公开(公告)号：US20070049635A1

公开(公告)日：2007-03-01

申请号：US10577653

申请日：2004-10-20

申请人： Koichi Ebihara ,  Kunihiko Morizane ,  Naofumi Tomura ,  Ryutaro Ezaki ,  Masako Yoshida ,  Yuko Osada

发明人： Koichi Ebihara ,  Kunihiko Morizane ,  Naofumi Tomura ,  Ryutaro Ezaki ,  Masako Yoshida ,  Yuko Osada

IPC分类号： A01N47/10 ,  C07C271/08 ,  C07C271/28

CPC分类号： C07D277/68 ,  A01N47/12 ,  C07C271/20 ,  C07D307/85

摘要： It is an object of the present invention to provide a diamine derivative, a process for producing the same, and a plant disease control agent containing the above-described compound as an active ingredient. According to the present invention, a diamine derivative represented by Formula (1), a process for producing the same, and a plant disease control agent containing the above-described compound as an active ingredient are provided. [In Formula, R1 represents, for example, a halogenated hydrocarbon having the carbon number of 1 to 6; R2 and R7 independently represent, for example, a hydrogen atom or a hydrocarbon having the carbon number of 1 to 6; R3 and R4 independently represent, for example, a hydrogen atom or a hydrocarbon which has the carbon number of 1 to 6 and which may be substituted, or represent a cycloalkyl group having the carbon number of 3 to 6 including a carbon atom bonding to R3 and R4; R5 and R6 independently represent, for example, a hydrogen atom or a hydrocarbon group having the carbon number of 1 to 6; and R8 represents an arylalkyl group which may be substituted, an aryl group which may be substituted, or a heteroaryl group which may be substituted.]

摘要翻译： 本发明的目的是提供二胺衍生物，其制备方法和含有上述化合物作为活性成分的植物病害防治剂。 根据本发明，提供由式（1）表示的二胺衍生物，其制备方法和含有上述化合物作为活性成分的植物病害防治剂。 [式中，R 1表示例如碳数为1〜6的卤代烃， R2和R7独立地表示例如氢原子或碳数为1至6的烃; R 3和R 4独立地表示例如氢原子或碳原子数1〜6的可以被取代的碳原子数为3〜6的环烷基，包括与R3结合的碳原子 和R4; R5和R6独立地表示例如氢原子或碳原子数为1〜6的烃基; R8表示可被取代的芳烷基，可被取代的芳基或可被取代的杂芳基。

公开(公告)号：US20090023667A1

公开(公告)日：2009-01-22

申请号：US11887152

申请日：2006-03-30

申请人： Naofumi Tomura ,  Kouichi Ebihara ,  Kunihiko Morizane ,  Ryutaro Ezaki ,  Nobuyuki Kawahara ,  Michikazu Nomura

发明人： Naofumi Tomura ,  Kouichi Ebihara ,  Kunihiko Morizane ,  Ryutaro Ezaki ,  Nobuyuki Kawahara ,  Michikazu Nomura

IPC分类号： A01N43/16 ,  A01N43/90 ,  A01N43/54 ,  A01N43/28 ,  A01N43/80 ,  A01N47/12 ,  A01P7/00 ,  A01N43/40 ,  A01N43/828 ,  A01N37/18 ,  A01N43/56 ,  A01N43/08

CPC分类号： A01N47/12 ,  A01N51/00 ,  A01N31/16 ,  A01N37/10 ,  A01N43/90 ,  A01N41/10 ,  A01N43/56 ,  A01N43/54 ,  A01N47/34 ,  A01N47/20 ,  A01N43/653 ,  A01N43/78 ,  A01N43/42 ,  A01N43/40 ,  A01N2300/00

摘要： An object of the present invention is to provide a composition for preventing harmful organisms exerting an excellent control effect against plant diseases and/or insecticidal effect. Disclosed is a composition for preventing harmful organisms comprising a diamine derivative represented by the formula (1), and one or more compounds selected from the group consisting of other fungicides, insecticides and acaricides as active ingredients, wherein, in the formula, R1 represents a hydrocarbon having 1 to 6 carbon atoms which is substituted with halogen or the like; R2 and R7 each independently represent a hydrogen atom, a hydrocarbon having 1 to 6 carbon atoms or the like; R3 and R4 each independently represent a hydrogen atom, a hydrocarbon having 1 to 6 carbon atoms which may be substituted or the like, or R3 and R4 represent a cycloalkyl group having 3 to 6 carbon atoms containing a carbon atom bonded thereto; R5 and R6 each independently represent a hydrogen atom, a hydrocarbon group having 1 to 6 carbon atoms or the like; and R8 represents an arylalkyl group which may be substituted, an aryl group which may be substituted or a heteroaryl group which may be substituted.

