公开(公告)号：US20060199801A1

公开(公告)日：2006-09-07

申请号：US10551810

申请日：2004-04-16

申请人： Jordi i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Maria Scherer ,  Reinhard Stierl

发明人： Jordi i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Oliver Wagner ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Maria Scherer ,  Reinhard Stierl

IPC分类号： A61K31/551 ,  A61K31/541 ,  A61K31/53 ,  A61K31/519

CPC分类号： C07D487/04 ,  A01N43/90

摘要： Bicyclic compounds of the formula I in which A1 or A5 is C and the other of the two variables A1, A5 is N, C or C—R3; A2, A3, A4 independently of one another are N or C—R3a, where one of the variables A2, A3 or A4 may also be S or a group N—R4 if A1 and A5 are both C, and where A4 is not N or C—R3a if A1 is N, A3 is C—R3a and A5 is C, and where A1 is attached to A2 and A3 to A4 or A2 is attached to A3 and A4 to A5 or A1 is attached to A5 and A2 to A3 or A1 is attached to A5 and A3 to A4 or A1 is attached to A2 and A4 to A5 by double bonds; n is 0, 1, 2, 3, 4 or 5; Ra is halogen, cyano, C1-C6-alkyl, C1-C6-alkoxy, C1-C6-haloalkyl, C1-C6-haloalkoxy, C2-C6-alkenyl, C2-C6-alkenyloxy or C(O)R5; R1 is halogen, cyano, C1-C10-alkyl, where a carbon atom of the C1-C10-alkyl radical may be replaced by a silicium atom, C1-C6-haloalkyl, C2-C10-alkenyl, C2-C6-haloalkenyl, C2-C6-alkynyl, C3-C8-cycloalkyl, C3-C8-cycloalkyl-C1-C4-alkyl, where the cycloalkyl moiety of the two last-mentioned groups may be unsubstituted or contain 1, 2, 3, 4, 5, or 6 radicals selected from the group consisting of C1-C4-alkylidene, C1-C4-alkyl, halogen, C1-C4-haloalkyl and hydroxy and the alkyl moiety of C3-C8-cycloalkyl-C1-C4-alkyl may be unsubstituted or contain 1, 2, 3, or 4 radicals selected from the group consisting of halogen, C1-C4-haloalkyl and hydroxy, C5-C8-cycloalkenyl which may be unsubstituted or contain 1, 2, 3 or 4 radicals selected from the group consisting of C1-C4-alkyl, halogen, C1-C4-haloalkyl and hydroxy, OR6, SR6, NR7R8, a radical of the formula —C(R11)(R12)C(═NOR13)(R14) or a radical of the formula —C(═NOR15)C(═NOR16)(R17); R2 is halogen, cyano, C1-C6-alkyl, C1-C6-haloalkyl, C2-C6-alkenyl, C2-C6-haloalkenyl, C2-C6-alkynyl, C3-C8-cycloalkyl, C5-C8-cycloalkenyl, OR6, SR6 or NR7R8; and the agriculturally acceptable salts of the compounds I, crop protection compositions comprising at least one compound of the formula I and/or an agriculturally acceptable salt of I and at least one solid or liquid carrier and a method for controlling phytopathogenic harmful fungi are described.

公开(公告)号：US20060241128A1

公开(公告)日：2006-10-26

申请号：US10532719

申请日：2003-11-04

申请人： Jordi Tormo I Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Jordi Tormo I Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  C07D487/04

CPC分类号： C07C69/65 ,  A01N43/90 ,  C07D487/04

摘要： Substituted 6-(2-halogenphenyl)-triazolopyrimidines of formula I in which R1 denote alkyl, alkenyl, alkynyl, alkadienyl, haloalkyl, haloalkenyl, cycloalkyl, phenyl, naphthyl, or a 5- or 6-membered saturated, unsaturated, or aromatic heterocycle, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, wherein R1 and R2 radicals may be substituted as defined in the description, R2 denote hydrogen, or a group mentioned for R1; or R1 and R2 together with the interjacent nitrogen atom represent a 5- or 6-membered heterocycle, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which ring may be substituted as defined in the description; Hal is halogen; L1, L3 independently denote hydrogen, halogen, or alkyl; L2 is hydrogen, halogen, haloalkyl, or NH2, NHRb, or N(Rb)2, wherein Rb is as defined in the description, wherein at least one from L1, L2, and L3 is not hydrogen; X is halogen, cyano, alkyl, alkoxy, haloalkoxy or alkenyloxy. processes for their preparation, compositions containing them and to their use for combating phytopathogenic fungi.

