公开(公告)号：US06767923B2

公开(公告)日：2004-07-27

申请号：US10282023

申请日：2002-10-29

申请人： Ingo Rose ,  Jordi Tormo i Blasco ,  Markus Gewehr ,  Wassilios Grammenos ,  Bernd Müller ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Thomas Grote ,  Andreas Gypser ,  Eberhard Ammermann ,  Gisela Lorenz ,  Reinhard Stierl ,  Siegfried Strathmann ,  Paul Carter ,  Jürgen Curtze

发明人： Ingo Rose ,  Jordi Tormo i Blasco ,  Markus Gewehr ,  Wassilios Grammenos ,  Bernd Müller ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Thomas Grote ,  Andreas Gypser ,  Eberhard Ammermann ,  Gisela Lorenz ,  Reinhard Stierl ,  Siegfried Strathmann ,  Paul Carter ,  Jürgen Curtze

IPC分类号： A61K31215

CPC分类号： C07C323/25 ,  A01N31/16 ,  C07C43/23 ,  C07C69/017

摘要： Benzhydryl derivatives of the formula I, where the index and the variables are as defined below: X is oxygen or sulfur; R1, R3 are halogen, cyano, nitro, hydroxyl, mercapto, amino, alkyl, alkenyl, alkynyl, alkoxy, alkenyloxy, alkynyloxy, alkylcarbonyloxy, formyloxy, alkylthio, alkenylthio, alkynylthio, alkylamino, dialkylamino, alkylcarbonyl or formyl, where the carbon atoms in the radicals mentioned may be partially or fully halogenated; R2 is halogen, cyano, nitro, hydroxyl, mercapto, amino, alkyl, alkoxy, haloalkyl or haloalkoxy, where the groups R2 may be different if n=2; R4 is alkyl, alkenyl or alkynyl, where the carbon atoms in these radicals may be unsubstituted or partially or fully halogenated; R5, R6 are hydroxyl, alkyl, alkenyl, haloalkyl, haloalkenyl, alkoxy, alkenyloxy, haloalkoxy, haloalkenyloxy, cycloalkyl, cycloalkylalkyl, cycloalkoxy or cycloalkylalkoxy; n is 0, 1 or 2; processes for preparing the compounds I, compositions comprising them and their use for controlling phytopathogenic harmful fungi are described.

摘要翻译： 式I的二苯甲基衍生物，其中指数和变量如下定义：X是氧或硫; R 1，R 3是卤素，氰基，硝基，羟基，巯基，氨基，烷基，烯基， 炔基，烷氧基，烯氧基，炔氧基，烷基羰基氧基，甲酰氧基，烷硫基，烯硫基，炔硫基，烷基氨基，二烷基氨基，烷基羰基或甲酰基，其中所述基团中的碳原子可以被部分或完全卤化; R 2是卤素，氰基， 硝基，羟基，巯基，氨基，烷基，烷氧基，卤代烷基或卤代烷氧基，其中如果n = 2，基团R 2可以不同; R 4是烷基，烯基或炔基，其中这些基团中的碳原子 R 5为羟基，烷基，烯基，卤代烷基，卤代烯基，烷氧基，烯氧基，卤代烷氧基，卤代烯氧基，环烷基，环烷基烷基，环烷氧基或环烷基烷氧基; n为0,1或 2;制备化合物I的方法，包含它们的组合物及其用途 描述了植物病原性有害真菌。

公开(公告)号：US20060211711A1

公开(公告)日：2006-09-21

申请号：US10550571

申请日：2004-03-30

申请人： Jordi Blasco ,  Carsten Blettner ,  Bernd Müller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Anja Schwögler ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schöfl ,  Reinhard Stierl

发明人： Jordi Blasco ,  Carsten Blettner ,  Bernd Müller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Anja Schwögler ,  Maria Scherer ,  Siegfried Strathmann ,  Ulrich Schöfl ,  Reinhard Stierl

IPC分类号： A61K31/519 ,  C07D487/04 ,  A01N43/90

CPC分类号： C07D487/04 ,  A01N43/90

摘要： 7-alkinylamino-triazolopyrimidins of formula (I), wherein the substituents have the following meanings: L=halogen, alkyl, halogenalkyl, alkoxy, amino, NHR, NR2, cyano, S(O)nA1 or C(O)A2; R=alkyl or alkylcarbonyl, A1=hydrogen, hydroxy, alkyl, alkylamino or aialkylamino; n=0, 1 or 2; A2=alkenyl, alkoxy, halogenalkoxy or one of the groups cited in A1; m=1, 2, 3, 4 or 5, whereby at least one group L is present in an ortho-position to the bond with the triazolopyrimidine skeleton; X=halogen, cyano, alkyl, halogenalkyl or alkoxy; R1=hydrogen or alkyl; R2=alkinyl which can be unsubstituted or substituted according to the description. The invention also relates to methods for the production of said compounds, agents containing said compounds and the use thereof to combat harmful phytopathogenic fungi.

