Drug efflux pump inhibitor
    51.
    发明申请
    Drug efflux pump inhibitor 审中-公开
    药物外排泵抑制剂

    公开(公告)号:US20060106034A1

    公开(公告)日:2006-05-18

    申请号:US11320229

    申请日:2005-12-29

    IPC分类号: A61K31/519

    摘要: A medicament for preventive and/or therapeutic treatment of a microbial infection which comprises as an active ingredient a compound represented by the following general formula (I): wherein, R1 and R2 represent hydrogen atom, a halogen atom, hydroxyl group or the like, W1 represents —CH═CH—, —CH2O—, —CH2CH2— or the like; R3 represents hydrogen atom, a halogen atom, hydroxyl group or an amino group; R4 represents hydrogen atom, a group of —OZ0-4R5 (Z0-4 represents an alkylene group, a fluorine-substituted alkylene group or a single bond, and R5 represents a cyclic alkyl group, an aryl group or the like); W2 represents a single bond or —C(R8)═C(R9)−(R8 and R9 represent hydrogen atom, a halogen atom, a lower alkyl group or the like, Q represents an acidic group, but W2 and Q may together form vinylidenethiazolidinedione or an equivalent heterocyclic ring; m and n represent an integer of 0 to 2, and q represents an integer of 0 to 3.

    摘要翻译: 一种用于预防和/或治疗微生物感染的药物,其包含作为活性成分的由以下通式(I)表示的化合物:其中R 1和R 2, SUP>表示氢原子,卤素原子,羟基等,W 1表示-CH-CH-,-CH 2 O - , - CH- 2 CH 2 - 或类似物; R 3表示氢原子,卤素原子,羟基或氨基; R 4表示氢原子,-OZ 0-4R 5(Z 0-4)的基团表示 亚烷基,氟取代的亚烷基或单键,R 5表示环状烷基,芳基等)。 -C(R 9) - (R 9) - (R 9) - (R 8) >和R 9表示氢原子,卤素原子,低级烷基等,Q表示酸性基团,但W 2和Q可以一起形成亚乙烯基乙二胺二酮或 等价杂环; m和n表示0〜2的整数,q表示0〜3的整数。

    Flat heating surface type gas stove
    52.
    发明授权
    Flat heating surface type gas stove 失效
    平面加热表面式燃气灶

    公开(公告)号:US06609513B2

    公开(公告)日:2003-08-26

    申请号:US10038908

    申请日:2002-01-08

    IPC分类号: F24C300

    CPC分类号: F24C3/067 Y02B40/166

    摘要: There is disclosed a novel flat heating surface type gas stove which is capable of heating a heating substance across a heat resistant glass at a practically applicable heating efficiency, thereby overcoming any inconvenience resulting from the exposure of flame and facilitating the cleaning of the gas stove. This gas stove 10 comprises a heat resistant glass top plate 12 which is disposed over a burner 15, wherein a gas-permeable porous body 40 is disposed below said top plate 12, and a space between said top plate 12 and a surface of said gas-permeable porous body 40 is assigned to a combustion space S. Combustion gas generated is designed to be discharged through said gas-permeable porous body 40. As high-temperature combustion gas passes through said gas-permeable porous body 40, radiant heat B is generated from the surface of said gas-permeable porous body 40. Since the heating substance 4 is heated by both of heat conduction and radiation, high heating efficiency can be achieved.

    摘要翻译: 公开了一种新颖的平面加热表面型燃气灶,其能够以实际适用的加热效率加热加热物质穿过耐热玻璃,从而克服由于火焰暴露而导致的任何不便,并且便于清洁燃气灶。 该燃气灶10包括设置在燃烧器15上方的耐热玻璃顶板12,其中透气性多孔体40设置在所述顶板12的下方,并且所述顶板12与所述气体的表面之间的空间 将透气性多孔体40分配给燃烧空间S.产生的燃烧气体被设计成通过所述透气性多孔体40排出。当高温燃烧气体通过所述透气性多孔体40时,辐射热B为 从所述透气性多孔体40的表面产生。由于加热物质4被热传导和辐射两者加热,因此可以实现高的加热效率。

