公开(公告)号：US5597939B1

公开(公告)日：2000-01-04

申请号：US63056996

申请日：1996-04-10

Applicant: BAYER AG

Inventor： MUELLER KLAUS-HELMUT ,  KOENIG KLAUS ,  KLUTH JOACHIM ,  LUERSSEN KLAUS ,  SANTEL HANS-JOACHIM ,  SCHMIDT ROBERT R

IPC: A01N47/38 ,  C07D249/12 ,  C07D403/12 ,  C07D405/12 ,  C07D409/12 ,  C07C275/70

CPC classification number: C07D403/12 ,  A01N47/38 ,  C07D249/12 ,  C07D405/12 ,  C07D409/12

公开(公告)号：US5262383A

公开(公告)日：1993-11-16

申请号：US90993992

申请日：1992-07-07

Applicant: BAYER AG

Inventor： FISCHER REINER ,  BRETSCHNEIDER THOMAS ,  KRUEGER BERND-WIELAND ,  BACHMANN JUERGEN ,  ERDELEN CHRISTOPH ,  WACHENDORFF-NEUMANN ULRIKE ,  SANTEL HANS-JOACHIM ,  LUERSSEN KLAUS ,  SCHMIDT ROBERT R

IPC: A01N43/08 ,  A01N20060101 ,  A01N43/06 ,  A01N43/10 ,  A01N47/06 ,  A01N47/18 ,  A01N57/08 ,  C07D20060101 ,  C07D307/60 ,  C07D307/94 ,  C07D333/32 ,  C07D333/50 ,  C07D401/12 ,  C07D405/12 ,  C07D407/12 ,  C07D409/12 ,  C07D497/10 ,  C07F20060101 ,  C07F9/655 ,  C07F9/6553 ,  C07D307/32

CPC classification number: C07D405/12 ,  A01N43/06 ,  A01N47/06 ,  A01N57/08 ,  C07D307/60 ,  C07D307/94 ,  C07D409/12 ,  C07F9/65515 ,  C07F9/65517

Abstract: The present invention relates to new 3-aryl-4-hydroxy- DELTA 3-dihydrofuranone and 3-aryl-4-hydroxy- DELTA 3-dihydrothiophenone derivatives, to a plurality of processes for their preparation, and to their use as insecticides, acaricides, herbicides and fungicides. The new 3-aryl-4-hydroxy- DELTA 3-dihydrofuranone and 3-aryl-4-hydroxy- DELTA 3-dihydrothiophenone derivatives have the general formula I (I) in which X represents alkyl, halogen, alkoxy or halogenoalkyl, G represents hydrogen (a) or the groups D represents oxygen or sulphur, E(+) represents a metal ion equivalent or an ammonium ion, L and M represent oxygen and/or sulphur, and the other variables have the meaning given in the text of the application, with the exception of the following compounds: 3-(2-methoxyphenyl)-4-hydroxy- DELTA 3-dihydrofuran-2-one, 3-(2-chlorophenyl)-4-hydroxy- DELTA 3-dihydrofuran-2-one, 3-(2-methoxyphenyl)-4-hydroxy- DELTA 3-dihydrofuran-2-one, 3-(2-fluorophenyl)-4-hydroxy- DELTA 3-dihydrofuran-2-one.

Abstract translation: 本发明涉及新的3-芳基-4-羟基-TATA3-二氢呋喃酮和3-芳基-4-羟基-TATA3-二氢噻吩酮衍生物，用于其制备的多个方法及其用作杀虫剂，杀螨剂 ，除草剂和杀真菌剂。 新的3-芳基-4-羟基-DTATA-二氢呋喃酮和3-芳基-4-羟基-DTATA-二氢噻吩酮衍生物具有通式I（I），其中X代表烷基，卤素，烷氧基或卤代烷基 ，G表示氢（a）或基团，其中D表示氧或硫，E（+）表示金属离子当量或铵离子，L和M表示氧和/或硫，其他变量 具有本申请文本中给出的含义，但以下化合物除外：3-（2-甲氧基苯基）-4-羟基-D-3,3-二氢呋喃-2-酮，3-（2-氯苯基）-4- （2-甲氧基苯基）-4-羟基-D-TA 3 - 二氢呋喃-2-酮，3-（2-氟苯基）-4-羟基-DDTA3-二氢呋喃-2-酮 -一。

公开(公告)号：US3920653A

公开(公告)日：1975-11-18

申请号：US33052473

申请日：1973-02-07

Applicant: BAYER AG

Inventor： WENZELBURGER JURGEN ,  JAGER GERHARD ,  EUE LUDWIG ,  SCHMIDT ROBERT R

IPC: A01N43/54 ,  A01N47/34 ,  A01P13/00 ,  C07D239/54 ,  C07D239/553 ,  C07D265/06 ,  C07D265/12 ,  C07D413/04 ,  C07D239/10

CPC classification number: C07D239/54 ,  C07D239/553 ,  C07D265/12

Abstract: 1-Aminouracil compounds of the formula IN WHICH R1 is an organic radical; R2 represents hydrogen, halogen, the thiocyanate radical, alkyl or optionally substituted aryl, and R3 represents alkyl or aralkyl optionally substituted in the aryl part, or R2 and R3 together represent a multi-membered methylene bridge which forms, with the two carbon atoms in the 5- and 6positions of the heterocyclic structure, a fused ring which is optionally substituted by alkyl; and agriculturally acceptable salts thereof; ARE OUTSTANDINGLY EFFECTIVE AS HERBICIDES, PARTICULARLY AS BROAD SPECTRUM TOTAL HERBICIDES.

