Substituted 5-Hetaryl-4-Aminopyrimidines
    51.
    发明申请

    公开(公告)号:US20110201496A1

    公开(公告)日:2011-08-18

    申请号:US12293432

    申请日:2007-03-26

    CPC分类号: A01N43/54

    摘要: The present invention relates to the use of 5-hetaryl-4-aminopyrimidines of the formula I and their salts for controlling plant-damaging fungi. The invention also relates to novel 5-hetaryl-4-aminopyrimidines and to crop protection compositions comprising at least one such compound as active component. Het is an optionally substituted 5- or 6-membered aromatic heterocycle which has 1, 2, 3 or 4 heteroatoms selected from the group consisting of nitrogen, oxygen and sulfur as ring members, where the 5- or 6-membered heteroaromatic radical may have 1, 2, 3 or 4 identical or different substituents L, R1, R2 are inter alia hydrogen, C1-C8-alkyl, C3-C8-cycloalkyl, C5-C10-bicycloalkyl, C2-C8-alkenyl, C4-C10-alkadienyl, C3-C6-cycloalkenyl, C2-C8-alkynyl, phenyl, naphthyl or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle which has one, two, three or four heteroatoms from the group consisting of O, N or S as ring members; or together form a ring; R3 is inter alia hydrogen, OH, halogen, cyano, NR31R32, C1-C8-alkyl, C1-C8-alkoxy, C1-C8-alkylthio, C1-C8-alkylsulfinyl, C1-C8-alkylsulfonyl, C2-C8-alkenyl or C2-C8-alkynyl, and R4 is halogen, cyano, hydroxyl, mercapto, N3, C1-C6-alkyl, C2-C8-alkenyl, C2-C8-alkynyl, C1-C6-haloalkyl, C1-C6-alkoxy, C3-C8-alkenyloxy, C3-C8-alkynyloxy, C1-C6-haloalkoxy, C1-C6-alkylthio, C3-C8-alkenylthio, C3-C8-alkinylthio, C1-C6-haloalkylthio, or is a radical of the formula C(═Z)OR41, C(═Z)NR42R43, C(═Z)NR44—NR42R43, C(═Z)R45, CR46R47—OR48, CR46R47—NR42R43, ON(═CR49R50), O—C(═Z)R45, NR42R43a, NR51(C(═Z)R45), NR51(C(═Z)OR41), NR51(C(═Z)—NR42R43), NR52a(N═CR49R50), NR52NR42R43, NR52OR41 or C(═N—X—R45)SR41.

    Azolylmethyloxiranes, Use Thereof for Controlling Plant Pathogenic Fungi, and Agents Containing the Same
    52.
    发明申请
    Azolylmethyloxiranes, Use Thereof for Controlling Plant Pathogenic Fungi, and Agents Containing the Same 失效
    唑基甲基环氧乙烷,其用途用于控制植物病原真菌和含有其的药剂

    公开(公告)号:US20090270256A1

    公开(公告)日:2009-10-29

    申请号:US12374710

    申请日:2007-07-18

    CPC分类号: C07D405/06

    摘要: The present invention relates to azolylmethyloxiranes of the general formula I in which A or B is phenyl which is substituted by one CN and optionally by one to three of the following substituents: halogen, NO2, amino, C1-C4-alkyl, C1-C4-alkoxy, C1-C4-haloalkyl, C1-C4-haloalkoxy, C1-C4-alkylamino, C1-C4-dialkylamino, thio or C1-C4-alkylthio, and the respective other substituent A or B is phenyl or 5-membered or 6-membered heteroaryl, these substituents optionally being substituted by one to three of the following substituents: halogen, CN, NO2, amino, C1-C4-alkyl, C1-C4-alkoxy, C1-C4-haloalkyl, C1-C4-haloalkoxy, C1-C4-alkylamino, C1-C4-dialkylamino, thio or C1-C4-alkylthio, and to the plant-compatible acid addition salts or metal salts thereof, to the use of the compounds of the formula I for controlling phytopathogenic fungi and to compositions comprising these compounds.

