公开(公告)号：US20070259919A1

公开(公告)日：2007-11-08

申请号：US11630569

申请日：2005-06-18

申请人： Joachim Rheinheimer ,  Frank Schieweck ,  Thomas Grote ,  Carsten Blettner ,  Anja Schwogler ,  Markus Gewehr ,  Wassilios Grammenos ,  Udo Hunger ,  Bernd Muller ,  Peter Schafer ,  John-Bryan Speakman ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Joachim Rheinheimer ,  Frank Schieweck ,  Thomas Grote ,  Carsten Blettner ,  Anja Schwogler ,  Markus Gewehr ,  Wassilios Grammenos ,  Udo Hunger ,  Bernd Muller ,  Peter Schafer ,  John-Bryan Speakman ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A01N43/40 ,  A01N43/86 ,  A01P3/00 ,  C07D213/22 ,  C07D401/04 ,  C07D417/04

CPC分类号： C07D401/04 ,  A01N43/40 ,  A01N43/54 ,  A01N43/56 ,  A01N43/653 ,  A01N43/78 ,  C07D213/61 ,  C07D213/70 ,  C07D213/74 ,  C07D213/78 ,  C07D213/84 ,  C07D213/86 ,  C07D417/04

摘要： The invention relates to 2-substituted pyridines of the formula I in which the index n and the substituents R1 to R4 and L are as defined in the description and in each case one of the two ring members X1, X2 is N, the other is C—H or C-halogen; Y is a group —CH—R1—, —N—R1—, —O— or —S— and  is five- or six-membered hetaryl comprising 1 to 3 heteroatoms selected from the group consisting of O, N and S or is phenyl, and to processes for their preparation, intermediates for their preparation, pesticidal compositions and methods for controlling harmful fungi and animal pests using the compounds according to the invention.

摘要翻译： 本发明涉及式I中的2-取代吡啶，其中指数n和取代基R 1至R 4和L如说明书和每一个中所定义 两个环成员X 1，X 2中的一个是N，另一个是CH或C-卤素; Y是基团-CH-R 1 - ，-NR 1 - ， - O-或-S-，并且是包含1至3个的五元或六元杂芳基 选自O，N和S的杂原子或为苯基，并且其制备方法，其制备中间体，杀虫组合物和使用本发明化合物控制有害真菌和动物害虫的方法。

公开(公告)号：US20070208038A1

公开(公告)日：2007-09-06

申请号：US10594738

申请日：2005-03-26

申请人： Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Bernd Muller ,  Matthias Niedenbruck ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Michael Rack ,  Barbara Nave ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Bernd Muller ,  Matthias Niedenbruck ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Michael Rack ,  Barbara Nave ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A61K31/519 ,  C07D487/04 ,  A01N43/90

CPC分类号： A01N43/90 ,  C07D487/04

摘要： 6-(2-Fluorophenyl)-triazolopyrimidines of the formula I in which the substituents are as defined below: R1 is C4-C8-alkyl, C4-C8-haloalkyl, substituted C3-C8-cycloalkyl, C3-C8-halocycloalkyl, C5-C8-alkenyl, C2-C8-haloalkenyl, C3-C6-cycloalkenyl, C3-C6-halocycloalkenyl, C2-C8-alkynyl, C2-C8-haloalkynyl or phenyl, naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S, R2 is hydrogen, C1-C3-alkyl or one of the groups mentioned under R1, R1 and R2 together with the nitrogen atom to which they are attached may also form a five- or six-membered heterocyclyl or heteroaryl which is attached via N and contain one to three further heteroatoms from the group consisting of O, N and S as ring member, except for piperidin-1-yl optionally substituted by methyl groups; R1 and/or R2 may be substituted according to the description; L1 is chlorine or fluorine; L2 is hydrogen, is, if L1 is fluorine, also fluorine; X is alkyl; processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

公开(公告)号：US20070191396A1

公开(公告)日：2007-08-16

申请号：US10591342

申请日：2005-03-17

申请人： Jordi Tormo i Blasco ,  Thomas Grote ,  Maria Scherer ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl ,  Markus Gewehr

