公开(公告)号：US20060135538A1

公开(公告)日：2006-06-22

申请号：US11340977

申请日：2006-01-30

申请人： Jordi Tormo Blasco ,  Klaus Ditrich ,  Hubert Sauter ,  Oliver Cullmann ,  Markus Gewehr ,  Wassilios Grammenos ,  Bernd Muller ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schafer ,  Frank Schieweck ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

发明人： Jordi Tormo Blasco ,  Klaus Ditrich ,  Hubert Sauter ,  Oliver Cullmann ,  Markus Gewehr ,  Wassilios Grammenos ,  Bernd Muller ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schafer ,  Frank Schieweck ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  C07D487/04

CPC分类号： C07D487/04 ,  A01N43/90

摘要： 7-(R)-Aminotriazolopyrimidines of the formula I where the substituents and the index are as defined below: R1 is hydrogen or methyl; R2 is methyl; R3 is C2-C1o-alkyl, C1-C4-alkoxymethyl, C3-C1o-cycloalkyl; R4 is halogen, Cl-C4-alkyl, C1-C4-haloalkyl or Cl-C4-alkoxy; n is a number from 1 to 5; Y is halogen, cyano, Cl-C4-alkyl or Cl-C4-alkoxy; where * is a center of chirality in the R configuration, processes for preparing these compounds, compositions comprising them and their use for controlling harmful fungi are described.

摘要翻译： 7-（R） - 取代基和指数如下所定义的式I的氨基三唑并嘧啶：R 1是氢或甲基; R 2是甲基; R 3是C 1 -C 2烷基，C 1 -C 4烷基，C 1 -C 4烷基，C 1 -C 4烷基， 亚烷基氧基甲基，C 3 -C 30环烷基; R 4是卤素，C 1 -C 4 - 烷基，C 1 -C 4 - 卤代烷基或C 1 -C 4 - C 4 - 烷氧基; n是从1到5的数字; Y是卤素，氰基，C 1 -C 4 - 烷基或C 1 -C 4 - 烷氧基; 其中*是R构型的手性中心，描述了制备这些化合物的方法，包含它们的组合物及其用于控制​​有害真菌的用途。

公开(公告)号：US06855718B2

公开(公告)日：2005-02-15

申请号：US10416467

申请日：2001-11-09

申请人： Jordi Tormo i Blasco ,  Klaus Ditrich ,  Hubert Sauter ,  Oliver Cullmann ,  Markus Gewehr ,  Wassilios Grammenos ,  Bernd Müller ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schäfer ,  Frank Schieweck ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

发明人： Jordi Tormo i Blasco ,  Klaus Ditrich ,  Hubert Sauter ,  Oliver Cullmann ,  Markus Gewehr ,  Wassilios Grammenos ,  Bernd Müller ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schäfer ,  Frank Schieweck ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  C07B53/00 ,  C07C209/62 ,  C07C211/03 ,  C07D487/04

CPC分类号： C07D487/04 ,  A01N43/90

摘要： A 7-(R)-Aminotriazolopyrimidines of formula I where the substituents and index are as defined below: R1 is hydrogen or methyl; R2 is methyl; R3 is C2-C10-alkyl, C1-C4-alkoxymethyl, C3-C10-cycloalkyl; Y is halogen, cyano, C1-C4-alkyl or C1-C4-alkoxy; where * is a center of chirality in the R configuration, processes for their preparation, compositions comprising them and their use for controlling harmful fungi.

摘要翻译： 式I的7-（R） - 氨基三唑并嘧啶，其中取代基和指数如下所定义：R 1是氢或甲基; R 2是甲基; R 3是C 2 -C 10 - 烷基，C 1 -C 4 - 烷氧基甲基，C 3 -C 10 - 环烷基; Y是卤素，氰基，C 1 -C 4 - 烷基或C 1 -C 4 - 烷氧基;其中*是R构型的手性中心，其制备方法，包含它们的组合物及其用途 用于控制有害真菌。

公开(公告)号：US20050261314A1

公开(公告)日：2005-11-24

申请号：US10484250

申请日：2002-07-16

申请人： Jordi i Blasco ,  Hubert Sauter ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schafer ,  Frank Schieweck ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

发明人： Jordi i Blasco ,  Hubert Sauter ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schafer ,  Frank Schieweck ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  C07D487/04

