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89 条记录 (耗时 0.026 秒)

    Herbicidal and phytohormonal amidoximes
    41.
    发明授权
    Herbicidal and phytohormonal amidoximes 失效
    除草和植物激素酰胺肟

    公开(公告)号：US4216006A

    公开(公告)日：1980-08-05

    申请号：US906863

    申请日：1978-05-17

    申请人： Daniel Farge ,  Jean Leboul ,  Yves Le Goff ,  Gilbert Poiget

    发明人： Daniel Farge ,  Jean Leboul ,  Yves Le Goff ,  Gilbert Poiget

    IPC分类号： C07C259/18 ,  C07D207/34 ,  C07D307/68 ,  C07D333/38 ,  A01N9/28

    CPC分类号： C07D333/38 ,  C07C259/18 ,  C07D207/34 ,  C07D307/68

    摘要： Amidoximes of the formula ##STR1## are disclosed. R represents a hydrogen atom or a hydrogen, lower alkyl (C.sub.1 -C.sub.4) or phenyl; R.sub.1 represents lower alkyl or a metal atom and Ar represents substituted or unsubstituted phenyl or a five-membered substituted or unsubstituted aromatic heterocyclic group where the hetero atom is selected from the group O, S and N. The compounds have phytohormonal activity at low dosages in plants and herbicidal activity at higher levels.

    摘要翻译： 公开了“IMAGE”公式的酰氨基。 R代表氢原子或氢原子，低级烷基（C1-C4）或苯基; R1表示低级烷基或金属原子，Ar表示取代或未取代的苯基或杂原子选自O，S和N的五元取代或未取代的芳族杂环基。该化合物在低剂量下具有植物激素活性 植物和除草活性较高。

    Dibenzo[de, h]quinoline derivatives
    46.
    发明授权
    Dibenzo[de, h]quinoline derivatives 失效
    Dibenzo {8 de，h {9 quinoline derivatives

    公开(公告)号：US4128650A

    公开(公告)日：1978-12-05

    申请号：US798139

    申请日：1977-05-18

    申请人： Jean-Louis Fabre ,  Daniel Farge ,  Claude James

    发明人： Jean-Louis Fabre ,  Daniel Farge ,  Claude James

    IPC分类号： A61K31/47 ,  A61K31/473 ,  A61P31/12 ,  C07D209/48 ,  C07D217/16 ,  C07D221/18 ,  C07D471/04 ,  C07D215/20

    CPC分类号： C07D209/48 ,  C07D209/49 ,  C07D217/16 ,  C07D221/18 ,  C07D471/04

    摘要： Compounds of the formula: ##STR1## wherein the symbols X each represent hydrogen or methoxy, R represents hydrogen or carboxymethyl, the symbols R.sub.1 each represent hydrogen or together represent a valency bond and the symbols R.sub.2 each represent hydrogen or together represent a valency bond, the pair of symbols R.sub.2 having the same significance as the pair of symbols R.sub.1, and when the symbols R.sub.1 and R.sub.2 represent hydrogen the symbol X also represents hydrogen, are new compounds possessing antiviral activity.

    摘要翻译： 其中符号X各自表示氢或甲氧基，R表示氢或羧甲基，符号R1各自表示氢或一起代表价键，符号R2各自表示氢或一起代表价键， 该对符号R2具有与该对符号R1相同的含义，并且当符号R1和R2表示氢时，符号X也表示氢，是具有抗病毒活性的新化合物。

    Process for preparing pyrrolo(1,2-A)azepinone derivatives
    48.
    发明授权
    Process for preparing pyrrolo(1,2-A)azepinone derivatives 失效
    制备吡咯（1,2-A）氮杂酮衍生物的方法

    公开(公告)号：US4826974A

    公开(公告)日：1989-05-02

    申请号：US116725

    申请日：1987-11-04

    申请人： Michel Barreau ,  Marie-Therese Comte ,  Daniel Farge ,  Jean-Luc Malleron ,  Gerard Ponsinet ,  Gerard Roussel