摘要翻译： 其中R 1表示烷基，烯基，炔基，链二烯基，卤代烷基，卤代烯基，环烷基，苯基，萘基或5-或6-元的取代的6-（2-卤代苯基） - 三唑并嘧啶， 含有1至4个氮原子或1至3个氮原子和1个硫或氧原子的饱和，不饱和或芳族杂环，其中R 1和R 2可以是 如说明书中所定义，R 2表示氢或R 1所提及的基团; 或R 1和R 2连同中间的氮原子代表含有1-4个氮原子或一至三个氮原子的一个或多个六元杂环，一个 硫或氧原子，该环可以如说明书中所定义取代; 卤素是卤素; L 1，L 3独立地表示氢，卤素或烷基; L 2是氢，卤素，卤代烷基或NH 2，NHR b或/或N（R b） 其中R b如描述中所定义，其中至少一个L 1，L 2， ，而L 3不是氢; X是卤素，氰基，烷基，烷氧基，卤代烷氧基或烯氧基。 其制备方法，含有它们的组合物及其用于对抗植物病原真菌的用途。

公开(公告)号：US20060079537A1

公开(公告)日：2006-04-13

申请号：US10531898

申请日：2003-11-14

申请人： Jordi Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Jordi Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A61K31/519 ,  C07D487/04

CPC分类号： C07D487/04 ,  A01N43/90

摘要： 2-Substituted triazolopyrimidines of the formula I, in which the substituents are as defined below: L are halogen, cyano, nitro, alkyl, alkenyl, alkynyl, haloalkyl, haloalkenyl, alkoxy, alkenyloxy, alkynyloxy, haloalkoxy, —C(═O)-A or S(═O)pA′; A and A′ are as defined in the description; p is 0, 1 or 2; m is 0, 1, 2, 3, 4 or 5; X is cyano, alkyl, haloalkyl, alkoxy or haloalkoxy; R1,R2 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, alkadienyl, haloalkenyl, cycloalkenyl, alkynyl, haloalkynyl or cycloalkynyl, phenyl, naphthyl or a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S, R1 and R2 together with the nitrogen atom to which they are attached may also form a five- or six-membered ring which may be interrupted by an atom from the group consisting of O, N and S, where R1 and/or R2 may be substituted as defined in the description; and R3 is cyano, hydroxyl, alkoxy, alkenyloxy, haloalkoxy, haloalkenyloxy, NR1R2 or S(O)nR31, where n and R31 are as defined in the description; Processes and intermediates for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi are described.

摘要翻译： 氰基，硝基，烷基，烯基，炔基，卤代烷基，卤代烯基，烷氧基，烯氧基，炔氧基，卤代烷氧基，-C（ - O） - 取代的取代基如下： -A或S（-O） A'; A和A'如说明书所定义; p为0,1或2; m为0,1,2,3,4或5; X是氰基，烷基，卤代烷基，烷氧基或卤代烷氧基; R 1，R 2是氢，烷基，卤代烷基，环烷基，卤代环烷基，烯基，链二烯基，卤代烯基，环烯基，炔基，卤代炔基或环炔基，苯基，萘基或五 - 至十元饱和的，部分不饱和的或芳族杂环，其含有一至四个由O，N和S组成的组的杂原子，R 1和R 2连同 它们所连接的氮原子也可以形成可被来自O，N和S的原子间隔的五元或六元环，其中R 1和/或 R 2可以如说明书中定义的取代; 和R 3是氰基，羟基，烷氧基，烯氧基，卤代烷氧基，卤代烯氧基，NR 1 R 2或S（O）n 其中n和R 31如在说明书中所定义的; 描述了制备这些化合物的方法和中间体，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US20060167017A1

公开(公告)日：2006-07-27

申请号：US10539039

申请日：2003-12-16

申请人： Bernd Muller ,  Jordi Blasco ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Bernd Muller ,  Jordi Blasco ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Wassilios Grammenos ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： C07D487/04 ,  A01N43/90

CPC分类号： C07D487/04

摘要： Triazolopyrimidines of the formula I where the index and the substituents are as defined below: R1 is C1-C10-alkyl, C2-C10-alkenyl, C2-C10-alkynyl, C3-C10-cycloalkyl, C3-C10-cycloalkenyl, phenyl, naphthyl, or a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle which is attached via carbon to the triazolopyrimidine and contains one to four heteroatoms from the group consisting of N, O and S; R2 is C1-C4-alkyl which may be substituted by halogen, cyano, nitro or C1-C2-alkoxy; n is 0 or an integer from 1 to 4; R is as defined in the description; X is SOm—Rx, NRxRy or NRx—(C═O)—Ry; m is 0 or an integer from 1 to 3; and processes for preparing these compounds, compositions comprising them and their use for controlling harmful fungi are described.

