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1.PROCESS FOR PREPARING DIASTEREOMERICALLY ENRICHED PHOSPHORAMIDATE DERIVATIVES OF NUCLEOSIDE COMPOUNDS FOR TREATMENT OF VIRAL INFECTIONS 审中-公开
Title translation: 制备用于治疗病毒感染的核苷类化合物的二异氰酸酯衍生物的方法公开(公告)号:US20150183818A1
公开(公告)日:2015-07-02
申请号:US14409523
申请日:2013-07-02
Applicant: BRISTOL-MYERS SQUIBB COMPANY
Inventor: Kristy Tran , Martin D. Eastgate , Jacob Janey , Ke Chen , Victor W. Rosso
CPC classification number: C07H19/20 , C07D471/08 , C07F9/2458 , C07F9/26 , C07F9/65586 , C07F9/65616 , C07H19/10 , C07H19/16
Abstract: The present invention is directed to a process for preparing diastereomerically enriched nucleoside phosphoramidates having the formula I:
Abstract translation: 本发明涉及一种制备具有式I的非对映体富集的核苷氨基磷酸酯的方法: