公开(公告)号：US07799334B2

公开(公告)日：2010-09-21

申请号：US11919588

申请日：2006-05-10

申请人： Markus Gewehr ,  Jochen Dietz ,  Thomas Grote ,  Wassilios Grammenos ,  Udo Hünger ,  Bernd Müller ,  Frank Schieweck ,  Anja Schwögler ,  Jan Klaas Lohmann ,  Joachim Rheinheimer ,  Jens Renner ,  Peter Schäfer

发明人： Markus Gewehr ,  Jochen Dietz ,  Thomas Grote ,  Wassilios Grammenos ,  Udo Hünger ,  Bernd Müller ,  Frank Schieweck ,  Anja Schwögler ,  Jan Klaas Lohmann ,  Joachim Rheinheimer ,  Jens Renner ,  Peter Schäfer

IPC分类号： A61K31/16 ,  A01N25/00 ,  C07D231/00 ,  A01N25/26 ,  A01N37/18

CPC分类号： A01N43/56 ,  C07D231/14

摘要： The present invention relates to pyrazolecarboxamides of the formula I in which the variables are as defined below: X is trifluoromethyl; R1 is F, Cl, Br, C1-C4-alkyl or C1-C4-haloalkyl; R2 is hydrogen, halogen or C1-C4-alkyl; R3 is hydrogen, C1-C4-alkyl, C1-C4-haloalkyl, C2-C4-alkenyl, C2-C4-alkynyl or C3-C6-cycloalkyl; W is O or S; with the proviso that, if R3 is hydrogen and W is oxygen, a) R1 and R2 are not simultaneously methyl and F, respectively; b) R1 and R2 are not simultaneously trifluoromethyl and hydrogen or fluorine, respectively. to processes for preparing these compounds, to seeds and compositions comprising them and to methods for controlling harmful fungi.

摘要翻译： 本发明涉及式I的吡唑酰胺，其中变量如下所定义：X是三氟甲基; R1是F，Cl，Br，C1-C4-烷基或C1-C4卤代烷基; R2是氢，卤素或C1-C4-烷基; R 3是氢，C 1 -C 4 - 烷基，C 1 -C 4卤代烷基，C 2 -C 4 - 烯基，C 2 -C 4 - 炔基或C 3 -C 6 - 环烷基; W为O或S; 条件是，如果R3是氢并且W是氧，则a）R1和R2分别不同时为甲基和F; b）R1和R2分别不同时为三氟甲基和氢或氟。 制备这些化合物的方法，包括它们的种子和组合物以及用于控制有害真菌的方法。

公开(公告)号：US20110004021A1

公开(公告)日：2011-01-06

申请号：US12876415

申请日：2010-09-07

申请人： Jochen DIETZ ,  Markus Gewehr ,  Thomas Grote ,  Wassilios Grammenos ,  Udo Hünger ,  Bernd Müller ,  Frank Schieweck ,  Anja Schwögler ,  Jan Klaas Lohmann ,  Joachim Rheinheimer ,  Jens Renner ,  Peter Schäfer

发明人： Jochen DIETZ ,  Markus Gewehr ,  Thomas Grote ,  Wassilios Grammenos ,  Udo Hünger ,  Bernd Müller ,  Frank Schieweck ,  Anja Schwögler ,  Jan Klaas Lohmann ,  Joachim Rheinheimer ,  Jens Renner ,  Peter Schäfer

IPC分类号： C07C211/52

CPC分类号： C07D277/56 ,  C07D277/587

摘要： Thiazolecarboxanilides of the formula I in which the variables are as defined below: A is X is halogen; Y is cyano, nitro, C1-C4-alkyl, C1-C4-haloalkyl, methoxy or methylthio; p is 0, 1; R1 is hydrogen, halogen, C1-C4-alkyl, C1-C4-haloalkyl; R2 is hydrogen, methyl, halogen; R3 is hydrogen, methyl, ethyl; W is O, S; and processes for preparing these compounds, compositions and seed comprising them and methods for controlling harmful fungi.