摘要翻译： 其中指数和取代基如下定义的式I的三唑并嘧啶：R 1是C 1 -C 10 - 烷基， C 1 -C 10亚烷基，C 2 -C 10 - 炔基，C 3 - 亚烷基 C 1 -C 10 - 环烷基，C 3 -C 10 - 环烯基，苯基，萘基或五至十元饱和的， 部分不饱和或芳族杂环，其通过碳连接到三唑并嘧啶并且包含一至四个由N，O和S组成的组的杂原子; R 2是可以被卤素，氰基，硝基或C 1 H 3取代的C 1 -C 4 - 烷基 -C 2 - 烷氧基; n为0或1至4的整数; R如说明书所定义; X是SO x，x，x，x，y，x，y，x， - （CO）-R y; m为0或1〜3的整数; 并描述了制备这些化合物的方法，包含它们的组合物及其用于控制​​有害真菌的用途。

公开(公告)号：US20050272748A1

公开(公告)日：2005-12-08

申请号：US10531980

申请日：2003-11-14

申请人： Jordi Tormo Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Jordi Tormo Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  C07D487/04 ,  A61K31/519

CPC分类号： C07D487/04 ,  A01N43/90

摘要： 2-Mercapto-substituted triazolopyrimidines of the formula I in which the substituents are as defined below: L is halogen, cyano, nitro, alkyl, alkenyl, alkynyl, haloalkyl, haloalkenyl, alkoxy, alkenyloxy, alkynyloxy, haloalkoxy or —C(═O)-A; A is hydrogen, hydroxyl, alkyl, alkenyl, alkoxy, haloalkoxy, alkylamino or dialkylamino; m is 0, 1, 2, 3, 4 or 5; X is halogen, cyano, alkyl, haloalkyl, alkoxy or haloalkoxy; R1, R2 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, alkadienyl, haloalkenyl, cycloalkenyl, alkynyl, haloalkynyl or cycloalkynyl, phenyl, naphthyl or a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle which contains one to four hetero atoms from the group consisting of O, N and S; R1 and R2 together with the nitrogen atom to which they are attached may also form a five- or six-membered ring which may be interrupted by an atom from the group consisting of O, N and S; where R1 and/or R2 may be substituted as stated in the description; processes for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi are described.

摘要翻译： 2-巯基取代的式Ⅰ的三唑并嘧啶，其中取代基如下：L是卤素，氰基，硝基，烷基，烯基，炔基，卤代烷基，卤代烯基，烷氧基，烯氧基，炔氧基，卤代烷氧基或-C ）-一个; A是氢，羟基，烷基，烯基，烷氧基，卤代烷氧基，烷基氨基或二烷基氨基; m为0,1,2,3,4或5; X是卤素，氰基，烷基，卤代烷基，烷氧基或卤代烷氧基; R 1，R 2是氢，烷基，卤代烷基，环烷基，卤代环烷基，烯基，链二烯基，卤代烯基，环烯基，炔基，卤代炔基或环炔基，苯基，萘基或五 至10元饱和，部分不饱和或芳族杂环，其含有一个至四个由O，N和S组成的组的杂原子; R 1和R 2与它们所连接的氮原子一起也可以形成五元或六元环，其可被来自基团的原子中断 由O，N和S组成; 其中R 1和/或R 2可以如描述中所述被取代; 描述了制备这些化合物的方法，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US20050176736A1

公开(公告)日：2005-08-11

申请号：US10508409

申请日：2003-03-19

申请人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl ,  Ulrich Schofl

发明人： Jordi Tormo i Blasco ,  Carsten Blettner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl ,  Ulrich Schofl

