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41.发明授权公开(公告)号：US08980931B1
公开(公告)日：2015-03-17
申请号：US14263293
申请日：2014-04-28
发明人： Takaaki Masuda , Hiroshi Yamaguchi
IPC分类号： A61K31/4178 , C07D409/06 , G01N30/02
CPC分类号： C07D409/06 , A61K9/08 , A61K31/4178 , A61K47/34 , G01N30/02 , G01N2030/027 , G01N2030/8813
摘要： Disclosed is a method of evaluating stability of a pharmaceutical preparation containing luliconazole. The method includes measuring an amount of production of an SE form of luliconazole represented by following formula (2), an amount of production of a Z form of luliconazole represented by following formula (3) and an amount of production of an amide form of luliconazole represented by following formula (1) after storage under a severe condition or an accelerated condition, and judging that the stability of the pharmaceutical preparation is high if each of the amount of production of the SE form, the amount of production of the Z form and the amount of production of the amide form is not more than 5% by weight with respect to a compounded amount of luliconazole.
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公开(公告)号：US08835479B2
公开(公告)日：2014-09-16
申请号：US13866876
申请日：2013-04-19
发明人： Hiroyasu Koga , Yasuko Nanjoh , Hideo Kaneda
IPC分类号： A61K31/4178 , C07D233/00 , A61K47/10 , A61K47/34 , A61K9/00 , C07D409/06 , A61K47/14 , A61K47/36
CPC分类号： A61K31/4178 , A61K9/0014 , A61K47/10 , A61K47/14 , A61K47/34 , A61K47/36 , C07D409/06
摘要： The invention provides a method for the treatment of fungal dermatitis. The treatment method involves administering an effective amount of luliconazole or a pharmaceutically acceptable salt thereof to a target in need of a treatment of fungal dermatitis.
摘要翻译： 本发明提供了一种治疗真菌性皮炎的方法。 治疗方法包括将有效量的利咯康唑或其药学上可接受的盐给予需要治疗真菌性皮炎的靶标。
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公开(公告)号：US6410574B2
公开(公告)日：2002-06-25
申请号：US36208799
申请日：1999-07-28
申请人： NIHON NOHYAKU CO LTD
IPC分类号： A01N43/42 , A01N43/54 , A01N43/653 , A01N43/82 , A01N43/828 , A01N43/90 , A01N47/04 , A01N47/14 , A01N47/18 , A01N47/34 , A01N47/38 , A01N47/44 , A01N57/20 , A01P3/00 , A01N37/00 , A01N43/00 , A01N47/00 , A01N55/02
CPC分类号： A01N43/82 , A01N61/00 , A01N59/20 , A01N47/38 , A01N43/90 , A01N43/653 , A01N43/54 , A01N43/28 , A01N2300/00
摘要： The present invention relates to a fungicidal composition obtained by mixing a 1,2,3-thiadiazole derivative of general formula (I) useful as a plant disease controller with at least one fungicide selected from the compounds having a fungicidal activity against plant diseases, and to a method for using the same:wherein R1 is hydrogen, alkyl or cycloalkyl and R2 is CO-Y-R3, wherein Y is O, S, NR4 or the like and R3 is hydrogen, alkyl, phenyl, 5- or 6-membered heterocycle or the like.
摘要翻译： 本发明涉及通过将可用作植物病害防治剂的通式（I）的1,2,3-噻二唑衍生物与至少一种选自对植物病害具有杀真菌活性的化合物的杀真菌剂混合而获得的杀真菌组合物，以及 涉及其使用方法：其中R1是氢，烷基或环烷基，R2是CO-Y-R3，其中Y是O，S，NR4等，R3是氢，烷基，苯基，5-或6- 元杂环等。
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公开(公告)号：US20230234951A1
公开(公告)日：2023-07-27
申请号：US17930882
申请日：2022-09-09
发明人： Bart HERLÉ , Hannes Fiepko KOOLMAN , Alan LONG , Robin MEIER , Ikki YONEMURA , Julien Gagnepain
IPC分类号： C07D471/04 , C07D487/04 , C07D413/04 , C07D413/14 , C07D498/04 , C07D401/04 , C07D513/04 , C07D417/04 , C07D401/14
CPC分类号： C07D471/04 , C07D487/04 , C07D413/04 , C07D413/14 , C07D498/04 , C07D401/04 , C07D513/04 , C07D417/04 , C07D401/14
摘要： The present invention relates to cyclopropyl-(hetero)aryl substituted ethylsulphonyl-pyridine derivatives of formula (I)
wherein the variables are as defined in the description and in the claims, which can be used as antiparasitic agents for the treatment, prevention and/or control of parasitic infections and/or infestations in animals.-
公开(公告)号：US20220287308A1
公开(公告)日：2022-09-15
申请号：US17631348
申请日：2020-08-06
IPC分类号： A01N43/90 , C07D498/14 , A01P7/04
摘要： A compound, or a salt thereof, is expressed by General Formula (1): wherein R represents a (C1-C6) alkoxy (C1-C6) alkyl group, which is useful as an agricultural and horticultural insecticide with reduced harmful effects to animals including humans in production of agricultural, horticultural and other crops.
