摘要:
Herbicidal substituted sulphonylaminotriazolinones of the formula ##STR1## in which R.sup.1 represents an optionally substituted radical from the group consisting of alkyl, aralkyl, aryl and heteroaryl,R.sup.2 represents hydrogen or the group --SO.sub.2 --R.sup.1 where R.sup.1 has the abovementioned meaning,R.sup.3 represents hydrogen, halogen, hydroxyl, mercapto, amino or an optionally substituted radical from the group consisting of alkyl, cycloalkyl, aralkyl, aryl, alkoxy, alkenyloxy, alkinyloxy, alkylthio, alkylsulphinyl, alkylsulphonyl, alkenylthio, alkinylthio, aralkoxy, aralkylthio, alkylamino and dialkylamino,R.sup.4 represents hydrogen, halogen, hydroxyl, amino or an optionally substituted radical from the group consisting of alkyl, alkoxy, alkylthio, alkylsulphinyl, alkylsulphonyl, alkylamino and dialkylamino,X represents nitrogen or a CH group,Y represents nitrogen or a CR.sup.5 group whereR.sup.5 represents hydrogen, halogen, cyano, alkyl, formyl, alkylcarbonyl or alkoxycarbonyl, andZ represents nitrogen or a CR.sup.6 group whereR.sup.6 represents hydrogen, halogen, hydroxyl, amino or an optionally substituted radical from the group consisting of alkyl, alkoxy, alkylthio, alkylsulphinyl, alkylsulphonyl, alkylamino and dialkylamino,and salts thereof. Intermediates of the formulas ##STR2## are also new.
摘要翻译:式(I)的除草取代的磺酰基氨基三唑啉酮,其中R 1表示由烷基,芳烷基,芳基和杂芳基组成的组中的任选取代的基团,R 2表示氢或基团-SO 2 -R 1,其中R 1具有上述含义, R 3表示氢,卤素,羟基,巯基,氨基或任选取代的基团,其由烷基,环烷基,芳烷基,芳基,烷氧基,烯氧基,烷氧基,烷硫基,烷基亚磺酰基,烷基磺酰基,链烯硫基,炔基硫基,芳烷氧基,芳烷硫基, 和二烷基氨基,R 4表示氢,卤素,羟基,氨基或任选取代的基团,其由烷基,烷氧基,烷硫基,烷基亚磺酰基,烷基磺酰基,烷基氨基和二烷基氨基,X表示氮或CH基,Y表示氮或CR 5 基团,其中R 5表示氢,卤素,氰基,烷基,甲酰基,烷基羰基或烷氧基羰基,Z表示氮或C R 6基团,其中R 6表示氢,卤素,羟基,氨基或任选取代的由烷基,烷氧基,烷硫基,烷基亚磺酰基,烷基磺酰基,烷基氨基和二烷基氨基组成的组的基团及其盐。 式(II)和(IMA)(IV)的中间体也是新的。
摘要:
Herbicidal substituted sulphonylaminotriazolinones of the formula ##STR1## in which R.sup.1 represents an optionally substituted radical from the group consisting of alkyl, aralkyl, aryl and heteroaryl,R.sup.2 represents hydrogen or the group --SO.sub.2 --R.sup.1 where R.sup.1 has the abovementioned meaning,R.sup.3 represents hydrogen, halogen, hydroxyl, mercapto, amino or an optionally substituted radical from the group consisting of alkyl, cycloalkyl, aralkyl, aryl, alkoxy, alkenyloxy, alkinyloxy, alkylthio, alkylsulphinyl, alkylsulphonyl, alkenylthio, alkinylthio, aralkoxy, aralkylthio, alkylamino and dialkylamino,R.sup.4 represents hydrogen, halogen, hydroxyl, amino or an optionally substituted radical from the group consisting of alkyl, alkoxy, alkylthio, alkylsulphinyl, alkylsulphonyl, alkylamino and dialkylamino,X represents nitrogen or a CH group,Y represents nitrogen or a CR.sup.5 group whereR.sup.5 represents hydrogen, halogen, cyano, alkyl, formyl, alkylcarbonyl or alkoxycarbonyl, andZ represents nitrogen or a CR.sup.6 group whereR.sup.6 represents hydrogen, halogen, hydroxyl, amino or an optionally substituted radical from the group consisting of alkyl, alkoxy, alkylthio, alkylsulphinyl, alkylsulphonyl, alkylamino and dialkylamino,and salts thereof. Intermediates of the formulas ##STR2## are also new.