    摘要翻译: 本发明涉及通式I的唑基甲基环氧乙烷,其中A或B是被一个CN和任选的一个到三个以下取代基取代的苯基:卤素,NO 2,氨基,C 1 -C 4烷基,C 1 -C 4 - 烷氧基,C 1 -C 4卤代烷基,C 1 -C 4卤代烷氧基,C 1 -C 4 - 烷基氨基,C 1 -C 4 - 二烷基氨基,硫代或C 1 -C 4 - 烷硫基,各自的其它取代基A或B是苯基或5元或 这些取代基任选被1-3个以下取代基取代:卤素,CN,NO 2,氨基,C 1 -C 4 - 烷基,C 1 -C 4 - 烷氧基,C 1 -C 4卤代烷基,C 1 -C 4 - 卤代烷氧基 C 1 -C 4 - 烷基氨基,C 1 -C 4 - 二烷基氨基,硫代或C 1 -C 4 - 烷硫基,以及与植物相容的酸加成盐或金属盐,用于控制植物病原真菌的式I化合物, 包含这些化合物的组合物。

    Fungicidal Mixtures Comprising a Substituted 3-Hydroxymethylpyridine and a Further Fungicidal Compound
    56.
    发明申请
    Fungicidal Mixtures Comprising a Substituted 3-Hydroxymethylpyridine and a Further Fungicidal Compound 审中-公开
    包含取代的3-羟甲基吡啶和另外的杀真菌化合物的杀真菌混合物

    公开(公告)号:US20100273650A1

    公开(公告)日:2010-10-28

    申请号:US12742717

    申请日:2008-11-14

    CPC分类号: A01N43/40 A01N2300/00

    摘要: The present invention relates to mixtures of fungicidally active compounds comprising at least one substituted 3-hydroxymethylpyridin compound formula I and at least one further fungicidally active compound II. wherein: X is O, S or NR4; R1 is C1-C6-alkyl, C1-C6-alkoxy-C1-C6-alkyl, C1-C6-haloalkyl, aryl-C1-C4-alkyl, aryloxy-C1-C4-alkyl, arylthio-C1-C4-alkyl, aryl or heteroaryl, wherein the cyclic moieties of the last five radicals are unsubstituted or substituted with 1, 2 or 3 radicals selected from halogen, C1-C4-alkyl, C2-C4-alkenyl, C2-C4-alkynyl, C1-C4-haloalkyl, C1-C4-alkoxy, C1-C4-alkylthio, C1-C4-haloalkoxy, C1-C4-haloalkylthio, cyano and nitro; R2 is H or C1-C4-alkyl; R3 is C1-C6-alkyl, C1-C6-alkoxy-C1-C6-alkyl, C1-C6-haloalkyl, aryl-C1-C4-alkyl, aryloxy-C1-C4-alkyl, arylthio-C1-C4-alkyl, aryl or heteroaryl, wherein the cyclic moieties of the last five radicals are unsubstituted or substituted with 1, 2 or 3 radicals selected from halogen, C1-C4-alkyl, C2-C4-alkenyl, C2-C4-alkynyl, C1-C4-haloalkyl, C1-C4-alkoxy, C1-C4-alkylthio, C1-C4-haloalkoxy, C1-C4-haloalkylthio, cyano and nitro; R4 is H, C1-C6-alkyl, C1-C6-alkoxy-C1-C6-alkyl, C1-C6-haloalkyl, aryl-C1-C4-alkyl, aryloxy-C1-C4-alkyl, arylthio-C1-C4-alkyl, aryl or heteroaryl, wherein the cyclic moieties of the last five radicals are unsubstituted or substituted with 1, 2 or 3 radicals selected from halogen, C1-C4-alkyl, C2-C4-alkenyl, C2-C4-alkynyl, C1-C4-haloalkyl, C1-C4-alkoxy, C1-C4-alkylthio, C1-C4-haloalkoxy, C1-C4-haloalkylthio, cyano and nitro;