CPC分类号： C07D487/04 ,  A01N43/90

摘要： The invention relates to 7-amino triazolopyrimidines of formula (I), in which the substituents have the following meanings: R1, R2 represent hydrogen, alkyl, alkenyl, alkynyl, cycloalkyl, phenyl, naphthyl; or 5-membered or 6-membered heterocyclyl containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom; or 5-membered or 6-membered heteroaryl containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or R1 and R2 can, together with the nitrogen atom, which binds them, form a 5-membered or 6-membered ring containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom; R3 represents alkyl, alkenyl, alkynyl, cycloalkyl, phenylalkyl and alkyl halide; whereby R3 and R2 can be unsubstituted or partially or completely substituted according to the description; X represents halogen, cyano, alkoxy, alkyl halide, phenyl or phenyl that is substituted by Ra. The invention also relates to methods and intermediate products for producing said compounds, to agents containing the same, and to their use.

摘要翻译： 本发明涉及式（I）的7-氨基三唑并嘧啶，其中取代基具有以下含义：R 1，R 2表示氢，烷基，烯基，炔基 ，环烷基，苯基，萘基; 或含有1至4个氮原子或1至3个氮原子和1个硫或氧原子的5元或6元杂环基; 或含有1至4个氮原子或1至3个氮原子和1个硫或氧原子的5元或6元杂芳基，或R 1和R 2可以， 与它们结合的氮原子一起形成含有一至四个氮原子或一至三个氮原子和一个硫或氧原子的五元或六元环; R 3表示烷基，烯基，炔基，环烷基，苯基烷基和烷基卤; 根据描述，R 3和R 2可以是未取代的或部分或完全取代的; X表示卤素，氰基，烷氧基，烷基卤，苯基或被R a取代的苯基。 本发明还涉及用于生产所述化合物的方法和中间产物，含有该化合物的试剂及其用途。

公开(公告)号：US20050090665A1

公开(公告)日：2005-04-28

申请号：US10482216

申请日：2002-07-03

申请人： Bernd Muller ,  Hubert Sauter ,  Markus Gewehr ,  Wassilios Grammenos ,  Jordi I Blasco ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schafer ,  Frank Schieweck ,  Michael Rack ,  Gisela Lorenz ,  Siegfried Strathmann ,  Eberhard Ammermann ,  Reinhard Stierl

发明人： Bernd Muller ,  Hubert Sauter ,  Markus Gewehr ,  Wassilios Grammenos ,  Jordi I Blasco ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schafer ,  Frank Schieweck ,  Michael Rack ,  Gisela Lorenz ,  Siegfried Strathmann ,  Eberhard Ammermann ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  C07D487/04

CPC分类号： C07D487/04 ,  A01N43/90

摘要： Triazolopyrimidines of formula (I), wherein the index and substituents have the following meaning: n=0 or a whole number of 1-5; R=halogen, cyano, hydroxy, cyanate, alkyl, alkenyl, alkinyl, halogenalkyl, halogenalkenyl, alkoxy, alkenyloxy, alkinyloxy, halogenalkoxy, cycloalkyl, cycloalkenyl, cycloalkoxy, alkoxycarbonyl, alkenyloxycarbonyl, alkinyloxycarbonyl, aminocarbonyl, alkylaminocarbonyl, dialkylaminocarbonyl, alkoximinoalkyl, alkenyloximinocarbonyl, alkinyloximinoalkyl, alkylcarbonyl, alkenylcarbonyl, alkinylcarbonyl, cycloalkylcarbonyl or a five to ten membered saturated, partially unsaturated or aromatic heterocycle, containing one to four heteroatoms from the group O, N or S; R1=alkyl, alkenyl, alkinyl, cycloalkyl, cycloalkenyl, phenyl, naphthyl or a five to ten membered saturated, partially unsaturated or aromatic heterocycle, containing one to four heteroatoms from the group O, N or S, R and/or R1 being able to be substituted according to the description; R2=alkyl, alkenyl or alkinyl which can be substituted by halogen, cyano, nitro, alkoxy or alkoxycarbonyl. The invention also relates to a method for the production of said compounds, agents containing same, and the use thereof in controlling noxious fungi.

