公开(公告)号：US07186861B2

公开(公告)日：2007-03-06

申请号：US10507605

申请日：2003-03-12

申请人： Wassilios Grammenos ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Andreas Gypser ,  Bernd Müller ,  Joachim Rheinheimer ,  Peter Schäfer ,  Anja Schwögler ,  Jordi Tormo i Blasco ,  Norbert Götz ,  Gisela Lorenz ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Reinhard Stierl

发明人： Wassilios Grammenos ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Andreas Gypser ,  Bernd Müller ,  Joachim Rheinheimer ,  Peter Schäfer ,  Anja Schwögler ,  Jordi Tormo i Blasco ,  Norbert Götz ,  Gisela Lorenz ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Reinhard Stierl

IPC分类号： C07C233/09 ,  A01N37/18

CPC分类号： C07C235/34 ,  A01N37/18 ,  A01N37/36 ,  A01N37/38 ,  C07C233/22 ,  C07C2601/02 ,  C07C2601/08 ,  C07C2601/14

摘要： Z-substituted acrylamides of formula (I), where the substituents have the following meanings: X═H, halogen, alkyl, haloalkyl, alkoxy, haloalkoxy, with X in the 3- or 4-position, n=1 or 2, where X can be different if n=2, R1=alkyl, haloalkyl, cycloalkyl, alkoxy, haloalkoxy, aziridine and oxirane and R2═H, alkyl, haloalkyl, allyl, propargyl or CH2C≡C-alkyl. Methods for production thereof, agents comprising the above and the use thereof for the treatment of plant-pathogenic fungal pests.

摘要翻译： 式（I）的Z-取代的丙烯酰胺，其中取代基具有以下含义：XH，卤素，烷基，卤代烷基，烷氧基，卤代烷氧基，其中X为3-或4-位，n = 1或2，其中X可以 如果n = 2，R 1 =烷基，卤代烷基，环烷基，烷氧基，卤代烷氧基，氮丙啶和环氧乙烷和R 2 -H，烷基，卤代烷基，烯丙基，炔丙基 或CH 2C≡C-烷基。 其制备方法，包含上述物质及其用于治疗植物致病性真菌害虫的用途。

公开(公告)号：US07300908B2

公开(公告)日：2007-11-27

申请号：US10482216

申请日：2002-07-03

申请人： Bernd Müller ,  Hubert Sauter ,  Markus Gewehr ,  Wassilios Grammenos ,  Jordi Tormo i Blasco ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schäfer ,  Frank Schieweck ,  Michael Rack ,  Gisela Lorenz ,  Siegfried Strathmann ,  Eberhard Ammermann ,  Reinhard Stierl

发明人： Bernd Müller ,  Hubert Sauter ,  Markus Gewehr ,  Wassilios Grammenos ,  Jordi Tormo i Blasco ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schäfer ,  Frank Schieweck ,  Michael Rack ,  Gisela Lorenz ,  Siegfried Strathmann ,  Eberhard Ammermann ,  Reinhard Stierl

IPC分类号： C07D487/04 ,  A01N43/48

CPC分类号： C07D487/04 ,  A01N43/90

摘要： Triazolopyrimidines of formula (I), wherein the index and substituents have the following meaning: n=0 or a whole number of 1-5; R=halogen, cyano, hydroxy, cyanate, alkyl, alkenyl, alkinyl, halogenalkyl, halogenalkenyl, alkoxy, alkenyloxy, alkinyloxy, halogenalkoxy, cycloalkyl, cycloalkenyl, cycloalkoxy, alkoxycarbonyl, alkenyloxycarbonyl, alkinyloxycarbonyl, aminocarbonyl, alkylaminocarbonyl, dialkylaminocarbonyl, alkoximinoalkyl, alkenyloximinocarbonyl, alkinyloximinoalkyl, alkylcarbonyl, alkenylcarbonyl, alkinylcarbonyl, cycloalkylcarbonyl or a five to ten membered saturated, partially unsaturated or aromatic heterocycle, containing one to four heteroatoms from the group O, N or S; R1=alkyl, alkenyl, alkinyl, cycloalkyl, cycloalkenyl, phenyl, naphthyl or a five to ten membered saturated, partially unsaturated or aromatic heterocycle, containing one to four heteroatoms from the group O, N or S, R and/or R1 being able to be substituted according to the description; R2=alkyl, alkenyl or alkinyl which can be substituted by halogen, cyano, nitro, alkoxy or alkoxycarbonyl. The invention also relates to a method for the production of said compounds, agents containing same, and the use thereof in controlling noxious fungi