    摘要翻译: 本发明涉及杀真菌活性化合物的混合物,其包含至少一种取代的3-羟甲基吡啶化合物式I和至少一种其它杀真菌活性化合物II。 其中:X是O,S或NR4; R 1是C 1 -C 6烷基,C 1 -C 6烷氧基-C 1 -C 6烷基,C 1 -C 6卤代烷基,芳基-C 1 -C 4烷基,芳氧基-C 1 -C 4烷基,芳硫基-C 1 -C 4烷基, 芳基或杂芳基,其中最后五个基团的环状部分是未取代的或被1,2或3个选自卤素,C 1 -C 4 - 烷基,C 2 -C 4 - 烯基,C 2 -C 4 - 炔基,C 1 -C 4 - 卤代烷基,C 1 -C 4 - 烷氧基,C 1 -C 4 - 烷硫基,C 1 -C 4卤代烷氧基,C 1 -C 4卤代烷硫基,氰基和硝基; R2是H或C1-C4-烷基; R 3是C 1 -C 6烷基,C 1 -C 6烷氧基-C 1 -C 6烷基,C 1 -C 6卤代烷基,芳基-C 1 -C 4烷基,芳氧基-C 1 -C 4烷基,芳硫基-C 1 -C 4烷基, 芳基或杂芳基,其中最后五个基团的环状部分是未取代的或被1,2或3个选自卤素,C 1 -C 4 - 烷基,C 2 -C 4 - 烯基,C 2 -C 4 - 炔基,C 1 -C 4 - 卤代烷基,C 1 -C 4 - 烷氧基,C 1 -C 4 - 烷硫基,C 1 -C 4卤代烷氧基,C 1 -C 4卤代烷硫基,氰基和硝基; R 4是H,C 1 -C 6烷基,C 1 -C 6烷氧基-C 1 -C 6烷基,C 1 -C 6卤代烷基,芳基-C 1 -C 4烷基,芳氧基-C 1 -C 4烷基,芳硫基-C 1 -C 4 - 烷基,芳基或杂芳基,其中最后五个基团的环状部分是未取代的或被1,2或3个选自卤素,C 1 -C 4 - 烷基,C 2 -C 4 - 烯基,C 2 -C 4 - 炔基,C 1 -C 4 - C 1 -C 4 - 卤代烷基,C 1 -C 4 - 烷氧基,C 1 -C 4 - 烷硫基,C 1 -C 4卤代烷氧基,C 1 -C 4卤代烷硫基,氰基和硝基;

    Fungicidal Mixtures III
    57.
    发明申请
    Fungicidal Mixtures III 审中-公开
    杀菌混合物III

    公开(公告)号:US20100273649A1

    公开(公告)日:2010-10-28

    申请号:US12742487

    申请日:2008-11-14

    摘要: The present invention relates to mixtures of fungicidally active compounds comprising at least one substituted 2-[hydroxyl(pyridine-3-yl)methyl]acrylate compound of the formula I wherein: R1 is H, C1-C6-alkyl, C1-C6-alkoxy-C1-C6-alkyl, C1-C6-haloalkyl, aryl or heteroaryl, wherein the cyclic moieties of the last two radicals are unsubstituted or substituted with 1, 2 or 3 radicals selected from halogen, C1-C4-alkyl, C2-C4-alkynyl, C1-C4-haloalkyl, C1-C4-alkoxy, C1-C4-alkylthio, C1-C4-haloalkoxy, cyano and nitro; A is a covalent bond or C1-C4-alkylen, which is unsubstituted or which may carry a substitutent selected from C1-C4-alkyl, C1-C4-haloalkyl, C1-C4-alkoxy and cyano; Ar is aryl or heteroaryl, wherein the cyclic moieties of the aromatic radicals are unsubstituted or substituted with 1, 2 or 3 radicals Ra, where the radicals Ra are identical or different and selected from halogen, C1-C4-alkyl, C2-C4-alkenyl, C2-C4-alkynyl, C1-C4-haloalkyl, C1-C4-alkoxy, C1-C4-alkylthio, C1-C4-haloalkoxy, C1-C4-haloalkylthio, cyano, nitro, aryl, hetaryl, aryloxy, hetaryloxy, aryloxy-C1-C4-alkyl and hetaryloxy-C1-C4-alkyl, wherein the cyclic moieties of the six last mentioned radicals are unsubstituted or substituted with 1, 2 or 3 radicals selected from halogen, C1-C4-alkyl, C1-C4-haloalkyl, C1-C4-alkoxy, C1-C4-alkylthio, C1-C4-haloalkoxy, cyano and nitro; or a salt thereof; and at least one further fungicidally active compound II.

