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10 条记录 (耗时 0.02 秒)

    Nitrothiophenes, fungicidal and/or bactericidal compositions containing nitrothiophenes, and use thereof
    1.
    发明授权
    Nitrothiophenes, fungicidal and/or bactericidal compositions containing nitrothiophenes, and use thereof 失效

    公开(公告)号：US4451660A

    公开(公告)日：1984-05-29

    申请号：US361758

    申请日：1982-03-25

    申请人： Hendrik Dolman ,  Johannes Kuipers

    发明人： Hendrik Dolman ,  Johannes Kuipers

    IPC分类号： C07D333/14 ,  A01N43/10 ,  A01N43/40 ,  A01P1/00 ,  A01P3/00 ,  C07D213/71 ,  C07D333/36 ,  C07D333/42 ,  C07D409/12 ,  C07D333/00 ,  A01N43/02

    CPC分类号： C07D333/42 ,  A01N43/10 ,  A01N43/40 ,  C07D213/71

    摘要： The invention relates to new nitrothiophenes of the general formula ##STR1## wherein R is an alkyl group having 1 to 12 carbon atoms, which alkyl group may be substituted with a phenyl group substituted, if desired, with nitro, halogen, alkyl with 1 to 4 carbon atoms or alkoxy with 1 to 4 carbon atoms, with an alkoxycarbonyl group having 2 to 5 carbon atoms, or with a thiocyanato group, orR is a phenyl group, a pyridyl group or an N-oxypyridyl group, which groups may be substituted with nitro, halogen, alkyl with 1 to 4 carbon atoms, or alkoxy with 1 to 4 carbon atoms;R.sub.1 is a hydrogen atom, a halogen atom, an alkyl group having 1 to 4 carbon atoms, or a phenyl group substituted or not substituted with nitro, halogen, alkyl with 1 to 4 carbon atoms, or alkoxy with 1 to 4 carbon atoms;R.sub.2 is a hydrogen atom, an alkyl group having 1 to 4 carbon atoms, a cyano group, an alkanoyl group having 1 to 5 carbon atoms, an .alpha.,.alpha.-dialkoxyalkyl- or .alpha.,.alpha.-alkylene-dioxyalkyl group having 3 to 10 carbon atoms, a carboxy group, an alkoxycarbonyl group having 2 to 5 carbon atoms, an .alpha.-hydroxyalkyl group having 1 to 4 carbon atoms, an .alpha.-haloalkyl group having 1 to 4 carbon atoms, an .alpha.-alkoxyalkyl group having 2 to 6 carbon atoms, an alkoxycarboximidoyl group having 2 to 5 carbon atoms, a sulpho group, an amino-, alkylamino- or dialkylamino- sulphonyl group, the alkyl group(s) of which has (have) 1 to 4 carbon atoms, or an alkoxysulphonyl group having 1 to 4 carbon atoms, andn is 0 to 2.The compositions are particularly suitable to prevent infections by phytophagous microorganisms in agriculture and horticulture. For this purpose, the seed is treated prior to sowing or the soil destined for sowing or planting is treated with the composition in a dosage from 100 to 1,500 mg of active substance per kg of seed and from 2 to 100 kg of active substance per hectare, respectively.

    New thiazole compounds having fungicidal activity
    2.
    发明授权
    New thiazole compounds having fungicidal activity 失效
    具有杀真菌活性的新噻唑化合物

