-
1.
公开(公告)号:US20080275056A1
公开(公告)日:2008-11-06
申请号:US12089420
申请日:2006-10-23
申请人: Alfonso De Dios , Cristina Garcia-Paredes , Beatriz Lopez Uralde Garmendia , Mary Margaret Mader , Mark Andrew Pobanz , Chuan Shih , Boyu Zhong
发明人: Alfonso De Dios , Cristina Garcia-Paredes , Beatriz Lopez Uralde Garmendia , Mary Margaret Mader , Mark Andrew Pobanz , Chuan Shih , Boyu Zhong
IPC分类号: A61K31/496 , C07D401/14 , A61K31/4725
CPC分类号: C07D403/12 , C07D403/14
摘要: The present invention provides kinase inhibitors of Formula (I) wherein R1, R2, and X are as described herein, or a pharmaceutically acceptable salt thereof.
摘要翻译: 本发明提供其中R1,R2和X如本文所述的式(I)的激酶抑制剂或其药学上可接受的盐。
-
2.
公开(公告)号:US07582638B2
公开(公告)日:2009-09-01
申请号:US12089420
申请日:2006-10-23
申请人: Alfonso De Dios , Cristina Garcia-Paredes , Beatriz López de Uralde Garmendia , Mary Margaret Mader , Mark Andrew Pobanz , Chuan Shih , Boyu Zhong
发明人: Alfonso De Dios , Cristina Garcia-Paredes , Beatriz López de Uralde Garmendia , Mary Margaret Mader , Mark Andrew Pobanz , Chuan Shih , Boyu Zhong
IPC分类号: A61K31/4725 , A61K31/496 , C07D403/141
CPC分类号: C07D403/12 , C07D403/14
摘要: The present invention provides kinase inhibitors of Formula (I) wherein R1, R2, and X are as described herein, or a pharmaceutically acceptable salt thereof.
摘要翻译: 本发明提供其中R1,R2和X如本文所述的式(I)的激酶抑制剂或其药学上可接受的盐。
-
公开(公告)号:US07652015B2
公开(公告)日:2010-01-26
申请号:US12088526
申请日:2006-10-25
申请人: Jolie Anne Bastian , Jesus Andres Blas de Blas , Alfonso De Dios , Kevin John Hudziak , Tiechao Li , Beatriz López De Uralde-Garmendia , Mary Margaret Mader , Michael Ray Myers , Mark Andrew Pobanz , Chuan Shih , Boyu Zhong
发明人: Jolie Anne Bastian , Jesus Andres Blas de Blas , Alfonso De Dios , Kevin John Hudziak , Tiechao Li , Beatriz López De Uralde-Garmendia , Mary Margaret Mader , Michael Ray Myers , Mark Andrew Pobanz , Chuan Shih , Boyu Zhong
IPC分类号: A61K31/4439 , A61K31/454 , C07D401/12 , C07D401/14 , C07D409/14
CPC分类号: C07D401/12 , C07D401/14
摘要: The present invention provides kinase inhibitors of Formula (I). Wherein R1, R2, X and Z are as described herein, or a pharmaceutically acceptable salt thereof.
摘要翻译: 本发明提供式(I)的激酶抑制剂。 其中R1,R2,X和Z如本文所述,或其药学上可接受的盐。
-
公开(公告)号:US20080269244A1
公开(公告)日:2008-10-30
申请号:US12088526
申请日:2006-10-25
申请人: Jolie Anne Bastian , Jesus Andres Blas de Blas , Alfonso De Dios , Kevin John Hudziak , Tiechao Li , Beatriz Lopez De Uralde-Garmendia , Mary Margaret Mader , Michael Ray Myers , Mark Andrew Pobanz , Chuan Shih , Boyu Zhong
发明人: Jolie Anne Bastian , Jesus Andres Blas de Blas , Alfonso De Dios , Kevin John Hudziak , Tiechao Li , Beatriz Lopez De Uralde-Garmendia , Mary Margaret Mader , Michael Ray Myers , Mark Andrew Pobanz , Chuan Shih , Boyu Zhong
IPC分类号: A61K31/496 , C07D401/14
CPC分类号: C07D401/12 , C07D401/14
摘要: The present invention provides kinase inhibitors of Formula (I). Wherein R1, R2, X and Z are as described herein, or a pharmaceutically acceptable salt thereof.