摘要翻译： 式I的噻唑甲酰苯胺，其中变量如下定义：A是X是卤素; Y是氰基，硝基，C 1 -C 4烷基，C 1 -C 4卤代烷基，甲氧基或甲硫基; p为0，1; R1是氢，卤素，C1-C4-烷基，C1-C4卤代烷基; R2是氢，甲基，卤素; R3是氢，甲基，乙基; W是O，S; 以及制备这些化合物，组合物和包含它们的种子的方法以及用于控制有害真菌的方法。

公开(公告)号：US20100087321A1

公开(公告)日：2010-04-08

申请号：US12519973

申请日：2007-12-04

申请人： Jens Renner ,  Thomas Grote ,  Bernd Müller ,  Jan Klaas Lohmann ,  Sarah Ulmschneider ,  Alice Glättli ,  Jochen Dietz

发明人： Jens Renner ,  Thomas Grote ,  Bernd Müller ,  Jan Klaas Lohmann ,  Sarah Ulmschneider ,  Alice Glättli ,  Jochen Dietz

IPC分类号： A01N43/653 ,  C07D249/08 ,  A01H5/00 ,  A01P3/00

CPC分类号： C07D405/06 ,  A01N43/653

摘要： The present invention relates to azolylmethyloxiranes of the general formula (I) in which A stands for phenyl which is optionally substituted by one to three of the following substituents: halogen, NO2, amino, C1-C4-alkyl, C1-C4-alkoxy, C1-C4-haloalkyl, C1-C4-haloalkoxy, C1-C4-alkylamino, C1-C4-dialkylamino, thio or C1-C4-alkylthio, with the proviso that A does not stand for 2-methylphenyl, and also their plant-compatible acid addition salts or metal salts, and also to the use of the compounds of the formula I for controlling phytopathogenic fungi, and to compositions comprising them.

摘要翻译： 本发明涉及通式（I）的唑基甲基环氧乙烷，其中A代表任选被一至三个以下取代基取代的苯基：卤素，NO 2，氨基，C 1 -C 4烷基，C 1 -C 4 - 烷氧基， C 1 -C 4卤代烷基，C 1 -C 4卤代烷氧基，C 1 -C 4烷基氨基，C 1 -C 4 - 二烷基氨基，硫代或C 1 -C 4 - 烷硫基，条件是A不代表2-甲基苯基， 并且还涉及用于控制植物病原真菌的式I化合物以及包含它们的组合物的用途。

公开(公告)号：US20090197929A1

公开(公告)日：2009-08-06

申请号：US12306339

申请日：2007-06-25

申请人： Jochen Dietz ,  Thomas Grote ,  Bernd Müller ,  Jan Klaas Lohmann ,  Jens Renner ,  Sarah Ulmschneider ,  Alice Glättli

发明人： Jochen Dietz ,  Thomas Grote ,  Bernd Müller ,  Jan Klaas Lohmann ,  Jens Renner ,  Sarah Ulmschneider ,  Alice Glättli

IPC分类号： A01N43/64 ,  C07D249/08 ,  A01P3/00

CPC分类号： C07D417/14 ,  C07D403/14 ,  C07D405/14 ,  C07D409/14 ,  C07D413/14

摘要： The present invention relates to azolylmethyloxiranes of the general formula I in which A or B is a 5-membered heteroaryl selected from the group consisting of thienyl, furyl, pyrrolyl, pyrazolyl, imidazolyl, oxazolyl, thiazolyl, isoxazolyl and isothiazolyl which is substituted by one to three of the following substituents: halogen, NO2, amino, C1-C4-alkyl, C1-C4-alkoxy, C1-C4-haloalkyl, C1-C4-haloalkoxy, C1-C4-alkylamino, C1-C4-dialkylamino, thio or C1-C4-alkylthio, and the respective other substituent A or B is phenyl which is optionally substituted by one to three of the following substituents: halogen, NO2, amino, C1-C4-alkyl, C1-C4-alkoxy, C1-C4-haloalkyl, C1-C4-haloalkoxy, C1-C4-alkylamino, C1-C4-dialkylamino, thio or C1-C4-alkylthio, and to the plant-compatible acid addition salts or metal salts thereof, to the use of the compounds of the formula I for controlling phytopathogenic fungi and to compositions comprising these compounds.