摘要翻译： 式（I）的三唑并嘧啶，其中指数和取代基具有以下含义：n = 0或整数1-5; 环烷氧基，烷氧基羰基，链烯氧基羰基，烷氧基羰基，氨基羰基，烷基氨基羰基，二烷基氨基羰基，肟基烷基，链烯基肟基羰基，烷氧基羰基，烷氧基羰基， 烷基羰基，链烯基羰基，炔基羰基，环烷基羰基或五至十元饱和，部分不饱和或芳族杂环，含有一至四个O，N或S基团的杂原子; R 1 =烷基，烯基，炔基，环烷基，环烯基，苯基，萘基或五至十元饱和，部分不饱和或芳族杂环，其含有一至四个O，N或S ，R和/或R 1能够根据描述进行取代; 可以被卤素，氰基，硝基，烷氧基或烷氧基羰基取代的烷基，烯基或炔基。 本发明还涉及生产所述化合物的方法，含有该化合物的试剂及其在控制有害真菌中的用途

公开(公告)号：US07071334B2

公开(公告)日：2006-07-04

申请号：US10474461

申请日：2002-04-06

申请人： Jordi Tormo i Blasco ,  Hubert Sauter ,  Bernd Müller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schäfer ,  Frank Schieweck ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

发明人： Jordi Tormo i Blasco ,  Hubert Sauter ,  Bernd Müller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schäfer ,  Frank Schieweck ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

IPC分类号： C07D487/04 ,  A01N43/90

CPC分类号： C07D487/04 ,  A01N43/90

摘要： 6-(2-Chloro-6-fluoro-phenyl)-triazolopyrimidines of formula (I), in which R1 and R2 independently denote hydrogen or alkyl, alkenyl, alkynyl, alkadienyl, or haloalkyl, cycloalkyl, bicycloalkyl, phenyl, naphthyl, or 5- or 6-membered heterocyclyl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or 5- or 6-membered heteroaryl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or where R1 and R2 radicals may be unsubstituted or partially or fully halogenated or may be substituted as defined in the description. R1 and R2 together with the interjacent nitrogen atom represent a 5- or 6-membered heterocyclic ring, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which may be substituted; X is cyano, alkoxy, haloalkoxy or alkenyloxy; processes for their preparation, compositions containing them and to their use for combating phytopathogenic fungi

摘要翻译： 式（I）的6-（2-氯-6-氟 - 苯基） - 三唑并嘧啶，其中R 1和R 2独立地表示氢或烷基，烯基， 炔基，链烯基或卤代烷基，环烷基，二环烷基，苯基，萘基或含有1-4个氮原子或1-3个氮原子和一个硫或氧原子的5-或6-元杂环基，或5-或6-元 含有一至四个氮原子或一至三个氮原子和一个硫或氧原子的杂芳基，或其中R 1和R 2基团可以是未取代的或部分或完全的 卤化的或可以如说明书中所定义的取代。 R 1和R 2与中间的氮原子一起表示含有1-4个氮原子或一至三个氮原子的一个5-或6-元杂环，一个 硫或氧原子，其可以被取代; X是氰基，烷氧基，卤代烷氧基或烯氧基; 其制备方法，含有它们的组合物及其用于对抗植物病原真菌的用途

公开(公告)号：US07449471B2

公开(公告)日：2008-11-11

申请号：US11677862

申请日：2007-02-22

申请人： Andreas Gypser ,  Thomas Grote ,  Anja Schwögler ,  Joachim Rheinheimer ,  Frank Schieweck ,  Jordi Tormo i Blasco ,  Ingo Rose ,  Peter Schäfer ,  Markus Gewehr ,  Wassilios Grammenos ,  Bernd Müller ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

发明人： Andreas Gypser ,  Thomas Grote ,  Anja Schwögler ,  Joachim Rheinheimer ,  Frank Schieweck ,  Jordi Tormo i Blasco ,  Ingo Rose ,  Peter Schäfer ,  Markus Gewehr ,  Wassilios Grammenos ,  Bernd Müller ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

