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    MICROBIOCIDES
    41.
    发明申请
    MICROBIOCIDES 失效

    公开(公告)号：US20090054496A1

    公开(公告)日：2009-02-26

    申请号：US12092338

    申请日：2005-11-13

    申请人： Harald Walter ,  Camilla Corsi ,  Josef Ehrenfreund ,  Hans Tobler

    发明人： Harald Walter ,  Camilla Corsi ,  Josef Ehrenfreund ,  Hans Tobler

    IPC分类号： A01N43/40 ,  C07D231/10 ,  A01N43/56 ,  C07D207/00 ,  A01N43/36 ,  C07D249/04 ,  A01N43/64 ,  C07D277/00 ,  A01N43/78 ,  C07D213/56

    CPC分类号： A01N43/36 ,  A01N43/40 ,  A01N43/56 ,  A01N43/78 ,  A01N43/84 ,  C07C211/45 ,  C07C211/52 ,  C07C2601/02 ,  C07C2601/04 ,  C07D207/34 ,  C07D213/82 ,  C07D231/14 ,  C07D249/04 ,  C07D277/56 ,  C07D327/06

    摘要： The invention relates to a fungicidally active compound of the general Formula (I): where Het is a 5- or 6-membered heterocyclic ring containing one to three heteroatoms, each independently selected from oxygen, nitrogen and sulphur, the ring being substituted by the groups R3, R4 and R5; R1 and R2 are independently H, halo, C1-4 alkyl or C1-4 haloalkyl; and R3, R4 and R5 are each, independently, H, halo, C1-4 alkyl, C1-4 haloalkyl or C1-4 haloalkoxy, provided that at least one of R3, R4 and R5 is not H; to the preparation of these compounds, to novel intermediates used in their preparation, to agrochemical compositions which comprise at least one of the novel compounds as an active ingredient, to the preparation of the compositions and to the use of the active ingredients or compositions in agriculture or horticulture for controlling or preventing infestations of plants by phytopathogenic microorganisms, especially fungi.

    摘要翻译： 本发明涉及通式（I）的杀真菌活性化合物：其中Het是含有一至三个杂原子的5-或6-元杂环，各自独立地选自氧，氮和硫，所述环被 基团R3，R4和R5; R 1和R 2独立地为H，卤素，C 1-4烷基或C 1-4卤代烷基; 并且R 3，R 4和R 5各自独立地为H，卤素，C 1-4烷基，C 1-4卤代烷基或C 1-4卤代烷氧基，条件是R 3，R 4和R 5中的至少一个不为H; 涉及这些化合物的制备，其制备中使用的新型中间体，包含至少一种新化合物作为活性成分的农用化学组合物，用于制备组合物以及在农业中使用活性成分或组合物 或园艺用于通过植物病原微生物，特别是真菌控制或预防植物侵染。

    3-carbonylaminothiophenes and their use as fungicides
    42.
    发明授权
    3-carbonylaminothiophenes and their use as fungicides 失效
    3-羰基氨基噻吩及其作为杀真菌剂的用途