IPC分类号： A01N43/90 ,  C07C255/57 ,  C07D487/04 ,  A61K31/519

CPC分类号： C07D487/04 ,  A01N43/90 ,  C07C255/57

摘要： The invention relates to triazolopyrimidines of formula (I), in which the substituents are defined as follows: L1 represents cyano, S(═O)nA1 or C(═O)A2, wherein A1 stands for hydrogen, hydroxy, alkyl, alkylamino or dialkylamino; A2 stands for C1-C8 alkoxy, C1-C6 haloalkoxy or one of the groups named in A1; and n stands for 0, 1 or 2; L2, L3 represent hydrogen or halogen; L4, L5 represent hydrogen, halogen or alkyl; X represents halogen, cyano, alkyl, haloalkyl, alkoxy or haloalkoxy; R1 represents alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, alkadienyl, haloalkenyl, cycloalkenyl, alkynyl, haloalkynyl or cycloalkynyl, phenyl, naphthyl, or a five to ten-membered saturated, partially unsaturated or aromatic heterocyclus containing between one and four heteroatoms from the group containing O, N or S; R2 represents hydrogen or R1; R1 and R2 can form, together with the nitrogen atom to which they are bonded, a five or six-membered ring, which can be interrupted and/or substituted by an atom from the group O, N and S; whereby R1 and/or R2 can be substituted in accordance with the description. The invention also relates to methods and intermediate products for producing said compounds, to agents containing the latter and to the use of said compounds for combating harmful fungi.

摘要翻译： 本发明涉及式（I）的三唑并嘧啶，其中取代基定义如下：L 1表示氰基，S（-O）n A 1 或其中A 1代表氢，羟基，烷基，烷基氨基或二烷基氨基;或C（= O） A 2代表C 1 -C 8烷氧基，C 1 -C 6烷基，C 1 -C 6 - >卤代烷氧基或在A 中命名的基团之一; 而n代表0,1或2; L 2，L 3表示氢或卤素; L 4，L 5代表氢，卤素或烷基; X表示卤素，氰基，烷基，卤代烷基，烷氧基或卤代烷氧基; R 1表示烷基，卤代烷基，环烷基，卤代环烷基，烯基，链烯基，卤代烯基，环烯基，炔基，卤代炔基或环炔基，苯基，萘基或五至十元饱和，部分不饱和或芳族杂环 含有一个至四个来自含有O，N或S的基团的杂原子; R 2表示氢或R 1; R 1和R 2可以与它们所键合的氮原子一起形成五元或六元环，其可被中断和/或被 来自O，N和S族的原子; 其中R 1和/或R 2可以根据描述被取代。 本发明还涉及用于生产所述化合物的方法和中间产物，含有后者的试剂和所述化合物用于防治有害真菌的用途。

公开(公告)号：US20050107401A1

公开(公告)日：2005-05-19

申请号：US10505146

申请日：2003-02-06

申请人： Frank Schieweck ,  Jordi Blasco ,  Thomas Grote ,  Andreas Gypser ,  Bernd Muller ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schafer ,  Wassilios Grammenos ,  Markus Gewehr ,  Anja Schwogler ,  Carsten Blettner ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

发明人： Frank Schieweck ,  Jordi Blasco ,  Thomas Grote ,  Andreas Gypser ,  Bernd Muller ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schafer ,  Wassilios Grammenos ,  Markus Gewehr ,  Anja Schwogler ,  Carsten Blettner ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

IPC分类号： A01N43/54 ,  C07D401/04 ,  A61K31/506 ,  C07D43/04

CPC分类号： C07D401/04

摘要： The invention relates to 2-(2-pyridyl)-5-phenyl-6-amninopyrimidines of formula I, wherein the substitutes and the index have the following meaning: R1 represents halogen, hydroxy, hyano, hxo, nitro, amino, mercapto, alkyl, halogenalkyl, alkenyl, alkinyl, cycloalkyl, alkoxy, halogenalkoxy, carboxyl, alkoxycarbonyl, carbamoyl, alkylaminocarbonyl, dialkylamincarbonyl, morpholinocarbonyl, pyrrolidinocarbonyl, alkylcarbonylamino, alkylamino. dialkylamino, alkylthio, alkylsulfinyl, alkylsulfonyl, hydroxysulfonyl, aminosulfonyl, alkylaminosulfonyl, dialkylaminosulfonyl; m=0 or 1-4; R2 represents hydrogen, halogen, cyano, alkyl, halogenalkyl or alkoxy; R3, R4 represents hydrogen, alkyl, halogenalkyl, cycloalkyl, halogencycloalkyl, alkenyl, halogenalkenyl, cycloalkenyl, alkinyl, halogenalkinyl or cycloalkinyl, R3 and R4 together with the nitrogen atom to which they are connected, form a five or six-membered ring which is interrupted by an atom from the group O, N or S and/or can be substituted according to the description; R5 represents halogen, alkyl or halogenalkyl; R6 represents hydrogen or one of the known groups in R5; R7, R8 represent hydrogen, halogen, alkyl or halogenalkyl; R9 represents hydrogen, halogen, hydroxy, cyano, alkyl, alkoxy, cycloalkoxy, halogenalkoxy, alkoxycarbonyl or alkylaminocarbonyl. The invention also relates to a method and intermediate product for the production of said compound in addition to the use thereof for combating undesirable plants.

