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20 条记录 (耗时 0.012 秒)

    Anthelmintic phosphonamidate and phosphoramidate compositions and methods of use
    2.
    发明授权
    Anthelmintic phosphonamidate and phosphoramidate compositions and methods of use 失效
    驱虫剂膦酰胺酸酯和氨基磷酸酯组合物和使用方法

    公开(公告)号：US4139614A

    公开(公告)日：1979-02-13

    申请号：US662744

    申请日：1976-03-01

    申请人： Edward E. Kilbourn ,  Ernest Weiler ,  William D. Weir

    发明人： Edward E. Kilbourn ,  Ernest Weiler ,  William D. Weir

    IPC分类号： C07F9/24 ,  C07F9/44 ,  C07F9/58 ,  C07F9/6509 ,  A61K31/66 ,  C07F9/38

    CPC分类号： C07F9/650988 ,  C07F9/2454 ,  C07F9/4461 ,  C07F9/588

    摘要： This invention relates to novel anthelmintic compositions containing as the essential active ingredient, a compound of the formula: ##STR1## wherein R.sup.1 is cylcoalkyl, or optionally substituted aralkyl, aryl, pyridyl, or pyrazinyl;R.sup.2 is hydrogen, alkyl, cycloalkyl, alkoxyalkyl, alkylthioalkyl, cyanoalkyl, alkenyl, or optionally substituted aralkyl or aryl;R.sup.1 and R.sup.2 taken together with the nitrogen atom to which they are attached form an optionally substituted morpholino or piperidino group;R.sup.3 is hydrogen, alkyl, cycloalkyl, alkenyl, or optionally substituted aralkyl or aryl;R.sup.4 is alkoxy, haloalkoxy, dialkylamino, alkylthio, phenoxy or phenylthio; andR.sup.5 is alkyl, alkoxy, haloalkoxy, dialkylamino, alkylthio, phenyl, phenoxy or phenylthio; andX is oxygen or sulfur;And pharmaceutically acceptable metal salts and metal salt complexes thereof, and to methods of employing them in the treatment of intestinal parasites in animals, e.g. mammals, fish, and birds.

    摘要翻译： 本发明涉及含有作为必需活性成分的下式化合物的新型驱肠剂组合物：其中R 1为环烷基或任选取代的芳烷基，芳基，吡啶基或吡嗪基; R2是氢，烷基，环烷基，烷氧基烷基，烷硫基烷基，氰基烷基，烯基或任选取代的芳烷基或芳基; R1和R2与它们所连接的氮原子一起形成任选取代的吗啉代或哌啶子基; R3是氢，烷基，环烷基，烯基或任选取代的芳烷基或芳基; R4是烷氧基，卤代烷氧基，二烷基氨基，烷硫基，苯氧基或苯硫基; R 5为烷基，烷氧基，卤代烷氧基，二烷基氨基，烷硫基，苯基，苯氧基或苯硫基; X为氧或硫; 和药学上可接受的金属盐和金属盐复合物，以及在处理动物肠内寄生虫的方法中的应用。 肉类，鱼类和禽类。

    3-Pyridylmethyl aryl urea rodenticides
    3.
    发明授权
    3-Pyridylmethyl aryl urea rodenticides 失效
    3-吡啶基甲基芳基脲杀鼠剂

    公开(公告)号：US3994905A

    公开(公告)日：1976-11-30

    申请号：US622914

    申请日：1975-10-16

    申请人： Edward E. Kilbourn ,  David L. Peardon ,  J. Edgar Ware

    发明人： Edward E. Kilbourn ,  David L. Peardon ,  J. Edgar Ware

    IPC分类号： A01N47/20 ,  C07D213/75

    CPC分类号： A01N47/20

    摘要： Novel 1-(3-pyridylmethyl)-3-(4'-substituted-phenyl or -naphthyl)-ureas and their acid addition salts. The 4'-substituent may be -NO.sub.2, -CN, -CF.sub.3, -C(O)R.sub.1, -SCN, SR.sub.2, -SO.sub.2 C.sub.6 H.sub.5 or -SO.sub.2 NR.sub.3 R.sub.4. These compounds are biologically active, and many are active rodenticides.