    公开(公告)号：US07582589B2

    公开(公告)日：2009-09-01

    申请号：US10554336

    申请日：2004-04-21

    申请人： Josef Ehrenfreund ,  Harald Walter ,  Hans Tobler ,  Clemens Lamberth

    发明人： Josef Ehrenfreund ,  Harald Walter ,  Hans Tobler ,  Clemens Lamberth

    IPC分类号： A01N43/56 ,  C07D231/10

    CPC分类号： C07D409/12 ,  A01N55/00 ,  C07D333/28 ,  C07D333/36 ,  C07D411/12 ,  C07D413/12 ,  C07D417/12

    摘要： The invention also relates to novel compounds of formula (1) where Het is a 5- or 6-membered heterocyclic ring containing one to three heteroatoms, each independently selected from oxygen, nitrogen and sulphur, the ring being substituted by one to three groups R4; R1 is hydrogen, optionally substituted (C1-4)alkyl, formyl, optionally substituted (C1-4)alkylC(═O), optionally substituted (C1-4)alkylC(═O)O, optionally substituted (C1-4)alkoxy(C1-4)alkyl, optionally substituted allyl, optionally substituted propargyl or optionally substituted allenyl; each R2 is, independently, halogen, optionally substituted (C1-4)alkyl, optionally substituted (C1-4)alkoxy or optionally substituted (C1-4)alkoxy(C1-4)alkyl; R3 is either at position 2 or at position 4 of the thiophene ring and is an organic group containing three to thirteen carbon atoms and at least one silicon atom and, optionally, one to three heteroatoms, each independently selected from oxygen, nitrogen and sulphur, and is optionally substituted by one to four independently selected halogen atoms; each R4 is, independently, halogen, C1-3 alkyl, C1-3 haloalkyl, C1-3alkoxy(C1-3)alkyl or cyano; r is 0, 1 or 2; and X is 0 or S; or an N-oxide thereof, to novel intermediates used in the preparation of these compounds, to agrochemical compositions which comprise at least one of the novel compounds as an active ingredient and to the use of the active ingredients or compositions in agriculture or horticulture for controlling or preventing infestation of plants by phytopathogenic microorganisms, preferably fungi.

    摘要翻译： 本发明还涉及式（1）的新化合物，其中Het是含有一至三个杂原子的5-或6-元杂环，各自独立地选自氧，氮和硫，该环被一至三个基团R 4取代 ; 任选取代的（C 1-4）烷基C（ - O），任选取代的（C 1-4）烷基C（ - O）O，任选取代的（C 1-4）烷氧基 （C 1-4）烷基，任选取代的烯丙基，任选取代的炔丙基或任选取代的烯丙基; 每个R 2独立地是卤素，任选取代的（C 1-4）烷基，任选取代的（C 1-4）烷氧基或任选取代的（C 1-4）烷氧基（C 1-4）烷基; R3位于噻吩环的2位或4位，是含有3至13个碳原子和至少一个硅原子的有机基团，以及任选的一至三个各自独立地选自氧，氮和硫的杂原子， 并且任选被一至四个独立选择的卤素原子取代; 每个R 4独立地是卤素，C 1-3烷基，C 1-3卤代烷基，C 1-3烷氧基（C 1-3）烷基或氰基; r为0,1或2; X为0或S; 或其N-氧化物，用于制备这些化合物的新型中间体，包含至少一种新化合物作为活性成分的农用化学组合物以及农业或园艺中的活性成分或组合物用于控制 或通过植物病原微生物，优选真菌来防止植物感染。

    3-Carbonylaminothiophenes and their use as fungicides
    45.
    发明申请
    3-Carbonylaminothiophenes and their use as fungicides 失效

