公开(公告)号：US3925386A

公开(公告)日：1975-12-09

申请号：US26687272

申请日：1972-06-28

Applicant: BAYER AG

Inventor： JAGER GERHARD ,  WENZELBURGER HANS JURGEN ,  SCHMIDT ROBERT R

IPC: C07D239/22 ,  C07D265/12 ,  C07D319/08 ,  C07D239/04

CPC classification number: C07D239/22 ,  C07D265/12 ,  C07D319/08

Abstract: Novel 6-hydroxy-dihydro-uracil compounds of the formula:

WHEREIN R1 is hydrocarbyl and substituted hydrocarbyl, both aliphatic and aromatic, R2 is hydrogen, alkyl, or optionally, substituted aryl, R3 is alkyl or aralkyl, and R2 and R3 together may be an alkylene bridge; ARE PREPARED BY REACTING A 2,3-DIHYDRO-1,3-OXAZINE-2,4-DIONE OF THE GENERAL FORMULA

IN WHICH R1, R2 and R3 have the above mentioned meanings, is reacted with ammonia at a temperature of -50*C to +50*C, optionally in the presence of a diluent, but in the substantial absence of water. These compounds are herbicidally active.

Abstract translation: 新型6-羟基 - 二氢尿嘧啶化合物，其具有下式：

公开(公告)号：US3870726A

公开(公告)日：1975-03-11

申请号：US34858173

申请日：1973-04-06

Applicant: BAYER AG

Inventor： JAGER GERHARD ,  PLEMPEL MANFRED ,  BUCHEL KARL HEINZ

IPC: C07C29/42 ,  C07D295/084 ,  C07D521/00 ,  C07D49/36

CPC classification number: C07D295/092 ,  C07C29/42 ,  C07D231/12 ,  C07D233/56 ,  C07D249/08 ,  C07C33/20 ,  C07C33/28

Abstract: 3-PHENYL-3-AZOLYLPROPYNES BEARING A LOWER ALKYL OR ARYL GROUP IN THE 3-POSITION AND OPTIONALLY SUBSTITUTED IN THE 1-POSITION BY HALOGENO, LOWER ALKYL, ARYL OR CERTAIN SUBSTITUTED LOWER ALKYL GROUPS ARE PREPARED BY TREATING THE CORRESPONDING 3HYDROXYPROPYNE WITH A THIONYL BISAZOLE. Certain of the 1substituted compounds can be prepared through substitution reactions utilizing the lithium salt. The compounds and their salts, of which 3,3-diphenyl-3-(imidazolyl-(1))-propyne is a typical embodiment, are antimycotic agents and can be employed alone or in the form of pharmaceutical compositions in the treatment of mycotic infections in animals.

Abstract translation: 3-苯基-3-丙烯酸酯在3位置上的低级烷基或亚芳基可以被卤代烷基，低级亚烷基，亚芳基或某些取代的低级烷基组成的1位置取代，通过用相应的3-羟基丙酸酯处理而制备 一个THIONYL BISAZOLE。 某些1-取代的化合物可以通过使用锂盐的取代反应来制备。 化合物及其盐，其中3,3-二苯基-3- [咪唑基 - （1）] - 丙炔是典型的实施方案，是抗真菌剂，并且可以单独使用或以药物组合物的形式用于治疗真菌病 动物感染

公开(公告)号：US3869490A

公开(公告)日：1975-03-04

申请号：US26592672

申请日：1972-06-23

Applicant: BAYER AG

Inventor： JAGER GERHARD ,  METZGER CARL ,  EUE LUDWIG ,  SCHMIDT ROBERT

IPC: A01N47/20 ,  A01P13/02 ,  C07C67/00 ,  C07C239/00 ,  C07C271/28 ,  C07C313/00 ,  C07C317/28 ,  C07C323/43 ,  C07C325/00 ,  C07C333/02 ,  C07C333/08 ,  C07D295/12 ,  C07D307/88 ,  C07C155/02

CPC classification number: C07D295/12 ,  A01N47/20 ,  C07C333/02 ,  C07D307/88

Abstract: Compounds of the formula:

ARE OUTSTANDINGLY EFFECTIVE HERBICIDES PARTICULARLY WHEN USED AS SELECTIVE HERBICIDES AND ARE OUTSTANDINGLY TOLERATED BY CROP PLANTS.

