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公开(公告)号:US20140107340A1
公开(公告)日:2014-04-17
申请号:US14050431
申请日:2013-10-10
Applicant: H. Lundbeck A/S
Inventor: John Paul Kilburn , Lars Kyhn Rasmussen , Mikkel Jessing , Eman Mohammed Eldemenky , Bin Chen , Yu Jiang , Allen T. Hopper
IPC: C07C233/78 , C07D213/40 , C07D211/26 , C07D405/04 , C07D239/26 , C07D405/06 , C07D237/08 , C07D233/64 , C07D241/12 , C07D403/06 , C07C233/75 , C07C233/66 , C07D309/04 , C07D401/06
CPC classification number: A61K31/505 , C07C233/66 , C07C233/73 , C07C233/75 , C07C233/78 , C07C2601/08 , C07D211/26 , C07D213/40 , C07D213/61 , C07D231/12 , C07D233/64 , C07D237/08 , C07D239/26 , C07D241/12 , C07D309/04 , C07D401/06 , C07D403/04 , C07D403/06 , C07D405/04 , C07D405/06
Abstract: The present invention is directed to benzamide containing compounds which inhibit the P2X7 receptor
Abstract translation: 本发明涉及抑制P2X7受体的含苯甲酰胺的化合物
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公开(公告)号:US20170202836A1
公开(公告)日:2017-07-20
申请号:US15479972
申请日:2017-04-05
Applicant: H. Lundbeck A/S
Inventor: John Paul Kilburn , Lars Kyhn Rasmussen , Mikkel Jessing , Eman Mohamed Eldemenky , Bin Chen , Yu Jiang , Allen T. Hopper
IPC: A61K31/505
CPC classification number: A61K31/505 , C07C233/66 , C07C233/73 , C07C233/75 , C07C233/78 , C07C2601/08 , C07D211/26 , C07D213/40 , C07D213/61 , C07D231/12 , C07D233/64 , C07D237/08 , C07D239/26 , C07D241/12 , C07D309/04 , C07D401/06 , C07D403/04 , C07D403/06 , C07D405/04 , C07D405/06
Abstract: The present invention is directed to benzamide-containing compounds of formula I or pharmaceutically acceptable salts thereof which inhibit the P2X7 receptor, and their use in the treatment of epilepsy.
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公开(公告)号:US20150283134A1
公开(公告)日:2015-10-08
申请号:US14744103
申请日:2015-06-19
Applicant: H. Lundbeck A/S
Inventor: John Paul Kilburn , Lars Kyhn Rasmussen , Mikkel Jessing , Eman Mohamed Eldemenky , Bin Chen , Yu Jiang , Allen T. Hopper
IPC: A61K31/505
CPC classification number: A61K31/505 , C07C233/66 , C07C233/73 , C07C233/75 , C07C233/78 , C07C2601/08 , C07D211/26 , C07D213/40 , C07D213/61 , C07D231/12 , C07D233/64 , C07D237/08 , C07D239/26 , C07D241/12 , C07D309/04 , C07D401/06 , C07D403/04 , C07D403/06 , C07D405/04 , C07D405/06
Abstract: The present invention is directed to benzamide containing compounds which inhibit the P2X7 receptor
Abstract translation: 本发明涉及抑制P2X7受体的含苯甲酰胺的化合物
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公开(公告)号:US09649308B2
公开(公告)日:2017-05-16
申请号:US14744103
申请日:2015-06-19
Applicant: H. Lundbeck A/S
Inventor: John Paul Kilburn , Lars Kyhn Rasmussen , Mikkel Jessing , Eman Mohamed Eldemenky , Bin Chen , Yu Jiang , Allen T. Hopper
IPC: A61K31/505 , C07C233/66 , C07C233/73 , C07C233/75 , C07C233/78 , C07D211/26 , C07D213/40 , C07D213/61 , C07D231/12 , C07D233/64 , C07D237/08 , C07D239/26 , C07D241/12 , C07D309/04 , C07D401/06 , C07D403/06 , C07D405/04 , C07D405/06 , C07D403/04
CPC classification number: A61K31/505 , C07C233/66 , C07C233/73 , C07C233/75 , C07C233/78 , C07C2601/08 , C07D211/26 , C07D213/40 , C07D213/61 , C07D231/12 , C07D233/64 , C07D237/08 , C07D239/26 , C07D241/12 , C07D309/04 , C07D401/06 , C07D403/04 , C07D403/06 , C07D405/04 , C07D405/06
Abstract: The present invention is directed to benzamide-containing compounds of formula I or pharmaceutically acceptable salts thereof which inhibit the P2X7 receptor, and their use in the treatment of pain.
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公开(公告)号:US09102591B2
公开(公告)日:2015-08-11
申请号:US14050431
申请日:2013-10-10
Applicant: H. Lundbeck A/S
Inventor: John Paul Kilburn , Lars Kyhn Rasmussen , Mikkel Jessing , Eman Mohammed Eldemenky , Bin Chen , Yu Jiang , Allen T. Hopper
IPC: C07D239/26 , C07D237/08 , C07D241/12 , C07D211/26 , C07D213/40 , C07D309/04 , C07D401/06 , C07C233/78 , C07C233/66 , C07C233/75 , C07D233/64 , C07D403/06 , C07D405/04 , C07D405/06 , C07D231/12 , C07D403/04 , C07C233/73 , C07D213/61
CPC classification number: A61K31/505 , C07C233/66 , C07C233/73 , C07C233/75 , C07C233/78 , C07C2601/08 , C07D211/26 , C07D213/40 , C07D213/61 , C07D231/12 , C07D233/64 , C07D237/08 , C07D239/26 , C07D241/12 , C07D309/04 , C07D401/06 , C07D403/04 , C07D403/06 , C07D405/04 , C07D405/06
Abstract: The present invention is directed to benzamide containing compounds which inhibit the P2X7 Receptor.
Abstract translation: 本发明涉及抑制P2X7受体的含苯甲酰胺的化合物。
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