    公开(公告)号：US20060276434A1

    公开(公告)日：2006-12-07

    申请号：US10554336

    申请日：2004-04-21

    申请人： Josef Ehrenfreund ,  Harald Walter ,  Hans Tobler ,  Clemens Lamberth

    发明人： Josef Ehrenfreund ,  Harald Walter ,  Hans Tobler ,  Clemens Lamberth

    IPC分类号： C07F7/02 ,  A01N43/54 ,  A01N43/40

    CPC分类号： C07D409/12 ,  A01N55/00 ,  C07D333/28 ,  C07D333/36 ,  C07D411/12 ,  C07D413/12 ,  C07D417/12

    摘要： The invention also relates to novel compounds of formula (I) where Het is a 5- or 6-membered heterocyclic ring containing one to three heteroatoms, each independently selected from oxygen, nitrogen and sulphur, the ring being substituted by one to three groups R4; R1 is hydrogen, optionally substituted (C1-4)alkyl, formyl, optionally substituted (C1-4)alkylC(═O), optionally substituted (C1-4)alkylC(═O)O, optionally substituted (C1-4)alkoxy(C1-4)alkyl, optionally substituted allyl, optionally substituted propargyl or optionally substituted allenyl; each R2 is, independently, halogen, optionally substitute (C1-4)alkyl, optionally substituted (C1-4)alkoxy or optionally substituted (C1-4)alkoxy(C1-4)alkyl; R3 is either position 2 or at position 4 of the thiophene ring and is an organic group containing three to thirteen carbon atoms and al least one silicon atom and, optionally, one to three heteroatoms, each independently selected from oxygen, nitrogen and sulphur, and is optionally substituted by one to four independently selected halogen atoms; each R4 is, independently, halogen, C1-3 alkyl, C1-3 haloalkyl, C1-3alkoxy(C1-3)alkyl or cyano; r is 0, 1 or 2; and X is O or S; or an N-oxide thereof, to novel intermediates used in the preparation of these compounds, to agrochemical compositions which comprise at least one of the novel compounds as an active ingredient and to the use of the active ingredients or compositions in agriculture or horticulture for controlling or preventing infestation of plants by phytopathogenic microorganisms, preferably fungi.

    Silicon compounds with microbiocidal activity
    46.
    发明授权
    Silicon compounds with microbiocidal activity 失效

    公开(公告)号：US07618952B2

    公开(公告)日：2009-11-17

    申请号：US10569343

    申请日：2004-09-08

    申请人： Josef Ehrenfreund ,  Clemens Lamberth ,  Hans Tobler ,  Harald Walter

    发明人： Josef Ehrenfreund ,  Clemens Lamberth ,  Hans Tobler ,  Harald Walter

    IPC分类号： A61K31/695 ,  C07F7/18 ,  C07F7/08 ,  C07F17/00

    CPC分类号： C07F7/0812 ,  A01N55/00

    摘要： Fungicidal compounds of formula (I): where X is O or S; RING is phenyl or thienyl; Het is a 5- or 6-membered heterocyclic ring containing one to three heteroatoms, each independently selected from oxygen, nitrogen and sulphur, the ring being substituted by one to four groups R4; R1 is hydrogen, optionally substituted (C1-4)alkyl, formyl, optionally substituted (C1-4)alkylC(═O), optionally substituted (C1-4)alkylC(═O)O, optionally substituted (C1-4)alkoxy(C1-4)alkyl, optionally substituted allyl, optionally substituted propargyl or optionally substituted allenyl; each R2 is, independently, halogen, optionally substituted (C1-4)alkyl, optionally substituted (C1-4)alkoxy or optionally substituted (C1-4)alkoxy(C1-4)alkyl; R3 is (CRaRb)m—Cy—(CRCRd)n—Y; each R4 is, independently, selected from halogen, C1-3 alkyl, C1-3 haloalkyl, C1-3alkoxy(C1-3)alkyl and cyano; Ra, Rb, Rc and Rd are each, independently, hydrogen or optionally substituted (C1-4)alkyl; Cy is an optionally substituted carbocyclic or heterocyclic 3-7 membered ring which may be saturated, unsaturated or aromatic and which optionally contains a silicon atom as a ring member; (CRaRb)m and (CRcRd)n may be bound either to the same carbon or silicon atom of Cy or to different atoms separated by 1, 2 or 3 ring members; Y is Si(OpZ1)(OqZ2)(OsZ) and provided that Cy contains a silicon atom as a ring member then Y may also be hydrogen; Z is C1-4 alkyl or C2-4 alkenyl (each of which is optionally interrupted by one heteroatom selected from O, S and N and is optionally substituted by one to three independently selected halogen atoms); Z1 and Z2 are, independently, methyl or ethyl; in and n are each, independently, 0, 1, 2 or 3; p, q and s are each, independently, 0 or 1; and r is 0, 1 or 2; or an N-oxide thereof; novel intermediates used in the preparation of these compounds, agrochemical compositions which comprise at least one of the novel compounds as active ingredient and the use of the active ingredients or compositions in agriculture or horticulture for controlling or preventing infestation of plants by phytopathogenic microorganisms, preferably fungi.

