘要翻译： 本发明涉及2-氰基-3-（卤代）烷氧基 - 苯磺酰胺化合物I，其中变量Alk和R1至R5如权利要求1所定义，和/或其农业上有用的盐。 此外，本发明涉及化合物I和/或其盐对抗动物害虫的用途; 包含至少一种式I化合物和/或至少一种农业上可用的I盐和至少一种惰性液体和/或其农业上可接受的载体的农药组合物，其具有杀虫作用，如果需要 ，至少一种表面活性剂; 以及一种对抗动物害虫的方法，包括使动物有害生物，其习惯，繁殖地，食物供应，植物，种子，土壤，区域，动物害虫生长或可能生长的区域，材料或环境，或材料，植物 ，防止动物攻击或侵染的种子，土壤，表面或空间与杀虫有效量的式I的至少一个2-氰基-3-（卤代）烷氧基 - 苯磺酰胺化合物和/或至少一种农业上可接受的盐 其中。 包括从土壤和叶面昆虫中保护种子免受土壤昆虫和所得植物的根和芽的方法，包括在种子播种前和/或后发芽后将种子与2-氰基-3-（卤代）烷氧基 - 苯磺酰胺 通式I的化合物

公开(公告)号：US20120149705A1

公开(公告)日：2012-06-14

申请号：US13400752

申请日：2012-02-21

申请人： Thomas SCHMIDT ,  Michael PUHL ,  Joachim DICKHAUT ,  Henricus Maria Martinus BASTIAANS ,  Michael RACK ,  Deborah L. CULBERTSON ,  Douglas D. Anspaugh ,  Franz-Josef BRAUN ,  Toni BUCCI ,  Henry Van Tuyl COTTER ,  David G. KUHN ,  Hassan OLOUMI-SADEGHI

发明人： Thomas SCHMIDT ,  Michael PUHL ,  Joachim DICKHAUT ,  Henricus Maria Martinus BASTIAANS ,  Michael RACK ,  Deborah L. CULBERTSON ,  Douglas D. Anspaugh ,  Franz-Josef BRAUN ,  Toni BUCCI ,  Henry Van Tuyl COTTER ,  David G. KUHN ,  Hassan OLOUMI-SADEGHI

IPC分类号： A01N43/56 ,  C07D401/14 ,  C07D413/14 ,  A01P5/00 ,  A01N43/84 ,  A01P7/04 ,  A01P7/02 ,  C07D401/04 ,  C07D409/14

CPC分类号： C07D401/04 ,  A01N43/56 ,  A01N43/84 ,  C07D401/14 ,  C07D409/14 ,  C07D413/14

摘要： N-Thio-anthranilamid compounds of formula (I) wherein A is a group selected from A1 and A2 wherein the variables and the indices are as defined per the description, processes for preparing the compounds I, pesticidal compositions comprising compounds I, use of compounds I for the control of insects, acarids or nematodes, and methods for treating, controlling, preventing or protecting animals against infestation or infection by parasites by use of compounds of formula I.

摘要翻译： 式（I）的N-硫代 - 邻氨基苯甲酰胺化合物，其中A是选自A1和A2的基团，其中变量和指数如说明书所定义，制备化合物I的方法，包含化合物I的杀虫组合物，化合物的用途 用于控制昆虫，螨虫或线虫的方法，以及通过使用式I化合物来治疗，控制，预防或保护动物免受寄生虫侵染或感染的方法。

公开(公告)号：US08143292B2

公开(公告)日：2012-03-27

申请号：US11994812

申请日：2006-06-30

申请人： Thomas Schmidt ,  Michael Puhl ,  Joachim Dickhaut ,  Henricus Maria Martinus Bastiaans ,  Michael Rack ,  Deborah L. Culbertson ,  Douglas D. Anspaugh ,  Franz-Josef Braun ,  Toni Bucci ,  Henry Van Tuyl Cotter ,  David G. Kuhn ,  Hassan Oloumi-Sadeghi