    摘要翻译: 本发明涉及包含至少一种式I的取代的2- [羟基(吡啶-3-基)甲基]丙烯酸酯化合物的杀真菌活性化合物的混合物,其中:R1是H,C1-C6-烷基,C1-C6- 烷氧基-C 1 -C 6 - 烷基,C 1 -C 6卤代烷基,芳基或杂芳基,其中最后两个基团的环状部分是未取代的或被1,2或3个选自卤素,C 1 -C 4 - 烷基, C 4 - 炔基,C 1 -C 4卤代烷基,C 1 -C 4 - 烷氧基,C 1 -C 4 - 烷硫基,C 1 -C 4卤代烷氧基,氰基和硝基; A是共价键或C1-C4-亚烷基,其是未取代的或可以携带选自C 1 -C 4 - 烷基,C 1 -C 4 - 卤代烷基,C 1 -C 4 - 烷氧基和氰基的取代基; Ar是芳基或杂芳基,其中芳族基团的环状部分是未取代的或被1,2或3个基团R a取代,其中基团R a相同或不同并且选自卤素,C 1 -C 4烷基,C 2 -C 4 - 烯基,C 2 -C 4 - 炔基,C 1 -C 4卤代烷基,C 1 -C 4 - 烷氧基,C 1 -C 4 - 烷硫基,C 1 -C 4卤代烷氧基,C 1 -C 4卤代烷硫基,氰基,硝基,芳基,杂芳基,芳氧基, 芳氧基-C 1 -C 4烷基和芳基氧基-C 1 -C 4烷基,其中六个最后提到的基团的环状部分是未取代的或被1,2或3个选自卤素,C 1 -C 4 - 烷基,C 1 -C 4 卤代烷基,C 1 -C 4 - 烷氧基,C 1 -C 4 - 烷硫基,C 1 -C 4卤代烷氧基,氰基和硝基; 或其盐; 和至少一种其它杀真菌活性化合物II。

    Fungicidal Mixtures
    58.
    发明申请
    Fungicidal Mixtures 审中-公开
    杀菌混合物

    公开(公告)号:US20100179059A1

    公开(公告)日:2010-07-15

    申请号:US12602790

    申请日:2008-06-05

    摘要: The present invention relates to mixtures comprising, as active components, 1) a fungicidal compound of formula (I) wherein: R1 is alkyl; alkoxyalkyl; haloalkyl; arylalkyl; aryl; or heteroaryl; R2 is alkyl; alkoxyalkyl; haloalkyl; arylalkyl; aryl; heteroaryl; 5-pyrimidinyl; or 2- or 5-thiazolyl; R3 is H; alkyl; alkoxyalkyl; haloalkyl; arylalkyl; aryloxyalkyl; arylthioalkyl; aryl; heteroaryl; or alkylsilyl; R4 is H; acyl; haloacyl, alkoxycarbonyl; aryloxycarbonyl; alkylaminocarbonyl; or dialkylaminocarbonyl; or a salt thereof; and 2) a fungicidal compound II selected from azoles, strobilurins, carboxamides, heterocylic compounds, carbamates, and other active compounds in synergistically effective amounts.

    摘要翻译: 本发明涉及包含作为活性成分的1)式(I)的杀真菌化合物的混合物,其中:R 1是烷基; 烷氧基烷基 卤代烷基 芳烷基 芳基; 或杂芳基; R2是烷基; 烷氧基烷基 卤代烷基 芳烷基 芳基; 杂芳基; 5-嘧啶基; 或2-或5-噻唑基; R3为H; 烷基; 烷氧基烷基 卤代烷基 芳烷基 芳氧基烷基; 芳硫基烷基 芳基; 杂芳基; 或烷基甲硅烷基; R4是H; 酰基; 卤代酰基,烷氧基羰基; 芳氧基羰基; 烷基氨基羰基; 或二烷基氨基羰基; 或其盐; 和2)协同有效量的选自吡唑,嗜球半胱氨酸,羧酰胺,杂环化合物,氨基甲酸酯和其它活性化合物的杀真菌化合物II。