摘要翻译： 式（I）的7-烷基氨基 - 三唑并嘧啶类，其中取代基具有以下含义：L =卤素，烷基，卤代烷基，烷氧基，氨基，NHR，NR 2，氰基，S（O） 或者C（O）A 2 O 2。 R =烷基或烷基羰基，A 1〜H 2，羟基，烷基，烷基氨基或亚烷基氨基; n = 0,1或2; 链烯基，烷氧基，卤代烷氧基或A 1中引用的基团之一; m = 1,2,3,4或5，其中至少一个基团L存在于与三唑并嘧啶骨架的键的邻位; X =卤素，氰基，烷基，卤代烷基或烷氧基; R 1 =氢或烷基; R 2 =炔基，其可以是未取代的或根据描述取代的。 本发明还涉及生产所述化合物的方法，含有所述化合物的试剂及其用于对抗有害植物病原真菌的用途。

公开(公告)号：US07820647B2

公开(公告)日：2010-10-26

申请号：US11596891

申请日：2005-05-17

申请人： Anja Schwögler ,  Frank Schieweck ,  Joachim Rheinheimer ,  Markus Gewehr ,  Bernd Müller ,  Thomas Grote ,  Wassilios Grammenos ,  Udo Hünger ,  Carsten Blettner ,  Peter Schäfer ,  Oliver Wagner ,  Reinhard Stierl ,  Ulrich Schöfl ,  Siegfried Strathmann ,  Maria Scherer

发明人： Anja Schwögler ,  Frank Schieweck ,  Joachim Rheinheimer ,  Markus Gewehr ,  Bernd Müller ,  Thomas Grote ,  Wassilios Grammenos ,  Udo Hünger ,  Carsten Blettner ,  Peter Schäfer ,  Oliver Wagner ,  Reinhard Stierl ,  Ulrich Schöfl ,  Siegfried Strathmann ,  Maria Scherer

IPC分类号： C07D239/48 ,  C07D403/04 ,  A01N43/54 ,  A01N43/58 ,  A01N43/34 ,  A01P3/00

CPC分类号： C07D401/04 ,  C07D403/04

摘要： The invention relates to 2-substituted pyrimidines of the formula I in which the index n and the substituents L and R1 to R3 are as defined in the description and X is a group —CH—Ra, —N—Rb—, —O— or —S—; Ra may be hydrogen, halogen, C1-C6-alkyl, C1-C6-alkoxy, cyano or C1-C6-alkoxycarbonyl; Rb is hydrogen, C1-C6-alkyl or C3-C6-cycloalkyl; T is a group —CH—Ra—; p is an integer from 1 to 4; Y is a group —CH—Ra— or —N—Rb—, o is 0 or 1; Z is O, S or a group N(Rc) Rc is hydrogen, C1-C6-alkyl or C1-C6-alkoxy, and to processes for their preparation, to pesticidal compositions comprising them and to their use as pesticides.

摘要翻译： 本发明涉及式I的2-取代嘧啶，其中指数n和取代基L和R1至R3如说明书中所定义，X为基团-CH-Ra，-N-Rb-，-O- 或-S-; R a可以是氢，卤素，C 1 -C 6 - 烷基，C 1 -C 6 - 烷氧基，氰基或C 1 -C 6 - 烷氧基羰基; R b是氢，C 1 -C 6 - 烷基或C 3 -C 6 - 环烷基; T是基团-CH-R a; p是1至4的整数; Y是基团-CH-R a或-N-R b - ，o是0或1; Z是O，S或基团N（R c）R c是氢，C 1 -C 6烷基或C 1 -C 6 - 烷氧基，并且其制备方法，包含它们的杀虫组合物和它们作为农药的用途。

公开(公告)号：US20050261314A1

公开(公告)日：2005-11-24

申请号：US10484250

申请日：2002-07-16

申请人： Jordi i Blasco ,  Hubert Sauter ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schafer ,  Frank Schieweck ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