摘要:
Novel herbicides of the formula ##STR1## in which R.sup.1 represents an organic radical,R.sup.2 represents hydrogen or an organic radical,R.sup.3 represents an organic radical or an amino radical,R.sup.4 represents hydrogen, an organic radical, an ether radical or an amino radical,X represents N or CH,Y and Z each represent N, CH or a substituted C radical, andM is H, a metal ion or an acyl radical, or a strong acid adduct thereof. Some intermediates are also new.
摘要:
Herbicidally active novel 1-(2-oxyaminosulphonylphenylsulphonyl)-3-heteroaryl-iso (thio)-ureas of the formula ##STR1## in which R is optionally substituted alkyl, alkenyl, alkinyl, cycloalkyl-alkyl, cycloalkyl, aralkyl, aryl or heteryl,R.sup.1 is optionally substituted alkyl, alkenyl, alkinyl, cycloalkyl, cycloalkyl-alkyl, aralkyl or aryl,R.sup.2 is hydrogen, or optionally substituted alkyl, alkenyl, alkinyl or aralkyl,R.sup.3 is an optionally substituted and/or optionally fused 6-membered aromatic heterocycle which contains at least one nitrogen atom, andQ is oxygen or sulphur,or strong acid-adducts thereof.
摘要:
The invention relates to novel sulphonylaminocarbonyltriazolinones of the formula (I), ##STR1## in which R.sup.1 represents hydrogen, hydroxyl, amino, alkylideneamino or a respectively optionally substituted radical from the group consisting of alkyl, alkenyl, alkinyl, alkylamino, dialkylamino, alkanoylamino, cycloalkyl, cycloalkylalkyl, cycloalkylamino, aryl, arylalkyl,R.sup.2 represents respectively halogen-substituted alkyl or alkenyl andR.sup.3 represents a respectively optionally substituted radical from the group consisting of alkyl, aralkyl, aryl, heteroaryl,and to salts of compounds of the formula (I), to processes and novel intermediates for preparing the compounds (I) and to their use as herbicides and/or fungicides.
摘要:
The invention relates to novel sulphonylaminocarbonyltriazolinones of the formula (I), ##STR1## in which R.sup.1 represents hydrogen, hydroxyl, amino, alkylideneamino or a respectively optionally substituted radical from the group consisting of alkyl, alkenyl, alkinyl, alkylamino, dialkylamino, alkanoylamino, cycloalkyl, cycloalkylalkyl, cycloalkylamino, aryl, arylalkyl,R.sup.2 represents respectively halogen-substituted alkyl or alkenyl andR.sup.3 represents a respectively optionally substituted radical from the group consisting of alkyl, aralkyl, aryl, heteroaryl,and to salts of compounds of the formula (I), to processes and novel intermediates for preparing the compounds (I) and to their use as herbicides and/or fungicides.
摘要:
The invention relates to novel sulphonylaminocarbonyltriazolinones having halogenoalkoxy substituents of the formula (I) ##STR1## in which R.sup.1 represents hydrogen, hydroxyl, amino, alkylideneamino or a respectively optionally substituted radical from the group consisting of alkyl, alkenyl, alkynyl, alkoxy, alkenyloxy, alkylamino, dialkylamino, alkanoylamino, cycloalkyl, cycloalkylalkyl, cycloalkylamino, aryl and arylalkyl,R.sup.2 represents respectively halogen-substituted alkyl or alkenyl, andR.sup.3 represents a respectively optionally substituted radical from the group consisting of alkyl, aralkyl, aryl and heteroaryl,and salts of compounds of the formula (I), and to processes and novel intermediates for preparing the compounds (I), and to their use as herbicides and/or fungicides.