摘要翻译： 本发明的目的是提供一种防止对植物病害和/或杀虫效果具有优异防除效果的有害生物的组合物。 本发明公开了一种防止包含由式（1）表示的二胺衍生物和一种或多种选自其它杀真菌剂，杀虫剂和杀螨剂作为活性成分的化合物的有害生物的组合物，其中，式中R1表示 被卤素等取代的具有1至6个碳原子的烃; R2和R7各自独立地表示氢原子，碳原子数为1〜6的烃等; R 3和R 4各自独立地表示氢原子，可以被取代的碳原子数为1〜6的烃基，或者R 3和R 4表示碳原子数3〜6的环烷基，其中， R 5和R 6各自独立地表示氢原子，碳原子数为1〜6的烃基等; R8表示可被取代的芳烷基，可被取代的芳基或可被取代的杂芳基。

公开(公告)号：US20090192167A1

公开(公告)日：2009-07-30

申请号：US11989293

申请日：2006-07-19

申请人： Michikazu Nomura ,  Naofumi Tomura ,  Ryutaro Ezaki ,  Nobuyuki Kawahara

发明人： Michikazu Nomura ,  Naofumi Tomura ,  Ryutaro Ezaki ,  Nobuyuki Kawahara

IPC分类号： A01N43/08 ,  A01N43/60 ,  A01P3/00

CPC分类号： A01N47/12 ,  A01N37/46 ,  A01N43/40 ,  A01N47/20 ,  A01N2300/00

摘要： An insecticidal and fungicidal composition capable of controlling crop diseases and insect pests at the same time by combining an insecticidal active ingredient and a fungicidal active ingredient is provided. The insecticidal and fungicidal composition is characterized by comprising as active ingredients a compound represented by the general formula (1) or (2) and a compound represented by the general formula (3) or (4). wherein, in the formula, A1, A2, A3, and A4 independently represent a carbon atom, a nitrogen atom or an oxidized nitrogen atom; G1 and G2 independently represent an oxygen atom or a sulfur atom; R1 and R2 independently a hydrogen atom or a C1-C4 alkyl group; Xs may be the same or different and represent a hydrogen atom, a halogen atom or a trifluoromethyl group; Q1 represents substituents such as a phenyl group, a heterocyclic group or the like; and Q2 represents substituents such as a phenyl group, a heterocyclic group or the like.

摘要翻译： 提供了通过组合杀虫活性成分和杀真菌活性成分同时控制作物病虫害的杀虫杀真菌组合物。 杀虫剂和杀真菌组合物的特征在于，含有通式（1）或（2）表示的化合物和通式（3）或（4）表示的化合物作为活性成分。 其中，在该式中，A1，A2，A3和A4独立地表示碳原子，氮原子或氧化氮原子; G1和G2独立地表示氧原子或硫原子; R1和R2独立地为氢原子或C1-C4烷基; X可以相同或不同，表示氢原子，卤原子或三氟甲基; Q1表示取代基，例如苯基，杂环基等; Q2表示取代基，例如苯基，杂环基等。

公开(公告)号：US5965774A

公开(公告)日：1999-10-12

申请号：US150170

申请日：1998-09-09

申请人： Yukihiro Yoshikawa ,  Kanji Tomiya ,  Naofumi Tomura ,  Hiroyuki Katsuta ,  Osamu Takahashi ,  Shunichi Inami ,  Yuji Yanase ,  Junro Kishi ,  Hideo Kawashima

发明人： Yukihiro Yoshikawa ,  Kanji Tomiya ,  Naofumi Tomura ,  Hiroyuki Katsuta ,  Osamu Takahashi ,  Shunichi Inami ,  Yuji Yanase ,  Junro Kishi ,  Hideo Kawashima

IPC分类号： C07D231/14 ,  A01N43/26 ,  A01N43/56 ,  A01N43/78 ,  C07C211/45 ,  C07D213/82 ,  C07D231/16 ,  C07D241/14 ,  C07D263/34 ,  C07D277/20 ,  C07D277/30 ,  C07D277/56 ,  C07D307/68 ,  C07D309/28 ,  C07D327/06 ,  C07D333/24

CPC分类号： A01N43/56 ,  A01N43/78 ,  C07C211/45 ,  C07D231/14 ,  C07D277/56

摘要： A substituted anilide derivative represented by the formula (2): ##STR1## wherein A and B are methyl, and X is a hydrogen atom. The substituted anilide can be used to prepare a substituted carboxanilide derivative that exhibits a disease control effect against Botrytis cinerea, Powdery mildew, Pyricularia oryzae of rice plant and other various plant diseases, is excellent in residual effect, has activity against strains that are resistant to conventional chemicals, is safe for crops, and thus is useful as a plant disease control agent.

