公开(公告)号：US06525211B1

公开(公告)日：2003-02-25

申请号：US09838812

申请日：2001-04-20

申请人： Klaus-Helmut Müller ,  Rolf Kirsten ,  Ernst Rudolf F. Gesing ,  Joachim Kluth ,  Mark Wilhelm Drewes ,  Kurt Findeisen ,  Johannes Rudolf Jansen ,  Klaus König ,  Hans-Jochem Riebel ,  Otto Schallner ,  Markus Dollinger ,  Hans-Joachim Santel

发明人： Klaus-Helmut Müller ,  Rolf Kirsten ,  Ernst Rudolf F. Gesing ,  Joachim Kluth ,  Mark Wilhelm Drewes ,  Kurt Findeisen ,  Johannes Rudolf Jansen ,  Klaus König ,  Hans-Jochem Riebel ,  Otto Schallner ,  Markus Dollinger ,  Hans-Joachim Santel

IPC分类号： C07C30941

CPC分类号： C07D263/34 ,  A01N43/74 ,  A01N43/76 ,  A01N43/82 ,  A01N47/38 ,  C07C249/12 ,  C07C309/87 ,  C07C311/29 ,  C07C311/65 ,  C07C331/32 ,  C07D249/12 ,  C07D249/14 ,  C07D263/42 ,  C07D271/06 ,  C07D271/10 ,  C07D487/04

摘要： The invention relates to novel sulphonylamino(thio)carbonyl compounds of the formula (I), in which A represents a single bond, oxygen, sulphur or the group N—R, in which R represents hydrogen, alkyl, alkenyl, alkinyl or cycloalkyl, Q represents oxygen or sulphur, R1 represents hydrogen or formyl or represents in each case optionally substituted alkyl, alkenyl, alkinyl, alkylcarbonyl, alkoxycarbonyl, alkylsulphonyl, cycloalkyl, cycloalkylcarbonyl or cycloalkylsulphonyl, R2 represents cyano or halogen or represents in each case optionally substituted alky, alkenyl, alkinyl, alkoxy, alkenyloxy or alkinyloxy, and R3 represents in each case optionally substituted heterocyclyl having 5 ring members of which at least one is oxygen, sulphur or nitrogen and from one to three further ring members can be nitrogen, and salts of compounds of the formula (I), the previously known compounds 4,5-dimethoxy-2-(2,5-dimethoxy-phenylsulphonylaminocarbonyl)-2,4-dihydro-3H-1,2,4-triazol-3-one, 4,5-diethoxy-2-(2,5-dimethoxy-phenylsulphonylaminocarbonyl)-2,4-dihydro-3H-1,2,4-triazol-3-one and N-(2,5-dimethoxy-phenylsulphonyl)-1,5-dimethyl-1H-pyrazole-3-carboxamide being excluded by disclaimer; and also to processes and novel intermediates for the preparation of the novel substances and to their use as herbicides.

摘要翻译： 本发明涉及式（I）的新型磺酰基氨基（硫代）羰基化合物，其中A表示单键，氧，硫或基团NR，其中R表示氢，烷基，烯基，炔基或环烷基，Q表示氧 或硫，R1表示氢或甲酰基，或表示在各种情况下任选取代的烷基，烯基，炔基，烷基羰基，烷氧基羰基，烷基磺酰基，环烷基，环烷基羰基或环烷基磺酰基，R2表示氰基或卤素，或表示在各情况下任选取代的烷基，烯基，炔基 ，烷氧基，烯氧基或烷氧基，R 3在各自的情况下表示具有5个环成员的任选取代的杂环基，其中至少一个是氧，硫或氮，并且一至三个其它的环成员可以是氮， I），先前已知的化合物4,5-二甲氧基-2-（2,5-二甲氧基 - 苯基磺酰基氨基羰基）-2,4-二氢-3H-1,2,4-三唑-3-酮，4,5-二乙氧基 -2-（2,5-二 甲氧基 - 苯基磺酰基氨基羰基）-2,4-二氢-3H-1,2,4-三唑-3-酮和N-（2,5-二甲氧基 - 苯基磺酰基）-1,5-二甲基-1H-吡唑-3-甲酰胺 被排除在免责声明之外;还涉及用于制备新物质和用作除草剂的方法和新型中间体。

公开(公告)号：US06251831B1

公开(公告)日：2001-06-26

申请号：US09223246

申请日：1998-12-30

申请人： Klaus-Helmut Müller ,  Rolf Kirsten ,  Ernst Rudolf F. Gesing ,  Joachim Kluth ,  Mark Wilhelm Drewes ,  Kurt Findeisen ,  Johannes Rudolf Jansen ,  Klaus König ,  Hans-Jochem Riebel ,  Otto Schallner ,  Markus Dollinger ,  Hans-Joachim Santel