    Silicon compounds with microbiocidal activity
    47.
    发明申请
    Silicon compounds with microbiocidal activity 失效

    公开(公告)号：US20060287328A1

    公开(公告)日：2006-12-21

    申请号：US10569343

    申请日：2004-09-08

    申请人： Josef Ehrenfreund ,  Clemens Lamberth ,  Hans Tobler ,  Harald Walter

    发明人： Josef Ehrenfreund ,  Clemens Lamberth ,  Hans Tobler ,  Harald Walter

    IPC分类号： C07D417/02 ,  C07D413/02 ,  C07D409/02 ,  C07D403/02 ,  A01N43/54 ,  A01N43/80 ,  A01N43/76 ,  A01N43/64

    CPC分类号： C07F7/0812 ,  A01N55/00

    摘要： Fungicidal compounds of formula (1): where X is O or S; RING is phenyl or thienyl; Het is a 5- or 6-membered heterocyclic ring containing one to three heteroatoms, each independently selected from oxygen, nitrogen and sulphur, the ring being substituted by one to four groups R4; R1 is hydrogen, optionally substituted (C1-4)alkyl, formyl, optionally substituted (C1-4)alkylC(═O), optionally substituted (C1-4)alkylC(═O)O, optionally substituted (C1-4)alkoxy(C1-4)alkyl, optionally substituted allyl, optionally substituted propargyl or optionally substituted allenyl; each R2 is, independently, halogen, optionally substituted (C1-4)alkyl, optionally substituted (C1-4)alkoxy or optionally substituted (C1-4)alkoxy(C1-4)alkyl; R3 is (CRaRb)m-Cy-(CRcRd)n—Y; each R4 is, independently, selected from halogen, C1-3 alkyl, C1-3 haloalkyl, C1-3alkoxy(C1-3)alkyl and cyano; Ra, Rb, Rc and Rd are each, independently, hydrogen or optionally substituted (C1-4)alkyl; Cy is an optionally substituted carbocyclic or heterocyclic 3-7 membered ring which may be saturated, unsaturated or aromatic and which optionally contains a silicon atom as a ring member; (CRaRb)m and (CRcRd), may be bound either to the same carbon or silicon atom of Cy or to different atoms separated by 1, 2 or 3 ring members; Y is Si(OpZ1)(OqZ2)(O5Z) and provided that Cy contains a silicon atom as a ring member then Y may also be hydrogen; Z is C1-4 alkyl or C2-4 alkenyl (each of which is optionally interrupted by one heteroatom selected from O, S and N and is optionally substituted by one to three independently selected halogen atoms); Z1 and Z2 are, independently, methyl or ethyl; in and n are each, independently, 0, 1, 2 or 3; p, q and s are each, independently, 0 or 1; and r is 0, 1 or 2; or an N-oxide thereof; novel intermediates used in the preparation of these compounds, agrochemical compositions which comprise at least one of the novel compounds as active ingredient and the use of the active ingredients or compositions in agriculture or horticulture for controlling or preventing infestation of plants by phytopathogenic microorganisms, preferably fungi.

    Heterocyclocarboxamide derivatives
    48.
    发明授权
    Heterocyclocarboxamide derivatives 有权
    杂环羧酰胺衍生物

    公开(公告)号：US07598395B2

    公开(公告)日：2009-10-06

    申请号：US10530737

    申请日：2003-10-14

    申请人： Josef Ehrenfreund ,  Hans Tobler ,  Harald Walter

    发明人： Josef Ehrenfreund ,  Hans Tobler ,  Harald Walter

    IPC分类号： C07D231/00 ,  C07D207/00 ,  C07D295/00 ,  C09B5/00 ,  A01N47/36 ,  A01N43/58 ,  A01N43/647 ,  A01N43/36

    CPC分类号： C07D213/82 ,  A01N43/32 ,  A01N43/36 ,  A01N43/40 ,  A01N43/56 ,  A01N43/76 ,  A01N43/78 ,  A01N43/90 ,  C07C211/61 ,  C07C2603/66 ,  C07D207/34 ,  C07D231/14 ,  C07D263/34 ,  C07D277/56 ,  C07D327/06 ,  C07D487/08 ,  C07D493/08 ,  C07D495/08