    发明人： Michel Barreau ,  Marie-Therese Comte ,  Daniel Farge ,  Jean-Luc Malleron ,  Gerard Ponsinet ,  Gerard Roussel

    IPC分类号： A61K31/55 ,  A61P25/18 ,  C07D487/04 ,  C07D487/06 ,  C07D403/14 ,  C07D413/14

    CPC分类号： C07D487/04

    摘要： Pyrrolo[1,2-a]azepinone derivatives of formula: ##STR1## in which R.sub.3 is H or halogen and either (A) R is benzyl or phenylthio in which the phenyls are optionally substituted by one or more halogens or hydroxy, alkyl, alkyloxy or alkylthio radicals, R.sub.1 and R.sub.2, which may be identical or different, denote alkyl optionally substituted by dialkylamino in which the alkyls are optionally joined to form a 1-pyrrolidinyl, piperidino, morpholino or 1-piperazinyl ring substituted by alkyl, or alternatively R.sub.1 and R.sub.2 form a heterocyclic ring chosen from pyrrolidine, piperidine, morpholine and piperazine, substituted by alkyl, alkenyl (2 to 4 C), benzyl or phenethyl optionally substituted by halogen, alkyl, alkyloxy, alkylthio, CF.sub.3, COOH, carboxyalkyl, alkyloxycarbonyl, alkyloxycarbonylalkyl, hydroxyalkyl, or alkylcarbonyloxyalkyl in which the alkylcarbonyl has 2 to 18 C, or (B) R is phenyl optionally substituted with one or more halogens or hydroxy, alkyl, alkyloxy or alkylthio radicals and R.sub.1 and R.sub.2 together form a piperazine or homopiperazine ring substituted by hydroxyalkyl (2 to 4 C), alkenyl (2 to 4 C), alkynyl (2 to 4 C), benzyl or phenethyl optionally substituted by halogen, alkyl, alkyloxy, alkylthio, CN, CF.sub.3, COOH, carboxyalkyl, alkyloxycarbonyl, alkyloxycarbonylalkyl, hydroxyalkyl, or alkylcarbonyloxyalkyl in which the alkylcarbonyl has 2 to 18 C, the said alkyls containing, except where otherwise stated, 1 to 4 C in a straight or branched chain, and the pharmaceutically acceptable salts thereof, are useful as antipsychotics.

    摘要翻译： 吡咯并[1,2-a]吖庚因酮衍生物，其中R 3为H或卤素，（A）R为苄基或苯硫基，其中苯基任选被一个或多个卤素或羟基取代 ，烷基，烷氧基或烷硫基，R 1和R 2可以相同或不同，表示任选被二烷基氨基取代的烷基，其中烷基任选地连接以形成被烷基取代的1-吡咯烷基，哌啶子基，吗啉代或1-哌嗪基环 或者R1和R2形成选自吡咯烷，哌啶，吗啉和哌嗪的杂环，被烷基，烯基（2至4 C），任选被卤素，烷基，烷氧基，烷硫基，CF 3，COOH取代的苄基或苯乙基取代， 羧基烷基，烷氧基羰基，烷氧基羰基烷基，羟基烷基或烷基羰氧基烷基，其中烷基羰基具有2至18个C，或（B）R是任选被一个或多个卤素或羟基，烷基，烷氧基或烷硫基取代的苯基， 和R2一起形成被羟烷基（2〜4 C），烯基（2〜4 C），炔基（2〜4 C），任选被卤素，烷基，烷氧基，烷硫基，CN取代的苄基或苯乙基取代的哌嗪或高哌嗪环 ，CF 3，COOH，羧基烷基，烷氧基羰基，烷氧基羰基烷基，羟基烷基或其中烷基羰基具有2〜18个碳原子的烷基羰氧基烷基，所述烷基除了另外说明的含有1〜4个C的直链或支链， 其盐可用作抗精神病药。