摘要翻译： 由式（2）表示的取代的酰苯胺衍生物：其中A和B是甲基，X是氢原子。 取代的酰苯胺可用于制备对灰葡萄孢，白粉病，稻瘟病菌和其他各种植物病害具有疾病防治作用的取代羧酰苯胺衍生物，其残留效果优异，具有抗抗性的菌株的活性 常规化学品对作物是安全的，因此可用作植物病害防治剂。

公开(公告)号：US5747518A

公开(公告)日：1998-05-05

申请号：US627929

申请日：1996-04-03

申请人： Yukihiro Yoshikawa ,  Kanji Tomiya ,  Hiroyuki Katsuta ,  Hideo Kawashima ,  Osamu Takahashi ,  Shunichi Inami ,  Yuji Yanase ,  Junro Kishi ,  Hitoshi Shimotori ,  Naofumi Tomura

发明人： Yukihiro Yoshikawa ,  Kanji Tomiya ,  Hiroyuki Katsuta ,  Hideo Kawashima ,  Osamu Takahashi ,  Shunichi Inami ,  Yuji Yanase ,  Junro Kishi ,  Hitoshi Shimotori ,  Naofumi Tomura

IPC分类号： A01N43/10 ,  A01N43/40 ,  A01N43/56 ,  A01N43/78 ,  C07D333/36 ,  C07D333/42 ,  C07D333/44 ,  C07D401/12 ,  C07D403/12 ,  C07D409/12 ,  C07D417/12 ,  A61K31/415 ,  A61K31/38 ,  A61K31/425 ,  A61K31/44

CPC分类号： C07D401/12 ,  A01N43/10 ,  A01N43/40 ,  A01N43/56 ,  A01N43/78 ,  C07D333/36 ,  C07D333/42 ,  C07D333/44 ,  C07D403/12 ,  C07D409/12 ,  C07D417/12

摘要： The substituted thiophene derivative of the invention which is represented by the general formula (1) has a broad disease spectrum for a pathogenic fungus of various crops, exhibits an excellent controlling effect on disease such as gray mold, powdery mildew and rust in particular, and is also effective for a resistant fungus of conventional fungicides which has become a serious problem, and consequently is useful for an agricultural and horticultural fungicide. ##STR1##

摘要翻译： 由通式（1）表示的本发明的取代噻吩衍生物对各种作物的致病真菌具有广泛的疾病谱，特别是对灰霉病，白粉病和锈病等疾病具有优异的防治效果， 对于已经成为严重问题的常规杀真菌剂的抗性真菌也是有效的，因此可用于农业和园艺杀真菌剂。 （1）

公开(公告)号：US5914344A

公开(公告)日：1999-06-22

申请号：US908187

申请日：1997-08-07

申请人： Yukihiro Yoshikawa ,  Kanji Tomiya ,  Naofumi Tomura ,  Hiroyuki Katsuta ,  Osamu Takahashi ,  Shunichi Inami ,  Yuji Yanase ,  Junro Kishi ,  Hideo Kawashima

发明人： Yukihiro Yoshikawa ,  Kanji Tomiya ,  Naofumi Tomura ,  Hiroyuki Katsuta ,  Osamu Takahashi ,  Shunichi Inami ,  Yuji Yanase ,  Junro Kishi ,  Hideo Kawashima

IPC分类号： C07D231/14 ,  A01N43/26 ,  A01N43/56 ,  A01N43/78 ,  C07C211/45 ,  C07D213/82 ,  C07D231/16 ,  C07D241/14 ,  C07D263/34 ,  C07D277/20 ,  C07D277/30 ,  C07D277/56 ,  C07D307/68 ,  C07D309/28 ,  C07D327/06 ,  C07D333/24 ,  A61K31/415