发明人： Jordi i Blasco ,  Hubert Sauter ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schafer ,  Frank Schieweck ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  C07D487/04

CPC分类号： C07D487/04 ,  A01N43/90

摘要： The invention relates to 7-amino triazolopyrimidines of formula (I), in which the substituents have the following meanings: R1, R2 represent hydrogen, alkyl, alkenyl, alkynyl, cycloalkyl, phenyl, naphthyl; or 5-membered or 6-membered heterocyclyl containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom; or 5-membered or 6-membered heteroaryl containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or R1 and R2 can, together with the nitrogen atom, which binds them, form a 5-membered or 6-membered ring containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom; R3 represents alkyl, alkenyl, alkynyl, cycloalkyl, phenylalkyl and alkyl halide; whereby R3 and R2 can be unsubstituted or partially or completely substituted according to the description; X represents halogen, cyano, alkoxy, alkyl halide, phenyl or phenyl that is substituted by Ra. The invention also relates to methods and intermediate products for producing said compounds, to agents containing the same, and to their use.

摘要翻译： 本发明涉及式（I）的7-氨基三唑并嘧啶，其中取代基具有以下含义：R 1，R 2表示氢，烷基，烯基，炔基 ，环烷基，苯基，萘基; 或含有1至4个氮原子或1至3个氮原子和1个硫或氧原子的5元或6元杂环基; 或含有1至4个氮原子或1至3个氮原子和1个硫或氧原子的5元或6元杂芳基，或R 1和R 2可以， 与它们结合的氮原子一起形成含有一至四个氮原子或一至三个氮原子和一个硫或氧原子的五元或六元环; R 3表示烷基，烯基，炔基，环烷基，苯基烷基和烷基卤; 根据描述，R 3和R 2可以是未取代的或部分或完全取代的; X表示卤素，氰基，烷氧基，烷基卤，苯基或被R a取代的苯基。 本发明还涉及用于生产所述化合物的方法和中间产物，含有该化合物的试剂及其用途。

公开(公告)号：US20050090665A1

公开(公告)日：2005-04-28

申请号：US10482216

申请日：2002-07-03

申请人： Bernd Muller ,  Hubert Sauter ,  Markus Gewehr ,  Wassilios Grammenos ,  Jordi I Blasco ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schafer ,  Frank Schieweck ,  Michael Rack ,  Gisela Lorenz ,  Siegfried Strathmann ,  Eberhard Ammermann ,  Reinhard Stierl

发明人： Bernd Muller ,  Hubert Sauter ,  Markus Gewehr ,  Wassilios Grammenos ,  Jordi I Blasco ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schafer ,  Frank Schieweck ,  Michael Rack ,  Gisela Lorenz ,  Siegfried Strathmann ,  Eberhard Ammermann ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  C07D487/04

CPC分类号： C07D487/04 ,  A01N43/90

摘要： Triazolopyrimidines of formula (I), wherein the index and substituents have the following meaning: n=0 or a whole number of 1-5; R=halogen, cyano, hydroxy, cyanate, alkyl, alkenyl, alkinyl, halogenalkyl, halogenalkenyl, alkoxy, alkenyloxy, alkinyloxy, halogenalkoxy, cycloalkyl, cycloalkenyl, cycloalkoxy, alkoxycarbonyl, alkenyloxycarbonyl, alkinyloxycarbonyl, aminocarbonyl, alkylaminocarbonyl, dialkylaminocarbonyl, alkoximinoalkyl, alkenyloximinocarbonyl, alkinyloximinoalkyl, alkylcarbonyl, alkenylcarbonyl, alkinylcarbonyl, cycloalkylcarbonyl or a five to ten membered saturated, partially unsaturated or aromatic heterocycle, containing one to four heteroatoms from the group O, N or S; R1=alkyl, alkenyl, alkinyl, cycloalkyl, cycloalkenyl, phenyl, naphthyl or a five to ten membered saturated, partially unsaturated or aromatic heterocycle, containing one to four heteroatoms from the group O, N or S, R and/or R1 being able to be substituted according to the description; R2=alkyl, alkenyl or alkinyl which can be substituted by halogen, cyano, nitro, alkoxy or alkoxycarbonyl. The invention also relates to a method for the production of said compounds, agents containing same, and the use thereof in controlling noxious fungi.