    摘要： The invention relates to a fungicidally active compound of formula (I): where Het is a 5- or 6-membered heterocyclic ring containing one to three heteroatoms, each independently selected from oxygen, nitrogen and sulphur, provided that the ring is not 1,2,3-triazole, the ring being substituted by groups R8, R9 and R10; X is a single or double bond; Y is O, S, N(R11) or (CR12R13)(CR14R15)m(CR16R17)n; m is 0 or 1; n is 0 or 1; and R1 to R17 each, independently, have a range of values; to the preparation of these compounds, to novel intermediates used in the preparation of these compounds, to agrochemical compositions which comprise at least one of the novel compounds as active ingredient, to the preparation of the compositions mentioned and to the use of the active ingredients or compositions in agriculture or horticulture for controlling or preventing infestation of plants by phytopathogenic microorganisms, preferably fungi.

    摘要翻译： 本发明涉及式（I）的杀真菌活性化合物：其中Het是含有一至三个杂原子的5-或6-元杂环，各自独立地选自氧，氮和硫，条件是环不为1， 该环被R8，R9和R10基团取代; X是单键或双键; Y是O，S，N（R11）或（CR12R13）（CR14R15）m（CR16R17）n; m为0或1; n为0或1; 并且R 1至R 17各自独立地具有一定范围的值; 涉及这些化合物的制备，用于制备这些化合物的新型中间体，包括至少一种新化合物作为活性成分的农用化学组合物，所述组合物的制备以及使用活性成分或 用于通过植物病原微生物，优选真菌控制或预防植物感染的农业或园艺成分。

    MICROBIOCIDAL (E.G. FUNGICIDAL) 1,2,3-TRIAZOLE DERIVATIVES
    49.
    发明申请
    MICROBIOCIDAL (E.G. FUNGICIDAL) 1,2,3-TRIAZOLE DERIVATIVES 有权
    MICROBIOCIDAL（E.G. Fungicidal）1,2,3-三唑衍生物

    公开(公告)号：US20090216027A1

    公开(公告)日：2009-08-27

    申请号：US12463449

    申请日：2009-05-11

    申请人： Josef Ehrenfreund ,  Hans Tobler ,  Harald Walter

    发明人： Josef Ehrenfreund ,  Hans Tobler ,  Harald Walter

    IPC分类号： C07D249/04 ,  C07D487/00

    CPC分类号： C07D401/12 ,  A01N43/647 ,  A01N55/00 ,  C07D249/04 ,  C07D333/36 ,  C07D405/12 ,  C07D409/12 ,  C07D409/14 ,  C07D411/12 ,  C07D413/12 ,  C07D417/12 ,  C07D487/08 ,  C07D493/08 ,  C07D495/08

    摘要： A compound of formula (I): where A is an ortho-substituted ring selected from a number of specified rings; R1 is halogen, cyano, nitro, C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy or C1-4 haloalkoxy or optionally substituted C2-4 alkenyl, optionally substituted C2-4 alkynyl or optionally substituted SO2(C1-4)alkyl (where the optionally substituted moieties may each have up to 3 substituents, each independently selected from halogen and C1-4 alkoxy); R2 is C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy(C1-4)alkyl or C1-4 alkylthio(C1-4)alkyl or [optionally substituted aryl](C1-4)alkyl- or [optionally substituted aryl]oxy(C1-4)alkyl-(where the optionally substituted aryl moieties may each have up to 3 substituents, each independently selected from halogen and C1-4 alkoxy); R3 is hydrogen, CH2C≡CR4, CH2CR4═C(H)R4, CH═C═CH2 or COR5 or optionally substituted C1-4 alkyl, optionally substituted C1-4 alkoxy or optionally substituted (C1-4) alkylC(═O)O (where the optionally substituted moieties may each have up to 3 substituents, each independently selected from halogen and C1-4 alkoxy, C1-4 alkyl, C1-2 haloalkoxy, hydroxy, cyano, carboxyl, methoxycarbonyl, ethoxycarbonyl, methylsulfonyl and ethylsulfonyl); each R4 is, independently, hydrogen, halogen, C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy or C1-4 alkoxy(C1-4)alkyl; and R5 is hydrogen or optionally substituted C1-6 alkyl, optionally substituted C1-4 alkoxy, optionally substituted C1-4 alkoxy(C1-4)alkyl, optionally substituted C1-4 alkylthio(C1-4)alkyl or optionally substituted aryl (where the optionally substituted moieties may each have up to 3 substituents, each independently selected from halogen, C1-6 alkoxy, C1-6 haloalkoxy, cyano, hydroxy, methoxycarbonyl and ethoxycarbonyl).

