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公开(公告)号：US20060019981A1
公开(公告)日：2006-01-26
申请号：US10530465
申请日：2003-11-18
IPC分类号： C07D471/02 , A61K31/4745
CPC分类号： C07D471/04
摘要： In one aspect, the present invention is directed to a one pot method of preparing intermediates of Formula (V), which are useful in making inhibitors of phosphodiesterase-4: The present invention is also directed to a method of preparing phosphodiesterase inhibitors comprising the Formula (IX, IXa)
摘要翻译： 一方面，本发明涉及一种制备式（V）中间体的一锅法，其可用于制备磷酸二酯酶-4的抑制剂：本发明还涉及一种制备磷酸二酯酶抑制剂的方法，其包含式 （IX，IXa）
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公开(公告)号：US07312334B2
公开(公告)日：2007-12-25
申请号：US10530465
申请日：2003-11-18
IPC分类号： C07D471/02
CPC分类号： C07D471/04
摘要： In one aspect, the present invention is directed to a one pot method of preparing intermediates of Formula (V), which are useful in making inhibitors of phosphodiesterase-4: The present invention is also directed to a method of preparing phosphodiesterase inhibitors comprising the Formula (IX, IXa).
摘要翻译： 一方面，本发明涉及一种制备式（V）中间体的一锅法，其可用于制备磷酸二酯酶-4的抑制剂：本发明还涉及一种制备磷酸二酯酶抑制剂的方法，其包含式 （IX，IXa）。
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公开(公告)号：US06909002B2
公开(公告)日：2005-06-21
申请号：US10690118
申请日：2003-10-21
IPC分类号： A61K31/4745 , C07D471/02 , C07D471/04
CPC分类号： C07D471/04
摘要： In one aspect, the present invention is directed to a one pot method of preparing intermediates of Formula V, which are useful in making inhibitors of phosphodiesterase-4: The present invention is also directed to a method of preparing phosphodiesterase inhibitors comprising the Formula
摘要翻译： 一方面，本发明涉及制备式V中间体的一锅法，其可用于制备磷酸二酯酶-4的抑制剂：本发明还涉及制备磷酸二酯酶抑制剂的方法，其包含式
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公开(公告)号：US08680294B2
公开(公告)日：2014-03-25
申请号：US13387619
申请日：2010-07-27
申请人： John Traverse , William M. Leong , Steven P. Miller , Jennifer Albaneze-Walker , Thomas J. Hunter , Lijun Wang , Hongbiao Liao , Ashok Arasappan , Scott T. Trzaska , Randi M. Smith , Azzeddine Lekhal , Stephane L. Bogen , Jianshe Kong , Frank Bennett , F. George Njoroge , Marc Poirier , Shen-Chun Kuo , Yonggang Chen , Kenneth S. Matthews , Patrice Demonchaux , Amadeo Ferreira
发明人： John Traverse , William M. Leong , Steven P. Miller , Jennifer Albaneze-Walker , Thomas J. Hunter , Lijun Wang , Hongbiao Liao , Ashok Arasappan , Scott T. Trzaska , Randi M. Smith , Azzeddine Lekhal , Stephane L. Bogen , Jianshe Kong , Frank Bennett , F. George Njoroge , Marc Poirier , Shen-Chun Kuo , Yonggang Chen , Kenneth S. Matthews , Patrice Demonchaux , Amadeo Ferreira
IPC分类号： C07D207/06
CPC分类号： C07D209/52 , C07C51/353 , C07C67/04 , C07C237/04 , C07C315/02 , C07C315/04 , C07C317/28 , C07C319/14 , C07C319/20 , C07C2601/02 , C07C2601/14 , C07K5/0202 , C07K5/06034 , C07C323/53 , C07C317/44 , C07C57/03 , C07C69/533
摘要： Processes useful for the preparation of a Compound of Formula I: Formula (I). Intermediates useful for the preparation of the compound of Formula I, and processes useful for preparing said intermediates are disclosed.
摘要翻译： 用于制备式I化合物的方法：式（I）。 公开了可用于制备式I化合物的中间体和用于制备所述中间体的方法。
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5.发明申请ENANTIO- AND STEREO-SPECIFIC SYNTHESES OF BETA-AMINO-ALPHA- HYDROXY AMIDES 有权氨基 - 氨基 - 羟丙基氨基酸的纯化和立体特异性合成公开(公告)号：US20120178942A1
公开(公告)日：2012-07-12
申请号：US13387619
申请日：2010-07-27
申请人： John Traverse , William M. Leong , Steven P. Miller , Jennifer Albaneze-Walker , Thomas J. Hunter , Lijun Wang , Hongbiao Liao , Ashok Arasappan , Scott T. Trzaska , Randi M. Smith , Azzeddine Lekhal , Stephane L. Bogen , Jianshe Kong , Frank Bennett , F. George Njoroge , Marc Poirier , Shen-Chun Kuo , Yonggang Chen , Kenneth S. Matthews , Patrice Demonchaux , Amadeo Ferreira
发明人： John Traverse , William M. Leong , Steven P. Miller , Jennifer Albaneze-Walker , Thomas J. Hunter , Lijun Wang , Hongbiao Liao , Ashok Arasappan , Scott T. Trzaska , Randi M. Smith , Azzeddine Lekhal , Stephane L. Bogen , Jianshe Kong , Frank Bennett , F. George Njoroge , Marc Poirier , Shen-Chun Kuo , Yonggang Chen , Kenneth S. Matthews , Patrice Demonchaux , Amadeo Ferreira
IPC分类号： C07D209/52 , C07C237/14 , C07C317/44 , C07C315/02 , C07C271/56 , C07C231/02 , C07C263/00 , C07C265/10 , C07C313/12 , C07C211/35 , C07C275/26 , C07C273/18
CPC分类号： C07D209/52 , C07C51/353 , C07C67/04 , C07C237/04 , C07C315/02 , C07C315/04 , C07C317/28 , C07C319/14 , C07C319/20 , C07C2601/02 , C07C2601/14 , C07K5/0202 , C07K5/06034 , C07C323/53 , C07C317/44 , C07C57/03 , C07C69/533
摘要： Processes useful for the preparation of a Compound of Formula I: Formula (I). Intermediates useful for the preparation of the compound of Formula I, and processes useful for preparing said intermediates are disclosed.
摘要翻译： 用于制备式I化合物的方法：式（I）。 公开了可用于制备式I化合物的中间体和用于制备所述中间体的方法。
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