    公开(公告)号：US4889863A

    公开(公告)日：1989-12-26

    申请号：US222907

    申请日：1988-07-22

    申请人： Hendrik Dolman ,  Johannes Kuipers

    发明人： Hendrik Dolman ,  Johannes Kuipers

    IPC分类号： C07D277/20 ,  A01N43/78 ,  C07D277/36 ,  C07D277/54 ,  C07D277/56 ,  C07D417/04 ,  C07D417/12

    CPC分类号： C07D417/04 ,  C07D277/36 ,  C07D277/54 ,  C07D277/56 ,  C07D417/12

    摘要： The invention relates to new thiazole compounds of the general formula ##STR1## wherein R is an C.sub.1 -C.sub.12 alkyl group or a phenyl group, which groups are unsubstituted or substituted with halogen, nitro or cyano;R.sub.1 is a cyano group; a formyl group; an alkylcarbonyl or alkoxycarbonyl group having 2-5 carbon atoms; or a substituted or non-substituted benzoyl group;R.sub.2 is a hydrogen atom; a halogen atom; an amino group; an amino group substituted with 1 or 2 substituents selected from the group consisting of C.sub.1 -C.sub.4 alkyl, C.sub.2 -C.sub.5 alkynyl, C.sub.2 -C.sub.5 alkylcarbonyl and C.sub.2 -C.sub.5 alkoxycarbonyl; an alkyl, alkoxy, alkylthio, alkylsulphinyl or alkyl-sulphonyl group having 1-4 carbon atoms; or a substituted or non-substituted aryl, aryloxy, arylthio, arylsulphinyl or arylsulphonyl group; andn is 1 or 2.The new compounds show a fungicidal activity and may be used in particular against plant pathogenic seed fungi and soil fungi.

    Fungicidal and/or bactericidal compositions containing nitrothiophenes, and use thereof
    3.
    发明授权
    Fungicidal and/or bactericidal compositions containing nitrothiophenes, and use thereof 失效
    含有硝基噻吩的杀真菌剂和/或杀菌组合物及其用途

    公开(公告)号：US4649154A

    公开(公告)日：1987-03-10

    申请号：US543895

    申请日：1983-10-20

    申请人： Hendrik Dolman ,  Johannes Kuipers

    发明人： Hendrik Dolman ,  Johannes Kuipers

    IPC分类号： C07D333/14 ,  A01N43/10 ,  A01N43/40 ,  A01P1/00 ,  A01P3/00 ,  C07D213/71 ,  C07D333/36 ,  C07D333/42 ,  C07D409/12 ,  A01N43/02

    CPC分类号： C07D333/42 ,  A01N43/10 ,  A01N43/40 ,  C07D213/71

    摘要： The invention relates to new nitrothiophenes of the general formula ##STR1## wherein R is an alkyl group having 1 to 12 carbon atoms, which alkyl group may be substituted with a phenyl group substituted, if desired, with nitro, halogen, alkyl with 1 to 4 carbon atoms or alkoxy with 1 to 4 carbon atoms, with an alkoxycarbonyl group having 2 to 5 carbon atoms, or with a thiocyanato group,or R is a phenyl group, a pyridyl group or an N-oxypyridyl group, which groups may be substituted with nitro, halogen, alkyl with 1 to 4 carbon atoms, or alkoxy with 1 to 4 carbon atoms;R.sub.1 is a hydrogen atom, a halogen atom, an alkyl group having 1 to 4 carbon atoms, or a phenyl group substituted or not substituted with nitro, halogen, alkyl with 1 to 4 carbon atoms, or alkoxy with 1 to 4 carbon atoms;R.sub.2 is a hydrogen atom, an alkyl group having 1 to 4 carbon atoms, a cyano group, an alkanoyl group having 1 to 5 carbon atoms, an .alpha.,.alpha.-dialkoxyalkyl- or .alpha.,.alpha.-alkylenedioxyalkyl group having 3 to 10 carbon atoms, a carboxy group, an alkoxycarbonyl group having 2 to 5 carbon atoms, an .alpha.-hydroxyalkyl group having 1 to 4 carbon atoms, an .alpha.-haloalkyl group having 1 to 4 carbon atoms, an .alpha.-alkoxyalkyl group having 2 to 6 carbon atoms, an alkoxycarboximidoyl group having 2 to 5 carbon atoms, a sulpho group, an amino-, alkylamino- or dialkylaminosulphonyl group, the alkyl group(s) of which has (have) 1 to 4 carbon atoms, or an alkoxysulphonyl group having 1 to 4 carbon atoms, andn is 0 to 2.The compositions are particularly suitable to prevent infections by phytophagous microorganisms in agriculture and horticulture. For this purpose, the seed is treated prior to sowing or the soil destined for sowing or planting is treated with the composition in a dosage from 100 to 1,500 mg of active substance per kg of seed and from 2 to 100 kg of active substance per hectare, respectively.

