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    INNOVATIVE FORMULATION
    3.
    发明申请
    INNOVATIVE FORMULATION 有权
    创新公式

    公开(公告)号：US20090130156A1

    公开(公告)日：2009-05-21

    申请号：US11912299

    申请日：2006-04-20

    申请人： Valerio Borzatta ,  Oreste Picolo ,  Elisa Capparella

    发明人： Valerio Borzatta ,  Oreste Picolo ,  Elisa Capparella

    IPC分类号： A01N65/00 ,  A01N25/00 ,  A01N57/00 ,  A01N37/34

    CPC分类号： A01N43/30 ,  A01N25/28 ,  A01N53/00 ,  A01N2300/00

    摘要： The present invention relates to a new formulation characterised by the presence of two components, one of which (A) possesses insecticidal, acaricidal, fungicidal, snailcidal or vermicidal activity and the other (B) exhibits synergistic activity with the first by enhancing its effectiveness, and in which the average release time of component (A) is 1 to 12 hours later than the average release time of component (B). The formulation is obtained by: a) separate microencapsulation of both components (A) and (B) within a multilayer system of specific polymers in which component (A) is in a more interior portion of the capsule than component (B), being separated from component (B) by a polymer layer of suitable thickness (FIG. 1); b) microencapsulation of both components within a single layer system (FIG. 2), combined with an immediate-release emulsion/microemulsion containing an additional amount of component (B).

    摘要翻译： 本发明涉及一种新的制剂，其特征在于两种成分的存在，其中一种成分（A）具有杀虫，杀螨，杀真菌，杀虫或杀虫活性，另一种（B）通过提高其有效性与第一种成分具有协同作用， 其中组分（A）的平均释放时间比组分（B）的平均释放时间晚1至12小时。 该制剂通过以下方法获得：a）在特定聚合物的多层体系内单独的组分（A）和（B）的微胶囊化，其中组分（A）在组分（B）的更多内部部分中，分离 由组分（B）通过合适厚度的聚合物层（图1）; b）在单层系统（图2）中的两种组分的微囊化，与含有额外量的组分（B）的立即释放乳液/微乳液组合。

    Substituted alkynyl phenoxy compounds as new synergists in pesticidal compositions
    5.
    发明授权
    Substituted alkynyl phenoxy compounds as new synergists in pesticidal compositions 有权
    取代炔基苯氧基化合物作为农药组合物中的新增效剂

    公开(公告)号：US08809389B2

    公开(公告)日：2014-08-19

    申请号：US13391496

    申请日：2010-08-18

    申请人： Valerio Borzatta ,  Elisa Capparella ,  Leni Moroni ,  Graham Moores ,  Despina Philippou

    发明人： Valerio Borzatta ,  Elisa Capparella ,  Leni Moroni ,  Graham Moores ,  Despina Philippou

    IPC分类号： A01N43/30 ,  A01N31/14 ,  C07C43/215 ,  C07C41/16

    CPC分类号： C07C41/16 ,  A01N43/30 ,  C07C43/215 ,  A01N51/00 ,  A01N53/00

    摘要： A composition comprising an alkynyl phenoxy compound of Formula (I) as a synergist and a pesticidal active ingredient is described, wherein R1 and R2, similar or different, are (C1-C4)alkyl or R1O— and R2O— together represent a group —O—CH2—O—, —O—CH(CH3)—O, —O—CH2—CH2—O—, —O—CH2—CH2—, R3 is (C1-C6)alkyl, (C3-C6)alkenyl or —B—(CH2—CH2—O)z-R6 where B is —CH2—O— or —O—, z is 0, 1 or 2 and R6 is (C1-C4)alkyl; R4 is hydrogen or methyl; R5 is hydrogen or methyl; x is an integer from 1 to 2; y is 0, 1 or 2; with the proviso that when R3 is —B—(CH2CH2—O)z-R6, y is 1 and 5-(propargyloxy)-benzo[1,3]dioxole is excluded.