    Equipment for filling flexible container with viscous material.
    53.
    发明授权
    Equipment for filling flexible container with viscous material. 有权
    用粘性材料填充柔性容器的设备。

    公开(公告)号:US06546973B2

    公开(公告)日:2003-04-15

    申请号:US10216231

    申请日:2002-08-12

    IPC分类号: B65D714

    摘要: The present invention is a system for filling a container main body at least whose drum body is made of a flexible film, with a viscous material. A viscous material is charged by the charging means into container main bodies conveyed by the container conveying means, the drum body of the container main body is pressed by the pressing means to cause the surface of the viscous material to bulge, and the opening of the reinforcing component of the container main body is capped by the capping means, allowing the opening to be capped in an air-tight manner with a lid member while virtually all of the air inside the container main body is evacuated, and preventing air from being left over in the container main body so as to prevent hardening, curing and deterioration in the quality of the viscous material that can be caused by such remaining air.

    摘要翻译: 本发明是一种用粘性材料填充容器主体至少其鼓体由柔性膜制成的系统。 通过充电装置将粘性材料装入由容器输送装置输送的容器主体中,容器主体的鼓体被加压装置按压使粘性材料的表面膨胀,并且打开 容器主体的增强部件被封盖装置盖住,允许开口用盖部件以气密方式被盖住,同时几乎所有的容器主体内的所有空气都被抽真空,并且防止空气被留下 在容器主体中,以防止由这种剩余空气引起的粘性物质的硬化,固化和劣化。

    Jointing device for a corrugated flexible conduit
    54.
    发明授权
    Jointing device for a corrugated flexible conduit 失效
    用于波纹软管的接合装置

    公开(公告)号:US5356181A

    公开(公告)日:1994-10-18

    申请号:US135292

    申请日:1993-10-12

    摘要: A jointing device, which permits quick connection and disconnection of a corrugated flexible conduit, comprises a joint body having a cylindrical connector section for receiving the conduit, the connector section being formed with receive holes arranged circumferentially thereof, and a clasp axially slidably mounted on the joint body. The clasp has an outer cylinder axially slidably fitted on the connector section and covering the receive holes formed in the connector section, an inner cylinder slidably fitted into the connector section for receiving the conduit, and locking members connected at their respective fixed ends with the inner cylinder. The outer and inner cylinders are connected with each other. The locking members each have a free end portion thereof formed with a claw engageable with and disengageable from the conduit. The free end portion of each locking member is received in a corresponding receive hole when the free end portion is pushed radially outward by the corrugated flexible conduit. Each locking member is engaged at its claw with a groove or depression of the corrugated flexible conduit when the free end portion thereof is pushed radially inward by a corresponding receive hole-defining face of the connector section.

    摘要翻译: 允许波纹柔性导管的快速连接和断开的连接装置包括具有用于容纳导管的圆柱形连接器部分的接头主体,连接器部分形成有沿圆周方向布置的接收孔,以及可轴向可滑动地安装在 关节体。 该卡扣具有轴向可滑动地装配在连接器部分上并覆盖形成在连接器部分中的接收孔的外筒,可滑动地装配到连接器部分中用于容纳导管的内筒,以及在其各自固定端连接的锁定件, 圆筒。 外筒和内筒相互连接。 锁定构件各自具有形成有可与导管接合并与导管分离的爪的自由端部。 当自由端部被波纹柔性导管径向向外推动时,每个锁定构件的自由端部被容纳在相应的接收孔中。 当其自由端被径向向内推动时,每个锁定构件在其爪处与波纹柔性导管的凹槽或凹陷接合,由连接器部分的相应接收孔限定面推动。

    Electrically driving system for foldable rearview mirrors of motor
vehicle
    56.
    发明授权
    Electrically driving system for foldable rearview mirrors of motor vehicle 失效
    机动车辆可折叠后视镜电驱动系统