摘要翻译： 本发明涉及通式I的唑基甲基环氧乙烷，其中A或B是选自噻吩基，呋喃基，吡咯基，吡唑基，咪唑基，恶唑基，噻唑基，异恶唑基和被一个取代基的异噻唑基的5元杂芳基 至三个以下取代基：卤素，NO 2，氨基，C 1 -C 4 - 烷基，C 1 -C 4 - 烷氧基，C 1 -C 4 - 卤代烷基，C 1 -C 4 - 卤代烷氧基，C 1 -C 4烷基氨基，C 1 -C 4二烷基氨基，硫代 或其它取代基A或B为任选被一至三个以下取代基取代的苯基：卤素，NO 2，氨基，C 1 -C 4 - 烷基，C 1 -C 4 - 烷氧基，C 1 -C 4 - 烷硫基， C 4-卤代烷基，C 1 -C 4卤代烷氧基，C 1 -C 4 - 烷基氨基，C 1 -C 4 - 二烷基氨基，硫代或C 1 -C 4 - 烷硫基，以及与植物相容的酸加成盐或其金属盐， 用于控制植物病原真菌的式I化合物和包含这些化合物的组合物。

公开(公告)号：US20120225777A1

公开(公告)日：2012-09-06

申请号：US13470426

申请日：2012-05-14

申请人： Jochen Dietz ,  Thomas Grote ,  Bernd Müller ,  Jan Klaas Lohmann ,  Jens Renner ,  Sarah Ulmschneider ,  Alice Glättli

发明人： Jochen Dietz ,  Thomas Grote ,  Bernd Müller ,  Jan Klaas Lohmann ,  Jens Renner ,  Sarah Ulmschneider ,  Alice Glättli

IPC分类号： A01N43/653 ,  A01C1/06 ,  A01P3/00 ,  C07D405/06

CPC分类号： C07D405/06

摘要： The present invention relates to azolylmethyloxiranes of the general formula I in which A is phenyl which is substituted by three F, B is unsubstituted pyridyl, thienyl, thiazolyl, oxazolyl or furyl or is phenyl which is substituted by one to three of the following substituents: halogen, NO2, amino, C1-C4-alkyl, C1-C4-alkoxy, C1-C4-haloalkyl, C1-C4-haloalkoxy, C1-C4-alkylamino, C1-C4-dialkylamino, thio or C1-C4-alkylthio, and to the plant-compatible acid addition salts or metal salts thereof, to the use of the compounds of the formula I for controlling phytopathogenic fungi and to compositions comprising these compounds.

摘要翻译： 本发明涉及通式I的唑基甲基环氧乙烷，其中A是被三个F取代的苯基，B是未取代的吡啶基，噻吩基，噻唑基，恶唑基或呋喃基，或是被一至三个以下取代基取代的苯基： 卤素，NO 2，氨基，C 1 -C 4 - 烷基，C 1 -C 4 - 烷氧基，C 1 -C 4卤代烷基，C 1 -C 4卤代烷氧基，C 1 -C 4烷基氨基，C 1 -C 4 - 二烷基氨基，硫代或C 1 -C 4烷硫基， 以及与植物相容的酸加成盐或其金属盐，用于控制植物病原真菌的式I化合物和包含这些化合物的组合物。

公开(公告)号：US20120220455A1

公开(公告)日：2012-08-30

申请号：US13470512

申请日：2012-05-14

申请人： Jochen DIETZ ,  Thomas Grote ,  Bernd Müller ,  Jan Klaas Lohmann ,  Jens Renner ,  Sarah Ulmschneider ,  Alice Glättli

发明人： Jochen DIETZ ,  Thomas Grote ,  Bernd Müller ,  Jan Klaas Lohmann ,  Jens Renner ,  Sarah Ulmschneider ,  Alice Glättli