    Composition for the treatment of soil or seed against phytophagous fungi
    4.
    发明授权
    Composition for the treatment of soil or seed against phytophagous fungi 失效
    用于处理土壤或种子的组合物用于植物性真菌

    公开(公告)号：US4221801A

    公开(公告)日：1980-09-09

    申请号：US965215

    申请日：1978-11-30

    申请人： Johannes Kuipers ,  Hendrik Dolman

    发明人： Johannes Kuipers ,  Hendrik Dolman

    IPC分类号： A01N33/22 ,  A01N43/78 ,  A01P3/00 ,  A01N9/12 ,  A01N9/20

    CPC分类号： A01N43/78

    摘要： The invention relates to a composition against phytophagous micro-organisms, comprising 2-cyano-5-nitro-thiazole. Infections by phytophagous micro-organisms in agriculture and horitculture can be prevented by treating the seed prior to sowing or the soil destined for sowing or planting with the composition in a dosage of from 100 to 600 mg of active substance per kg of seed and from 2 to 100 kg of active substance per hextare, respectively.

    摘要翻译： 本发明涉及包含2-氰基-5-硝基 - 噻唑的抗食性微生物的组合物。 可以通过在播种之前处理种子或用组合物播种或种植的土壤，每千克种子的活性物质为100-600毫克，以及2 至100公斤活性物质。

    Thio compounds having fungicidal activity
    7.
    发明授权
    Thio compounds having fungicidal activity 失效
    硫代化合物具有杀菌活性

    公开(公告)号：US4994485A

    公开(公告)日：1991-02-19

    申请号：US566868

    申请日：1990-08-14

    申请人： Hendrik Dolman ,  Johannes Kuipers

    发明人： Hendrik Dolman ,  Johannes Kuipers

    IPC分类号： A01N37/34 ,  A01N41/10 ,  A01N43/10 ,  C07D333/34 ,  C07D333/38 ,  C07D409/04

    CPC分类号： C07D409/04 ,  A01N37/34 ,  A01N43/10 ,  C07C323/00 ,  C07D333/34 ,  C07D333/38

    摘要： The invention relates to new thio compounds of the general formula ##STR1## wherein R is an alkyl group substituted or not substituted with halogen and having 1-12 carbon atoms, an alkenyl or alkynyl group having 2-4 carbon atoms, an alkadienyl group having 3 or 4 carbon atoms or a substituted or unsubstituted phenyl or phenyl(C.sub.1 -C.sub.4)alkyl group;R.sub.1 is a cyano group, a formyl group, an alkylcarbonyl or alkoxycarbonyl group substituted or unsubstituted with halogen and having 2-5 carbon atoms, a substituted or unsubstituted benzoyl group, or an alkylsulphonyl group having 1-4 carbon atoms;R.sub.2 is a hydrogen atom, a halogen atom, an amino group unsubstituted or substituted with one or two groups selected from C.sub.1 -C.sub.4 alkyl and C.sub.2 -C.sub.5 alkylcarbonyl, an amino group forming part of a heterocyclic ring which may comprise 1 or 2 additional heteroatoms selected from N, O and S, an alkyl or alkoxy group having 1-4 carbon atoms and optionally substituted with C.sub.2 -C.sub.5 alkylcarbonyl, or a substituted or unsubstituted phenyl, phenoxy or phenylthio group;or whereinR.sub.1 and R.sub.2, together with the vinylene group to which they are bound, constitute a substituted or unsubstituted phenyl group;X is a cyano group or a formyl group;n is 1 or 2;Y is an alkylthio group having 1-4 carbon atoms; andZ is a hydrogen atom, a halogen atom, a nitro group, or an alkyl or alkoxy group having 1-4 carbon atoms and optionally substituted with halogen;or wherein Y and Z together constitute a sulphur atom; with the proviso that, when Y and Z do not together constitute a sulphur atom, R.sub.1 and R.sub.2, together with the vinylene group to which they are bound, constitute a substituted or unsubstituted phenyl group.The new compounds show a fungicidal and/or bactericidal activity and may be used in particular against plantpathogenic seed fungi and soil fungi and/or bacteria.

