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公开(公告)号:US20120122862A1
公开(公告)日:2012-05-17
申请号:US13361134
申请日:2012-01-30
申请人: Haiyan Jia , Ian Zachary , Michelle Tickner , Lili Cheng , Chris Chapman , Katie Ellard , Basil Hartzoulakis , Ashley Jarvis , Rosemary Lynch , Jamie Nally , David Selwood , Mark Stewart
发明人: Haiyan Jia , Ian Zachary , Michelle Tickner , Lili Cheng , Chris Chapman , Katie Ellard , Basil Hartzoulakis , Ashley Jarvis , Rosemary Lynch , Jamie Nally , David Selwood , Mark Stewart
IPC分类号: A61K31/538 , A61K31/197 , C07D333/38 , A61K31/381 , C07C311/46 , C07D277/56 , A61K31/426 , C07D307/68 , A61K31/341 , C07D417/12 , A61K31/433 , C07D409/12 , A61K31/4436 , C07D409/14 , C07D413/12 , C07D498/04 , A61K31/5383 , A61P25/00 , A61P25/28 , A61P35/00 , A61P37/02 , C07C279/14
CPC分类号: C07D333/38 , C07C279/12 , C07D277/56 , C07D307/68 , C07D409/12 , C07D409/14 , C07D413/12 , C07D413/14 , C07D417/12
摘要: The present invention is a compound of formula (I) or formula (II) which are suitable as NP-1 antagonists.
摘要翻译: 本发明是适合作为NP-1拮抗剂的式(I)或式(II)的化合物。
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公开(公告)号:US20120269864A1
公开(公告)日:2012-10-25
申请号:US13493110
申请日:2012-06-11
申请人: Haiyan Jia , Ian ZACHARY , Michelle TICKNER , Lili CHENG , Chris CHAPMAN , Katie ELLARD , Basil HARTZOULAKIS , Ashley JARVIS , Rosemary LYNCH , Jamie NALLY , David SELWOOD , Mark STEWART
发明人: Haiyan Jia , Ian ZACHARY , Michelle TICKNER , Lili CHENG , Chris CHAPMAN , Katie ELLARD , Basil HARTZOULAKIS , Ashley JARVIS , Rosemary LYNCH , Jamie NALLY , David SELWOOD , Mark STEWART
IPC分类号: A61K31/433 , A61K31/381 , C07D417/12 , C07D409/14 , A61K31/4436 , C07D413/12 , A61K31/538 , A61K31/506 , C07D498/04 , A61K31/5383 , A61K31/4245 , C07F5/02 , A61K31/69 , A61P25/28 , A61P25/00 , A61P35/00 , A61P37/02 , C07D409/12 , C07C279/14 , A61K31/197 , C07D277/56 , A61K31/4168 , C07D333/38
CPC分类号: C07D333/38 , C07C279/12 , C07D277/56 , C07D307/68 , C07D409/12 , C07D409/14 , C07D413/12 , C07D413/14 , C07D417/12
摘要: The present invention is a compound of formula (I) or formula (II) which are suitable as NP-1 antagonists.
摘要翻译: 本发明是适合作为NP-1拮抗剂的式(I)或式(II)的化合物。
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公开(公告)号:US08227606B2
公开(公告)日:2012-07-24
申请号:US13361134
申请日:2012-01-30
申请人: Haiyan Jia , Ian Zachary , Michelle Tickner , Lili Cheng , Chris Chapman , Katie Ellard , Basil Hartzoulakis , Ashley Jarvis , Rosemary Lynch , Jamie Nally , David Selwood , Mark Stewart
发明人: Haiyan Jia , Ian Zachary , Michelle Tickner , Lili Cheng , Chris Chapman , Katie Ellard , Basil Hartzoulakis , Ashley Jarvis , Rosemary Lynch , Jamie Nally , David Selwood , Mark Stewart
IPC分类号: C07D417/14
CPC分类号: C07D333/38 , C07C279/12 , C07D277/56 , C07D307/68 , C07D409/12 , C07D409/14 , C07D413/12 , C07D413/14 , C07D417/12
摘要: The present invention is a compound of formula (I) or formula (II) which are suitable as NP-1 antagonists.
摘要翻译: 本发明是适合作为NP-1拮抗剂的式(I)或式(II)的化合物。
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公开(公告)号:US08158789B2
公开(公告)日:2012-04-17
申请号:US12439523
申请日:2007-10-04
申请人: Haiyan Jia , Ian Zachary , Michelle Tickner , Lili Cheng , Chris Chapman , Katie Ellard , Basil Hartzoulakis , Ashley Jarvis , Rosemary Lynch , Jamie Nally , David Selwood , Mark Stewart
发明人: Haiyan Jia , Ian Zachary , Michelle Tickner , Lili Cheng , Chris Chapman , Katie Ellard , Basil Hartzoulakis , Ashley Jarvis , Rosemary Lynch , Jamie Nally , David Selwood , Mark Stewart
IPC分类号: C07D409/14
CPC分类号: C07D333/38 , C07C279/12 , C07D277/56 , C07D307/68 , C07D409/12 , C07D409/14 , C07D413/12 , C07D413/14 , C07D417/12
摘要: The present invention is a compound of formula (I) or formula (II) which are suitable as NP-1 antagonists.
摘要翻译: 本发明是适合作为NP-1拮抗剂的式(I)或式(II)的化合物。
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公开(公告)号:US20100022525A1
公开(公告)日:2010-01-28
申请号:US12439523
申请日:2007-10-04
申请人: Haiyan Jia , Ian Zachary , Michelle Tickner , Lili Cheng , Chris Chapman , Katie Ellard , Basil Hartzoulakis , Ashley Jarvis , Rosemary Lynch , Jamie Nally , David Selwood , Mark Stewart
发明人: Haiyan Jia , Ian Zachary , Michelle Tickner , Lili Cheng , Chris Chapman , Katie Ellard , Basil Hartzoulakis , Ashley Jarvis , Rosemary Lynch , Jamie Nally , David Selwood , Mark Stewart
IPC分类号: A61K31/538 , A61K31/4436 , A61K31/41 , A61K31/381 , C07D265/36 , C07D409/12 , C07D285/10 , C07D333/36
CPC分类号: C07D333/38 , C07C279/12 , C07D277/56 , C07D307/68 , C07D409/12 , C07D409/14 , C07D413/12 , C07D413/14 , C07D417/12
摘要: The present invention is a compound of formula (I) or formula (II) which are suitable as NP-1 antagonists.
摘要翻译: 本发明是适合作为NP-1拮抗剂的式(I)或式(II)的化合物。
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