摘要翻译： 本发明涉及式I的2-（2-吡啶基）-5-苯基-6-脒嘧啶，其中取代基和指数具有以下含义：R 1表示卤素，羟基，杂环基， 烷氧基，烷氧基羰基，氨基甲酰基，烷基氨基羰基，二烷基氨基羰基，吗啉代羰基，吡咯烷基羰基，烷基羰基氨基，烷基氨基。 二烷基氨基，烷硫基，烷基亚磺酰基，烷基磺酰基，羟基磺酰基，氨基磺酰基，烷基氨基磺酰基，二烷基氨基磺酰基; m = 0或1-4; R 2表示氢，卤素，氰基，烷基，卤代烷基或烷氧基; R 3，R 4表示氢，烷基，卤代烷基，环烷基，卤代烷基，烯基，卤代烯基，环烯基，炔基，卤代炔基或环炔基，R 3 O 和R 4与它们连接的氮原子一起形成5或6元环，其被来自基团O，N或S的原子和/或可被取代 根据说明; R 5表示卤素，烷基或卤代烷基; R 6表示氢或R 5中的已知基团之一; R 7，R 8表示氢，卤素，烷基或卤代烷基; R 9表示氢，卤素，羟基，氰基，烷基，烷氧基，环烷氧基，卤代烷氧基，烷氧基羰基或烷基氨基羰基。 本发明还涉及用于生产所述化合物的方法和中间产物，除了其用于对抗不期望的植物之外。

公开(公告)号：US20050272749A1

公开(公告)日：2005-12-08

申请号：US10531981

申请日：2003-11-04

申请人： Jordi Tormo Blasco ,  Carsten Bletner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

发明人： Jordi Tormo Blasco ,  Carsten Bletner ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Peter Schafer ,  Frank Schieweck ,  Anja Schwogler ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Ulrich Schofl ,  Reinhard Stierl

IPC分类号： C07D487/04 ,  A61K31/519

CPC分类号： C07D487/04

摘要： 5-Alkyl-7-aminotriazolopyrimidines of the formula I, where: R1, R2 are hydrogen, alkyl, alkenyl, alkynyl, haloalkyl, cycloalkyl, phenyl, naphthyl; 5- or 6-membered saturated, unsaturated or aromatic heterocyclyl which contains one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom; or R1 and R2 together with the bridging nitrogen atom can form a 5- or 6-membered ring which contains one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom; R3 is cycloalkyl or bicycloalkyl; where R1, R2 and R3 may be substituted as outlined in the description; X is alkyl or haloalkyl; and their salts; processes and intermediates for their preparation, compositions comprising them and their use for controlling phytopathogenic harmful fungi are described.

摘要翻译： 式I的5-烷基-7-氨基三唑并嘧啶，其中：R 1，R 2是氢，烷基，烯基，炔基，卤代烷基，环烷基，苯基，萘基; 含有1-4个氮原子或一至三个氮原子和一个硫或氧原子的5-或6-元饱和，不饱和或芳族杂环基; 或R 1和R 2与桥连氮原子一起可以形成含有1-4个氮原子或一至三个氮原子的5-或6-元环，并且 一个硫或氧原子; R 3是环烷基或双环烷基; 其中R 1，R 2和R 3可以如说明书中概述的那样被取代; X是烷基或卤代烷基; 和它们的盐; 描述了其制备方法和中间体，包含它们的组合物及其用于控制​​植物病原性有害真菌的用途。

公开(公告)号：US20050107619A1

公开(公告)日：2005-05-19

申请号：US10507605

申请日：2003-03-12

申请人： Wassilios Grammenos ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Andreas Gypser ,  Bernd Muller ,  Joachim Rheinheimer ,  Peter Schafer ,  Anja Schwogler ,  Jordi Blasco ,  Norbert Gotz ,  Gisela Lorenz ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Reinhard Stierl