发明人： Jordi Tormo i Blasco ,  Thomas Grote ,  Maria Scherer ,  Reinhard Stierl ,  Siegfried Strathmann ,  Ulrich Schofl ,  Markus Gewehr

IPC分类号： A01N43/90 ,  A01N37/52 ,  A01N37/34

CPC分类号： A01N43/90 ,  A01N2300/00

摘要： The invention relates to fungicidal mixtures, containing the following in a synergistically effective quantity as active components: 1) the triazolopyrimidine derivative of formula (I); and 2) a phenylamidine derivative of formula (II), in which the variables are defined as follows: R1, R4, R5 represent alkyl, alkenyl or alkynyl; R2, R3 represent cyano, alkyl, alkenyl, alkynyl, alkoxy, alkoxyalkyl, benzyloxy or alkylcarbonyl; m represents 0 or 1; A represents a direct bond, —O—, —S—, NRd, CHRe or —O—CHRe; R6 represents phenyl or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle, containing between one and four heteroatoms from the group comprising O, N or S, whereby the groups can be substituted according to the description. The invention also relates to a method for controlling pathogenic fungi using mixtures of compounds (I) and (II), to the use of compounds (I) and (II) for producing mixtures of this type and to agents that contain said mixtures.

摘要翻译： 本发明涉及杀真菌混合物，其具有协同有效量作为活性成分：1）式（I）的三唑并嘧啶衍生物; 和2）式（II）的苯基脒衍生物，其中变量定义如下：R 1，R 4，R 5， 代表烷基，烯基或炔基; R 2，R 3代表氰基，烷基，烯基，炔基，烷氧基，烷氧基烷基，苄氧基或烷基羰基; m表示0或1; A表示直接键，-O-，-S-，NR d，CHR e或-O-CHR e; R 6表示苯基或五元或六元饱和，部分不饱和或芳族杂环，其含有一个至四个来自O，N或S的基团的杂原子，其中基团可以根据 的描述。 本发明还涉及使用化合物（I）和（II）的混合物来控制致病真菌的方法，用于制备这种类型的混合物和含有所述混合物的试剂的化合物（I）和（II）。

公开(公告)号：US20070149551A1

公开(公告)日：2007-06-28

申请号：US11677862

申请日：2007-02-22

申请人： Andreas GYPSER ,  Thomas Grote ,  Anja Schwogler ,  Joachim Rheiheimer ,  Frank Schieweck ,  Jordi Blasco ,  Ingo Rose ,  Peter Schafer ,  Markus Gewehr ,  Wassilios Grammenos ,  Bernd Muller ,  Eberhard Ammernann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

发明人： Andreas GYPSER ,  Thomas Grote ,  Anja Schwogler ,  Joachim Rheiheimer ,  Frank Schieweck ,  Jordi Blasco ,  Ingo Rose ,  Peter Schafer ,  Markus Gewehr ,  Wassilios Grammenos ,  Bernd Muller ,  Eberhard Ammernann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

IPC分类号： A61K31/506 ,  C07D403/02

CPC分类号： C07D239/42 ,  C07D239/47 ,  C07D239/48 ,  C07D239/52 ,  C07D403/12

摘要： 5-Phenylpyrimidines of the formula I in which the substituents and the index are as defined below: R1,R2 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, alkynyl or haloalkynyl, and R1 and R2 together with the nitrogen atom to which they are attached may also form a saturated or unsaturated ring which may be interrupted by an ether, thio, sulfoxyl or sulfonyl group and may be substituted by one to four groups Ra and/or Rb; R3 is hydrogen, halogen, cyano, alkyl, haloalkyl, alkoxy, haloalkoxy or alkenyloxy; R4 is hydrogen, halogen, cyano, hydroxyl, mercapto, azido, alkyl, alkenyl, alkynyl, haloalkyl, alkoxy, alkenyloxy, alkynyloxy, haloalkoxy, alkylthio, alkenylthio, alkynylthio, haloalkylthio, —ON═CRNaRb, —CRc═NORa, —NRcN═CRaRb, —NRaRb, —NRcNRaRb, —NORa, —NRcC (═NRc′)NRaRb, —NRcC(═O)NRaRb, —NRaC(═O)Rc, —NRaC(═NORc)Rc′, —OC (═O)Rc, —C(═NORc)NRaRb, —CRc(═NNRaRb), —C (═O)NRaRb or —C(═O) Rc; in which Ra, Rb and Rc are as defined in the description; X is halogen, alkyl, alkoxy or haloalkyl; and m is an integer from 1 to 5; processes for preparing these compounds, compositions comprising them and their use for controlling harmful fungi are described.

