专利检索 ap:("GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO. 2) LIMITED") AND inv:"Simon Christopher Cranko Lucas" 第 1 页

1.

发明授权
2,3-dihydrobenzohurans as bromodomain inhibitors 有权

公开(公告)号：US11319307B2

公开(公告)日：2022-05-03

申请号：US16753543

申请日：2018-10-04

申请人： GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO.2) LIMITED

发明人： Stephen John Atkinson , Emmanuel Hubert Demont , Lee Andrew Harrison , Simon Christopher Cranko Lucas , Alexander G. Preston , Jonathan Thomas Seal , Ian David Wall , Robert J. Watson , James Michael Woolven

IPC分类号： C07D413/12 , C07D307/80 , C07D405/12 , C07D407/12 , A61K45/06

摘要： The present invention relates to compounds of formula (I) and salts thereof, pharmaceutical compositions containing such compounds and to their use in therapy.

2.

发明授权
Benzofuran derivatives and their use as bromodomain inhibitors 有权

公开(公告)号：US11273146B2

公开(公告)日：2022-03-15

申请号：US16753544

申请日：2018-10-04

申请人： GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO. 2) LIMITED

发明人： Stephen John Atkinson , Emmanuel Hubert Demont , Lee Andrew Harrison , Simon Christopher Cranko Lucas , Alexander G. Preston , Jonathan Thomas Seal , Ian David Wall , Robert J. Watson , James Michael Woolven

IPC分类号： A61K31/4025 , A61K31/343 , A61K31/351 , A61K31/397 , A61K31/4155 , A61K31/4192 , A61K31/4196 , A61K31/443 , A61K31/4525 , A61K31/501 , A61K31/506 , A61K45/06 , C07D307/79 , C07D405/10 , C07D405/12 , C07D405/14 , C07D407/12 , C07D407/14 , C07D413/12 , C07D471/04

摘要： The present invention relates to compounds of formula (I) and salts thereof, pharmaceutical compositions containing such compounds and to their use in therapy.

3.

发明授权
Pyrazole derivatives as bromodomain inhibitors 有权

公开(公告)号：US10966961B2

公开(公告)日：2021-04-06

申请号：US16489859

申请日：2018-02-27

申请人： GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO.2) LIMITED

发明人： Stephen John Atkinson , Emmanuel Hubert Demont , Lee Andrew Harrison , Gemma Michele Liwicki , Simon Christopher Cranko Lucas , Alexander G. Preston , Jonathan Thomas Seal , Ian David Wall , Robert J. Watson

IPC分类号： A61K31/4155 , C07D405/12 , A61K31/415 , C07D231/14 , C07D403/12 , C07D471/04 , A61K31/437 , A61K31/4439 , C07D401/12 , A61K31/422 , C07D413/12 , A61K31/5377 , C07D405/14 , C07D417/12 , A61K31/4192 , A61K31/4184 , A61K31/4245 , A61K31/433

摘要： The present invention is directed to pyrazole derivatives, pharmaceutical compositions comprising the compounds and the use of the compounds or the compositions in the treatment of various diseases.