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公开(公告)号:US20080269244A1
公开(公告)日:2008-10-30
申请号:US12088526
申请日:2006-10-25
申请人: Jolie Anne Bastian , Jesus Andres Blas de Blas , Alfonso De Dios , Kevin John Hudziak , Tiechao Li , Beatriz Lopez De Uralde-Garmendia , Mary Margaret Mader , Michael Ray Myers , Mark Andrew Pobanz , Chuan Shih , Boyu Zhong
发明人: Jolie Anne Bastian , Jesus Andres Blas de Blas , Alfonso De Dios , Kevin John Hudziak , Tiechao Li , Beatriz Lopez De Uralde-Garmendia , Mary Margaret Mader , Michael Ray Myers , Mark Andrew Pobanz , Chuan Shih , Boyu Zhong
IPC分类号: A61K31/496 , C07D401/14
CPC分类号: C07D401/12 , C07D401/14
摘要: The present invention provides kinase inhibitors of Formula (I). Wherein R1, R2, X and Z are as described herein, or a pharmaceutically acceptable salt thereof.
摘要翻译: 本发明提供式(I)的激酶抑制剂。 其中R 1,R 2,X和Z如本文所述,或其药学上可接受的盐。
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公开(公告)号:US07652015B2
公开(公告)日:2010-01-26
申请号:US12088526
申请日:2006-10-25
申请人: Jolie Anne Bastian , Jesus Andres Blas de Blas , Alfonso De Dios , Kevin John Hudziak , Tiechao Li , Beatriz López De Uralde-Garmendia , Mary Margaret Mader , Michael Ray Myers , Mark Andrew Pobanz , Chuan Shih , Boyu Zhong
发明人: Jolie Anne Bastian , Jesus Andres Blas de Blas , Alfonso De Dios , Kevin John Hudziak , Tiechao Li , Beatriz López De Uralde-Garmendia , Mary Margaret Mader , Michael Ray Myers , Mark Andrew Pobanz , Chuan Shih , Boyu Zhong
IPC分类号: A61K31/4439 , A61K31/454 , C07D401/12 , C07D401/14 , C07D409/14
CPC分类号: C07D401/12 , C07D401/14
摘要: The present invention provides kinase inhibitors of Formula (I). Wherein R1, R2, X and Z are as described herein, or a pharmaceutically acceptable salt thereof.
摘要翻译: 本发明提供式(I)的激酶抑制剂。 其中R1,R2,X和Z如本文所述,或其药学上可接受的盐。
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公开(公告)号:US20080306068A1
公开(公告)日:2008-12-11
申请号:US11569809
申请日:2005-06-15
申请人: Tiechao Li , Mark Andrew Pobanz , Chuan Shih , Yong Wang , Boyu Zhong , Jesus Andres Blas , Alfonso De Dios , Beatriz Lopez De Uralde-Garmendia , Luisa Maria Martin Cabrejas
发明人: Tiechao Li , Mark Andrew Pobanz , Chuan Shih , Yong Wang , Boyu Zhong , Jesus Andres Blas , Alfonso De Dios , Beatriz Lopez De Uralde-Garmendia , Luisa Maria Martin Cabrejas
IPC分类号: A61K31/5377 , C07D401/02 , A61K31/454 , C07D401/14 , A61P29/00 , A61P37/02 , A61P25/00 , A61K31/4545 , A61K31/496 , C07D295/00
CPC分类号: C07D401/12 , C07D401/14 , C07D409/14 , C07D413/14
摘要: The present invention provides kinase inhibitors of Formula I:
摘要翻译: 本发明提供式I的激酶抑制剂:
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公开(公告)号:US07767674B2
公开(公告)日:2010-08-03
申请号:US11569809
申请日:2005-06-15
申请人: Tiechao Li , Mark Andrew Pobanz , Chuan Shih , Yong Wang , Boyu Zhong , Jesus Andres Blas , Alfonso De Dios , Beatriz Lopez De Uralde-Garmendia , Luisa Maria Martin Cabrejas
发明人: Tiechao Li , Mark Andrew Pobanz , Chuan Shih , Yong Wang , Boyu Zhong , Jesus Andres Blas , Alfonso De Dios , Beatriz Lopez De Uralde-Garmendia , Luisa Maria Martin Cabrejas
IPC分类号: A61K31/5377 , A61K31/496 , A61K31/415 , A61K31/4439 , C07D231/40 , C07D401/12 , C07D413/14
CPC分类号: C07D401/12 , C07D401/14 , C07D409/14 , C07D413/14
摘要: The present invention provides kinase inhibitors of Formula I:
摘要翻译: 本发明提供式I的激酶抑制剂:
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公开(公告)号:US07084170B2
公开(公告)日:2006-08-01
申请号:US10490935
申请日:2002-10-15
申请人: Cora Sue Grossman , Philip Arthur Hipskind , Ho-Shen Lin , Karen Lynn Lobb , Beatriz Lopez de Uralde Garmendia , Jose Eduardo Lopez , Mary Margaret Mader , Michael Enrico Richett , Chuan Shih , Alfonso De Dios
发明人: Cora Sue Grossman , Philip Arthur Hipskind , Ho-Shen Lin , Karen Lynn Lobb , Beatriz Lopez de Uralde Garmendia , Jose Eduardo Lopez , Mary Margaret Mader , Michael Enrico Richett , Chuan Shih , Alfonso De Dios
IPC分类号: A61K31/381 , C07D333/34
CPC分类号: C07D277/36 , C07D333/34 , C07D333/38
摘要: The present invention provides antineoplastic compounds of the formula: and antineoplastic methods.