IPC分类号： C07D239/42 ,  C07D239/30 ,  A61K31/505 ,  A61K31/506 ,  A01N43/54

CPC分类号： C07D239/42 ,  C07D239/47 ,  C07D239/48 ,  C07D239/52 ,  C07D403/12

摘要： 5-Phenylpyrimidines of the formula I in which the substituents and the index are as defined below: R1,R2 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, alkynyl or haloalkynyl, and R1 and R2 together with the nitrogen atom to which they are attached may also form a saturated or unsaturated ring which may be interrupted by an ether, thio, sulfoxyl or sulfonyl group and may be substituted by one to four groups Ra and/or Rb; R3 is hydrogen, halogen, cyano, alkyl, haloalkyl, alkoxy, haloalkoxy or alkenyloxy; R4 is hydrogen, halogen, cyano, hydroxyl, mercapto, azido, alkyl, alkenyl, alkynyl, haloalkyl, alkoxy, alkenyloxy, alkynyloxy, haloalkoxy, alkylthio, alkenylthio, alkynylthio, haloalkylthio, —ON═CRaRb, —CRc═NORa, —NRcN═CRaRb, —NRaRb, —NRcNRaRb, —NORa, —NRcC(═NRc′)NRaRb, —NRcC(═O)NRaRb, —NRaC(═O)Rc, —NRaC(═NORc)Rc′, —OC(═O)Rc, —C(═NORc)NRaRb, —CRc(═NNRaRb), —C (═O)NRaRb or —C(═O)Rc; in which Ra, Rb and Rc are as defined in the description; X is halogen, alkyl, alkoxy or haloalkyl; and m is an integer from 1 to 5 ; processes for preparing these compounds, compositions comprising them and their use for controlling harmful fungi are described.

公开(公告)号：US06855718B2

公开(公告)日：2005-02-15

申请号：US10416467

申请日：2001-11-09

申请人： Jordi Tormo i Blasco ,  Klaus Ditrich ,  Hubert Sauter ,  Oliver Cullmann ,  Markus Gewehr ,  Wassilios Grammenos ,  Bernd Müller ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schäfer ,  Frank Schieweck ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

发明人： Jordi Tormo i Blasco ,  Klaus Ditrich ,  Hubert Sauter ,  Oliver Cullmann ,  Markus Gewehr ,  Wassilios Grammenos ,  Bernd Müller ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schäfer ,  Frank Schieweck ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  C07B53/00 ,  C07C209/62 ,  C07C211/03 ,  C07D487/04

CPC分类号： C07D487/04 ,  A01N43/90

摘要： A 7-(R)-Aminotriazolopyrimidines of formula I where the substituents and index are as defined below: R1 is hydrogen or methyl; R2 is methyl; R3 is C2-C10-alkyl, C1-C4-alkoxymethyl, C3-C10-cycloalkyl; Y is halogen, cyano, C1-C4-alkyl or C1-C4-alkoxy; where * is a center of chirality in the R configuration, processes for their preparation, compositions comprising them and their use for controlling harmful fungi.

摘要翻译： 式I的7-（R） - 氨基三唑并嘧啶，其中取代基和指数如下所定义：R 1是氢或甲基; R 2是甲基; R 3是C 2 -C 10 - 烷基，C 1 -C 4 - 烷氧基甲基，C 3 -C 10 - 环烷基; Y是卤素，氰基，C 1 -C 4 - 烷基或C 1 -C 4 - 烷氧基;其中*是R构型的手性中心，其制备方法，包含它们的组合物及其用途 用于控制有害真菌。

公开(公告)号：US07465735B2

公开(公告)日：2008-12-16

申请号：US10495280

申请日：2002-11-15

申请人： Andreas Gypser ,  Thomas Grote ,  Anja Schwögler ,  Joachim Rheinheimer ,  Frank Schieweck ,  Jordi Tormo i Blasco ,  Ingo Rose ,  Peter Schäfer ,  Markus Gewehr ,  Wassilios Grammenos ,  Bernd Müller ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

发明人： Andreas Gypser ,  Thomas Grote ,  Anja Schwögler ,  Joachim Rheinheimer ,  Frank Schieweck ,  Jordi Tormo i Blasco ,  Ingo Rose ,  Peter Schäfer ,  Markus Gewehr ,  Wassilios Grammenos ,  Bernd Müller ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

IPC分类号： C07D239/42 ,  C07D239/46 ,  C07D239/48 ,  C07D239/52 ,  C07D401/12 ,  C07D403/12 ,  A61K31/505 ,  A61K31/506 ,  A01N43/54