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公开(公告)号：US11311013B2
公开(公告)日：2022-04-26
申请号：US17057563
申请日：2019-05-22
发明人： Hirokazu Fujihara , Yutaka Abe , Ryosuke Tanaka , Shunsuke Fuchi
IPC分类号： A01N43/52 , A61P33/10 , C07D401/04
摘要： The present invention has an object to develop and provide a novel agricultural and horticultural insecticidal and acaricidal agent due to the factors such as serious damages caused by pests and the like and growing resistant pests against existing drugs in the crop production such as agriculture and horticulture.
The present invention provides an agricultural and horticultural insecticidal and acaricidal agent having as an active ingredient a benzimidazole compound represented by general formula (1) wherein R represents an alkyl group or the like, R1 represents a haloalkyl group or the like, X represents an oxygen atom or the like, m and n represent 0 or the like, or a salt thereof, and a method for using the same.-
公开(公告)号：US20210204545A1
公开(公告)日：2021-07-08
申请号：US17057563
申请日：2019-05-22
发明人： Hirokazu FUJIHARA , Yutaka ABE , Ryosuke TANAKA , Shunsuke FUCHI
IPC分类号： A01N43/52 , C07D401/04 , A61P33/10
摘要： The present invention has an object to develop and provide a novel agricultural and horticultural insecticidal and acaricidal agent due to the factors such as serious damages caused by pests and the like and growing resistant pests against existing drugs in the crop production such as agriculture and horticulture.
The present invention provides an agricultural and horticultural insecticidal and acaricidal agent having as an active ingredient a benzimidazole compound represented by general formula (1) wherein R represents an alkyl group or the like, R1 represents a haloalkyl group or the like, X represents an oxygen atom or the like, m and n represent 0 or the like, or a salt thereof, and a method for using the same.-
公开(公告)号：US20210000111A1
公开(公告)日：2021-01-07
申请号：US16976436
申请日：2019-03-01
发明人： Keiichi Yamada , Yutaka Abe , Yutaka Kato , Ayuko Nakauchi , Yuki Saito , Shunsuke Fuchi
IPC分类号： A01N43/10 , C07D307/66 , C07D333/36 , A01N43/08 , C07D307/68 , C07D409/04 , A01N43/40 , C07D207/34 , A01N43/36
摘要： An amide compound represented by the general formula [I]: or a salt thereof, an agricultural and horticultural microbicide comprising the compound or the salt as an active ingredient, and a method for using the agricultural and horticultural microbicide.
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公开(公告)号：US10575525B2
公开(公告)日：2020-03-03
申请号：US16077978
申请日：2017-02-24
发明人： Soichiro Matsuo , Ikki Yonemura , Akiyuki Suwa , Shunpei Fujie
IPC分类号： A01N43/76 , C07D413/14 , C07D413/04 , A01N47/02 , A61K31/4439
摘要： In crop production in the fields of agriculture, horticulture and the like, the damage caused by insect pests etc. is still immense, and insect pests resistant to existing insecticides have emerged. To solve the problems, the present invention has been made, and an object of the present invention is to develop and provide a novel agricultural and horticultural insecticide.The present invention provides a benzoxazole compound represented by the general formula (1): {wherein R1 represents a trifluoromethoxy group or a trifluoromethylsulfinyl group, R2 represents a hydrogen atom, and m represents 2}, or a salt thereof; an agricultural and horticultural insecticide comprising the compound or a salt thereof as an active ingredient; and a method for using the insecticide.
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公开(公告)号：US20200048247A1
公开(公告)日：2020-02-13
申请号：US16340661
申请日：2017-10-12
发明人： Ikki Yonemura , Naoto Shimizu , Akiyuki Suwa , Shunpei Fujie
IPC分类号： C07D471/04 , A01N43/40
摘要： In crop production in the fields of agriculture, horticulture and the like, the damage caused by insect pests etc. is still immense, and insect pests resistant to existing insecticides have emerged. Under such circumstances, the development of novel agricultural and horticultural insecticides is desired. The present invention provides an agricultural and horticultural insecticide comprising a 1H-pyrrolo-condensed heterocyclic compound represented by the general formula (1): {wherein A and A1 each represent a nitrogen atom, R3 and R4 each represent a haloalkyl group, R2 represents a hydrogen atom or an acetyl group, R1 represents a halogen atom, and m represents 0 or 2}, an N-oxide thereof or a salt thereof as an active ingredient, and a method for using the insecticide.
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