    公开(公告)号:US4973146A

    公开(公告)日:1990-11-27

    申请号:US203735

    申请日:1988-06-07

    申请人: Kiyoshi Nakayama

    发明人: Kiyoshi Nakayama

    IPC分类号: B60R1/06 B60R1/074 G02B5/08

    CPC分类号: B60R1/074

    摘要: An electrically driving system for the rearview mirrors, wherein the incorporated motors are rotated normally or reversibly in response to the operation of a operational switch, thereby erecting or folding the mirror bodies. The system comprises a momentary operational switch, a relay circuit, a group of limit switches for cutting off the relay circuit and motor circuit respectively by detecting erected and folded positions of the mirror bodies, and a circuit for judging a folded state. When the operational switch is pushed, any folded mirror is detected within delay time of the circuit for judging a folded state. And only when both of the left and right mirror bodies are in the fold positions, the erecting relay is actuated to rotate the motors in the erecting direction.

    Multi-position electrical switch
    57.
    发明授权
    Multi-position electrical switch 失效
    多位置电气开关

    公开(公告)号:US4947461A

    公开(公告)日:1990-08-07

    申请号:US322779

    申请日:1989-03-03

    IPC分类号: H01H25/04

    摘要: A multiple electrical switch comprising a casing, a control knob supported on the top edge of the casing for tiltable movement in four directions, a retainer horizontally mounted within the casing and a conversion knob tiltably supported by the retainer and having an upper portion projecting through the central aperture of the control knob. Upper and lower base plates are disposed on respective opposite sides of the retainer, with each of the upper and lower base plates defining a printed circuit board and having a plurality of fixed connecting contacts. The switch further comprise an insulating elastic sheet having a central portion for covering the upper portion of the conversion knob and opposite side peripheral portions for covering respective top surfaces of the upper base plate and each portion including a swell including a movable connecting contact corresponding to a respective one of the plurality of fixed connecting contacts of the upper base plate.

    摘要翻译: 一种多重电气开关,包括壳体,支撑在壳体的顶部边缘上的用于在四个方向上可倾斜运动的控制旋钮,水平安装在壳体内的保持器和由保持器可倾斜地支撑的转换旋钮, 控制旋钮的中心孔径。 上基板和下基板设置在保持器的相对的相对侧上,每个上基板和下基板限定印刷电路板并具有多个固定的连接触头。 开关还包括绝缘弹性片,其具有用于覆盖转换旋钮的上部的中心部分和用于覆盖上基板的各个顶表面的相对侧周边部分,并且每个部分包括包括对应于 上基板的多个固定连接触头中的一个。

    Process for producing methylol urea solution and process for producing
slow-releasing nitrogenous fertilizer using the same
    58.
    发明授权
    Process for producing methylol urea solution and process for producing slow-releasing nitrogenous fertilizer using the same 失效
    制备羟甲基脲溶液的方法和使用该方法生产缓释氮肥的方法

    公开(公告)号:US4895983A

    公开(公告)日:1990-01-23

    申请号:US338444

    申请日:1989-04-13

    CPC分类号: C05C9/02

    摘要: A process for producing a methylol urea solution which comprises carrying out addition reaction between urea and formaldehyde in the presence of water and an alkali, wherein said alkali is a polyphosphoric acid salt; and a process for producing a slow-releasing nitrogenous fertilizer which comprises subjecting the resulting methylol urea solution to dehydration condensation and drying the resulting condensate are disclosed. The methylol urea solution undergoes no substantial pH variation with time either during or after the addition reaction, and the fertilizer obtained therefrom is excellent in slow-releasing properties.