    摘要翻译： 描述了包含式（I）的炔基苯氧基化合物作为增效剂和杀虫活性成分的组合物，其中相同或不同的是（C1-C4）烷基或R1O-和R2O-一起代表基团 - O-CH 2 -O - ， - O-CH（CH 3）-O，-O-CH 2 -CH 2 -O-，-O-CH 2 -CH 2 - ，R 3是（C 1 -C 6）烷基，（C 3 -C 6） 或-B-（CH2-CH2-O）z-R6，其中B是-CH2-O-或-O-，z是0,1或2，R6是（C1-C4）烷基; R4是氢或甲基; R5是氢或甲基; x是1到2的整数; y为0,1或2; 条件是当R3为-B-（CH2CH2-O）z-R6时，y为1，排除5-（炔丙氧基） - 苯并[1,3]间二氧杂环戊烯。

    Biologically Active Formulation
    6.
    发明申请
    Biologically Active Formulation 有权
    生物活性配方

    公开(公告)号：US20090130155A1

    公开(公告)日：2009-05-21

    申请号：US11912136

    申请日：2006-04-21

    申请人： Oreste Piccolo ,  Valerio Borzatta ,  Giovanna Delogu ,  Elisa Capparella ,  Cristina De Candia ,  Carlotta Gobbi ,  Giovanna Di Blasi

    发明人： Oreste Piccolo ,  Valerio Borzatta ,  Giovanna Delogu ,  Elisa Capparella ,  Cristina De Candia ,  Carlotta Gobbi ,  Giovanna Di Blasi

    IPC分类号： A01N43/04 ,  C08B30/18 ,  C08B37/16

    CPC分类号： A01N25/10

    摘要： The present invention provides a formulation characterised by the simultaneous presence in cyclodextrin based supramolecular complexes, of two components, one of which possesses insecticidal, acaricidal, fungicidal, snailcidal or vermicidal activity and the other possesses an activity synergistic with the first, enhancing its effectiveness. The biologically active substance is chosen from the following classes of chemical products: carbamates, organophosphates, thioureas, pentatomic or hexatomic heterocycles in which 1, 2 or 3 nitrogen atoms are present. The synergistic substance can be chosen from components containing at least one aromatic or non aromatic carbocyclic ring, such as piperonyl butoxide, sesamol, verbutin or MGK 264. For the same dose, the activity of the present formulations is greater than that of the mixture of the two active components alone or separately complexed with cyclodextrin. The process for preparing said formulation and its use for the activities herein indicated are further aspects of the present invention.

    摘要翻译： 本发明提供了一种制剂，其特征在于同时存在两种组分的基于环糊精的超分子复合物，其中一种具有杀虫，杀螨，杀真菌，杀虫或杀虫活性，另一种具有与第一种协同增效的活性，提高其有效性。 生物活性物质选自以下类别的化学产品：其中存在1,2或3个氮原子的氨基甲酸酯，有机磷酸酯，硫脲，五原子或六原子杂环。 协同物质可以选自含有至少一个芳族或非芳族碳环的组分，例如胡椒基丁醚，芝麻酚，鸟嘌呤或MGK 264.对于相同的剂量，本发明制剂的活性大于 两种活性组分单独或分别与环糊精复合。 制备所述制剂的方法及其用于本文所述活性的用途是本发明的另外的方面。

    Process for synthesizing heliotropine and its derivatives
    7.
    发明授权
    Process for synthesizing heliotropine and its derivatives 失效
    合成天葵及其衍生物的方法