Abstract translation: 式Ⅰ的1-氨尿嘧啶化合物，其中R1是有机基团; R 2表示氢，卤素，硫氰酸酯基，烷基或任选取代的芳基，R 3表示在芳基部分任选取代的烷基或芳烷基，或者R 2和R 3一起表示多元亚甲基桥，其与两个碳原子形成 杂环结构的5-和6-位，任选被烷基取代的稠合环; 和其农业上可接受的盐; 作为除草剂特别有效，特别是作为广谱光谱杀草剂。

公开(公告)号：US3925386A

公开(公告)日：1975-12-09

申请号：US26687272

申请日：1972-06-28

Applicant: BAYER AG

Inventor： JAGER GERHARD ,  WENZELBURGER HANS JURGEN ,  SCHMIDT ROBERT R

IPC: C07D239/22 ,  C07D265/12 ,  C07D319/08 ,  C07D239/04

CPC classification number: C07D239/22 ,  C07D265/12 ,  C07D319/08

Abstract: Novel 6-hydroxy-dihydro-uracil compounds of the formula:

WHEREIN R1 is hydrocarbyl and substituted hydrocarbyl, both aliphatic and aromatic, R2 is hydrogen, alkyl, or optionally, substituted aryl, R3 is alkyl or aralkyl, and R2 and R3 together may be an alkylene bridge; ARE PREPARED BY REACTING A 2,3-DIHYDRO-1,3-OXAZINE-2,4-DIONE OF THE GENERAL FORMULA

IN WHICH R1, R2 and R3 have the above mentioned meanings, is reacted with ammonia at a temperature of -50*C to +50*C, optionally in the presence of a diluent, but in the substantial absence of water. These compounds are herbicidally active.

Abstract translation: 新型6-羟基 - 二氢尿嘧啶化合物，其具有下式：

公开(公告)号：US3894074A

公开(公告)日：1975-07-08

申请号：US33540073

申请日：1973-02-23

Applicant: BAYER AG

Inventor： WAGNER KLAUS ,  EUE LUDWIG ,  SCHMIDT ROBERT R ,  ROOS ERNST

IPC: A01N47/06 ,  A01N33/22 ,  A01N37/02 ,  A01N37/44 ,  A01N41/04 ,  A01N41/08 ,  A01N47/22 ,  C07C67/00 ,  C07C201/00 ,  C07C205/26 ,  C07C205/37 ,  C07C205/43 ,  C07C205/48 ,  C07C239/00 ,  C07C271/08 ,  C07C301/00 ,  C07C303/28 ,  C07C309/63 ,  C07C309/66 ,  C07C125/06

CPC classification number: C07C205/26 ,  C07C205/37 ,  C07C205/43 ,  C07C205/48 ,  C07C309/66

Abstract: Novel 2,4-bis-(trifluoromethyl)-6-nitrophenol compounds of the formula

IN WHICH X is hydrogen; M; HNR 1R2R3; -COR4; -COOR5; N,Ndimethylaminocarbonyl; -SO2R6 or -CO-NH-R7; M is an equivalent of an alkali metal or alkaline earth metal, R1, R2 and R3 (individually) are hydrogen, alkyl, alkoxyalkyl, alkenyl, hydroxyalkyl, cycloalkyl, phenyalkyl, phenyl or substituted phenyl, R4 and R5 individually are alkyl, substituted alkyl, alkenyl, phenyl or substituted phenyl, R6 is alkyl, substituted alkyl, phenyl, substituted phenyl or dimethylamino, and R is alkyl, alkenyl, cycloalkyl, phenyl or substituted phenyl; ARE OUTSTANDINGLY EFFECTIVE SELECTIVE HERBICIDES.

Abstract translation: 新型的2,4-二（三氟甲基）-6-硝基苯酚化合物，其中X是氢; M; HNR + 1R2R3; -COR4; -COOR5; N，N-二甲基氨基羰基; -SO 2 R 6或-CO-NH-R 7; M是碱金属或碱土金属的当量，R 1，R 2和R 3（各自）是氢，烷基，烷氧基烷基，烯基，羟基烷基，环烷基，苯烷基，苯基或取代的苯基，R4和R5分别是烷基， ，烯基，苯基或取代的苯基，R 6是烷基，取代的烷基，苯基，取代的苯基或二甲基氨基，R是烷基，烯基，环烷基，苯基或取代的苯基; 是非常有效的选择性除草剂。