CPC分类号： C07D239/42 ,  C07D239/47 ,  C07D239/48 ,  C07D239/52 ,  C07D403/12

摘要： 5-Phenylpyrimidines, their preparation, compositions comprising them and their use 5-Phenylpyrimidines of the formula I in which the substituents and the index are as defined below: R1,R2 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, alkynyl or haloalkynyl, and R1 and R2 together with the nitrogen atom to which they are attached may also form a saturated or unsaturated ring which may be interrupted by an ether, thio, sulfoxyl or sulfonyl group and may be substituted by one to four groups Ra and/or Rb; R3 is hydrogen, halogen, cyano, alkyl, haloalkyl, alkoxy, haloalkoxy or alkenyloxy; R4 is hydrogen, halogen, cyano, hydroxyl, mercapto, azido, alkyl, alkenyl, alkynyl, haloalkyl, alkoxy, alkenyloxy, alkynyloxy, haloalkoxy, alkylthio, alkenylthio, alkynylthio, haloalkylthio, —ON═CRaRb, —CRc═NORa, —NRcN═CRaRb, —NRaRb, —NRcNRaRb, —NORa, —NRcC(═NRc′)NRaRb, —NRcC(═O)NRaRb, —NRaC(═O)Rc, —NRaC(═NORc)Rc′, —OC(═O)Rc, —C(═NORc)NRaRb, —CRc(═NNRaRb), —C(═O)NRaRb or —C(═O)Rc; in which Ra, Rb and Rc are as defined in the description; X is halogen, alkyl, alkoxy or haloalkyl; and m is an integer from 1 to 5; processes for preparing these compounds, compositions comprising them and their use for controlling harmful fungi are described.

摘要翻译： 其中取代基和指数如下定义的式I的5-苯基嘧啶：R1，R2是氢，烷基，卤代烷基，环烷基，卤代环烷基，烯基，卤代烯基，炔基或卤代炔基，R1和R2与氮原子一起 它们所连接的也可以形成可被醚，硫代，亚砜基或磺酰基中断的饱和或不饱和环，并且可以被一至四个基团R a和/或R b取代; R3是氢，卤素，氰基，烷基，卤代烷基，烷氧基，卤代烷氧基或烯氧基; R4是氢，卤素，氰基，羟基，巯基，叠氮基，烷基，烯基，炔基，卤代烷基，烷氧基，烯氧基，炔氧基，卤代烷氧基，烷硫基，烯硫基，炔硫基，卤代烷硫基，-ON-CRaRb，-CRc-NORa，-NRcN -CRaRb，-NRaRb，-NRcNRaRb，-NORa，-NRcC（-NRc'）NRaRb，-NRcC（-O）NRaRb，-NRaC（-O）Rc，-NRaC（-NORc）Rc'，-OC（ - O）R c，-C（-NOR c）NR a R b，-CR c（-NNR a R b）， - C（-O）NR a R b或-C（-O）R c; 其中Ra，Rb和Rc如说明书中所定义; X是卤素，烷基，烷氧基或卤代烷基; m为1〜5的整数。 描述了制备这些化合物的方法，包含它们的组合物及其用于控制​​有害真菌的用途。

公开(公告)号：US07307172B2

公开(公告)日：2007-12-11

申请号：US10484250

申请日：2002-07-16

申请人： Jordi Tormo i Blasco ,  Hubert Sauter ,  Bernd Müller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schäfer ,  Frank Schieweck ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl ,  Günter Krummel

发明人： Jordi Tormo i Blasco ,  Hubert Sauter ,  Bernd Müller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schäfer ,  Frank Schieweck ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl ,  Günter Krummel

IPC分类号： A61K31/41 ,  A01N43/653 ,  C07D249/00

CPC分类号： C07D487/04 ,  A01N43/90

摘要： The invention relates to 7-amino triazolopyrimidines of formula (I), in which the substituents have the following meanings: R1, R2 represent hydrogen, alkyl, alkenyl, alkynyl, cycloalkyl, phenyl, naphthyl; or 5-membered or 6-membered heterocyclyl containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom; or 5-membered or 6-membered heteroaryl containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or R1 and R2 can, together with the nitrogen atom, which binds them, form a 5-membered or 6-membered ring containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom; R3 represents alkyl, alkenyl, alkynyl, cycloalkyl, phenylalkyl and alkyl halide; whereby R3 and R2 can be unsubstituted or partially or completely substituted according to the description; X represents halogen, cyano, alkoxy, alkyl halide, phenyl or phenyl that is substituted by Ra. The invention also relates to methods and intermediate products for producing said compounds, to agents containing the same, and to their use.