摘要翻译： 式（I）的三唑并嘧啶，其中指数和取代基具有以下含义：n = 0或整数1-5; 环烷氧基，烷氧基羰基，链烯氧基羰基，烷氧基羰基，氨基羰基，烷基氨基羰基，二烷基氨基羰基，肟基烷基，链烯基肟基羰基，烷氧基羰基，烷氧基羰基， 烷基羰基，链烯基羰基，炔基羰基，环烷基羰基或五至十元饱和，部分不饱和或芳族杂环，含有一至四个O，N或S基团的杂原子; R 1 =烷基，烯基，炔基，环烷基，环烯基，苯基，萘基或五至十元饱和，部分不饱和或芳族杂环，其含有一至四个O，N或S ，R和/或R 1能够根据描述进行取代; 可以被卤素，氰基，硝基，烷氧基或烷氧基羰基取代的烷基，烯基或炔基。 本发明还涉及生产所述化合物的方法，含有该化合物的试剂及其在控制有害真菌中的用途。

公开(公告)号：US20060135538A1

公开(公告)日：2006-06-22

申请号：US11340977

申请日：2006-01-30

申请人： Jordi Tormo Blasco ,  Klaus Ditrich ,  Hubert Sauter ,  Oliver Cullmann ,  Markus Gewehr ,  Wassilios Grammenos ,  Bernd Muller ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schafer ,  Frank Schieweck ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

发明人： Jordi Tormo Blasco ,  Klaus Ditrich ,  Hubert Sauter ,  Oliver Cullmann ,  Markus Gewehr ,  Wassilios Grammenos ,  Bernd Muller ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schafer ,  Frank Schieweck ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  C07D487/04

CPC分类号： C07D487/04 ,  A01N43/90

摘要： 7-(R)-Aminotriazolopyrimidines of the formula I where the substituents and the index are as defined below: R1 is hydrogen or methyl; R2 is methyl; R3 is C2-C1o-alkyl, C1-C4-alkoxymethyl, C3-C1o-cycloalkyl; R4 is halogen, Cl-C4-alkyl, C1-C4-haloalkyl or Cl-C4-alkoxy; n is a number from 1 to 5; Y is halogen, cyano, Cl-C4-alkyl or Cl-C4-alkoxy; where * is a center of chirality in the R configuration, processes for preparing these compounds, compositions comprising them and their use for controlling harmful fungi are described.

摘要翻译： 7-（R） - 取代基和指数如下所定义的式I的氨基三唑并嘧啶：R 1是氢或甲基; R 2是甲基; R 3是C 1 -C 2烷基，C 1 -C 4烷基，C 1 -C 4烷基，C 1 -C 4烷基， 亚烷基氧基甲基，C 3 -C 30环烷基; R 4是卤素，C 1 -C 4 - 烷基，C 1 -C 4 - 卤代烷基或C 1 -C 4 - C 4 - 烷氧基; n是从1到5的数字; Y是卤素，氰基，C 1 -C 4 - 烷基或C 1 -C 4 - 烷氧基; 其中*是R构型的手性中心，描述了制备这些化合物的方法，包含它们的组合物及其用于控制​​有害真菌的用途。

公开(公告)号：US20060217400A1

公开(公告)日：2006-09-28

申请号：US10539559

申请日：2003-12-17

申请人： Bernd Müller ,  Jordi Blasco ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Anja Schwögler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schöfl ,  Reinhard Stierl

发明人： Bernd Müller ,  Jordi Blasco ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Anja Schwögler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schöfl ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  C07D487/04

CPC分类号： C07D487/04 ,  A01N43/90

摘要： Triazolopyrimidines of the formula I in which the index n and the substituents R1, R2 and R3 are as defined in the description, and processes for preparing these compounds, compositions comprising them and their use for controlling harmful fungi are described.

摘要翻译： 其中指数n和取代基R 1，R 2和R 3的式I的三唑并嘧啶如说明书中所定义，以及 描述了制备这些化合物的方法，包含它们的组合物及其用于控制​​有害真菌的用途。

公开(公告)号：US06593315B2

公开(公告)日：2003-07-15

申请号：US09896971

申请日：2001-07-02

申请人： Andreas Gypser ,  Thomas Grote ,  Joachim Rheinheimer ,  Ingo Rose ,  Oliver Cullmann ,  Markus Gewehr ,  Wassilios Grammenos ,  Jordi Tormo i Blasco ,  Bernd Müller ,  Hubert Sauter ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