公开(公告)号：US20070142404A1

公开(公告)日：2007-06-21

申请号：US10590924

申请日：2005-03-29

申请人： Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Bernd Muller ,  Matthias Niedenbruck ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Michael Rack ,  Barbara Nave ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Udo Hunger ,  Bernd Muller ,  Matthias Niedenbruck ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Michael Rack ,  Barbara Nave ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A61K31/519 ,  C07D487/04

CPC分类号： A01N43/90 ,  C07D487/04

摘要： 6-(2,6-Dichlorophenyl)triazolopyrimidines of the formula I in which the substituents are as defined below: R1, R2 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S, R1 and R2 together with the nitrogen atom to which they are attached may also form a five- or six-membered heterocyclyl or heteroaryl which is attached via N and may contain one to three further heteroatoms from the group consisting of O, N and S as ring member and which is substituted according to the description; X is alkyl, cyano, alkoxy, haloalkoxy, alkenyloxy or haloalkenyloxy; processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

摘要翻译： 其中取代基如下定义的式I的6-（2,6-二氯苯基）三唑并嘧啶：R 1，R 2是氢，烷基，卤代烷基，环烷基 ，卤代环烷基，烯基，卤代烯基，环烯基，卤代环烯基，炔基，卤代炔基或苯基，萘基或五元或六元饱和的部分不饱和或芳族杂环，其含有一至四个由O，N和S组成的组的杂原子 R 1和R 2连同它们所连接的氮原子一起也可以形成通过N连接的五元或六元杂环基或杂芳基，并且可以 含有一个至三个由O，N和S组成的组的另外的杂原子作为环成员，并且根据描述被取代; X是烷基，氰基，烷氧基，卤代烷氧基，烯氧基或卤代烯氧基; 制备这些化合物的方法，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US20070135453A1

公开(公告)日：2007-06-14

申请号：US10579395

申请日：2004-12-14

申请人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  C07D487/04

CPC分类号： C07D487/04 ,  A01N43/90

摘要： The present invention relates to 6-(2,4,6-trihalophenyl)triazolopyrimidines of the formula I in which the substituents are as defined below: R1 is alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl or a five- or six-member saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S, R2 is hydrogen or one of the groups mentioned under R1, R1 and R2 together with the nitrogen atom to which they are attached may also form a five- or six-membered heterocyclyl or heteroaryl which is attached via N and may contain one to three further heteroatoms from the group consisting of O, N and S as ring members; R1 and/or R2 may be substituted as defined in the description; L1, L2, L3 are chlorine or fluorine, where at least one group is chlorine; X is cyano, alkyl, alkoxy, alkenyloxy, haloalkoxy or haloalkenyloxy; processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.

摘要翻译： 本发明涉及式I的6-（2,4,6-三卤代苯基）三唑并嘧啶，其中取代基如下：R 1是烷基，卤代烷基，环烷基，卤代环烷基，烯基， 卤代烯基，环烯基，卤代环烯基，炔基，卤代炔基或苯基，萘基或五或六元饱和的部分不饱和或芳族杂环，其含有一至四个由O，N和S组成的组的杂原子，R 2 R 1是氢或R 1，R 2和R 2中所提及的基团之一，与它们的氮原子一起 还可以形成通过N连接的五元或六元杂环基或杂芳基，并且可以含有一个至三个其它由O，N和S组成的组的杂原子作为环成员; R 1和/或R 2可以如说明书中所定义的取代; L 1，L 2，L 3 3是氯或氟，其中至少一个基团是氯; X是氰基，烷基，烷氧基，烯氧基，卤代烷氧基或卤代烯氧基; 制备这些化合物的方法，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US20060241128A1