发明人： Thomas Schmidt ,  Michael Puhl ,  Joachim Dickhaut ,  Henricus Maria Martinus Bastiaans ,  Michael Rack ,  Deborah L. Culbertson ,  Douglas D. Anspaugh ,  Franz-Josef Braun ,  Toni Bucci ,  Henry Van Tuyl Cotter ,  David G. Kuhn ,  Hassan Oloumi-Sadeghi

IPC分类号： A01N43/40 ,  C07D401/04

CPC分类号： C07D401/04 ,  A01N43/56 ,  A01N43/84 ,  C07D401/14 ,  C07D409/14 ,  C07D413/14

摘要： N-Thio-anthranilamid compounds of formula (I) wherein A is a group selected from A1 and A2 wherein the variables and the indices are as defined per the description, processes for preparing the compounds I, pesticidal compositions comprising compounds I, use of compounds I for the control of insects, acarids or nematodes, and methods for treating, controlling, preventing or protecting animals against infestation or infection by parasites by use of compounds of formula I.

公开(公告)号：US08338419B2

公开(公告)日：2012-12-25

申请号：US13400752

申请日：2012-02-21

申请人： Thomas Schmidt ,  Michael Puhl ,  Joachim Dickhaut ,  Henricus Maria Martinus Bastiaans ,  Michael Rack ,  Deborah L. Culbertson ,  Douglas D. Anspaugh ,  Franz-Josef Braun ,  Toni Bucci ,  Henry Van Tuyl Cotter ,  David G. Kuhn ,  Hassan Oloumi-Sadeghi

发明人： Thomas Schmidt ,  Michael Puhl ,  Joachim Dickhaut ,  Henricus Maria Martinus Bastiaans ,  Michael Rack ,  Deborah L. Culbertson ,  Douglas D. Anspaugh ,  Franz-Josef Braun ,  Toni Bucci ,  Henry Van Tuyl Cotter ,  David G. Kuhn ,  Hassan Oloumi-Sadeghi

IPC分类号： A01N43/84 ,  A01N43/56 ,  C07D401/14 ,  C07D413/14 ,  C07D401/04 ,  C07D409/14

CPC分类号： C07D401/04 ,  A01N43/56 ,  A01N43/84 ,  C07D401/14 ,  C07D409/14 ,  C07D413/14

摘要： N-Thio-anthranilamid compounds of formula (I) wherein A is a group selected from A1 and A2 wherein the variables and the indices are as defined per the description, processes for preparing the compounds I, pesticidal compositions comprising compounds I, use of compounds I for the control of insects, acarids or nematodes, and methods for treating, controlling, preventing or protecting animals against infestation or infection by parasites by use of compounds of formula I.

摘要翻译： 式（I）的N-硫代 - 邻氨基苯甲酰胺化合物，其中A是选自A1和A2的基团，其中变量和指数如说明书所定义，制备化合物I的方法，包含化合物I的杀虫组合物，化合物的用途 I用于控制昆虫，螨虫或线虫，以及通过使用式I化合物治疗，控制，预防或保护动物免受寄生虫感染或侵害的方法。

公开(公告)号：US09125414B2

公开(公告)日：2015-09-08

申请号：US13386473

申请日：2010-07-15

申请人： Ronan Le Vezouet ,  Sebastian Soergel ,  Christian Defieber ,  Steffen Gross ,  Karsten Koerber ,  Deborah L. Culbertson ,  Douglas D. Anspaugh

发明人： Ronan Le Vezouet ,  Sebastian Soergel ,  Christian Defieber ,  Steffen Gross ,  Karsten Koerber ,  Deborah L. Culbertson ,  Douglas D. Anspaugh

IPC分类号： A01N43/40 ,  A01P7/04 ,  A01N43/80 ,  A01N43/50 ,  A01N43/76 ,  A01N43/78 ,  C07D401/12 ,  C07D413/12 ,  C07D417/12

