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1.
公开(公告)号:US3462440A
公开(公告)日:1969-08-19
申请号:US3462440D
申请日:1965-12-03
Applicant: AMERICAN HOME PROD
Inventor: CHILDRESS SCOTT J , ARCHIBALD JOHN L
IPC: C07D401/06 , C07D401/14 , C07D403/06 , C07D403/14 , C07D57/00 , A61K27/00
CPC classification number: C07D401/14 , C07D401/06 , C07D403/06 , C07D403/14
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2.1,4-bis-(3-indoleglyoxyloyl) piperazines and derivatives thereof 失效
Title translation: 1,4-BIS-(3-INDOLEGLYOXYLOYL)PIPERAZINES AND DERIVATIVES WITHOFOF公开(公告)号:US3577423A
公开(公告)日:1971-05-04
申请号:US3577423D
申请日:1969-06-26
Applicant: AMERICAN HOME PROD
Inventor: ARCHIBALD JOHN L , FREED MEIER E
IPC: C07D401/06 , C07D401/14 , C07D403/06 , C07D403/14
CPC classification number: C07D401/14 , C07D401/06 , C07D403/06 , C07D403/14
Abstract: THE COMPOUNDS ARE 1,4-BIS (3-INDOLEGLYOXYLOYL) PIPERAZINES. SAID COMPOUNDS ARE USEFUL AS INTERMEDIATES IN THE PREPARATION OF CORRESPONDING 1,4-BIS(2-INDOL-3-YLETHYL)PIPERAZINES AND THEIR SALTS, WHICH ARE PHARMACOLOGICALLY ACTIVE AS HYPOTENSIVES.
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3.Certain decahydro and dodecahydro-5h-pyrido(1,2-a) - 1,6 - naphthyridine - 5 - ones,the corresponding - 5 - ols and derivatives thereof 失效
Title translation: 某些十氢化萘和十五氢-5H-吡啶(1,2-A)-1,6-萘啶-5-胺,相应的5-OLS及其衍生物公开(公告)号:US3557100A
公开(公告)日:1971-01-19
申请号:US3557100D
申请日:1969-06-11
Applicant: AMERICAN HOME PROD
Inventor: FREED MEIER E , ARCHIBALD JOHN L
IPC: C07D471/14 , C07D39/10
CPC classification number: C07D471/14
Abstract: THIS INVENTION RELATES TO DECAHYDRO AND DODECAHYDRO5H-PYRIDO(1,2-A)-1,6-NAPHTHYRIDINE COMPOUNDS, THEIR SUBSTITUTENTS, AND A PROCESS FOR THEIR PREPARATION. THE COMPOUNDS ARE USEFUL IN PHARMACOLOGY AS ANTIANDROGENIC, ANALGESIC AND CENTRAL NERVOUS SYSTEM DEPRESSANT AGENTS.
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4.Bis(pyridylethyl)- and bis(piperidylethyl)-indoles 失效
Title translation: BIS(PYRIDYLETHYL)和BIS(PIPERIDYLETHYL)-INDOLES公开(公告)号:US3462441A
公开(公告)日:1969-08-19
申请号:US3462441D
申请日:1966-01-03
Applicant: AMERICAN HOME PROD
Inventor: FREED MEIER E , ARCHIBALD JOHN L
IPC: C07D401/06 , C07D401/14 , C07D403/06 , C07D403/14 , C07D57/00 , A61K27/00
CPC classification number: C07D401/14 , C07D401/06 , C07D403/06 , C07D403/14
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公开(公告)号:US3471499A
公开(公告)日:1969-10-07
申请号:US3471499D
申请日:1965-12-03
Applicant: AMERICAN HOME PROD
Inventor: ARCHIBALD JOHN L , FREED MEIER E
IPC: C07D401/06 , C07D401/14 , C07D403/06 , C07D403/14 , C07D57/00 , A61K27/00
CPC classification number: C07D401/14 , C07D401/06 , C07D403/06 , C07D403/14
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公开(公告)号:US3431268A
公开(公告)日:1969-03-04
申请号:US3431268D
申请日:1965-10-19
Applicant: AMERICAN HOME PROD
Inventor: ARCHIBALD JOHN L
IPC: C07D401/14 , C07D57/00
CPC classification number: C07D401/14
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公开(公告)号:US3501481A
公开(公告)日:1970-03-17
申请号:US3501481D
申请日:1966-12-22
Applicant: AMERICAN HOME PROD
Inventor: ARCHIBALD JOHN L , FREED MEIER E
IPC: C07D455/03 , C07D471/04 , C07D33/38
CPC classification number: C07D455/00 , C07D471/04
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公开(公告)号:US3458515A
公开(公告)日:1969-07-29
申请号:US3458515D
申请日:1966-07-21
Applicant: AMERICAN HOME PROD
Inventor: ARCHIBALD JOHN L , FREED MEIER E
IPC: C07D207/32 , C07D207/335 , C07D207/337 , C07D57/00 , C07D27/22 , C07D51/00
CPC classification number: C07D207/335 , C07D207/337
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9.
公开(公告)号:US3445472A
公开(公告)日:1969-05-20
申请号:US3445472D
申请日:1965-12-03
Applicant: AMERICAN HOME PROD
Inventor: ARCHIBALD JOHN L
IPC: C07D401/06 , C07D401/14 , C07D403/06 , C07D403/14 , C07D57/00 , C07D29/34 , C07D31/40
CPC classification number: C07D401/14 , C07D401/06 , C07D403/06 , C07D403/14
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公开(公告)号:US3429885A
公开(公告)日:1969-02-25
申请号:US3429885D
申请日:1965-10-22
Applicant: AMERICAN HOME PROD
Inventor: ARCHIBALD JOHN L
CPC classification number: A61K31/00
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