Aniline type compounds
    1.
    发明授权
    Aniline type compounds 有权
    苯胺型化合物

    公开(公告)号:US09006485B2

    公开(公告)日:2015-04-14

    申请号:US14236362

    申请日:2012-08-10

    摘要: The present invention relates to compounds of the formula (I) wherein R1 and R2 independently of one another are hydrogen, C1-C10-alkyl, C1-C10-haloalkyl, C3-C10-cycloalkyl, C3-C10-halocycloalkyl, C2-C10-alkenyl, C2-C10-haloalkenyl or together represent an aliphatic chain, or the like; R3 is halogen, cyano, C1-C8-alkyl, C1-C8-haloalkyl, C3-C8-cycloalkyl, C3-C8-halocycloalkyl, C2-C8-alkenyl, C2-C8-haloalkenyl, C1-C8-alkoxy, phenyl, or the like; R4 is hydrogen, C1-C10-alkyl, C1-C10-haloalkyl, C3-C8-cycloalkyl, C3-C8-halocycloalkyl, C2-C10-alkenyl, C2-C10-haloalkenyl, phenyl, or the like; t is 0 or 1; p is 0, 1, 2, 3 or 4. The present invention also relates to a process for preparing a compound of the formula (I) which comprises reacting a compound of the formula II with a compound of the formulae III or IV: where t, p, R1 R3, R3 and R4 are as defined in any of claims 1 to 6 and where A− is an equivalent of an anion having a pKB of at least 10 (determined under standard conditions in water).

    摘要翻译: 本发明涉及式(I)化合物,其中R 1和R 2彼此独立地是氢,C 1 -C 10 - 烷基,C 1 -C 10 - 卤代烷基,C 3 -C 10 - 环烷基,C 3 -C 10 - 卤代环烷基,C 2 -C 10 烯基,C 2 -C 10 - 卤代链烯基或一起代表脂族链等; R3是卤素,氰基,C1-C8-烷基,C1-C8-卤代烷基,C3-C8-环烷基,C3-C8-卤代环烷基,C2-C8-烯基,C2-C8-卤代烯基,C1-C8-烷氧基,苯基, 或类似物; R4是氢,C1-C10-烷基,C1-C10-卤代烷基,C3-C8-环烷基,C3-C8-卤代环烷基,C2-C10-烯基,C2-C10-卤代烯基,苯基等; t为0或1; 本发明还涉及制备式(I)化合物的方法,其包括使式II化合物与式III或IV化合物反应:其中 t,p,R 1,R 3,R 3和R 4如权利要求1至6中任一项所定义,其中A-是pKB为至少10(在水中标准条件下测定)的阴离子的当量。

    Pesticidal Active Mixtures Comprising Aminothiazoline Compounds
    2.
    发明申请
    Pesticidal Active Mixtures Comprising Aminothiazoline Compounds 失效
    包括氨基噻唑啉化合物的杀虫活性混合物