摘要:
The invention relates to novel substituted arylsulphonyl(thio)ureas in which A represents nitrogen or a CH grouping, Q represents oxygen or sulphur, R1 represents hydrogen, halogen or respectively optionally substituted alkyl, alkoxy, alkylthio, alkylamino, dialkylamino, cycloalkyl, cycloalkyloxy or heterocyclyloxy, R2 represents hydrogen, halogen or respectively optionally substituted alkyl, alkoxy, alkylthio, alkylamino, dialkylamino, cycloalkyl, cycloalkyloxy or heterocyclyloxy, R3 represents hydrogen or optionally substituted alkyl, R4 represents respectively optionally substituted alkyl, alkoxy, alkenyl, alkinyl, alkenyloxy, alkinyloxy, cycloalkyl, cycloalkyloxy or cycloalkylalkyl, and R5 represents hydrogen, formyl or respectively optionally substituted alkyl, alkylcarbonyl, alkoxycarbonyl, alkylsulphonyl, alkenyl, alkinyl, cycloalkyl, cycloalkylcarbonyl, cycloalkylsulphonyl or heterocyclyl, and to salts of compounds of the formula (I), except for the compound N-(4,6-dimethyl-pyrimidin-2-yl)-N′-[2-(1,1,2,2-tetrafluoro-ethoxy)-6-methyl-phenylsulphonyl]-urea, to processes for preparing the novel compounds and to their use as herbicides.
摘要:
A process for the preparation of a 1-(2-oxyaminosulphonyl-phenylsulphonyl)-urea of the formula ##STR1## in which R.sup.1 is an optionally substituted radical from the series comprising alkyl, alkenyl, alkinyl, cycloalkyl, cycloalkylalkyl, aralkyl and aryl,R.sup.2 is hydrogen or an optionally substituted radical from the series comprising alkyl, alkenyl, alkinyl and aralkyl, andR.sup.3 is an optionally substituted and/or optionally fused six-membered aromatic heterocyclic radical containing at least one nitrogen atom,comprising reacting water with a benzodisultam of the formula ##STR2## at a temperature between 0.degree. C. and 100.degree. C. The products are herbicidally active.
摘要翻译:一种制备式(IMAGE)的1-(2-氧氨基磺酰基 - 苯基磺酰基) - 脲的方法,其中R 1是包含烷基,链烯基,炔基,环烷基,环烷基烷基,芳烷基和芳基的任意取代的基团, R 2是氢或任选取代的基团,其包含烷基,链烯基,炔基和芳烷基,并且R 3是任选被取代的和/或任选地稠合的含有至少一个氮原子的六元芳族杂环基团,包括使水与苯并二枯基 在0℃至100℃之间的温度下,该产物具有除草活性。
摘要:
A process for the preparation of a sulphonyliso(thio)urea of the formula ##STR1## in which R.sup.1 represents an optionally substituted radical from the group consisting of alkyl, aralkyl, aryl and heteroaryl,R.sup.2 represents an optionally substituted and/or optionally fused, six-membered aromatic heterocycle containing at least one nitrogen atom,R.sup.3 represents an optionally substituted radical from the group consisting of alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkyl-alkyl and aralkyl, andQ represents oxygen or sulphur,comprising reacting a sulphonylguanidine of the formula ##STR2## in which R.sup.4 represents an optionally substituted hydrocarbon radical,with a compound of the formulaH--Q--R.sup.3at a temperature between 0.degree. C. and 150.degree. C. The products are known herbicides.