摘要翻译: 本发明提供式(I)的激酶抑制剂。 其中R 1,R 2,X和Z如本文所述,或其药学上可接受的盐。
-
公开(公告)号:US07767674B2
公开(公告)日:2010-08-03
申请号:US11569809
申请日:2005-06-15
申请人: Tiechao Li , Mark Andrew Pobanz , Chuan Shih , Yong Wang , Boyu Zhong , Jesus Andres Blas , Alfonso De Dios , Beatriz Lopez De Uralde-Garmendia , Luisa Maria Martin Cabrejas
发明人: Tiechao Li , Mark Andrew Pobanz , Chuan Shih , Yong Wang , Boyu Zhong , Jesus Andres Blas , Alfonso De Dios , Beatriz Lopez De Uralde-Garmendia , Luisa Maria Martin Cabrejas
IPC分类号: A61K31/5377 , A61K31/496 , A61K31/415 , A61K31/4439 , C07D231/40 , C07D401/12 , C07D413/14
CPC分类号: C07D401/12 , C07D401/14 , C07D409/14 , C07D413/14
摘要: The present invention provides kinase inhibitors of Formula I:
摘要翻译: 本发明提供式I的激酶抑制剂:
-
公开(公告)号:US20080306068A1
公开(公告)日:2008-12-11
申请号:US11569809
申请日:2005-06-15
申请人: Tiechao Li , Mark Andrew Pobanz , Chuan Shih , Yong Wang , Boyu Zhong , Jesus Andres Blas , Alfonso De Dios , Beatriz Lopez De Uralde-Garmendia , Luisa Maria Martin Cabrejas
发明人: Tiechao Li , Mark Andrew Pobanz , Chuan Shih , Yong Wang , Boyu Zhong , Jesus Andres Blas , Alfonso De Dios , Beatriz Lopez De Uralde-Garmendia , Luisa Maria Martin Cabrejas
IPC分类号: A61K31/5377 , C07D401/02 , A61K31/454 , C07D401/14 , A61P29/00 , A61P37/02 , A61P25/00 , A61K31/4545 , A61K31/496 , C07D295/00
CPC分类号: C07D401/12 , C07D401/14 , C07D409/14 , C07D413/14
摘要: The present invention provides kinase inhibitors of Formula I:
摘要翻译: 本发明提供式I的激酶抑制剂:
-
公开(公告)号:USRE43878E1
公开(公告)日:2012-12-25
申请号:US13374053
申请日:2011-12-08
申请人: Tiechao Li , Mark Andrew Pobanz , Chuan Shih , Zhipei Wu , Wei Jennifer Yang , Boyu Zhong
发明人: Tiechao Li , Mark Andrew Pobanz , Chuan Shih , Zhipei Wu , Wei Jennifer Yang , Boyu Zhong
IPC分类号: A61K31/416 , A61K31/4439 , A61K31/444 , A61K31/501 , C07D401/14 , C07D413/14 , C07D403/12
CPC分类号: C07D401/14 , C07D401/12 , C07D403/12 , C07D403/14 , C07D405/14
摘要: The present invention provides amidophenoxyindazole compounds useful in the treatment of cancer.
摘要翻译: 本发明提供了可用于治疗癌症的氨基苯氧基吲唑化合物。
-
公开(公告)号:US08030302B2
公开(公告)日:2011-10-04
申请号:US12503223
申请日:2009-07-15
申请人: Tiechao Li , Mark Andrew Pobanz , Chuan Shih , Zhipei Wu , Wei Jennifer Yang , Boyu Zhong
发明人: Tiechao Li , Mark Andrew Pobanz , Chuan Shih , Zhipei Wu , Wei Jennifer Yang , Boyu Zhong
IPC分类号: A61K31/416 , A61K31/4439 , A61K31/444 , A61K31/501 , C07D401/14 , C07D413/14 , C07D403/12
CPC分类号: C07D401/14 , C07D401/12 , C07D403/12 , C07D403/14 , C07D405/14
摘要: The present invention provides amidophenoxyindazole compounds useful in the treatment of cancer.
摘要翻译: 本发明提供了可用于治疗癌症的氨基苯氧基吲唑化合物。
-
公开(公告)号:US07666879B2
公开(公告)日:2010-02-23
申请号:US11816416
申请日:2006-02-23
申请人: David Anthony Barda , Timothy Paul Burkholder , Joshua Ryan Clayton , Yan Hao , James Robert Henry , John Monte Knobeloch , Johnathan Alexander McLean , David Mendel , Mark Edward Rempala , Zhao-Qing Wang , Yvonne Yee Mai Yip , Boyu Zhong
发明人: David Anthony Barda , Timothy Paul Burkholder , Joshua Ryan Clayton , Yan Hao , James Robert Henry , John Monte Knobeloch , Johnathan Alexander McLean , David Mendel , Mark Edward Rempala , Zhao-Qing Wang , Yvonne Yee Mai Yip , Boyu Zhong
IPC分类号: A01N43/42 , A61K31/44 , C07D471/02 , C07D491/02 , C07D498/02 , C07D513/02 , C07D515/02 , C07D401/00
CPC分类号: C07D471/04
摘要: The present invention provides compounds that are inhibitors of VEGF-R2 of the formula: (I) and methods of using these compounds.
摘要翻译: 本发明提供了下式所示的VEGF-R2抑制剂的化合物:(I)和使用这些化合物的方法。
-
10.
公开(公告)号:US20090227622A1
公开(公告)日:2009-09-10
申请号:US11816416
申请日:2006-02-23
申请人: David Anthony Barda , Timothy Paul Burkholder , Joshua Ryan Clayton , Yan Hao , James Robert Henry , John Monte Knobeloch , Johnathan Alexander Mclean , David Mendel , Mark Edward Rempala , Zhao-Qing Wang , Yvonne Yee Yip , Boyu Zhong
发明人: David Anthony Barda , Timothy Paul Burkholder , Joshua Ryan Clayton , Yan Hao , James Robert Henry , John Monte Knobeloch , Johnathan Alexander Mclean , David Mendel , Mark Edward Rempala , Zhao-Qing Wang , Yvonne Yee Yip , Boyu Zhong
IPC分类号: A61K31/437 , C07D471/04
CPC分类号: C07D471/04
摘要: The present invention provides compounds that are inhibitors of VEGF-R2 of the formula: (I) and methods of using these compounds.
摘要翻译: 本发明提供了下式所示的VEGF-R2抑制剂的化合物:(I)和使用这些化合物的方法。
-
-
-
-
-
-
-
-
-