    公开(公告)号：US07402709B2

    公开(公告)日：2008-07-22

    申请号：US10577846

    申请日：2004-10-28

    申请人： Valerio Borzatta ,  Elisa Capparella ,  Carlotta Gobbi ,  Elisa Poluzzi

    发明人： Valerio Borzatta ,  Elisa Capparella ,  Carlotta Gobbi ,  Elisa Poluzzi

    IPC分类号： C07C45/90

    CPC分类号： C07D317/54

    摘要： A new high-yield, easily industrialized process for synthesizing compounds of formula (IV), in which X1 and X2, the same or different, are linear or branched C1-C8 alkyls, n and m are 0, 1 or 2, with the proviso that n and m are not simultaneously 0; or (OX1)n and (OX2)m taken together form an O-T-O group where T is chosen from —CH2—, —CH2CH2, —CH2CH2CH2—, —C(CH3)2—. The process comprises treating a chloromethyl derivative (I) with an alkaline acetate to form the intermediate acetylderivative (II); the intermediate (II) is to hydrolysed to form the alcohol (III); the alcohol (III) is then oxidised in the presence of air and catalysts to obtain the desired derivative (IV). The process runs its course within a short period of time, with high yields and high selectivity; in addition, the process does not require purification and separation of the intermediates and can therefore be favourably conducted in a single batch.

    摘要翻译： 合成式（IV）化合物的新的高产率，易于工业化的方法，其中相同或不同的X 1和X 2是直链或支链C1 -C 8烷基，n和m为0,1或2，条件是n和m不同时为0; 或（OX 1）n和（OX 2 N）m一起形成OTO基团，其中T选自-CH 2 - ， - CH 2 CH 2，CH 2 CH 2 CH 2 - ， - CH 2 CH 2 CH 2， - CH 2 CH 2 CH 2 - ， - C（CH 3）2 - 。 该方法包括用碱性乙酸盐处理氯甲基衍生物（I）以形成中间体乙酰衍生物（II）; 中间体（II）被水解形成醇（III）; 然后在空气和催化剂的存在下将醇（III）氧化以获得所需的衍生物（IV）。 该过程在短时间内运行，产量高，选择性高; 此外，该方法不需要中间体的纯化和分离，因此可以在单次批次中有利地进行。

    Innovative formulation
    8.
    发明授权
    Innovative formulation 有权
    创新配方

    公开(公告)号：US08025894B2

    公开(公告)日：2011-09-27

    申请号：US11912299

    申请日：2006-04-20

    申请人： Valerio Borzatta ,  Oreste Picolo ,  Elisa Capparella

    发明人： Valerio Borzatta ,  Oreste Picolo ,  Elisa Capparella

    IPC分类号： A01N25/28

    CPC分类号： A01N43/30 ,  A01N25/28 ,  A01N53/00 ,  A01N2300/00

    摘要： The present invention relates to a new formulation characterised by the presence of two components, one of which (A) possesses insecticidal, acaricidal, fungicidal, snailcidal or vermicidal activity and the other (B) exhibits synergistic activity with the first by enhancing its effectiveness, and in which the average release time of component (A) is 1 to 12 hours later than the average release time of component (B). The formulation is obtained by: a) separate microencapsulation of both components (A) and (B) within a multilayer system of specific polymers in which component (A) is in a more interior portion of the capsule than component (B), being separated from component (B) by a polymer layer of suitable thickness (FIG. 1); b) microencapsulation of both components within a single layer system (FIG. 2), combined with an immediate-release emulsion/microemulsion containing an additional amount of component (B).

    摘要翻译： 本发明涉及一种新的制剂，其特征在于两种成分的存在，其中一种成分（A）具有杀虫，杀螨，杀真菌，杀虫或杀虫活性，另一种（B）通过提高其有效性与第一种成分具有协同作用， 其中组分（A）的平均释放时间比组分（B）的平均释放时间晚1至12小时。 该制剂通过以下方法获得：a）在特定聚合物的多层体系内单独的组分（A）和（B）的微胶囊化，其中组分（A）在组分（B）的更多内部部分中，分离 由组分（B）通过合适厚度的聚合物层（图1）; b）在单层系统（图2）中的两种组分的微囊化，与含有额外量的组分（B）的立即释放乳液/微乳液组合。