摘要翻译： 式（I）的三唑并嘧啶，其中指数和取代基具有以下含义：n = 0或整数1-5; 环烷氧基，烷氧基羰基，链烯氧基羰基，烷氧基羰基，氨基羰基，烷基氨基羰基，二烷基氨基羰基，肟基烷基，链烯基肟基羰基，烷氧基羰基，烷氧基羰基， 烷基羰基，链烯基羰基，炔基羰基，环烷基羰基或五至十元饱和，部分不饱和或芳族杂环，含有一至四个O，N或S基团的杂原子; R 1 =烷基，烯基，炔基，环烷基，环烯基，苯基，萘基或五至十元饱和，部分不饱和或芳族杂环，其含有一至四个O，N或S ，R和/或R 1能够根据描述进行取代; 可以被卤素，氰基，硝基，烷氧基或烷氧基羰基取代的烷基，烯基或炔基。 本发明还涉及生产所述化合物的方法，含有该化合物的试剂及其在控制有害真菌中的用途。

公开(公告)号：US20050107401A1

公开(公告)日：2005-05-19

申请号：US10505146

申请日：2003-02-06

申请人： Frank Schieweck ,  Jordi Blasco ,  Thomas Grote ,  Andreas Gypser ,  Bernd Muller ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schafer ,  Wassilios Grammenos ,  Markus Gewehr ,  Anja Schwogler ,  Carsten Blettner ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

发明人： Frank Schieweck ,  Jordi Blasco ,  Thomas Grote ,  Andreas Gypser ,  Bernd Muller ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schafer ,  Wassilios Grammenos ,  Markus Gewehr ,  Anja Schwogler ,  Carsten Blettner ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

IPC分类号： A01N43/54 ,  C07D401/04 ,  A61K31/506 ,  C07D43/04

CPC分类号： C07D401/04

摘要： The invention relates to 2-(2-pyridyl)-5-phenyl-6-amninopyrimidines of formula I, wherein the substitutes and the index have the following meaning: R1 represents halogen, hydroxy, hyano, hxo, nitro, amino, mercapto, alkyl, halogenalkyl, alkenyl, alkinyl, cycloalkyl, alkoxy, halogenalkoxy, carboxyl, alkoxycarbonyl, carbamoyl, alkylaminocarbonyl, dialkylamincarbonyl, morpholinocarbonyl, pyrrolidinocarbonyl, alkylcarbonylamino, alkylamino. dialkylamino, alkylthio, alkylsulfinyl, alkylsulfonyl, hydroxysulfonyl, aminosulfonyl, alkylaminosulfonyl, dialkylaminosulfonyl; m=0 or 1-4; R2 represents hydrogen, halogen, cyano, alkyl, halogenalkyl or alkoxy; R3, R4 represents hydrogen, alkyl, halogenalkyl, cycloalkyl, halogencycloalkyl, alkenyl, halogenalkenyl, cycloalkenyl, alkinyl, halogenalkinyl or cycloalkinyl, R3 and R4 together with the nitrogen atom to which they are connected, form a five or six-membered ring which is interrupted by an atom from the group O, N or S and/or can be substituted according to the description; R5 represents halogen, alkyl or halogenalkyl; R6 represents hydrogen or one of the known groups in R5; R7, R8 represent hydrogen, halogen, alkyl or halogenalkyl; R9 represents hydrogen, halogen, hydroxy, cyano, alkyl, alkoxy, cycloalkoxy, halogenalkoxy, alkoxycarbonyl or alkylaminocarbonyl. The invention also relates to a method and intermediate product for the production of said compound in addition to the use thereof for combating undesirable plants.

摘要翻译： 本发明涉及式I的2-（2-吡啶基）-5-苯基-6-脒嘧啶，其中取代基和指数具有以下含义：R 1表示卤素，羟基，杂环基， 烷氧基，烷氧基羰基，氨基甲酰基，烷基氨基羰基，二烷基氨基羰基，吗啉代羰基，吡咯烷基羰基，烷基羰基氨基，烷基氨基。 二烷基氨基，烷硫基，烷基亚磺酰基，烷基磺酰基，羟基磺酰基，氨基磺酰基，烷基氨基磺酰基，二烷基氨基磺酰基; m = 0或1-4; R 2表示氢，卤素，氰基，烷基，卤代烷基或烷氧基; R 3，R 4表示氢，烷基，卤代烷基，环烷基，卤代烷基，烯基，卤代烯基，环烯基，炔基，卤代炔基或环炔基，R 3 O 和R 4与它们连接的氮原子一起形成5或6元环，其被来自基团O，N或S的原子和/或可被取代 根据说明; R 5表示卤素，烷基或卤代烷基; R 6表示氢或R 5中的已知基团之一; R 7，R 8表示氢，卤素，烷基或卤代烷基; R 9表示氢，卤素，羟基，氰基，烷基，烷氧基，环烷氧基，卤代烷氧基，烷氧基羰基或烷基氨基羰基。 本发明还涉及用于生产所述化合物的方法和中间产物，除了其用于对抗不期望的植物之外。