    摘要翻译： 新型1-（3-吡啶基甲基）-3-（4'-取代 - 苯基或 - 萘基） - 脲及其酸加成盐。 4'-取代基可以是-NO 2，-CN，-CF 3，-C（O）R 1，-SSCN，SR 2，-SO 2 C 6 H 5或-SO 2 NR 3 R 4。 这些化合物具有生物活性，许多是活性杀鼠剂。

    Arthropodicidal and nematocidal phosphoramidates
    5.
    发明授权
    Arthropodicidal and nematocidal phosphoramidates 失效
    节肢动物和杀线虫的氨基磷酸酯

    公开(公告)号：US4087521A

    公开(公告)日：1978-05-02

    申请号：US662743

    申请日：1976-03-01

    申请人： Harold E. Aller ,  Edward E. Kilbourn ,  Ernest D. Weiler ,  William D. Weir

    发明人： Harold E. Aller ,  Edward E. Kilbourn ,  Ernest D. Weiler ,  William D. Weir

    IPC分类号： C07F9/24 ,  C07F9/44 ,  C07F9/58 ,  C07F9/6509 ,  A01N9/36

    CPC分类号： C07F9/650988 ,  C07F9/2454 ,  C07F9/4461 ,  C07F9/588

    摘要： This invention relates to novel phosphoramidates of the formula: ##STR1## wherein R.sup.1 is (C.sub.6 -C.sub.10) aryl optionally substituted with alkyl, alkoxy, alkylthio, alkylsulfinyl, alkylsulfonyl, dialkylamino, haloalkyl, hydroxyalkyl, cyano, nitro, hydroxy, or halogen;R.sup.2 is hydrogen, alkyl, cycloalkyl, alkenyl, or optionally substituted aralkyl or aryl;R.sup.3 is (C.sub.1 -C.sub.6) alkyl;R.sup.4 is (C.sub.3 -C.sub.4) alkyl; andX, y and Z are independently oxygen or sulfur;And the agronomically acceptable metal salts and metal salt complexes thereof; to compositions containing them; and to methods of using them to control certain harmful pests, e.g. arthropods and nematodes.

    摘要翻译： 本发明涉及下式的新型氨基磷酸酯：其中R 1为任选被烷基，烷氧基，烷硫基，烷基亚磺酰基，烷基磺酰基，二烷基氨基，卤代烷基，羟烷基，氰基，硝基，羟基或卤素取代的（C6-C10） R2是氢，烷基，环烷基，烯基或任选取代的芳烷基或芳基; R3是（C1-C6）烷基; R4是（C3-C4）烷基; X，Y和Z独立地为氧或硫; 和其农业上可接受的金属盐和金属盐复合物; 包含他们的组合物; 以及使用它们来控制某些有害物质的方法，E.G. 神经元和神经元。

    Nematocidal phosphoramidates
    7.
    发明授权
    Nematocidal phosphoramidates 失效
    杀线虫的氨基磷酸酯

    公开(公告)号：US4259330A

    公开(公告)日：1981-03-31

    申请号：US662751

    申请日：1976-03-01

    申请人： Harold E. Aller ,  Edward E. Kilbourn ,  Ernest D. Weiler ,  William D. Weir

    发明人： Harold E. Aller ,  Edward E. Kilbourn ,  Ernest D. Weiler ,  William D. Weir

    IPC分类号： C07F9/24 ,  C07F9/44 ,  C07F9/58 ,  C07F9/6509 ,  A01N57/28 ,  A01N57/32

    CPC分类号： C07F9/650988 ,  C07F9/2454 ,  C07F9/4461 ,  C07F9/588

    摘要： This invention relates to novel phosphoramidates of the formula: ##STR1## wherein R.sup.1 is hydrogen, alkyl, cycloalkyl, or optionally substituted aralkyl, aryl, pyridyl, pyridylmethyl, pyridylethyl or pyrazinyl;R.sup.2 is hydrogen provided R.sup.1 is other than optionally substituted aryl; alkyl; cycloalkyl; alkoxyalkyl; alkylthioalkyl; cyanoalkyl; alkenyl; optionally substituted aralylky; or optionally substituted aryl, provided R.sup.1 is other than hydrogen;R.sup.1 and R.sup.2 taken together with the nitrogen to which they are attached form an optionally substituted morpholino or piperidino group;R.sup.3 is hydrogen, alkyl, cycloalkyl, alkenyl, or optionally substituted aralkyl or aryl;R.sup.4 is (C.sub.1 -C.sub.6) alkyl;R.sup.5 is (C.sub.3 -C.sub.4) alkyl; andX, Y and Z are independently oxygen or sulfur;the agronomically acceptable metal salts and metal salt complexes thereof; and to methods of using them to control nematodes.

    摘要翻译： 本发明涉及下式的新型氨基磷酸酯：其中R 1为氢，烷基，环烷基或任选取代的芳烷基，芳基，吡啶基，吡啶基甲基，吡啶基乙基或吡嗪基; R2是氢，只要R1不是任选取代的芳基; 烷基; 环烷基 烷氧基烷基 烷硫基烷基; 氰基烷基 烯基; 任选取代的芳酰基; 或任选取代的芳基，条件是R 1不是氢; R1和R2与它们所连接的氮一起形成任选取代的吗啉代或哌啶子基; R3是氢，烷基，环烷基，烯基或任选取代的芳烷基或芳基; R4是（C1-C6）烷基; R5是（C3-C4）烷基; X，Y和Z独立地为氧或硫; 其农艺学上可接受的金属盐和金属盐络合物; 以及使用它们来控制线虫的方法。