IN WHICH R and R4 are, e.g., optionally substituted aliphatic hydrocarbyl; R1, R2, and R3 represent hydrogen, alkyl, cycloalkyl, alkoxy, haloalkyl and/or halogen; Furthermore R2 and R3 conjointly may represent a -(CH)4grouping to form a fused benzene ring with the adjacent atoms of the phenyl ring shown in the formula X is sulfur; Y is oxygen, sulfur or a group of the formula

D R A W I N G

Abstract translation: 下式的化合物：

公开(公告)号：US3920727A

公开(公告)日：1975-11-18

申请号：US26590972

申请日：1972-06-23

Applicant: BAYER AG

Inventor： METZGER CARL ,  JAGER GERHARD ,  LURSSEN KLAUS

IPC: A01N47/20 ,  C07C271/06 ,  C07D307/88 ,  C07C125/06

CPC classification number: C07D307/88 ,  A01N47/20 ,  C07C271/06

Abstract: New N-arylcarbamic acid esters of the formula

wherein R4 is hydrogen or is defined as R4 is defined above, and Y and Y'' are oxygen or sulfur, ARE OUTSTANDINGLY EFFECTIVE IN REGULATING THE GROWTH OF PLANTS, I.E., TO INHIBIT, STIMULATE OR ALTER THE GROWTH OF PLANTS.

IN WHICH R is lower aliphatic hydrocarbyl, optionally substituted, R1, R2 and R3, which may be identical or different, are each hydrogen, alkyl, cycloalkyl, alkoxy, haloalkyl or halogen, R4 is alkyl, alkenyl, alkynyl, cycloalkenyl, haloalkyl, haloalkenyl, haloalkynyl, alkoxyalkyl or alkylthioalkyl, acylalkyl (i.e., alkanoyloxyalkyl), alkoxycarbonylalkyl, carbalkoxyalkyl, carbalkoxyalkenyl, or an optionally substituted cycloalkyl, aryl, aralkyl, aryloxyalkyl or arylthioalkyl radical, or the grouping

公开(公告)号：US3920653A

公开(公告)日：1975-11-18

申请号：US33052473

申请日：1973-02-07

Applicant: BAYER AG

Inventor： WENZELBURGER JURGEN ,  JAGER GERHARD ,  EUE LUDWIG ,  SCHMIDT ROBERT R

IPC: A01N43/54 ,  A01N47/34 ,  A01P13/00 ,  C07D239/54 ,  C07D239/553 ,  C07D265/06 ,  C07D265/12 ,  C07D413/04 ,  C07D239/10

CPC classification number: C07D239/54 ,  C07D239/553 ,  C07D265/12

Abstract: 1-Aminouracil compounds of the formula IN WHICH R1 is an organic radical; R2 represents hydrogen, halogen, the thiocyanate radical, alkyl or optionally substituted aryl, and R3 represents alkyl or aralkyl optionally substituted in the aryl part, or R2 and R3 together represent a multi-membered methylene bridge which forms, with the two carbon atoms in the 5- and 6positions of the heterocyclic structure, a fused ring which is optionally substituted by alkyl; and agriculturally acceptable salts thereof; ARE OUTSTANDINGLY EFFECTIVE AS HERBICIDES, PARTICULARLY AS BROAD SPECTRUM TOTAL HERBICIDES.

Abstract translation: 式Ⅰ的1-氨尿嘧啶化合物，其中R1是有机基团; R 2表示氢，卤素，硫氰酸酯基，烷基或任选取代的芳基，R 3表示在芳基部分任选取代的烷基或芳烷基，或者R 2和R 3一起表示多元亚甲基桥，其与两个碳原子形成 杂环结构的5-和6-位，任选被烷基取代的稠合环; 和其农业上可接受的盐; 作为除草剂特别有效，特别是作为广谱光谱杀草剂。

公开(公告)号：US3895933A

公开(公告)日：1975-07-22

申请号：US37006773

申请日：1973-06-14

Applicant: BAYER AG

Inventor： JAGER GERHARD ,  LURSSEN KLAUS

IPC: C07D405/06 ,  A01N43/40 ,  C07D213/04 ,  C07D213/20 ,  C07D213/61 ,  A01N9/22

CPC classification number: C07D213/20 ,  C07D213/61

Abstract: wherein R is optionally substituted phenyl, furyl or thienyl, N IS 1, 2 OR 3 R1 is hydrogen, alkyl of up to 6 carbon atoms or halogen, wherein the substituents R1 are selected independently of one another when n is 2 or 3; and X is a halide or perchlorate ion; THE ACTIVE INGREDIENT IS AN ADMIXTURE WITH A SOLID OR LIQUEFIED GASEOUS DILUENT OR CARRIER OR IN ADMIXTURE WITH A LIQUID DILUENT OR CARRIER AND CONTAINS A SURFACE-ACTIVE AGENT.
Plant growth regulant compositions containing as an active ingredient a 2-hydroxyethyl-1-pyridinium-(1) salt of the formula

Abstract translation: 含有式 - + CH 2 -CH-R X - 的2-羟乙基-1-吡啶鎓 - （1）盐作为活性成分的植物生长调节剂组合物，其中R为任选取代的苯基，呋喃基或噻吩基 当N为2或3时，取代基R 1彼此独立地选择; R 1为氢，最多6个碳原子的烷基或卤素。 X - 是卤化物或高氯酸根离子; 活性成分是具有固体或液体气相稀释剂或载体的混合物，或与液体稀释剂或载体混合并含有表面活性剂。