CPC分类号： A01N43/80 ,  A01N43/50 ,  A01N43/76 ,  A01N43/78 ,  C07D401/12 ,  C07D413/12 ,  C07D417/12

摘要： The present invention relates to methods and uses of compounds of formulae I or II and the salts and N-oxides thereof, wherein A is a substituted or unsubstituted 5-membered heterocyclic radical; X1 is S, O or NR1a, wherein R1a is selected from H, C1-C10-alkyl and the like; X2 is OR2a, NR2bR2c, S(O)mR2d; X2 is OR2a, NR2bR2c, S(O)mR2d, wherein m is 0, 1 or 2, R2a is C1-C4-alkyl, C1-C4-haloalkyl and the like, R2b, R2c are H, C1-C4-alkyl, C1-C4-haloalkyl and the like; X3 is a lone pair or oxygen; R1, R2 and R3 are, inter alia, hydrogen, and R1 is H, C1-C10-alkyl and the like. The present invention further relates to a method for controlling invertebrate pests, to a method for protecting plant propagation material and/or the plants which grow therefrom, to plant propagation material, comprising at least one compound according to the present invention, to a method for treating or protecting an animal from infestation or infection by parasites and to an agricultural composition containing at least one compound according to the present invention.

摘要翻译： 本发明涉及式I或II化合物及其盐和N-氧化物的方法和用途，其中A是取代或未取代的5元杂环基; X1是S，O或NR1a，其中R1a选自H，C1-C10-烷基等; X2是OR2a，NR2bR2c，S（O）mR2d; X2是OR2a，NR2bR2c，S（O）mR2d，其中m是0,1或2，R2a是C1-C4-烷基，C1-C4-卤代烷基等，R2b，R2c是H，C1-C4-烷基， C1-C4卤代烷基等; X3是孤对或氧气; R1，R2和R3尤其是氢，R1是H，C1-C10-烷基等。 本发明还涉及一种控制无脊椎害虫的方法，一种用于保护植物繁殖材料和/或从其生长的植物的方法，包括至少一种根据本发明的化合物的植物繁殖材料的方法， 治疗或保护动物免受寄生虫侵袭或感染，以及含有至少一种本发明化合物的农药组合物。

公开(公告)号：US20130203821A1

公开(公告)日：2013-08-08

申请号：US13821745

申请日：2011-09-12

申请人： Sebastian Soergel ,  Christian Defieber ,  Ronan Le Vezouet ,  Steffen Gross ,  Karsten Koerber ,  Deborah L. Culbertson ,  Douglas D. Anspaugh

发明人： Sebastian Soergel ,  Christian Defieber ,  Ronan Le Vezouet ,  Steffen Gross ,  Karsten Koerber ,  Deborah L. Culbertson ,  Douglas D. Anspaugh

IPC分类号： A01N43/82 ,  A01N43/653 ,  A01N43/647 ,  C07D417/12 ,  C07D401/12

CPC分类号： A01N43/82 ,  A01N43/40 ,  A01N43/50 ,  A01N43/56 ,  A01N43/647 ,  A01N43/653

摘要： The present invention relates to novel pyridine compounds of the formulae I and II, to their salts, to their tautomers, to their N-oxides, and to the salts of these N-oxides or tautomers. The compounds are useful for combating or controlling invertebrate pests, in particular arthropod pests. The invention also relates to a method for controlling in-vertebrate pests by using these compounds. The invention further relates to plant propagation material and to agricultural compositions comprising said compounds. wherein A is a radical of the formulae A1, A2, A3, A4, A5 or A6 wherein # denotes the binding site to the remainder of formulae I or II; Z is O, S or N—RN; X1 is S, O or NR1a; X2 is OR2a, NR2bR2c, S(O)mR2d; X3 is a lone pair or oxygen; R1, R2 and R3 are, inter alia, hydrogen, and RA1, RA2RA3RA4, RA5, RA6 and RN, are as defined in claim 1.

