Fungicidal agents
    31.
    发明授权
    Fungicidal agents 失效
    杀真菌剂

    公开(公告)号:US4845111A

    公开(公告)日:1989-07-04

    申请号:US193437

    申请日:1988-05-12

    摘要: A fungicidal composition comprising a fungicidally effective amount of (i) a substituted 1-hydroxyethyl-triazole of the formula ##STR1## in which A is --CH.sub.2 CH.sub.2 -- or --CH.dbd.CH--or an addition product thereof with an acid or metal salt, and (ii) at least one member selected from the group consisting of(A) wettable sulphur(B) a polyhalogenoalkylthio derivative,(C) a guanidine derivative,(D) an aromatic carboxylic acid derivative,(E) a dithiocarbamate,(F) a benzimidazole derivative,(G) an imidazole or triazole derivative,(H) a phosphoric acid ester,(I) a tetrahydroquinoline derivative,(J) an S,N-heterocyclene compound,(K) a urea derivative,(L) a sulphonamide derivative,(M) a polyhydroxy ether derivative,(N) a triazine derivative,(O) a copper complex salt,(P) an N-formyl derivative,(Q) a morpholine derivative,(R) a quinoxaline derivative, and(S) a dicarboximide derivative.

    摘要翻译: 一种杀真菌组合物,其包含杀真菌有效量的(i)式​​为“IMAGE”的取代的1-羟乙基三唑,其中A为-CH 2 CH 2 - 或-CH = CH-或其与酸或金属盐的加成产物, 和(ii)选自(A)可湿性硫(B),多卤代烷硫基衍生物,(C)胍衍生物,(D)芳族羧酸衍生物,(E)二硫代氨基甲酸酯(F) )苯并咪唑衍生物,(G)咪唑或三唑衍生物,(H)磷酸酯,(I)四氢喹啉衍生物,(J)S,N-杂环烯化合物,(K)脲衍生物,(L) 磺酰胺衍生物,(M)多羟基醚衍生物,(N)三嗪衍生物,(O)铜络合盐,(P)N-甲酰基衍生物,(Q)吗啉衍生物,(R)喹喔啉衍生物, 和(S)二羧酰亚胺衍生物。

    Process for the preparation of 5-acylpyrimidines
    32.
    发明授权
    Process for the preparation of 5-acylpyrimidines 失效
    5-酰基嘧啶的制备方法

    公开(公告)号:US4806644A

    公开(公告)日:1989-02-21

    申请号:US33433

    申请日:1987-04-01

    摘要: A process for the preparation of a 5-acylpyrimidine of the formula ##STR1## in which R is an organic radical comprising reacting a methyl ketone of the formulaR--CO--Ch.sub.3 in a first stage with a formylating reagent in the presence of a base to form an enolketone of the formulaR--CO--CH.dbd.CH--OR.sup.10in whichR.sup.10 represents hydrogen or a base radical, thereafter reacting the enolketone in 2nd and 3rd stages with formamidine or a formamidine salt, and with an amino-formylating agent, and, in a 4th stage heating to cyclize the compound formed.The end products, some of which are new, are intermediates for making herbicides.

    摘要翻译: 制备式“IMAGE”的5-酰基嘧啶的方法,其中R是有机基团,其包括使第一阶段的式R-CO-Ch 3的甲基酮与甲酰化试剂在碱的存在下反应 形成式R-CO-CH = CH-OR10的烯醇,其中R 10表示氢或碱基,然后使第二和第三阶段的烯醇与甲脒或甲脒盐反应,并与氨基甲酰化试剂反应, 并且在第四阶段加热以使所形成的化合物环化。 最终产品,其中一些是新的,是制造除草剂的中间体。

    Process for the preparation of 5-acylpyrimidines
    33.
    发明授权
    Process for the preparation of 5-acylpyrimidines 失效
    5-酰基嘧啶的制备方法

    公开(公告)号:US4713456A

    公开(公告)日:1987-12-15

    申请号:US769639

    申请日:1985-08-26

    摘要: A process for the preparation of a 5-acylpyrimidine of the formula ##STR1## in which R is an organic radical comprising reacting a methyl ketone of the formulaR--CO--CH.sub.3in a first stage with a formylating reagent in the presence of a base to form an enolketone of the formulaR--CO--CH.dbd.CH--OR.sup.10in which R.sup.10 represents hydrogen or a base radical, thereafter reacting the enolketone in 2nd and 3rd stages with formamidine or a formamidine salt, and with an amino-formylating agent, and, in a 4th stage heating to cyclize the compound formed.The end products, some of which are new, are intermediates for making herbicides.