发明人： Wassilios Grammenos ,  Thomas Grote ,  Carsten Blettner ,  Markus Gewehr ,  Andreas Gypser ,  Bernd Muller ,  Joachim Rheinheimer ,  Peter Schafer ,  Anja Schwogler ,  Jordi Blasco ,  Norbert Gotz ,  Gisela Lorenz ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Reinhard Stierl

IPC分类号： A01N37/18 ,  A01N37/36 ,  A01N37/38 ,  C07B61/00 ,  C07C231/12 ,  C07C233/22 ,  C07C235/34 ,  C07C233/73

CPC分类号： C07C235/34 ,  A01N37/18 ,  A01N37/36 ,  A01N37/38 ,  C07C233/22 ,  C07C2601/02 ,  C07C2601/08 ,  C07C2601/14

摘要： Z-substituted acrylamides of formula (I), where the substituents have the following meanings: X=H, halogen, alkyl, haloalkyl, alkoxy, haloalkoxy, with X in the 3- or 4-position, n=1 or 2, where X can be different if n=2, R1=alkyl, haloalkyl, cycloalkyl, alkoxy, haloalkoxy, aziridine and oxirane and R2=H, alkyl, haloalkyl, allyl, propargyl or CH2C≡C-alkyl. Methods for production thereof, agents comprising the above and the use thereof for the treatment of plant-pathogenic fungal pests.

摘要翻译： 式（I）的Z-取代的丙烯酰胺，其中取代基具有以下含义：X = H，卤素，烷基，卤代烷基，烷氧基，卤代烷氧基，其中X为3-或4-位，n = 1或2，其中 如果n = 2，则X可以不同，R 1 =烷基，卤代烷基，环烷基，烷氧基，卤代烷氧基，氮丙啶和环氧乙烷，R 2 = H，烷基，卤代烷基，烯丙基 炔丙基或CH 2C≡C-烷基。 其制备方法，包含上述物质及其用于治疗植物致病性真菌害虫的用途。

公开(公告)号：US20050261314A1

公开(公告)日：2005-11-24

申请号：US10484250

申请日：2002-07-16

申请人： Jordi i Blasco ,  Hubert Sauter ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schafer ,  Frank Schieweck ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

发明人： Jordi i Blasco ,  Hubert Sauter ,  Bernd Muller ,  Markus Gewehr ,  Wassilios Grammenos ,  Thomas Grote ,  Andreas Gypser ,  Joachim Rheinheimer ,  Ingo Rose ,  Peter Schafer ,  Frank Schieweck ,  Eberhard Ammermann ,  Siegfried Strathmann ,  Gisela Lorenz ,  Reinhard Stierl

IPC分类号： A01N43/90 ,  C07D487/04

CPC分类号： C07D487/04 ,  A01N43/90

摘要： The invention relates to 7-amino triazolopyrimidines of formula (I), in which the substituents have the following meanings: R1, R2 represent hydrogen, alkyl, alkenyl, alkynyl, cycloalkyl, phenyl, naphthyl; or 5-membered or 6-membered heterocyclyl containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom; or 5-membered or 6-membered heteroaryl containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or R1 and R2 can, together with the nitrogen atom, which binds them, form a 5-membered or 6-membered ring containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom; R3 represents alkyl, alkenyl, alkynyl, cycloalkyl, phenylalkyl and alkyl halide; whereby R3 and R2 can be unsubstituted or partially or completely substituted according to the description; X represents halogen, cyano, alkoxy, alkyl halide, phenyl or phenyl that is substituted by Ra. The invention also relates to methods and intermediate products for producing said compounds, to agents containing the same, and to their use.

摘要翻译： 本发明涉及式（I）的7-氨基三唑并嘧啶，其中取代基具有以下含义：R 1，R 2表示氢，烷基，烯基，炔基 ，环烷基，苯基，萘基; 或含有1至4个氮原子或1至3个氮原子和1个硫或氧原子的5元或6元杂环基; 或含有1至4个氮原子或1至3个氮原子和1个硫或氧原子的5元或6元杂芳基，或R 1和R 2可以， 与它们结合的氮原子一起形成含有一至四个氮原子或一至三个氮原子和一个硫或氧原子的五元或六元环; R 3表示烷基，烯基，炔基，环烷基，苯基烷基和烷基卤; 根据描述，R 3和R 2可以是未取代的或部分或完全取代的; X表示卤素，氰基，烷氧基，烷基卤，苯基或被R a取代的苯基。 本发明还涉及用于生产所述化合物的方法和中间产物，含有该化合物的试剂及其用途。