摘要翻译: 本发明提供下式的抗肿瘤化合物和抗肿瘤方法。
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公开(公告)号:US07250430B2
公开(公告)日:2007-07-31
申请号:US11447457
申请日:2006-06-06
申请人: Cora Sue Grossman , Philip Arthur Hipskind , Ho-Shen Lin , Karen Lynn Lobb , Beatriz Lopez de Uralde Garmendia , Jose Eduardo Lopez , Mary Margaret Mader , Michael Enrico Richett , Chuan Shih , Alfonso De Dios
发明人: Cora Sue Grossman , Philip Arthur Hipskind , Ho-Shen Lin , Karen Lynn Lobb , Beatriz Lopez de Uralde Garmendia , Jose Eduardo Lopez , Mary Margaret Mader , Michael Enrico Richett , Chuan Shih , Alfonso De Dios
IPC分类号: A61K31/381 , A61K31/426
CPC分类号: C07D277/36 , C07D333/34 , C07D333/38
摘要: The present invention provides antineoplastic compounds of the formula: and antineoplastic methods.
摘要翻译: 本发明提供下式的抗肿瘤化合物和抗肿瘤方法。
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7.
公开(公告)号:US20080275056A1
公开(公告)日:2008-11-06
申请号:US12089420
申请日:2006-10-23
申请人: Alfonso De Dios , Cristina Garcia-Paredes , Beatriz Lopez Uralde Garmendia , Mary Margaret Mader , Mark Andrew Pobanz , Chuan Shih , Boyu Zhong
发明人: Alfonso De Dios , Cristina Garcia-Paredes , Beatriz Lopez Uralde Garmendia , Mary Margaret Mader , Mark Andrew Pobanz , Chuan Shih , Boyu Zhong
IPC分类号: A61K31/496 , C07D401/14 , A61K31/4725
CPC分类号: C07D403/12 , C07D403/14
摘要: The present invention provides kinase inhibitors of Formula (I) wherein R1, R2, and X are as described herein, or a pharmaceutically acceptable salt thereof.
摘要翻译: 本发明提供其中R1,R2和X如本文所述的式(I)的激酶抑制剂或其药学上可接受的盐。
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8.
公开(公告)号:US07582638B2
公开(公告)日:2009-09-01
申请号:US12089420
申请日:2006-10-23
申请人: Alfonso De Dios , Cristina Garcia-Paredes , Beatriz López de Uralde Garmendia , Mary Margaret Mader , Mark Andrew Pobanz , Chuan Shih , Boyu Zhong
发明人: Alfonso De Dios , Cristina Garcia-Paredes , Beatriz López de Uralde Garmendia , Mary Margaret Mader , Mark Andrew Pobanz , Chuan Shih , Boyu Zhong
IPC分类号: A61K31/4725 , A61K31/496 , C07D403/141
CPC分类号: C07D403/12 , C07D403/14
摘要: The present invention provides kinase inhibitors of Formula (I) wherein R1, R2, and X are as described herein, or a pharmaceutically acceptable salt thereof.
摘要翻译: 本发明提供其中R1,R2和X如本文所述的式(I)的激酶抑制剂或其药学上可接受的盐。
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公开(公告)号:US20060223871A1
公开(公告)日:2006-10-05
申请号:US11447457
申请日:2006-06-06
申请人: Cora Grossman , Philip Hipskind , Ho-Shen Lin , Karen Lobb , Beatriz Lopez de Uralde Garmendia , Jose Lopez , Mary Mader , Michael Richett , Chuan Shih , Alfonso De Dios
发明人: Cora Grossman , Philip Hipskind , Ho-Shen Lin , Karen Lobb , Beatriz Lopez de Uralde Garmendia , Jose Lopez , Mary Mader , Michael Richett , Chuan Shih , Alfonso De Dios
IPC分类号: A61K31/426 , A61K31/381 , C07D333/34
CPC分类号: C07D277/36 , C07D333/34 , C07D333/38
摘要: The present invention provides antineoplastic compounds of the formula: and antineoplastic methods.
摘要翻译: 本发明提供下式的抗肿瘤化合物和抗肿瘤方法。
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公开(公告)号:US08030302B2
公开(公告)日:2011-10-04
申请号:US12503223
申请日:2009-07-15
申请人: Tiechao Li , Mark Andrew Pobanz , Chuan Shih , Zhipei Wu , Wei Jennifer Yang , Boyu Zhong
发明人: Tiechao Li , Mark Andrew Pobanz , Chuan Shih , Zhipei Wu , Wei Jennifer Yang , Boyu Zhong
IPC分类号: A61K31/416 , A61K31/4439 , A61K31/444 , A61K31/501 , C07D401/14 , C07D413/14 , C07D403/12
CPC分类号: C07D401/14 , C07D401/12 , C07D403/12 , C07D403/14 , C07D405/14
摘要: The present invention provides amidophenoxyindazole compounds useful in the treatment of cancer.
摘要翻译: 本发明提供了可用于治疗癌症的氨基苯氧基吲唑化合物。
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