CPC分类号： A01N43/56 ,  A01N43/78 ,  C07C211/45 ,  C07D231/14 ,  C07D277/56

摘要： A substituted carboxanilide derivative represented by the formula (1): ##STR1## wherein A is a hydrogen atom or methyl, B is a methyl or ethyl, and Het is 1-methyl-3-substituted-4-pyrazolyl or 2-methyl-4-substituted-5-triazoyl group, exhibits a disease control effect against Botrytis cinerea, Powdery mildew, Pyricularia oryzae of rice plant and other various plant diseases, is excellent in residual effect, has also activity against resistant strain for conventional chemicals, particularly exerts control effects against Botrytis cinerea at a lower dosage as compared with a prior art, is also safe for crops, and thus is useful as a plant control agent.

摘要翻译： 由式（1）表示的取代的羧酰苯胺衍生物：其中A是氢原子或甲基，B是甲基或乙基，Het是1-甲基-3-取代-4-吡唑基或2-甲基-4-取代的 -5-三唑酰基对植物灰葡萄孢，白粉病，稻瘟病等多种植物病害具有防治效果，残留效果优异，对常规化学品的抗性菌株也具有抗菌活性，特别是对抗 与现有技术相比，较低剂量的灰葡萄孢属对于作物也是安全的，因此可用作植物控制剂。

公开(公告)号：US5869427A

公开(公告)日：1999-02-09

申请号：US962331

申请日：1997-10-31

申请人： Yukihiro Yoshikawa ,  Kanji Tomiya ,  Toshio Kitajima ,  Hiroyuki Katsuta ,  Osamu Takahashi ,  Shunichi Inami ,  Yuji Yanase ,  Naofumi Tomura ,  Junro Kishi ,  Hideo Kawasima

发明人： Yukihiro Yoshikawa ,  Kanji Tomiya ,  Toshio Kitajima ,  Hiroyuki Katsuta ,  Osamu Takahashi ,  Shunichi Inami ,  Yuji Yanase ,  Naofumi Tomura ,  Junro Kishi ,  Hideo Kawasima

IPC分类号： C07D409/12 ,  C07D417/12 ,  C04D333/22 ,  A01N43/10

CPC分类号： C07D409/12 ,  C07D417/12

摘要： A novel substituted thiophene derivatives represented by the formula (1) in the invention: ##STR1## wherein R is a straight or branched alkyl group having 3-12 carbon atoms, straight or branched halogenoalkyl group having 3-12 carbon atoms, straight or branched alkenyl group having 3-10 carbon atoms, straight or branched halogenoalkenyl group having 3-10 carbon atoms, or cycloalkyl group having 3-10 carbon atoms, the cycloalkyl group being unsubstituted or substituted with an alkyl group having 1-4 carbon atoms, R and --NHCOAr are adjacent to each other, and Ar is a heterocyclic group; have excellent control activity on various plant disease such as Gray mold, Powdery mildew, Blast and Rust, and are useful as a plant disease control agent due to outstanding residual effect on Botrytis cinerea and excellent effect on Gibberella zeae.

摘要翻译： 在本发明中由式（1）表示的新型取代噻吩衍生物：其中R是具有3-12个碳原子的直链或支链烷基，具有3-12个碳原子的直链或支链卤代烷基， 具有3-10个碳原子的直链或支链烯基，具有3-10个碳原子的直链或支链卤代烯基或具有3-10个碳原子的环烷基，所述环烷基是未取代的或被具有1-4个碳原子的烷基取代 原子，R和-NHCOAr彼此相邻，Ar是杂环基; 对灰霉病，白粉病，爆破和锈病等各种植物病害具有优异的防治作用，由于对灰葡萄孢的突出残留效果，对玉米赤霉菌有极好的效果，可用作植物病害防治剂。

公开(公告)号：US20070244153A1

公开(公告)日：2007-10-18

申请号：US11658098

申请日：2005-07-19

申请人： Takeshi Kakimoto ,  Hisato Kamekawa ,  Yutaka Chiba ,  Toshiyuki Kohno ,  Yumi Kobayashi ,  Naofumi Tomura ,  Natsuko Araki ,  Masako Yoshida ,  Yoji Aoki ,  Shinichi Banba

发明人： Takeshi Kakimoto ,  Hisato Kamekawa ,  Yutaka Chiba ,  Toshiyuki Kohno ,  Yumi Kobayashi ,  Naofumi Tomura ,  Natsuko Araki ,  Masako Yoshida ,  Yoji Aoki ,  Shinichi Banba