    公开(公告)号:US20110224075A1

    公开(公告)日:2011-09-15

    申请号:US12934461

    申请日:2009-03-24

    摘要: The present invention relates to pesticidal mixtures comprising as active compounds 1) at least one aminothiazoline compound I of formula I: wherein R1 is selected from hydrogen, COCH3, COCH2CH3 or COCH2C(CH3)3; R2 and R3 together with the carbon atoms of the phenyl ring to which they are attached form a ring which, depending on the tautomeric formula I a) or b) is depicted as: a benzene ring, a saturated 5-, 6-, or 7-membered carbocycle, a partially unsaturated 5-, 6-, or 7-membered carbocycle, a 5-, 6-, or 7-membered saturated heterocycle, a partially unsaturated 5-, 6-, or 7-membered heterocycle, which heterocycles contain 1, 2, or 3 heteroatoms selected from O, S and N as ring members, and a 5- or 6-membered heteroaromatic ring which contains 1, 2, or 3 heteroatoms selected from O, S and N as ring members, and wherein the ring is unsubstituted or may carry any combination of 1, 2, 3, or 4 radicals selected from the group consisting of halogen, CH3, CH2CH3, CF3, CH3O, cyano and (═O) (oxo); R4 is selected from hydrogen, fluoro, chloro, bromo, CF3, CH3O or CH3; R5, R6 are selected from hydrogen, chloro, fluoro, bromo, CH3, CH3O or CF3, wherein at least one of R5 or R6 is not hydrogen; with the proviso that R2 and R3 together do not form a —OCH2—O— or a —OCF2O-group; or the tautomers, enantiomers, diastereomers or salts thereof, and 2) at least one active compound II selected from group A as defined in the description, use of these mixtures for combating insects, acarids, or nematodes, and a method for treating, controlling, preventing or protecting animals against infestation or infection by parasites using these mixtures.

    摘要翻译: 本发明涉及包含作为活性化合物的杀虫混合物1)至少一种式I的氨基噻唑啉化合物I:其中R 1选自氢,COCH 3,COCH 2 CH 3或COCH 2 C(CH 3)3; R2和R3与它们所连接的苯环的碳原子一起形成环,其取决于互变异构体式a a)或b)被描述为:苯环,饱和的5-,6-或 7元碳环,部分不饱和5-,6-或7-元碳环,5-,6-或7-元饱和杂环,部分不饱和5-,6-或7-元杂环,其中 杂环含有选自O,S和N作为环成员的1,2或3个杂原子,以及含有1,2或3个选自O,S和N作为环成员的杂原子的5或6元杂芳环, 并且其中所述环是未取代的或可以携带选自卤素,CH 3,CH 2 CH 3,CF 3,CH 3 O,氰基和(= O)(氧代)的1,2,3或4个基团的任何组合。 R4选自氢,氟,氯,溴,CF 3,CH 3 O或CH 3; R5,R6选自氢,氯,氟,溴,CH3,CH3O或CF3,其中R5或R6中的至少一个不是氢; 条件是R2和R3一起不形成-OCH2-O-或-OCF2O-基团; 或其互变异构体,对映异构体,非对映异构体或其盐,以及2)选自如说明书中定义的组A的至少一种活性化合物II,这些混合物用于防治昆虫,螨虫或线虫的用途,以及治疗,控制 ,防止或保护动物免受使用这些混合物的寄生虫的感染或感染。

    Indanyl- and Tetrahydronaphthyl-Amino-Azoline Compounds for Combating Animal Pests
    8.
    发明申请
    Indanyl- and Tetrahydronaphthyl-Amino-Azoline Compounds for Combating Animal Pests 失效
    茚基和四氢萘基 - 氨基 - 唑啉化合物,用于防治动物害虫

    公开(公告)号:US20080293569A1

    公开(公告)日:2008-11-27

    申请号:US12094854

    申请日:2006-11-15

    摘要: The present invention relates to Indanyl- and Tetrahydronaphthyl-amino-azoline compounds of formula I wherein the variables R1 and R2 are as defined in description.The invention relates also to methods of combating or controlling insects, arachnids or nematodes, to methods for protecting growing plants from attack or infestation by insects, arachnids or nematodes, to methods for the protection of seeds from soil insects and of the seedlings' roots and shoots from soil and foliar insects and to methods for treating, controlling, preventing or protecting animals against infestation or infection by parasites.

    摘要翻译: 本发明涉及式I的茚满基和四氢萘基 - 氨基 - 唑啉化合物,其中变量R1和R2如描述中所定义。 本发明还涉及防治昆虫,蜘蛛或线虫的方法,用于保护生长植物免受昆虫,蜘蛛或线虫侵袭或侵染的方法,用于保护种子免受土壤昆虫和幼苗根部和 来自土壤和叶面昆虫的芽,以及用于治疗,控制,预防或保护动物免受寄生虫感染或感染的方法。