    摘要翻译： 式（I）的化合物：其中A是选自多个指定环的邻位取代的环; R 1是卤素，氰基，硝基，C 1-4烷基，C 1-4卤代烷基，C 1-4烷氧基或C 1-4卤代烷氧基或任选取代的C 2-4烯基，任选取代的C 2-4炔基或任选取代的SO 2（C 1-4） 烷基（其中任选取代的部分可各自具有至多3个取代基，各自独立地选自卤素和C 1-4烷氧基）; R 2是C 1-4烷基，C 1-4卤代烷基，C 1-4烷氧基（C 1-4）烷基或C 1-4烷硫基（C 1-4）烷基或[任意取代的芳基]（C 1-4）烷基 - 或[ 芳基]氧基（C 1-4）烷基 - （其中任选取代的芳基部分可各自具有至多3个取代基，各自独立地选自卤素和C 1-4烷氧基）; R 3是氢，CH 2C≡CR4，CH 2 CR 4 -C（H）R 4，CH-C-CH 2或COR 5或任选取代的C 1-4烷基，任选取代的C 1-4烷氧基或任选取代的（C 1-4）烷基C（O） O（其中任选取代的部分可以各自具有至多3个取代基，各自独立地选自卤素和C 1-4烷氧基，C 1-4烷基，C 1-2卤代烷氧基，羟基，氰基，羧基，甲氧基羰基，乙氧基羰基，甲基磺酰基和乙基磺酰基） ; 每个R 4独立地是氢，卤素，C 1-4烷基，C 1-4卤代烷基，C 1-4烷氧基或C 1-4烷氧基（C 1-4）烷基; 并且R 5为氢或任选取代的C 1-6烷基，任选取代的C 1-4烷氧基，任选取代的C 1-4烷氧基（C 1-4）烷基，任选取代的C 1-4烷硫基（C 1-4）烷基或任选取代的芳基（其中 任选取代的部分各自可具有至多3个取代基，各自独立地选自卤素，C 1-6烷氧基，C 1-6卤代烷氧基，氰基，羟基，甲氧基羰基和乙氧基羰基）。

    Fungicidal 1,2,3 triazole derivatives
    50.
    发明授权
    Fungicidal 1,2,3 triazole derivatives 失效
    杀真菌剂1,2,3三唑衍生物

    公开(公告)号：US07531559B2

    公开(公告)日：2009-05-12

    申请号：US10524721

    申请日：2003-08-18

    申请人： Josef Ehrenfreund ,  Hans Tobler ,  Harald Walter

    发明人： Josef Ehrenfreund ,  Hans Tobler ,  Harald Walter

    IPC分类号： A61K31/41 ,  C07D249/00

    CPC分类号： C07D401/12 ,  A01N43/647 ,  A01N55/00 ,  C07D249/04 ,  C07D333/36 ,  C07D405/12 ,  C07D409/12 ,  C07D409/14 ,  C07D411/12 ,  C07D413/12 ,  C07D417/12 ,  C07D487/08 ,  C07D493/08 ,  C07D495/08