IPC分类号： A01N37/12 ,  A01N43/06 ,  A01N43/08 ,  A01N43/32 ,  A01N43/40 ,  A01N43/42 ,  C07C233/01

CPC分类号： C07D405/12 ,  C07C209/42 ,  C07C269/04 ,  C07C269/06 ,  C07C271/22 ,  C07C271/34 ,  C07C271/54 ,  C07C311/16 ,  C07C317/44 ,  C07C323/41 ,  C07C333/04 ,  C07C2601/08 ,  C07C2601/14

摘要： It is an object of the invention to provide a novel fungicide which exhibits a wide controlling spectrum against pathogens of various crops, and solves the toleration problem. The diamine derivative represented by the formula (1) and a process for preparation of the same, fungicides comprising the same as an active ingredient are disclosed: [wherein R1 is substituents such as an alkyl group having 1 to 6 carbon atoms and the like, R2 and R5 are each independently substituents such as hydrogen atom, an alkyl group having 1 to 6 carbon atoms and the like, R3 and R4 are each independently substituents such as hydrogen atom, an alkyl group having 1 to 6 carbon atoms and the like, or R3 and R4 may be bonded to each other to form a hydrocarbon ring having 3 to 6 carbon atoms, R6, R7, R8 and R9 are each independently substituents such as hydrogen atom, an alkyl group having 1 to 6 carbon atoms and the like, R10 is a substituent such as hydrogen atom, an alkyl group having 1 to 6 carbon atoms and the like, A is an oxygen atom or a sulfur atom, and Q is an aryl group or a heterocycle].

摘要翻译： 本发明的目的是提供一种对各种作物的病原体具有广泛控制谱的新型杀真菌剂，并解决了耐受性问题。 公开了式（1）表示的二胺衍生物及其制备方法：其中R1为具有1-6个碳原子的烷基等的取代基， R 2和R 5各自独立地为氢原子，碳原子数为1〜6的烷基等取代基，R 3和R 4各自独立地为氢原子，碳原子数1〜6的烷基等取代基， 或者R 3和R 4可以彼此键合形成具有3至6个碳原子的烃环，R 6，R 7，R 8和R 9各自独立地为氢原子，具有1至6个碳原子的烷基等取代基 中，R 10为氢原子，碳原子数为1〜6的烷基等取代基，A为氧原子或硫原子，Q为芳基或杂环。

公开(公告)号：US5240951A

公开(公告)日：1993-08-31

申请号：US761217

申请日：1991-09-19

申请人： Hitoshi Shimotori ,  Yuji Yanase ,  Takeshi Sekino ,  Katsutoshi Ishikawa ,  Toshiaki Kuwatsuka ,  Hiroharu Tanikawa ,  Hideo Kawashima ,  Naofumi Tomura ,  Yoshiro Kanemoto

发明人： Hitoshi Shimotori ,  Yuji Yanase ,  Takeshi Sekino ,  Katsutoshi Ishikawa ,  Toshiaki Kuwatsuka ,  Hiroharu Tanikawa ,  Hideo Kawashima ,  Naofumi Tomura ,  Yoshiro Kanemoto

IPC分类号： A01N43/80 ,  C07D275/02 ,  C07D275/03

CPC分类号： C07D275/03 ,  A01N43/80

摘要： Application of a rice blast control agent containing an isothiazolecarboxylic acid derivative of the below-described formula, which shows excellent activity against rice blast (Pyricularia oryzae) in rice cultivation, to the water surface of a paddy rice field results in the absorption of the derivative through roots of rice plants, so that the resistance of the rice plants can be enhanced. ##STR1## wherein R.sup.1 and R.sup.2 independently mean a hydrogen or halogen atom or a particular group, and Y stands for an OR.sub.3 group (R.sup.3 being a hydrogen or alkali metal atom or a particular group), an NHR.sup.4 group (R.sup.4 being a hydrogen atom or a particular group), or a morpholino group.

摘要翻译： 在水稻栽培中将含有对稻瘟病稻瘟病（Pyricularia oryzae）具有优异活性的下述式的异噻唑羧酸衍生物的稻瘟病控制剂施用于水稻田的水面，导致衍生物的吸收 通过水稻根系，可以提高水稻的抗性。 其中R1和R2独立地表示氢或卤素原子或特定基团，Y表示OR3基团（R3表示氢或碱金属原子或特定基团），NHR4基团（R4表示氢原子 或特定组）或吗啉基。