公开(公告)号：US20050272749A1

公开(公告)日：2005-12-08

申请号：US10531981

申请日：2003-11-04

申请人： Jordi Tormo Blasco ,  Carsten Bletner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Jordi Tormo Blasco ,  Carsten Bletner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： C07D487/04 ,  A61K31/519

CPC分类号： C07D487/04

摘要： 5-Alkyl-7-aminotriazolopyrimidines of the formula I, where: R1, R2 are hydrogen, alkyl, alkenyl, alkynyl, haloalkyl, cycloalkyl, phenyl, naphthyl; 5- or 6-membered saturated, unsaturated or aromatic heterocyclyl which contains one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom; or R1 and R2 together with the bridging nitrogen atom can form a 5- or 6-membered ring which contains one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom; R3 is cycloalkyl or bicycloalkyl; where R1, R2 and R3 may be substituted as outlined in the description; X is alkyl or haloalkyl; and their salts; processes and intermediates for their preparation, compositions comprising them and their use for controlling phytopathogenic harmful fungi are described.

摘要翻译： 式I的5-烷基-7-氨基三唑并嘧啶，其中：R 1，R 2是氢，烷基，烯基，炔基，卤代烷基，环烷基，苯基，萘基; 含有1-4个氮原子或一至三个氮原子和一个硫或氧原子的5-或6-元饱和，不饱和或芳族杂环基; 或R 1和R 2与桥连氮原子一起可以形成含有1-4个氮原子或一至三个氮原子的5-或6-元环，并且 一个硫或氧原子; R 3是环烷基或双环烷基; 其中R 1，R 2和R 3可以如说明书中概述的那样被取代; X是烷基或卤代烷基; 和它们的盐; 描述了其制备方法和中间体，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US20050272748A1

公开(公告)日：2005-12-08

申请号：US10531980

申请日：2003-11-14

申请人： Jordi Tormo Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Jordi Tormo Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  C07D487/04 ,  A61K31/519

CPC分类号： C07D487/04 ,  A01N43/90

摘要： 2-Mercapto-substituted triazolopyrimidines of the formula I in which the substituents are as defined below: L is halogen, cyano, nitro, alkyl, alkenyl, alkynyl, haloalkyl, haloalkenyl, alkoxy, alkenyloxy, alkynyloxy, haloalkoxy or —C(═O)-A; A is hydrogen, hydroxyl, alkyl, alkenyl, alkoxy, haloalkoxy, alkylamino or dialkylamino; m is 0, 1, 2, 3, 4 or 5; X is halogen, cyano, alkyl, haloalkyl, alkoxy or haloalkoxy; R1, R2 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, alkadienyl, haloalkenyl, cycloalkenyl, alkynyl, haloalkynyl or cycloalkynyl, phenyl, naphthyl or a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle which contains one to four hetero atoms from the group consisting of O, N and S; R1 and R2 together with the nitrogen atom to which they are attached may also form a five- or six-membered ring which may be interrupted by an atom from the group consisting of O, N and S; where R1 and/or R2 may be substituted as stated in the description; processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi are described.