    摘要： A compound of formula (I):, where A is an ortho-substituted ring selected from a number of specified rings; R1 is halogen, cyano, nitro, C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy or C1-4 haloalkoxy or optionally substituted C2-4 alkenyl, optionally substituted C2-4 alkynyl or optionally substituted SO2(C1-4 alkyl) (where the optionally substituted moieties may each have up to 3 substituents, each independently selected from halogen and C1-4 alkoxy); R2 is C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy(C1-4)alkyl or C1-4 alkylthio(C1-4)alkyl or [optionally substituted aryl](C1-4)alkyl- or [optionally substituted aryl]oxy(C1-4)alkyl (where the optionally substituted aryl moieties may each have up to 3 substituents, each independently selected from halogen and C1-4 alkoxy); R3 is hydrogen, CH2C≡CR4, CH2CR4═C(H)R4, CH═C═CH2 or COR5 or optionally substituted C1-4 alkyl, optionally substituted C1-4 alkoxy or optionally substituted (C1-4)alkylC(═O)O (where the optionally substituted moieties may each have up to 3 substituents, each independently selected from halogen and C1-4 alkoxy, C1-4 alkyl, C1-2 haloalkoxy, hydroxy, cyano, carboxyl, methoxycarbonyl, ethoxycarbonyl, methylsulfonyl and ethylsulfonyl); each R4 is, independently, hydrogen, halogen, C1-4 alkyl, C1-4 haloalkyl, C1-4 alkoxy or C1-4 alkoxy(C1-4)alkyl; and R5 is hydrogen or optionally substituted C1-6 alkyl, optionally substituted C1-4 alkoxy, optionally substituted C1-4 alkoxy(C1-4)alkyl, optionally substituted C1-4 alkylthio(C1-4)alkyl or optionally substituted aryl (where the optionally substituted moieties may each have up to 3 substituents, each independently selected from halogen, C1-6 alkoxy, C1-6 haloalkoxy, cyano, hydroxy, methoxycarbonyl and ethoxycarbonyl).

    摘要翻译： 式（I）的化合物：其中A是选自若干指定环的邻位取代的环; R 1是卤素，氰基，硝基，C 1-4烷基，C 1-4卤代烷基，C 1-4烷氧基或C 1-4卤代烷氧基或任选取代的C 2-4烯基，任选取代的C 2-4炔基或任选取代的SO 2（C 1-4烷基 ）（其中任选取代的部分可各自具有至多3个取代基，各自独立地选自卤素和C 1-4烷氧基）; R 2是C 1-4烷基，C 1-4卤代烷基，C 1-4烷氧基（C 1-4）烷基或C 1-4烷硫基（C 1-4）烷基或[任意取代的芳基]（C 1-4）烷基 - 或[ 芳基]氧基（C 1-4）烷基（其中任选取代的芳基部分可各自具有至多3个取代基，各自独立地选自卤素和C 1-4烷氧基）; R 3是氢，CH 2C≡CR4，CH 2 CR 4 -C（H）R 4，CH-C-CH 2或COR 5或任选取代的C 1-4烷基，任选取代的C 1-4烷氧基或任选取代的（C 1-4）烷基C（O） O（其中任选取代的部分可以各自具有至多3个取代基，各自独立地选自卤素和C 1-4烷氧基，C 1-4烷基，C 1-2卤代烷氧基，羟基，氰基，羧基，甲氧基羰基，乙氧基羰基，甲基磺酰基和乙基磺酰基） ; 每个R 4独立地是氢，卤素，C 1-4烷基，C 1-4卤代烷基，C 1-4烷氧基或C 1-4烷氧基（C 1-4）烷基; 并且R 5为氢或任选取代的C 1-6烷基，任选取代的C 1-4烷氧基，任选取代的C 1-4烷氧基（C 1-4）烷基，任选取代的C 1-4烷硫基（C 1-4）烷基或任选取代的芳基（其中 任选取代的部分各自可具有至多3个取代基，各自独立地选自卤素，C 1-6烷氧基，C 1-6卤代烷氧基，氰基，羟基，甲氧基羰基和乙氧基羰基）。