摘要翻译： 本发明涉及式（I）的7-氨基三唑并嘧啶，其中取代基具有以下含义：R 1，R 2表示氢，烷基，烯基，炔基 ，环烷基，苯基，萘基; 或含有1至4个氮原子或1至3个氮原子和1个硫或氧原子的5元或6元杂环基; 或含有1至4个氮原子或1至3个氮原子和1个硫或氧原子的5元或6元杂芳基，或R 1和R 2可以， 与它们结合的氮原子一起形成含有一至四个氮原子或一至三个氮原子和一个硫或氧原子的五元或六元环; R 3表示烷基，烯基，炔基，环烷基，苯基烷基和烷基卤; 根据描述，R 3和R 2可以是未取代的或部分或完全取代的; X表示卤素，氰基，烷氧基，烷基卤，苯基或被R a取代的苯基。 本发明还涉及用于生产所述化合物的方法和中间产物，含有该化合物的试剂及其用途。

公开(公告)号：US07038047B2

公开(公告)日：2006-05-02

申请号：US10483599

申请日：2002-07-08

申请人： Jordi Tormo i Blasco ,  Hubert Sauter ,  Bernd Müller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schäfer ,  Frank Schieweck ,  Michael Rack ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

发明人： Jordi Tormo i Blasco ,  Hubert Sauter ,  Bernd Müller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schäfer ,  Frank Schieweck ,  Michael Rack ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

IPC分类号： C07D487/04 ,  C07C69/612 ,  A01N43/90

CPC分类号： C07D487/04 ,  A01N43/90

摘要： Substituted 6-(2-methoxy-phenyl)-triazolopyrimidines of formula I in which R1 and R2 independently denote hydrogen or alkyl, alkenyl, alkynyl, or alkadienyl, haloalkyl, haloalkenyl, cycloalkyl, phenyl, naphthyl, or 5- or 6-membered heterocyclyl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or 5- or 6-membered heteroaryl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or where R1 and R2 radicals may be unsubstituted or substituted as defined in the description, or R1 and R2 together with the interjacent nitrogen atom represent a 5- or 6-membered heterocyclic ring, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which may be substituted; L1, L2 independently denote hydrogen or halogen, provided that at least one from L1 or L2 is halogen; X is halogen, cyano, alkyl, alkoxy, haloalkoxy or alkenyloxy; processes for their preparation, compositions containing them and to their use for combating phytopathogenic fungi.

摘要翻译： 其中R 1和R 2的取代的6-（2-甲氧基 - 苯基） - 三唑并嘧啶独立地表示氢或烷基，烯基，炔基或链二烯基，卤代烷基 含有1-4个氮原子或一至三个氮原子和一个硫或氧原子的卤代烯基，环烷基，苯基，萘基或5-或6-元杂环基，或含有一至四个的5-或6-元杂芳基 氮原子或一至三个氮原子和一个硫或氧原子，或其中R 1和R 2基团可以是未取代的或如说明书中定义的取代的，或R R 1和R 2与中间的氮原子一起表示含有1-4个氮原子或一至三个氮原子和一个硫原子的5-或6-元杂环 或氧原子，其可以被取代; L 1，L 2，L 2独立地表示氢或卤素，条件是至少一个L 1或L 2， 是卤素; X是卤素，氰基，烷基，烷氧基，卤代烷氧基或烯氧基; 其制备方法，含有它们的组合物及其用于对抗植物病原真菌的用途。

公开(公告)号：US06576595B1

公开(公告)日：2003-06-10

申请号：US10251783

申请日：2002-09-23

申请人： Ingo Rose ,  Jordi Tormo i Blasco ,  Markus Gewehr ,  Wassilios Grammenos ,  Bernd Müller ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Thomas Grote ,  Andreas Gypser ,  Eberhard Ammermann ,  Gisela Lorenz ,  Reinhard Stierl ,  Siegfried Strathmann

发明人： Ingo Rose ,  Jordi Tormo i Blasco ,  Markus Gewehr ,  Wassilios Grammenos ,  Bernd Müller ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Thomas Grote ,  Andreas Gypser ,  Eberhard Ammermann ,  Gisela Lorenz ,  Reinhard Stierl ,  Siegfried Strathmann

IPC分类号： A01N4316

CPC分类号： C07D311/86 ,  A01N43/16 ,  C07C45/46 ,  C07C45/54 ,  C07C49/84

摘要： Xanthone derivatives of the formula I where the index and the variables are as defined below: n is 0, 1 or 2; R1 is alkyl or haloalkyl; R2,R3 are alkoxy, alkenyloxy or alkynyloxy, or R2 and R3 together form an unsubstituted or substituted oxyalkyleneoxy group; R4 is halogen, cyano, hydroxyl, amino, mercapto, alkyl, haloalkyl, alkoxy, haloalkoxy, alkylthio, haloalkylthio, alkylcarbonyloxy or alkylcarbonylthio; R5 is a group R4, where the groups R5 may be different if n=2; X, Y are oxygen or sulfur; Processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi are described.