IPC分类号： A01N43/653 ,  A01P3/00 ,  C07D407/06

CPC分类号： C07D405/06

摘要： The present invention relates to azolylmethyloxiranes of the general formula I in which A is phenyl which is substituted by an F and another substituent selected from the group consisting of Cl, C1-C4-alkyl, C1-C4-haloalkyl and C1-C4-alkoxy, B is unsubstituted pyridyl, thienyl, thiazolyl, oxazolyl or furyl or is phenyl which is substituted by one to three of the following substituents: halogen, NO2, amino, C1-C4-alkyl, C1-C4-alkoxy, C1-C4-haloalkyl, C1-C4-haloalkoxy, C1-C4-alkylamino, C1-C4-dialkylamino, thio or C1-C4-alkylthio, with the proviso that B is not o-methylphenyl if A is 2-chloro-4-fluorophenyl, and to the plant-compatible acid addition salts or metal salts thereof, to the use of the compounds of the formula I for controlling phytopathogenic fungi and to compositions comprising these compounds.

摘要翻译： 本发明涉及通式I的唑基甲基环氧烷，其中A是被F取代的苯基，另一个选自Cl，C 1 -C 4 - 烷基，C 1 -C 4卤代烷基和C 1 -C 4 - 烷氧基的取代基 B是未取代的吡啶基，噻吩基，噻唑基，恶唑基或呋喃基，或被一至三个以下取代基取代的苯基：卤素，NO 2，氨基，C 1 -C 4烷基，C 1 -C 4烷氧基，C 1 -C 4 - 卤代烷基，C 1 -C 4 - 卤代烷氧基，C 1 -C 4 - 烷基氨基，C 1 -C 4 - 二烷基氨基，硫代或C 1 -C 4 - 烷硫基，条件是如果A是2-氯-4-氟苯基，则B不是邻甲基苯基， 涉及与植物相容的酸加成盐或其金属盐，用于控制植物病原真菌的式I化合物和包含这些化合物的组合物。

公开(公告)号：US20100179058A1

公开(公告)日：2010-07-15

申请号：US12303652

申请日：2007-06-15

申请人： Jochen Dietz ,  Thomas Grote ,  Bernd Müller ,  Jan Klaas Lohmann ,  Jens Renner ,  Sarah Ulmschneider ,  Alice Glättli

发明人： Jochen Dietz ,  Thomas Grote ,  Bernd Müller ,  Jan Klaas Lohmann ,  Jens Renner ,  Sarah Ulmschneider ,  Alice Glättli

IPC分类号： A01N43/653 ,  C07D405/06 ,  A01N25/00 ,  A01P3/00

CPC分类号： C07D405/06 ,  A01N43/653 ,  C07D405/14 ,  C07D409/14 ,  C07D413/14 ,  C07D417/14

摘要： The present invention relates to azolylmethyloxiranes of the general formula I in which A is phenyl which is substituted by two F, B is unsubstituted pyridyl, thienyl, thiazolyl, oxazolyl or furyl or is phenyl which is optionally substituted by one to three of the following substituents: halogen, NO2, amino, C1-C4-alkyl, C1-C4alkoxy, C1-C4-haloalkyl, C1-C4-haloalkoxy, C1-C4-alkylamino, thio or C1-C4-alkylthio, with the proviso that B is not o-methylphenyl if A is 2,4-difluorophenyl, and to the plant-compatible acid addition salts or metal salts thereof, to the use of the compounds of the formula I for controlling phytopathogenic fungi and to compositions comprising these compounds.

摘要翻译： 本发明涉及通式I的唑基甲基环氧乙烷，其中A是被两个F取代的苯基，B是未取代的吡啶基，噻吩基，噻唑基，恶唑基或呋喃基，或是任选被一至三个以下取代基取代的苯基 ：卤素，NO 2，氨基，C 1 -C 4烷基，C 1 -C 4烷氧基，C 1 -C 4卤代烷基，C 1 -C 4卤代烷氧基，C 1 -C 4烷基氨基，硫代或C 1 -C 4烷硫基，条件是B不为 如果A是2,4-二氟苯基，以及与植物相容的酸加成盐或金属盐，使用式I化合物来控制植物病原性真菌，以及包含这些化合物的组合物。

公开(公告)号：US20090270256A1

公开(公告)日：2009-10-29

申请号：US12374710

申请日：2007-07-18

申请人： Jochen Dietz ,  Thomas Grote ,  Bernd Muller ,  Jan Klaas Lohmann ,  Jens Renner ,  Sarah Ulmschneider ,  Alice Glattli