摘要翻译： 2-巯基取代的式Ⅰ的三唑并嘧啶，其中取代基如下：L是卤素，氰基，硝基，烷基，烯基，炔基，卤代烷基，卤代烯基，烷氧基，烯氧基，炔氧基，卤代烷氧基或-C ）-一个; A是氢，羟基，烷基，烯基，烷氧基，卤代烷氧基，烷基氨基或二烷基氨基; m为0,1,2,3,4或5; X是卤素，氰基，烷基，卤代烷基，烷氧基或卤代烷氧基; R 1，R 2是氢，烷基，卤代烷基，环烷基，卤代环烷基，烯基，链二烯基，卤代烯基，环烯基，炔基，卤代炔基或环炔基，苯基，萘基或五 至10元饱和，部分不饱和或芳族杂环，其含有一个至四个由O，N和S组成的组的杂原子; R 1和R 2与它们所连接的氮原子一起也可以形成五元或六元环，其可被来自基团的原子中断 由O，N和S组成; 其中R 1和/或R 2可以如描述中所述被取代; 描述了制备这些化合物的方法，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US20070088026A1

公开(公告)日：2007-04-19

申请号：US11548864

申请日：2006-10-12

申请人： Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schafer ,  Frank Schieweck ,  Hubert Sauter ,  Markus Gewehr ,  Bernd Muller ,  Jordi i Blasco ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

发明人： Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schafer ,  Frank Schieweck ,  Hubert Sauter ,  Markus Gewehr ,  Bernd Muller ,  Jordi i Blasco ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

IPC分类号： A61K31/541 ,  A61K31/5377 ,  A61K31/506 ,  C07D417/04 ,  C07D403/04 ,  C07D413/04

CPC分类号： C07D239/42 ,  A01N43/54 ,  A01N43/56 ,  A01N43/60 ,  A01N43/647 ,  A01N43/653 ,  A01N43/713 ,  A01N43/90 ,  C07D231/12 ,  C07D233/56 ,  C07D249/08 ,  C07D403/04 ,  C07D473/06 ,  C07D487/04

摘要： 5-Phenylpyrimidines of the formula I, in which the substituents have the following meanings: R1 is a five- to ten-membered saturated, partially unsaturated or aromatic mono- or bicyclic heterocycle comprising one to four hetero atoms selected from the group consisting of O, N or S, which heterocycle can be substituted as defined in the description, R2 is hydrogen, halogen, cyano, alkyl, haloalkyl or alkoxy; R3, R4 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, alkynyl, haloalkynyl or cycloalkynyl, R3 and R4 together with the nitrogen atom to which they are bonded may also form a five- or six-membered ring which can be interrupted by a hetero atom and have attached to it one or more substituents; R5, R6 are hydrogen, halogen, alkyl, haloalkyl or alkoxy; R7, R8 are hydrogen, halogen, alkyl or haloalkyl; R9 is hydrogen, halogen, alkyl, alkoxy, cycloalkoxy, haloalkoxy or alkoxycarbonyl, Processes and intermediates for the preparation of these compounds, and their use for controlling harmful fungi.

摘要翻译： 式I的5-苯基嘧啶，其中取代基具有以下含义：R 1是5至10元饱和的，部分不饱和的或芳族的单环或双环杂环，其包含一至四个杂 选自O，N或S的原子，该杂环可以如描述中所定义而被取代，R 2是氢，卤素，氰基，烷基，卤代烷基或烷氧基; R 3，R 4是氢，烷基，卤代烷基，环烷基，卤代环烷基，烯基，卤代烯基，环烯基，炔基，卤代炔基或环炔基，R 3 O 和R 4与它们所键合的氮原子一起也可以形成五元或六元环，其可被杂原子间隔并且与其连接一个或多个取代基; R 5，R 6是氢，卤素，烷基，卤代烷基或烷氧基; R 7，R 8是氢，卤素，烷基或卤代烷基; R 9是氢，卤素，烷基，烷氧基，环烷氧基，卤代烷氧基或烷氧羰基。用于制备这些化合物的方法和中间体及其用于控制​​有害真菌的用途。

公开(公告)号：US06455515B2

公开(公告)日：2002-09-24

申请号：US09879902

申请日：2001-06-14

申请人： Andreas Gypser ,  Thomas Grote ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schäfer ,  Oliver Cullmann ,  Markus Gewehr ,  Wassilios Grammenos ,  Jordi Tormo i Blasco ,  Bernd Müller ,  Hubert Sauter ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

发明人： Andreas Gypser ,  Thomas Grote ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schäfer ,  Oliver Cullmann ,  Markus Gewehr ,  Wassilios Grammenos ,  Jordi Tormo i Blasco ,  Bernd Müller ,  Hubert Sauter ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