摘要翻译： 本发明涉及式I和II的新型吡啶化合物，其盐，其互变异构体，其N-氧化物，以及这些N-氧化物或互变异构体的盐。 这些化合物可用于对抗或控制无脊椎害虫，特别是节肢动物害虫。 本发明还涉及通过使用这些化合物来控制脊椎动物害虫的方法。 本发明还涉及植物繁殖材料和包含所述化合物的农业组合物。 其中A是式A1，A2，A3，A4，A5或A6的基团，其中＃表示与式I或II的其余部分的结合位点; Z是O，S或N-RN; X1是S，O或NR1a; X2是OR2a，NR2bR2c，S（O）mR2d; X3是孤对或氧气; R1，R2和R3尤其是氢，RA1，RA2RA3RA4，RA5，RA6和RN如权利要求1中所定义。

公开(公告)号：US08710056B2

公开(公告)日：2014-04-29

申请号：US13382229

申请日：2010-07-01

申请人： Ronan Le Vezouet ,  Sebastian Soergel ,  Christian Defieber ,  Steffen Gross ,  Karsten Koerber ,  Deborah L. Culbertson ,  Douglas D. Anspaugh

发明人： Ronan Le Vezouet ,  Sebastian Soergel ,  Christian Defieber ,  Steffen Gross ,  Karsten Koerber ,  Deborah L. Culbertson ,  Douglas D. Anspaugh

IPC分类号： A01N43/58 ,  A61K31/50 ,  A01N43/80 ,  A01N25/00 ,  A01N43/08 ,  A01N43/10 ,  C07D207/20 ,  C07D327/02 ,  C07D275/02 ,  C07D277/18 ,  C07D417/12 ,  C07D261/18 ,  C07D261/02 ,  A61K31/42

CPC分类号： C07D417/12 ,  A01N43/80 ,  A01N53/00 ,  C07D413/12

摘要： The present invention relates to pyridazine compounds of formulae I or II and the salts and N-oxides thereof, wherein A is a substituted or unsubstituted isoxazole or isothiazole radical; V is C(Rv) or N; W is C(Rw) or N; with the proviso that either V or W is N; Rt, Ru, Rv, Rw are H, halogen, C1-C4-alkyl and the like; X1 is S, O or NR1a, wherein R1a is selected H, C1-C10-alkyl and the like; X2 is OR2a, NR2bR2c, S(O)mR2d, wherein m is 0, 1 or 2, R2a is C1-C4-alkyl, C1-C4-haloalkyl and the like, R2b, R2c are H, C1-C4-alkyl, C1-C4-haloalkyl and the like, or R2b and R2c together with the nitrogen atom to which they are bound form a heterocycle, and R2d is C1-C4-alkyl, C1-C4-haloalkyl, C3-C6-cycloalkyl and the like; and R1 is H, CN, C1-C10-alkyl and the like. The present invention further relates to a method for controlling invertebrate pests, to a method for protecting plant propagation material and/or the plants which grow therefrom, to plant propagation material, comprising at least one compound according to the present invention, to a method for treating or protecting an animal from infestation or infection by parasites and to an agricultural composition containing at least one compound according to the present invention.

摘要翻译： 本发明涉及式I或II的哒嗪化合物及其盐和N-氧化物，其中A是取代或未取代的异恶唑或异噻唑基; V是C（Rv）或N; W是C（Rw）或N; 条件是V或W为N; R 1，R u，R v，R w为H，卤素，C 1 -C 4 - 烷基等; X1是S，O或NR1a，其中R1a选自H，C1-C10-烷基等; X2是OR2a，NR2bR2c，S（O）mR2d，其中m是0,1或2，R2a是C1-C4-烷基，C1-C4-卤代烷基等，R2b，R2c是H，C1-C4-烷基， C1-C4卤代烷基等，或R2b和R2c与它们所结合的氮原子一起形成杂环，R2d是C1-C4-烷基，C1-C4卤代烷基，C3-C6-环烷基等 ; R1为H，CN，C1-C10-烷基等。 本发明还涉及一种控制无脊椎害虫的方法，一种用于保护植物繁殖材料和/或从其生长的植物的方法，包括至少一种根据本发明的化合物的植物繁殖材料的方法， 治疗或保护动物免受寄生虫侵袭或感染，以及含有至少一种本发明化合物的农药组合物。