    Process for preparing 3,4-dioxo-substituted aromatic aldehydes
    9.
    发明授权
    Process for preparing 3,4-dioxo-substituted aromatic aldehydes 失效
    制备3,4-二氧代取代的芳族醛的方法

    公开(公告)号：US07544843B2

    公开(公告)日：2009-06-09

    申请号：US11996723

    申请日：2006-07-25

    申请人： Elisa Capparella ,  Elisa Poluzzi ,  Valerio Borzatta

    发明人： Elisa Capparella ,  Elisa Poluzzi ,  Valerio Borzatta

    IPC分类号： C07C45/29

    CPC分类号： C07C45/29 ,  C07C45/68 ,  C07D317/54 ,  C07C47/575

    摘要： A new process for synthesizing 3,4-dioxo-substituted aromatic aldehydes by Oppenauer oxidation of the corresponding benzyl alcohols is described. The process, which specifically uses formaldehyde as hydrogen acceptor, proceeds with unexpectedly high yields and conversion percentages, allowing low cost access to finished and intermediate products of high industrial interest in the field of pharmaceutical products and fragrances.

    摘要翻译： 描述了通过相应的苄醇的Oppenauer氧化合成3,4-二氧代取代的芳族醛的新方法。 特别使用甲醛作为氢受体的方法，出乎意料地高产率和转化率，允许低成本进入医药产品和香料领域具有高工业意义的成品和中间产品。

    Process for synthesizing heliotropine and its derivatives
    10.
    发明申请
    Process for synthesizing heliotropine and its derivatives 失效
    合成天葵及其衍生物的方法

    公开(公告)号：US20070100167A1

    公开(公告)日：2007-05-03

    申请号：US10577846

    申请日：2004-10-28

    申请人： Valerio Borzatta ,  Elisa Capparella ,  Carlotta Gobbi ,  Elisa Poluzzi

    发明人： Valerio Borzatta ,  Elisa Capparella ,  Carlotta Gobbi ,  Elisa Poluzzi

    IPC分类号： C07C45/90

    CPC分类号： C07D317/54

    摘要： A new high-yield, easily industrialized process for synthesizing compounds of formula (IV), in which X1 and X2, the same or different, are linear or branched C1-C8 alkyls, n and m are 0, 1 or 2, with the proviso that n and m are not simultaneously 0; or (OX1)n and (OX2)m taken together form an O-T-O group where T is chosen from —CH2—, —CH2CH2, —CH2CH2CH2—, —C(CH3)2—. The process comprises treating a chloromethyl derivative (I) with an alkaline acetate to form the intermediate acetylderivative (II); the intermediate (II) is to hydrolysed to form the alcohol (III); the alcohol (III) is then oxidised in the presence of air and catalysts to obtain the desired derivative (IV). The process runs its course within a short period of time, with high yields and high selectivity; in addition, the process does not require purification and separation of the intermediates and can therefore be favourably conducted in a single batch.

    摘要翻译： 合成式（IV）化合物的新的高产率，易于工业化的方法，其中相同或不同的X 1和X 2是直链或支链C1 -C 8烷基，n和m为0,1或2，条件是n和m不同时为0; 或（OX 1）n和（OX 2 N）m一起形成OTO基团，其中T选自-CH 2 - ， - CH 2 CH 2，CH 2 CH 2 CH 2 - ， - CH 2 CH 2 CH 2， - CH 2 CH 2 CH 2 - ， - C（CH 3）2 - 。 该方法包括用碱性乙酸盐处理氯甲基衍生物（I）以形成中间体乙酰衍生物（II）; 中间体（II）被水解形成醇（III）; 然后在空气和催化剂的存在下将醇（III）氧化以获得所需的衍生物（IV）。 该过程在短时间内运行，产量高，选择性高; 此外，该方法不需要中间体的纯化和分离，因此可以在单次批次中有利地进行。