发明人： Andreas Gypser ,  Thomas Grote ,  Joachim Rheinheimer ,  Ingo Rose ,  Oliver Cullmann ,  Markus Gewehr ,  Wassilios Grammenos ,  Jordi Tormo i Blasco ,  Bernd Müller ,  Hubert Sauter ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

IPC分类号： A01N3736

CPC分类号： C07C251/86 ,  A01N37/50

摘要： Salicylic acid derivatives of the formula I, where the index and the substituents have the following meanings: X is halogen, NO2, cyano, alkyl or alkoxy; m is 0, 1, 2 or 3, it being possible for the substituents X to be different from each other if n is greater than 1; A is OH, alkoxy, NH2, NHCH3 or N(CH3)2; R1 is phenyl, naphthyl, cycloalkyl, 5-membered or 6-membered hetaryl or 5-membered or 6-membered heterocyclyl, comprising one to three N atoms and/or one O or S atom or one or two O and/or S atoms, the ring systems being unsubstituted or substituted; R2 is hydrogen, cyano, alkyl, alkenyl, alkynyl, haloalkyl, alkoxy or alkylthio, processes for the preparation of these compounds, compositions comprising them, and their use for controlling harmful fungi.

摘要翻译： 式I的水杨酸衍生物，其中指数和取代基具有以下含义：X是卤素，NO 2，氰基，烷基或烷氧基; m是0,1,2或3，取代基X可以是 如果n大于1，A是不同的; A是OH，烷氧基，NH2，NHCH3或N（CH3）2; R1是苯基，萘基，环烷基，5元或6元杂芳基或5元或6- 包括一至三个N原子和/或一个O或S原子或一个或两个O和/或S原子，所述环系是未取代或取代的; R2是氢，氰基，烷基，烯基，炔基，卤代烷基， 烷氧基或烷硫基，制备这些化合物的方法，包含它们的组合物及其用于控制​​有害真菌的用途。

公开(公告)号：US06455515B2

公开(公告)日：2002-09-24

申请号：US09879902

申请日：2001-06-14

申请人： Andreas Gypser ,  Thomas Grote ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schäfer ,  Oliver Cullmann ,  Markus Gewehr ,  Wassilios Grammenos ,  Jordi Tormo i Blasco ,  Bernd Müller ,  Hubert Sauter ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

发明人： Andreas Gypser ,  Thomas Grote ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schäfer ,  Oliver Cullmann ,  Markus Gewehr ,  Wassilios Grammenos ,  Jordi Tormo i Blasco ,  Bernd Müller ,  Hubert Sauter ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

IPC分类号： A01N3740

CPC分类号： C07C255/66 ,  A01N37/40 ,  A01N37/46 ,  A01N47/20 ,  A01N47/30 ,  C07C251/86

摘要： Salicylohydrazide derivatives of the formula I in which the index and the substituents have the following meanings: X is halogen, NO2, cyano, alkyl or alkoxy; m is 0, 1, 2 or 3, it being possible for the substituents X to differ from each other if n is greater than 1; R1 is NO2, NH2 or NH—CO—A; A is hydrogen, alkyl, alkoxy, NH2, NHCH3 or N(CH3)2; R2 is hydrogen, cyano, alkyl, alkenyl, alkynyl, haloalkyl, alkoxy or alkylthio; it being possible for the hydrocarbon radicals to be unsubstituted or substituted, R3 is phenyl, naphthyl, cycloalkyl, 5-membered or 6-membered hetaryl or 5-membered or 6-membered heterocyclyl containing one to three N atoms and/or one O or S atom or one or two O and/or S atoms, the ring systems being unsubstituted or substituted; the preparation of these compounds, compositions comprising them, and their use for controlling harmful fungi.

摘要翻译： 指数和取代基具有以下含义的式Iin的磺酰肼衍生物：X是卤素，NO 2，氰基，烷基或烷氧基; m是0,1,2或3，取代基X可能与每个 另外，如果n大于1，则R1为NO2，NH2或NH-CO-A; A为氢，烷基，烷氧基，NH2，NHCH3或N（CH3）2; R2为氢，氰基，烷基，烯基，炔基， 卤代烷基，烷氧基或烷硫基;烃基可以是未取代的或取代的，R3是苯基，萘基，环烷基，含有1至3个N原子的5元或6元杂芳基或5元或6元杂环基 和/或一个O或S原子或一个或两个O和/或S原子，所述环系是未取代或取代的;这些化合物的制备，包含它们的组合物及其用于控制​​有害真菌的用途。