    摘要翻译: 一种制备式“IMAGE”的5-酰基嘧啶的方法,其中R是有机基团,其包括使第一阶段的式R-CO-CH 3的甲基酮与甲酰化试剂在碱的存在下反应 形成式R-CO-CH = CH-OR10的烯醇,其中R 10表示氢或碱基,然后使第二和第三阶段的烯醇与甲脒或甲脒盐反应,并与氨基甲酰化试剂反应, 并且在第四阶段加热以使所形成的化合物环化。 最终产品,其中一些是新的,是制造除草剂的中间体。

    Fungicidal agents
    38.
    发明授权
    Fungicidal agents 失效
    杀真菌剂

    公开(公告)号:US5250560A

    公开(公告)日:1993-10-05

    申请号:US968029

    申请日:1992-10-29

    摘要: A fungicidal composition comprising a fungicidally effective amount of (i) a substituted 1-hydroxyethyl-triazole of the formula ##STR1## in which A is --CH.sub.2 CH.sub.2 -- or --CH.dbd.CH--,or an addition product thereof with an acid or metal salt, and (ii) at least one member selected from the group consisting ofA) wettable sulphur,B) a polyhalogenoalkylthio derivative,C) a quanidine derivative,D) an aromatic carboxylic acid derivative,E) a dithiocarbamate,F) a benzimidazole derivative,G) an imidazole or triazole derivative,H) a phosphoric acid ester,I) a tetrahydroquinoline derivative,J) an S,N-heterocyclene compound,K) a urea derivative,L) a sulphonamide derivative,M) a polyhydroxy ether derivative,N) a triazine derivative,O) a copper complex salt,P) an N-formyl derivative,Q) a morpholine derivative,R) a quinoxaline derivative, andS) a dicarboximide derivative.

    摘要翻译: 一种杀真菌组合物,其包含杀真菌有效量的(i)其中A是-CH 2 CH 2 - 或-CH = CH-的式“IMAGE”的取代的1-羟乙基三唑或其与酸或金属盐的加成产物 ,和(ii)至少一种选自A)可湿性硫,B)多卤代烷硫基衍生物,C)喹啉衍生物,D)芳族羧酸衍生物,E)二硫代氨基甲酸酯,F)苯并咪唑衍生物 ,G)咪唑或三唑衍生物,H)磷酸酯,I)四氢喹啉衍生物,J)S,N-杂环烯化合物,K)脲衍生物,L)磺酰胺衍生物,M)多羟基醚衍生物 ,N)三嗪衍生物,O)铜络合盐,P)N-甲酰基衍生物,Q)吗啉衍生物,R)喹喔啉衍生物和S)二羧酰亚胺衍生物。

    Fungicidal agents
    40.
    发明授权
    Fungicidal agents 失效
    杀真菌剂

    公开(公告)号:US5137903A

    公开(公告)日:1992-08-11

    申请号:US762274

    申请日:1991-09-19

    摘要: A fungicidal composition comprising a fungicidally effective amount of (i) a substituted 1-hydroxyethyl-triazole of the formula ##STR1## in whichA is --CH.sub.2 CH.sub.2 -- or CH.dbd.CH--,or an addition product thereof with an acid or metal salt, and (ii) at least one member selected from the group consisting ofA) wettable sulphur,B) a polyhalogenoalkylthio derivative,C) a quanidine derivative,D) an aromatic carboxylic acid derivative,E) a dithiocarbamate,F) a benzimidazole derivative,G) an imidazole or triazole derivative,H) a phosphoric acid ester,I) a tetrahydroquinoline derivative,J) an S,N-heterocyclene compound,K) a urea derivative,L) a sulphonamide derivative,M) a polyhydroxy ether derivative,N) a triazine derivative,O) a copper complex salt,P) an N-formyl derivative,Q) a morpholine derivative,R) a quinoxaline derivative, andS) a dicarboximide derivative.

    摘要翻译: 一种杀真菌组合物,其包含杀真菌有效量的(i)其中A是-CH 2 CH 2 - 或CH = CH-的式IMAMA的取代的1-羟乙基三唑或其与酸或金属盐的加成产物, 和(ii)至少一种选自A)可湿性硫,B)多卤代烷硫基衍生物,C)喹啉衍生物,D)芳族羧酸衍生物,E)二硫代氨基甲酸酯,F)苯并咪唑衍生物, G)咪唑或三唑衍生物,H)磷酸酯,I)四氢喹啉衍生物,J)S,N-杂环烯化合物,K)脲衍生物,L)磺酰胺衍生物,M)多羟基醚衍生物, N)三嗪衍生物,O)铜络合盐,P)N-甲酰基衍生物,Q)吗啉衍生物,R)喹喔啉衍生物,和S)二羧酰亚胺衍生物。