公开(公告)日：2006-10-26

申请号：US10532719

申请日：2003-11-04

申请人： Jordi Tormo I Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Jordi Tormo I Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  C07D487/04

CPC分类号： C07C69/65 ,  A01N43/90 ,  C07D487/04

摘要： Substituted 6-(2-halogenphenyl)-triazolopyrimidines of formula I in which R1 denote alkyl, alkenyl, alkynyl, alkadienyl, haloalkyl, haloalkenyl, cycloalkyl, phenyl, naphthyl, or a 5- or 6-membered saturated, unsaturated, or aromatic heterocycle, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, wherein R1 and R2 radicals may be substituted as defined in the description, R2 denote hydrogen, or a group mentioned for R1; or R1 and R2 together with the interjacent nitrogen atom represent a 5- or 6-membered heterocycle, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which ring may be substituted as defined in the description; Hal is halogen; L1, L3 independently denote hydrogen, halogen, or alkyl; L2 is hydrogen, halogen, haloalkyl, or NH2, NHRb, or N(Rb)2, wherein Rb is as defined in the description, wherein at least one from L1, L2, and L3 is not hydrogen; X is halogen, cyano, alkyl, alkoxy, haloalkoxy or alkenyloxy. processes for their preparation, compositions containing them and to their use for combating phytopathogenic fungi.

摘要翻译： 其中R 1表示烷基，烯基，炔基，链二烯基，卤代烷基，卤代烯基，环烷基，苯基，萘基或5-或6-元的取代的6-（2-卤代苯基） - 三唑并嘧啶， 含有1至4个氮原子或1至3个氮原子和1个硫或氧原子的饱和，不饱和或芳族杂环，其中R 1和R 2可以是 如说明书中所定义，R 2表示氢或R 1所提及的基团; 或R 1和R 2连同中间的氮原子代表含有1-4个氮原子或一至三个氮原子的一个或多个六元杂环，一个 硫或氧原子，该环可以如说明书中所定义取代; 卤素是卤素; L 1，L 3独立地表示氢，卤素或烷基; L 2是氢，卤素，卤代烷基或NH 2，NHR b或/或N（R b） 其中R b如描述中所定义，其中至少一个L 1，L 2， ，而L 3不是氢; X是卤素，氰基，烷基，烷氧基，卤代烷氧基或烯氧基。 其制备方法，含有它们的组合物及其用于对抗植物病原真菌的用途。

公开(公告)号：US20060217400A1

公开(公告)日：2006-09-28

申请号：US10539559

申请日：2003-12-17

申请人： Bernd Müller ,  Jordi Blasco ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Anja Schwögler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schöfl ,  Reinhard Stierl

发明人： Bernd Müller ,  Jordi Blasco ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Anja Schwögler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schöfl ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  C07D487/04

CPC分类号： C07D487/04 ,  A01N43/90

摘要： Triazolopyrimidines of the formula I in which the index n and the substituents R1, R2 and R3 are as defined in the description, and processes for preparing these compounds, compositions comprising them and their use for controlling harmful fungi are described.