公开(公告)号：US07786043B2

公开(公告)日：2010-08-31

申请号：US11632342

申请日：2005-07-22

申请人： Wassilios Grammenos ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Udo Hünger ,  Bernd Müller ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Anja Schwögler ,  Ulrich Schöfl ,  Harald Köhle ,  Siegfried Strathmann ,  Maria Scherer ,  Reinhard Stierl ,  Jan Rether

发明人： Wassilios Grammenos ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Udo Hünger ,  Bernd Müller ,  Joachim Rheinheimer ,  Peter Schäfer ,  Frank Schieweck ,  Anja Schwögler ,  Ulrich Schöfl ,  Harald Köhle ,  Siegfried Strathmann ,  Maria Scherer ,  Reinhard Stierl ,  Jan Rether

IPC分类号： C07D239/74 ,  C07D239/70 ,  C07D401/04 ,  C07D403/04 ,  A01N43/54 ,  C07D213/16 ,  C07D213/84 ,  C07D213/53 ,  C07D213/61 ,  C07D213/26

CPC分类号： C07D401/04

摘要： The invention relates to 2-(pyridin-2-yl)-pyrimidine compounds of general formula (I) and their use for controlling pathogenic fungi and as plant protection products that, as an active constituent, contain compounds of this type: In general formula (I), k represents 0, 1, 2, 3; m represents 0, 1, 2, 3, 4 or 5; n represents 1, 2, 3, 4 or 5; R1, independent of one another, represents halogen, OH, CN, NO2, C1-C4 alkyl, C1-C4 alkyl halide, C1-C4 alkoxy, C1-C4 alkoxy halide, C2-C4 alkenyl, C2-C4 alkynyl, C3-C8 cycloalkyl, C1-C4 alkoxy-C1-C4 alkyl, amino, phenoxy, which is optionally substituted by halogen or C1-C4 alkyl, NHR, NR2, C(Ra)═N—ORb, S(═O)pA1 or C(═O)A2, or two radicals R1 bound to adjacent carbon atoms can, together, also represent a group —O-Alk-O—, wherein Alk represents a linear or branched C1-C4 alkylene, and 1, 2, 3 or 4 hydrogen atoms can also be replaced by halogen; R2 represents C1-C4 alkyl halide, C1-C4 alkoxy, C1-C4 alkoxy halide, hydroxy, halogen, CN or NO2; whereby R2 can also represent hydrogen or C1-C4 alkyl when at least one of the three following conditions is fulfilled: n represents 3, 4 or 5; k represents 1, 2 or 3; if m is not equal to 0, at least one of the radicals R1 represents a radical that differs from halogen, C1-C4 alkyl, C1-C4 alkoxy and C1-C4 alkyl halide, and; R3 represents C1-C4 alkyl.

摘要翻译： 本发明涉及通式（I）的2-（吡啶-2-基） - 嘧啶化合物及其用于控制​​致病真菌的用途，作为作为活性成分的植物保护产品含有这种化合物：通式 （I）中，k表示0,1,2,3; m表示0,1,2,3,4或5; n表示1,2,3,4或5; R 1彼此独立地表示卤素，OH，CN，NO 2，C 1 -C 4烷基，C 1 -C 4烷基卤，C 1 -C 4烷氧基，C 1 -C 4烷氧基卤化物，C 2 -C 4烯基，C 2 -C 4炔基， C8环烷基，C1-C4烷氧基-C1-C4烷基，氨基，苯氧基，其任选被卤素或C 1 -C 4烷基取代，NHR，NR 2，C（R a）= N-OR b，S（= O）p A1或C （ΟO）A2或与相邻碳原子结合的两个基团R1一起也可以代表基团-O-Alk-O-，其中Alk表示直链或支链C 1 -C 4亚烷基，和1,2,3或 4个氢原子也可以被卤素取代; R2代表C1-C4烷基卤，C1-C4烷氧基，C1-C4烷氧基卤化物，羟基，卤素，CN或NO2; 其中当满足以下三个条件中的至少一个时，R2还可以表示氢或C1-C4烷基：n表示3,4或5; k表示1,2或3; 如果m不等于0，则基团R1中的至少一个表示与卤素，C 1 -C 4烷基，C 1 -C 4烷氧基和C 1 -C 4烷基卤化物不同的基团， R3表示C1-C4烷基。