    摘要翻译: 一种制备羟甲基脲溶液的方法,其包括在水和碱的存在下进行尿素和甲醛之间的加成反应,其中所述碱是多磷酸盐; 以及一种生产缓释氮肥的方法,其包括使得到的羟甲基脲溶液进行脱水缩合并干燥所得的冷凝物。 羟甲基脲溶液在加成反应期间或之后不会随时间发生显着的pH变化,并且由此获得的肥料具有优异的缓释性能。

    Rate sensor with coaxially mounted scanning antenna
    59.
    发明授权
    Rate sensor with coaxially mounted scanning antenna 失效
    速率传感器同轴安装的扫描天线

    公开(公告)号:US4675688A

    公开(公告)日:1987-06-23

    申请号:US899744

    申请日:1986-08-22

    IPC分类号: F41G7/22 H01Q3/08 H01Q3/00

    摘要: A rate sensor, preferably comprised of a tuned gyro, has a generally cylindrical outer housing and an inner, large diameter rotary cylindrical support defining the gyro's rotary axis. The rate sensing apparatus is mounted in the volume between the outer housing and the rotary cylindrical support whereby the interior of the rotary cylindrical support defines a large diameter hollow for receiving and supporting apparatus, other than rate sensing components of the rate sensor. The rate sensor may be advantageously used with a homing device, the seeker apparatus of the device being mounted in said hollow. This produces a homing device with a high packing density and, as the rotary axis of the gyro gimbals and that of the seeker coincide, detrimental unbalance and unwanted increase in inertial movement is eliminated.

    摘要翻译: 优选地由调谐陀螺仪组成的速率传感器具有大致圆柱形的外壳体和限定陀螺仪的旋转轴线的内部,大直径的旋转圆柱形支撑件。 速率检测装置安装在外壳和旋转圆柱形支撑件之间的体积中,由此旋转圆柱形支撑件的内部限定了用于接收和支撑装置的大直径中空部分,而不是速率传感器的速率感测部件。 速率传感器可以有利地与归位装置一起使用,该装置的引导装置安装在所述中空部分中。 这产生具有高填充密度的回原点装置,并且随着陀螺仪万向节的旋转轴线和探针的旋转轴重合,消除了有害的不平衡和不期望的惯性运动的增加。

    Multi-position electric switch
    60.
    发明授权
    Multi-position electric switch 失效
    多位置电开关

    公开(公告)号:US4499342A

    公开(公告)日:1985-02-12

    申请号:US471477

    申请日:1983-03-03

    申请人: Kiyoshi Nakayama

    发明人: Kiyoshi Nakayama

    IPC分类号: H01H25/04 H01H9/26

    CPC分类号: H01H25/041 H01H2300/012

    摘要: A switch suitable for use in the remote control of electrically driven rearview mirrors of a motor vehicle. The switch is adapted to close and open a plurality of switch elements by means of a single or divided operation member. The switch occupies only a small space in an instrument panel, etc. of a motor vehicle because the switch is thin and small. Fixed contact pairs (3a, 4a) to (3f', 4f') forming fixed contact components are printed approximately point symmetrically around a specific center on an insulating base plate. Movable contact means is disposed on top of the fixed contact components, said movable contact means being adapted to electrically connect each of the fixed contact pairs (3a, 4a) to (3f', 4') when said means is pushed. Said operation member is provided with pressing surfaces for pressing said switch elements comprising the fixed contact pairs (3a, 4a) to (3f', 4') and the movable contact means, and with means for automatically returning said operation member to its original position when it is not pushed.

    摘要翻译: 适用于遥控车用电动后视镜的开关。 开关适于通过单个或分开的操作构件封闭并打开多个开关元件。 由于开关薄而小,所以开关仅占用机动车辆仪表板等的较小空间。 形成固定接触部件的固定接触对(3a,4a)至(3f',4f')围绕绝缘基板上的特定中心大致点对称地打印。 可移动接触装置设置在固定接触部件的顶部上,当所述装置被推动时,所述可动接触装置适于将每个固定接触对(3a,4a)电连接到(3f',4')上。 所述操作构件设置有用于将包括固定接触对(3a,4a)至(3f',4')和可动接触装置的所述开关元件按压的按压表面,以及用于将所述操作构件自动返回到其原始位置的装置 当它不被推