摘要翻译： 其中指数n和取代基R 1，R 2和R 3的式I的三唑并嘧啶如说明书中所定义，以及 描述了制备这些化合物的方法，包含它们的组合物及其用于控制​​有害真菌的用途。

公开(公告)号：US20060211573A1

公开(公告)日：2006-09-21

申请号：US10548690

申请日：2004-03-24

申请人： Jordi Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schalfer ,  Frank Schieweck ,  Anja Schwogler ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Jordi Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schalfer ,  Frank Schieweck ,  Anja Schwogler ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  C07D487/04

CPC分类号： C07D487/04 ,  A01N43/90

摘要： 7-(Alkenylamino)triazolopyrimidines of the formula I wherein the substituents have the following meanings: L is halogen, alkyl, haloalkyl, alkoxy, amino, NHR or NR2; R is alkyl or alkyl-carbonyl; m is 1, 2, 3, 4 or 5; X is halogen, cyano, alkyl, haloalkyl or alkoxy; R1 is alkyl or haloalkyl; R2 is hydrogen, alkyl or haloalkyl; R3 is alkenyl, which can be unsubstituted or partially or completely halogenated or can be substituted according to the Description; R4 is hydrogen or alkyl, R3 and R4 can also, together with the nitrogen atom to which they are bonded, form a five- or six-membered unsaturated ring which can be interrupted by an atom from the group consisting of O, N and S and/or can carry one or more sub-stituents. Processes for the preparation of these compounds, preparations comprising them and their use in the control of harmful phytopathogenic fungi.

摘要翻译： 式（I）的7-（烯基氨基）三唑并嘧啶，其中取代基具有以下含义：L是卤素，烷基，卤代烷基，烷氧基，氨基，NHR或NR 2。 R是烷基或烷基 - 羰基; m为1,2,3,4或5; X是卤素，氰基，烷基，卤代烷基或烷氧基; R 1是烷基或卤代烷基; R 2是氢，烷基或卤代烷基; R 3是烯基，其可以是未取代的或部分的或完全卤化的或可以根据描述被取代; R 4是氢或烷基，R 3和R 4也可以与它们所键合的氮原子一起形成五元环 - 或六元不饱和环，其可以被来自O，N和S的原子中断，和/或可以携带一个或多个亚取代基。 制备这些化合物的方法，包含它们的制剂及其在控制有害植物病原真菌中的用途。

公开(公告)号：US07071334B2

公开(公告)日：2006-07-04

申请号：US10474461

申请日：2002-04-06

申请人： Jordi Tormo i Blasco ,  Hubert Sauter ,  Bernd Müller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schäfer ,  Frank Schieweck ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

发明人： Jordi Tormo i Blasco ,  Hubert Sauter ,  Bernd Müller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schäfer ,  Frank Schieweck ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

IPC分类号： C07D487/04 ,  A01N43/90

CPC分类号： C07D487/04 ,  A01N43/90

摘要： 6-(2-Chloro-6-fluoro-phenyl)-triazolopyrimidines of formula (I), in which R1 and R2 independently denote hydrogen or alkyl, alkenyl, alkynyl, alkadienyl, or haloalkyl, cycloalkyl, bicycloalkyl, phenyl, naphthyl, or 5- or 6-membered heterocyclyl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or 5- or 6-membered heteroaryl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or where R1 and R2 radicals may be unsubstituted or partially or fully halogenated or may be substituted as defined in the description. R1 and R2 together with the interjacent nitrogen atom represent a 5- or 6-membered heterocyclic ring, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which may be substituted; X is cyano, alkoxy, haloalkoxy or alkenyloxy; processes for their preparation, compositions containing them and to their use for combating phytopathogenic fungi

摘要翻译： 式（I）的6-（2-氯-6-氟 - 苯基） - 三唑并嘧啶，其中R 1和R 2独立地表示氢或烷基，烯基， 炔基，链烯基或卤代烷基，环烷基，二环烷基，苯基，萘基或含有1-4个氮原子或1-3个氮原子和一个硫或氧原子的5-或6-元杂环基，或5-或6-元 含有一至四个氮原子或一至三个氮原子和一个硫或氧原子的杂芳基，或其中R 1和R 2基团可以是未取代的或部分或完全的 卤化的或可以如说明书中所定义的取代。 R 1和R 2与中间的氮原子一起表示含有1-4个氮原子或一至三个氮原子的一个5-或6-元杂环，一个 硫或氧原子，其可以被取代; X是氰基，烷氧基，卤代烷氧基或烯氧基; 其制备方法，含有它们的组合物及其用于对抗植物病原真菌的用途