发明人： Jochen Dietz ,  Thomas Grote ,  Bernd Muller ,  Jan Klaas Lohmann ,  Jens Renner ,  Sarah Ulmschneider ,  Alice Glattli

IPC分类号： A01N25/26 ,  C07D405/06 ,  A01N43/653 ,  A01N43/54 ,  C07D405/14 ,  A01P3/00

CPC分类号： C07D405/06

摘要： The present invention relates to azolylmethyloxiranes of the general formula I in which A or B is phenyl which is substituted by one CN and optionally by one to three of the following substituents: halogen, NO2, amino, C1-C4-alkyl, C1-C4-alkoxy, C1-C4-haloalkyl, C1-C4-haloalkoxy, C1-C4-alkylamino, C1-C4-dialkylamino, thio or C1-C4-alkylthio, and the respective other substituent A or B is phenyl or 5-membered or 6-membered heteroaryl, these substituents optionally being substituted by one to three of the following substituents: halogen, CN, NO2, amino, C1-C4-alkyl, C1-C4-alkoxy, C1-C4-haloalkyl, C1-C4-haloalkoxy, C1-C4-alkylamino, C1-C4-dialkylamino, thio or C1-C4-alkylthio, and to the plant-compatible acid addition salts or metal salts thereof, to the use of the compounds of the formula I for controlling phytopathogenic fungi and to compositions comprising these compounds.

摘要翻译： 本发明涉及通式I的唑基甲基环氧乙烷，其中A或B是被一个CN和任选的一个到三个以下取代基取代的苯基：卤素，NO 2，氨基，C 1 -C 4烷基，C 1 -C 4 - 烷氧基，C 1 -C 4卤代烷基，C 1 -C 4卤代烷氧基，C 1 -C 4 - 烷基氨基，C 1 -C 4 - 二烷基氨基，硫代或C 1 -C 4 - 烷硫基，各自的其它取代基A或B是苯基或5元或 这些取代基任选被1-3个以下取代基取代：卤素，CN，NO 2，氨基，C 1 -C 4 - 烷基，C 1 -C 4 - 烷氧基，C 1 -C 4卤代烷基，C 1 -C 4 - 卤代烷氧基 C 1 -C 4 - 烷基氨基，C 1 -C 4 - 二烷基氨基，硫代或C 1 -C 4 - 烷硫基，以及与植物相容的酸加成盐或金属盐，用于控制植物病原真菌的式I化合物， 包含这些化合物的组合物。

公开(公告)号：US07910614B2

公开(公告)日：2011-03-22

申请号：US12374877

申请日：2007-07-17

申请人： Jochen Dietz ,  Thomas Grote ,  Bernd Müller ,  Jan Klaas Lohmann ,  Jens Renner ,  Sarah Ulmschneider ,  Alice Glättli

发明人： Jochen Dietz ,  Thomas Grote ,  Bernd Müller ,  Jan Klaas Lohmann ,  Jens Renner ,  Sarah Ulmschneider ,  Alice Glättli

IPC分类号： A61K31/4196 ,  C07D405/14

CPC分类号： C07D405/14 ,  A01N43/653 ,  C07D409/14

摘要： The present invention relates to azolylmethyloxiranes of the general formula I in which A or B is benzodioxolyl which is optionally substituted by one to five of the following substituents: halogen, CN, NO2, amino, C1-C4-alkyl, C1-C4-alkoxy, C1-C4-haloalkyl, C1-C4-haloalkoxy, C1-C4-alkylamino, C1-C4-dialkylamino, thio or C1-C4-alkylthio, and the respective other substituent A or B is phenyl or 5-membered or 6-membered heteroaryl, these substituents optionally being substituted by one to three of the following substituents: halogen, CN, NO2, amino, C1-C4-alkyl, C1-C4-alkoxy, C1-C4-haloalkyl, C1-C4-haloalkoxy, C1-C4-alkylamino, C1-C4-dialkylamino, thio or C1-C4-alkylthio, and to the plant-compatible acid addition salts or metal salts thereof, to the use of the compounds of the formula I for controlling phytopathogenic fungi and to compositions comprising these compounds.