IPC分类号： A01N3740

CPC分类号： C07C255/66 ,  A01N37/40 ,  A01N37/46 ,  A01N47/20 ,  A01N47/30 ,  C07C251/86

摘要： Salicylohydrazide derivatives of the formula I in which the index and the substituents have the following meanings: X is halogen, NO2, cyano, alkyl or alkoxy; m is 0, 1, 2 or 3, it being possible for the substituents X to differ from each other if n is greater than 1; R1 is NO2, NH2 or NH—CO—A; A is hydrogen, alkyl, alkoxy, NH2, NHCH3 or N(CH3)2; R2 is hydrogen, cyano, alkyl, alkenyl, alkynyl, haloalkyl, alkoxy or alkylthio; it being possible for the hydrocarbon radicals to be unsubstituted or substituted, R3 is phenyl, naphthyl, cycloalkyl, 5-membered or 6-membered hetaryl or 5-membered or 6-membered heterocyclyl containing one to three N atoms and/or one O or S atom or one or two O and/or S atoms, the ring systems being unsubstituted or substituted; the preparation of these compounds, compositions comprising them, and their use for controlling harmful fungi.

摘要翻译： 指数和取代基具有以下含义的式Iin的磺酰肼衍生物：X是卤素，NO 2，氰基，烷基或烷氧基; m是0,1,2或3，取代基X可能与每个 另外，如果n大于1，则R1为NO2，NH2或NH-CO-A; A为氢，烷基，烷氧基，NH2，NHCH3或N（CH3）2; R2为氢，氰基，烷基，烯基，炔基， 卤代烷基，烷氧基或烷硫基;烃基可以是未取代的或取代的，R3是苯基，萘基，环烷基，含有1至3个N原子的5元或6元杂芳基或5元或6元杂环基 和/或一个O或S原子或一个或两个O和/或S原子，所述环系是未取代或取代的;这些化合物的制备，包含它们的组合物及其用于控制​​有害真菌的用途。

公开(公告)号：US06593315B2

公开(公告)日：2003-07-15

申请号：US09896971

申请日：2001-07-02

申请人： Andreas Gypser ,  Thomas Grote ,  Joachim Rheinheimer ,  Ingo Rose ,  Oliver Cullmann ,  Markus Gewehr ,  Wassilios Grammenos ,  Jordi Tormo i Blasco ,  Bernd Müller ,  Hubert Sauter ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

发明人： Andreas Gypser ,  Thomas Grote ,  Joachim Rheinheimer ,  Ingo Rose ,  Oliver Cullmann ,  Markus Gewehr ,  Wassilios Grammenos ,  Jordi Tormo i Blasco ,  Bernd Müller ,  Hubert Sauter ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

IPC分类号： A01N3736

CPC分类号： C07C251/86 ,  A01N37/50

摘要： Salicylic acid derivatives of the formula I, where the index and the substituents have the following meanings: X is halogen, NO2, cyano, alkyl or alkoxy; m is 0, 1, 2 or 3, it being possible for the substituents X to be different from each other if n is greater than 1; A is OH, alkoxy, NH2, NHCH3 or N(CH3)2; R1 is phenyl, naphthyl, cycloalkyl, 5-membered or 6-membered hetaryl or 5-membered or 6-membered heterocyclyl, comprising one to three N atoms and/or one O or S atom or one or two O and/or S atoms, the ring systems being unsubstituted or substituted; R2 is hydrogen, cyano, alkyl, alkenyl, alkynyl, haloalkyl, alkoxy or alkylthio, processes for the preparation of these compounds, compositions comprising them, and their use for controlling harmful fungi.

摘要翻译： 式I的水杨酸衍生物，其中指数和取代基具有以下含义：X是卤素，NO 2，氰基，烷基或烷氧基; m是0,1,2或3，取代基X可以是 如果n大于1，A是不同的; A是OH，烷氧基，NH2，NHCH3或N（CH3）2; R1是苯基，萘基，环烷基，5元或6元杂芳基或5元或6- 包括一至三个N原子和/或一个O或S原子或一个或两个O和/或S原子，所述环系是未取代或取代的; R2是氢，氰基，烷基，烯基，炔基，卤代烷基， 烷氧基或烷硫基，制备这些化合物的方法，包含它们的组合物及其用于控制​​有害真菌的用途。