公开(公告)号：US20140315967A1

公开(公告)日：2014-10-23

申请号：US14359449

申请日：2012-11-16

Applicant: Kureha Corporation

Inventor： Nobuyuki Araki ,  Taiji Miyake ,  Emiko Obata

IPC: C07D249/08 ,  A01N43/653

CPC classification number: C07D249/08 ,  A01N43/50 ,  A01N43/653

Abstract: In order to provide a compound which exhibits a high controlling effect against plant diseases and is able to reduce phytotoxicity, the present invention is a triazole derivative represented by General Formula (I), the azole derivative being a (−)-enantiomer or (+)-enantiomer having an —R1 group, hydroxy group, and substituted or unsubstituted benzyl group bonded to a cyclopentane ring in cis-form.

Abstract translation: 本发明为通式（I）表示的三唑衍生物，为（ - ） - 对映异构体或（+） - 对映异构体的唑类衍生物，为了提供对植物病害具有高控制效果且能够降低植物毒性的化合物， ） - 对映异构体，其具有-R1基团，羟基和与顺式环戊烷环键合的取代或未取代的苄基。

公开(公告)号：US09440933B2

公开(公告)日：2016-09-13

申请号：US14691279

申请日：2015-04-20

Applicant: KUREHA CORPORATION

Inventor： Nobuyuki Araki ,  Taiji Miyake ,  Eiyu Imai ,  Emiko Obata

IPC: C07D249/08 ,  C07D249/12 ,  C07D233/56 ,  A01N43/653 ,  C07D233/60 ,  C07D405/06 ,  A01N43/50 ,  A01N43/80 ,  C07D405/04

CPC classification number: C07D249/12 ,  A01N43/50 ,  A01N43/653 ,  A01N43/80 ,  C07D233/56 ,  C07D233/60 ,  C07D249/08 ,  C07D405/04 ,  C07D405/06 ,  A01N25/04 ,  A01N25/28

Abstract: Provided is an azole derivative superior in disease-controlling activity contained as an active ingredient in agricultural or horticultural chemical agents.The azole derivative according to the present invention is represented by the following General Formula (I): (in Formula (I), R1 represents an unsubstituted or substituted C1-C6-alkyl group; R2 represents a carbonyl group-containing functional group, wherein the carbon atom in the carbonyl group is bound to the carbon atom in the cyclopentane ring substituted with R1 and to a hydrogen atom, a hydroxyl group, R3, OR3, or NR3R4; R3 and R4 each represent a C1-C6-alkyl group, a C2-C6-alkenyl group, or a C2-C6-alkynyl group; Y represents a halogen atom, a C1-C4-alkyl group, a C1-C4-haloalkyl group, a C1-C4-alkoxy group, a C1-C4-haloalkoxy group, a phenyl group, a cyano group, or a nitro group; m is 0 to 5; and A represents a nitrogen atom or a methine group).

公开(公告)号：US09278941B2

公开(公告)日：2016-03-08

申请号：US14359449

申请日：2012-11-16

Applicant: Kureha Corporation

Inventor： Nobuyuki Araki ,  Taiji Miyake ,  Emiko Obata

IPC: A01N43/653 ,  C07D249/08 ,  A01N43/50

CPC classification number: C07D249/08 ,  A01N43/50 ,  A01N43/653

Abstract: In order to provide a compound which exhibits a high controlling effect against plant diseases and is able to reduce phytotoxicity, the present invention is a triazole derivative represented by General Formula (I), the azole derivative being a (−)-enantiomer or (+)-enantiomer having an —R1 group, hydroxy group, and substituted or unsubstituted benzyl group bonded to a cyclopentane ring in cis-form.

Abstract translation: 本发明为通式（I）表示的三唑衍生物，为（ - ） - 对映异构体或（+） - 对映异构体的唑类衍生物，为了提供对植物病害具有高控制效果且能够降低植物毒性的化合物， ） - 对映异构体，其具有-R1基团，羟基和与顺式环戊烷环键合的取代或未取代的苄基。