摘要翻译： 本发明涉及通式I的唑基甲基环氧乙烷，其中A或B是苯并二恶唑基，其任选被一至五个以下取代基取代：卤素，CN，NO 2，氨基，C 1 -C 4 - 烷基，C 1 -C 4 - 烷氧基 ，C 1 -C 4卤代烷基，C 1 -C 4卤代烷氧基，C 1 -C 4烷基氨基，C 1 -C 4 - 二烷基氨基，硫代或C 1 -C 4 - 烷硫基，各自的取代基A或B为苯基或5元或6- 这些取代基任选被1-3个以下取代基取代：卤素，CN，NO 2，氨基，C 1 -C 4 - 烷基，C 1 -C 4 - 烷氧基，C 1 -C 4卤代烷基，C 1 -C 4 - 卤代烷氧基，C 1 -C 1-4 - 烷基氨基，C 1 -C 4 - 二烷基氨基，硫代或C 1 -C 4 - 烷硫基，以及与植物相容的酸加成盐或金属盐，用于控制植物病原真菌和组合物的式I化合物 包括这些化合物。

公开(公告)号：US20090203700A1

公开(公告)日：2009-08-13

申请号：US12306322

申请日：2007-06-27

申请人： Jochen Dietz ,  Thomas Grote ,  Bernd Müller ,  Jan Klaas Lohmann ,  Jens Renner ,  Sarah Ulmschneider ,  Alice Glättli

发明人： Jochen Dietz ,  Thomas Grote ,  Bernd Müller ,  Jan Klaas Lohmann ,  Jens Renner ,  Sarah Ulmschneider ,  Alice Glättli

IPC分类号： A01N43/40 ,  C07D405/14 ,  A01N43/64 ,  A01N43/58 ,  A01P3/00

CPC分类号： C07D405/14 ,  A01N43/653

摘要： The present invention relates to azolylmethyloxiranes of the general formula I in which A or B is a 6-membered heteroaryl selected from the group consisting of pyridinyl, pyrimidinyl, pyrazinyl, pyridazinyl and triazinyl which is substituted by one to three of the following substituents: halogen, NO2, amino, C1-C4-alkyl, C1-C4-alkoxy, C1-C4-haloalkyl, C1-C4-haloalkoxy, C1-C4-alkylamino, C1-C4-dialkylamino, thio or C1-C4-alkylthio, and the respective other substituent A or B is phenyl which is optionally substituted by one to three of the following substituents: halogen, NO2, amino, C1-C4-alkyl, C1-C4-alkoxy, C1-C4-haloalkyl, C1-C4-haloalkoxy, C1-C4-alkylamino, C1-C4-dialkylamino, thio or C1-C4-alkylthio, and to the plant-compatible acid addition salts or metal salts thereof, to the use of the compounds of the formula I for controlling phytopathogenic fungi and to compositions comprising these compounds.

摘要翻译： 本发明涉及通式Ⅰ的唑基甲基环氧烷，其中A或B是选自吡啶基，嘧啶基，吡嗪基，哒嗪基和三嗪基的6元杂芳基，其被一至三个以下取代基取代：卤素 ，NO 2，氨基，C 1 -C 4 - 烷基，C 1 -C 4 - 烷氧基，C 1 -C 4卤代烷基，C 1 -C 4卤代烷氧基，C 1 -C 4烷基氨基，C 1 -C 4 - 二烷基氨基，硫代或C 1 -C 4烷硫基， 相应的其它取代基A或B是任选被一至三个以下取代基取代的苯基：卤素，NO 2，氨基，C 1 -C 4 - 烷基，C 1 -C 4 - 烷氧基，C 1 -C 4卤代烷基，C 1 -C 4 - 卤代烷氧基，C 1 -C 4 - 烷基氨基，C 1 -C 4 - 二烷基氨基，硫代或C 1 -C 4 - 烷硫基，以及与植物相容的酸加成盐或金属盐，用于控制植物病原真菌的式I化合物 以及包含这些化合物的组合物。