公开(公告)号：US10562921B2

公开(公告)日：2020-02-18

申请号：US15590159

申请日：2017-05-09

申请人： Anacor Pharmaceuticals, Inc.

发明人： Tsutomu Akama ,  David Scott Carter ,  Jason S. Halladay ,  Robert T. Jacobs ,  Yang Liu ,  Jacob J. Plattner ,  Yong-Kang Zhang ,  Michael John Witty

IPC分类号： A61K31/166 ,  C07F5/02 ,  A61K31/443 ,  A61K31/4525 ,  A61K31/69 ,  A61K31/4178 ,  A61K31/431 ,  A61K31/47 ,  A61K31/5377

摘要： The present invention provides oxaborole ester compounds and compositions thereof which are useful to treat diseases associated with parasites, such as Chagas Disease and African Animal Trypanosomosis.

公开(公告)号：US11578087B2

公开(公告)日：2023-02-14

申请号：US17108066

申请日：2020-12-01

申请人： Anacor Pharmaceuticals, Inc.

发明人： Tsutomu Akama ,  David Scott Carter ,  Jason S. Halladay ,  Robert T. Jacobs ,  Yang Liu ,  Jacob J. Plattner ,  Yong-Kang Zhang ,  Michael John Witty

IPC分类号： C07F5/00 ,  C07F5/02 ,  A61K31/166 ,  A61K31/443 ,  A61K31/4525 ,  A61K31/69 ,  A61K31/4178 ,  A61K31/431 ,  A61K31/47 ,  A61K31/5377

摘要： The present invention provides oxaborole ester compounds and compositions thereof which are useful to treat diseases associated with parasites, such as Chagas Disease and African Animal Trypanosomosis.

公开(公告)号：US20180072760A1

公开(公告)日：2018-03-15

申请号：US15562099

申请日：2016-04-08

申请人： ANACOR PHARMACEUTICALS, INC.

发明人： Yong-Kang ZHANG ,  Jacob J. Plattner ,  Robert T. Jacobs

IPC分类号： C07F5/02

CPC分类号： C07F5/025 ,  C07D241/18

摘要： This invention provides, among other things, novel compounds useful for treating protozoal infections, pharmaceutical compositions containing such compounds, as well as combinations of these compounds with at least one additional therapeutically effective agent. Formula (I) and (II)

公开(公告)号：US10882872B2

公开(公告)日：2021-01-05

申请号：US16580676

申请日：2019-09-24

申请人： Anacor Pharmaceuticals, Inc.

发明人： Tsutomu Akama ,  David Scott Carter ,  Jason S. Halladay ,  Robert T. Jacobs ,  Yang Liu ,  Jacob J. Plattner ,  Yong-Kang Zhang ,  Michael John Witty

IPC分类号： C07F5/00 ,  C07F5/02 ,  A61K31/166 ,  A61K31/443 ,  A61K31/4525 ,  A61K31/69 ,  A61K31/4178 ,  A61K31/431 ,  A61K31/47 ,  A61K31/5377

摘要： The present invention provides oxaborole ester compounds and compositions thereof which are useful to treat diseases associated with parasites, such as Chagas Disease and African Animal Trypanosomosis.