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公开(公告)号:US3553332A
公开(公告)日:1971-01-05
申请号:US3553332D
申请日:1967-06-27
Applicant: HOFFMANN LA ROCHE
Inventor: GRUNBERG EMANUEL
IPC: A61K31/135 , A61K27/00
CPC classification number: A61K31/135
Abstract: BENZOPHENONE DERIVATIVES HAVING A DI-SUBSTITUTED AMINO-ALKOXY SUBSTITUTENT ON ONE PHENYL RING AND HALO OR NITRO SUBSTITUTENT ON THE OTHER WERE FOUND TOBE USEFUL AGAINST MYCOBACTERIAL INFECTIONS, PARTICULARLY MYCOBACTERIUM TUBERCULOSIS.
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2.2,4-Diamino-5-(3-alkoxy-4,5-methylenedioxybenzyl)pyrimidine 失效
Title translation: 2,4-二氨基-5-(3-烷氧基-4,5-亚甲二氧基苄基)嘧啶公开(公告)号:US3867527A
公开(公告)日:1975-02-18
申请号:US40495373
申请日:1973-10-10
Applicant: HOFFMANN LA ROCHE
Inventor: GRUNBERG EMANUEL , HOFFER MAX
IPC: C07D405/06 , A61K31/505 , A61P31/04 , C07D239/49 , C07D317/60 , C07D317/64 , A61K27/00
CPC classification number: C07D317/60 , C07D317/64
Abstract: 2,4-Diamino-5-(3-alkoxy-4,5-methylenedioxybenzyl)pyrimidines, such as, for example, 2,4-diamino-5-(3-methoxy-4,5methylenedioxybenzyl)pyrimidine, prepared from the corresponding benzaldehydes, are described. The end products are useful as potentiators of the antibacterial activity of sulfonamides, as well as antibiotics.
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3.Antibacterial composition containing 5-methyl - 3 - sulfanilamidoisoxazole and trimethoxybenzyl pyrimidine 失效
Title translation: 含有5-甲基-3-磺酰氨基恶唑酮和三甲氧基苄基嘧啶的抗菌组合物公开(公告)号:US3515783A
公开(公告)日:1970-06-02
申请号:US3515783D
申请日:1967-10-20
Applicant: HOFFMANN LA ROCHE
Inventor: GRUNBERG EMANUEL
IPC: A61K31/635 , A01N9/16
CPC classification number: A61K31/635 , A61K31/505 , A61K2300/00
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公开(公告)号:US3657436A
公开(公告)日:1972-04-18
申请号:US3657436D
申请日:1970-02-09
Applicant: HOFFMANN LA ROCHE
Inventor: BERGER LEO , GRUNBERG EMANUEL , STERNBACH LEO HENRYK , STEMPEL ARTHUR
IPC: A61K31/19 , A61K31/535 , A61K27/00
CPC classification number: A61K31/19 , A61K31/535
Abstract: ANTHRANILIC ACID DERIVATIVES WHICH ARE USEFUL IN COMBATTING VIRAL INFECTIONS CAUSED BY COL-SK AND COMPOSITIONS CONTAINING THESE DERIVATIVES.
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5.Anthelmintic method using 6-methoxy-1-phenazinol 5,10-dioxide 失效
Title translation: 使用6-甲氧基-1-苯乙烯醇5,10-二氧化物的方法公开(公告)号:US3502774A
公开(公告)日:1970-03-24
申请号:US3502774D
申请日:1967-05-26
Applicant: HOFFMANN LA ROCHE
Inventor: GRUNBERG EMANUEL
CPC classification number: A61K31/70
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6.Method for controlling ectoparasite trichomonal infestation with 6-methoxy-1-phenazinol-5,10-dioxide 失效
Title translation: 用6-甲氧基-1-苯乙烯醇5,10-二氧化物控制蓖麻毒素诱导的方法公开(公告)号:US3502773A
公开(公告)日:1970-03-24
申请号:US3502773D
申请日:1967-05-26
Applicant: HOFFMANN LA ROCHE
Inventor: GRUNBERG EMANUEL
IPC: A61K27/00
CPC classification number: A61K31/70
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