摘要翻译： 式I的呫吨酮衍生物，其中指数和变量如下：n为0,1或2; R 1为烷基或卤代烷基; R 2为烷氧基，烯氧基或炔氧基，或者R 2和R 3一起形成未取代或取代的 氧基亚烷基氧基; R4是卤素，氰基，羟基，氨基，巯基，烷基，卤代烷基，烷氧基，卤代烷氧基，烷硫基，卤代烷硫基，烷基羰基氧基或烷基羰基硫基; R5是R4基团，其中如果n = 2，基团R5可以不同; X ，Y为氧或硫;制备这些化合物的方法，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US06767923B2

公开(公告)日：2004-07-27

申请号：US10282023

申请日：2002-10-29

申请人： Ingo Rose ,  Jordi Tormo i Blasco ,  Markus Gewehr ,  Wassilios Grammenos ,  Bernd Müller ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Thomas Grote ,  Andreas Gypser ,  Eberhard Ammermann ,  Gisela Lorenz ,  Reinhard Stierl ,  Siegfried Strathmann ,  Paul Carter ,  Jürgen Curtze

发明人： Ingo Rose ,  Jordi Tormo i Blasco ,  Markus Gewehr ,  Wassilios Grammenos ,  Bernd Müller ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Thomas Grote ,  Andreas Gypser ,  Eberhard Ammermann ,  Gisela Lorenz ,  Reinhard Stierl ,  Siegfried Strathmann ,  Paul Carter ,  Jürgen Curtze

IPC分类号： A61K31215

CPC分类号： C07C323/25 ,  A01N31/16 ,  C07C43/23 ,  C07C69/017

摘要： Benzhydryl derivatives of the formula I, where the index and the variables are as defined below: X is oxygen or sulfur; R1, R3 are halogen, cyano, nitro, hydroxyl, mercapto, amino, alkyl, alkenyl, alkynyl, alkoxy, alkenyloxy, alkynyloxy, alkylcarbonyloxy, formyloxy, alkylthio, alkenylthio, alkynylthio, alkylamino, dialkylamino, alkylcarbonyl or formyl, where the carbon atoms in the radicals mentioned may be partially or fully halogenated; R2 is halogen, cyano, nitro, hydroxyl, mercapto, amino, alkyl, alkoxy, haloalkyl or haloalkoxy, where the groups R2 may be different if n=2; R4 is alkyl, alkenyl or alkynyl, where the carbon atoms in these radicals may be unsubstituted or partially or fully halogenated; R5, R6 are hydroxyl, alkyl, alkenyl, haloalkyl, haloalkenyl, alkoxy, alkenyloxy, haloalkoxy, haloalkenyloxy, cycloalkyl, cycloalkylalkyl, cycloalkoxy or cycloalkylalkoxy; n is 0, 1 or 2; processes for preparing the compounds I, compositions comprising them and their use for controlling phytopathogenic harmful fungi are described.

摘要翻译： 式I的二苯甲基衍生物，其中指数和变量如下定义：X是氧或硫; R 1，R 3是卤素，氰基，硝基，羟基，巯基，氨基，烷基，烯基， 炔基，烷氧基，烯氧基，炔氧基，烷基羰基氧基，甲酰氧基，烷硫基，烯硫基，炔硫基，烷基氨基，二烷基氨基，烷基羰基或甲酰基，其中所述基团中的碳原子可以被部分或完全卤化; R 2是卤素，氰基， 硝基，羟基，巯基，氨基，烷基，烷氧基，卤代烷基或卤代烷氧基，其中如果n = 2，基团R 2可以不同; R 4是烷基，烯基或炔基，其中这些基团中的碳原子 R 5为羟基，烷基，烯基，卤代烷基，卤代烯基，烷氧基，烯氧基，卤代烷氧基，卤代烯氧基，环烷基，环烷基烷基，环烷氧基或环烷基烷氧基; n为0,1或 2;制备化合物I的方法，包含它们的组合物及其用途 描述了植物病原性有害真菌。