    摘要翻译： 本发明涉及通式为“IMAGE”的新的硫代化合物，其中R是被卤素取代或未被卤素取代或具有1-12个碳原子的烷基，具有2-4个碳原子的链烯基或炔基， 3或4个碳原子或取代或未取代的苯基或苯基（C 1 -C 4）烷基; 取代或未取代的苯甲酰基或具有1-4个碳原子的烷基磺酰基; R 1为氰基，甲酰基，被卤素取代或未取代的，具有2-5个碳原子的烷基羰基或烷氧基羰基。 R2是氢原子，卤素原子，未取代或被选自C1-C4烷基和C2-C5烷基羰基的一个或两个基团取代的氨基，形成杂环的一部分的氨基，其可以包含1或2个另外的杂原子 选自N，O和S，具有1-4个碳原子并且任选被C 2 -C 5烷基羰基取代的烷基或烷氧基，或取代或未取代的苯基，苯氧基或苯硫基; 或其中R 1和R 2与它们所结合的亚乙烯基一起构成取代或未取代的苯基; X是氰基或甲酰基; n为1或2; Y是具有1-4个碳原子的烷硫基; Z是氢原子，卤素原子，硝基或具有1-4个碳原子并任选被卤素取代的烷基或烷氧基; 或其中Y和Z一起构成硫原子; 条件是当Y和Z不在一起构成硫原子时，R 1和R 2与它们所结合的亚乙烯基一起构成取代或未取代的苯基。 新化合物显示出杀真菌和/或杀菌活性，特别可用于植物致病种子真菌和土壤真菌和/或细菌。

    2-Arylimino-imidazolidines, compositions containing same, and method of use thereof
    9.
    发明授权
    2-Arylimino-imidazolidines, compositions containing same, and method of use thereof 失效
    2-芳基亚胺基咪唑啉，含有它们的组合物及其使用方法

    公开(公告)号：US4374143A

    公开(公告)日：1983-02-15

    申请号：US264460

    申请日：1981-05-18

    申请人： Hendrik Dolman ,  Johannes Kuipers

    发明人： Hendrik Dolman ,  Johannes Kuipers

    IPC分类号： A01N43/50 ,  A01N43/54 ,  A01P3/00 ,  A61K31/415 ,  A61K31/505 ,  A61P31/04 ,  C07D233/50 ,  C07D239/14 ,  C07D333/00 ,  C07D405/12 ,  C07D409/12 ,  C07F3/00

    CPC分类号： C07D239/14 ,  A01N43/50 ,  A01N43/54 ,  C07D233/50 ,  C07F3/003

    摘要： The invention relates to novel 2-aryliminohexahydropyrimidines and imidazolidines, of the formula ##STR1## as well as to salts and complexes thereof, having fungicidal activity. These compounds are particularly active against rust of beans, brown rust of wheat and mildew on cereals. After having been processed into compositions, the compounds of the invention can successfully be used to prevent or control mould infections in agriculture and horticulture in a dosage of 200-1000 g of active substance per hectare.Very active fungicides are, for example, 2-(4-cyclohexyl-phenyl) iminohexahydropyrimidine and 2-(4-n-hexyl-phenyl) iminohexahydropyrimidine, as well as the sulphuric acid salts of these compounds and complexes with zinc salts.

    摘要翻译： 本发明涉及具有杀真菌活性的新颖的2-芳基亚氨基六氢嘧啶和咪唑烷，其具有式“IMAGE”以及其盐和络合物。 这些化合物特别有效防止豆类的生锈，小麦的褐锈病和谷物上的霉变。 在加工成组合物后，本发明的化合物可以成功地用于预防或控制农业和园艺中的霉菌感染，剂量为每公顷200-1000克活性物质。 非常活性的杀真菌剂是例如2-（4-环己基 - 苯基）亚氨基六氢嘧啶和2-（4-正己基 - 苯基）亚氨基六氢嘧啶，以及这些化合物的硫酸盐和与锌盐的络合物。