发明人： Klaus-Helmut Müller ,  Rolf Kirsten ,  Ernst Rudolf F. Gesing ,  Joachim Kluth ,  Mark Wilhelm Drewes ,  Kurt Findeisen ,  Johannes Rudolf Jansen ,  Klaus König ,  Hans-Jochem Riebel ,  Otto Schallner ,  Markus Dollinger ,  Hans-Joachim Santel

IPC分类号： A01N43653

CPC分类号： C07D263/34 ,  A01N43/74 ,  A01N43/76 ,  A01N43/82 ,  A01N47/38 ,  C07C249/12 ,  C07C309/87 ,  C07C311/29 ,  C07C311/65 ,  C07C331/32 ,  C07D249/12 ,  C07D249/14 ,  C07D263/42 ,  C07D271/06 ,  C07D271/10 ,  C07D487/04

摘要： The invention relates to novel sulphonylamino(thio)carbonyl compounds of the formula (I), in which A represents a single bond, oxygen, sulphur or the group N—R, in which R represents hydrogen, alkyl, alkenyl, alkinyl or cycloalkyl, Q represents oxygen or sulphur, R1 represents hydrogen or formyl or represents in each case optionally substituted alkyl, alkenyl, alkinyl, alkylcarbonyl, alkoxycarbonyl, alkylsulphonyl, cycloalkyl, cycloalkylcarbonyl or cycloalkylsulphonyl, R2 represents cyano or halogen or represents in each case optionally substituted alkyl, alkenyl, alkinyl, alkoxy, alkenyloxy or alkinyloxy, and R3 represents in each case optionally substituted heterocyclyl having 5 ring members of which at least one is oxygen, sulphur or nitrogen and from one to three further ring members can be nitrogen, and salts of compounds of the formula (I), the previously known compounds 4,5-dimethoxy-2-(2,5-dimethoxy-phenylsulphonylaminocarbonyl)-2,4-dihydro-3H-1,2,4-triazol-3-one, 4,5-diethoxy-2-(2,5-dimethoxy-phenylsulphonylaminocarbonyl)-2,4-dihydro-3H-1,2,4-triazol-3-one and N-(2,5-dimethoxy-phenylsulphonyl)-1,5-dimethyl-1H-pyrazole-3-carboxamide being excluded by disclaimer; and also to processes and novel intermediates for the preparation of the novel substances and to their use as herbicides.

摘要翻译： 本发明涉及式（I）的新型磺酰基氨基（硫代）羰基化合物，其中A表示单键，氧，硫或基团NR，其中R表示氢，烷基，烯基，炔基或环烷基，Q表示氧 或硫，R 1表示氢或甲酰基或在每种情况下表示任选取代的烷基，烯基，炔基，烷基羰基，烷氧基羰基，烷基磺酰基，环烷基，环烷基羰基或环烷基磺酰基，R 2表示氰基或卤素，或表示在各种情况下任选取代的烷基，烯基， ，烷氧基，烯氧基或烷氧基，R 3在各自的情况下表示具有5个环成员的任选取代的杂环基，其中至少一个是氧，硫或氮，并且一至三个其它的环成员可以是氮， I），先前已知的化合物4,5-二甲氧基-2-（2,5-二甲氧基 - 苯基磺酰基氨基羰基）-2,4-二氢-3H-1,2,4-三唑-3-酮，4,5-二乙氧基 -2-（2,5-d 苯并磺酰基氨基羰基）-2,4-二氢-3H-1,2,4-三唑-3-酮和N-（2,5-二甲氧基 - 苯基磺酰基）-1,5-二甲基-1H-吡唑-3-甲酰胺 由免责声明排除;以及用于制备新物质和用作除草剂的方法和新型中间体。

公开(公告)号：US06200934B1

公开(公告)日：2001-03-13

申请号：US09142272

申请日：1998-09-03

申请人： Klaus-Helmut Müller ,  Mark Wilhelm Drewes ,  Ernst Rudolf F. Gesing ,  Johannes Rudolf Jansen ,  Rolf Kirsten ,  Joachim Kluth ,  Klaus König ,  Hans-Jochem Riebel ,  Otto Schallner ,  Kurt Findeisen ,  Markus Dollinger

发明人： Klaus-Helmut Müller ,  Mark Wilhelm Drewes ,  Ernst Rudolf F. Gesing ,  Johannes Rudolf Jansen ,  Rolf Kirsten ,  Joachim Kluth ,  Klaus König ,  Hans-Jochem Riebel ,  Otto Schallner ,  Kurt Findeisen ,  Markus Dollinger

IPC分类号： A01N43653

CPC分类号： A01N47/38 ,  C07D249/12

摘要： The invention relates to novel substituted arylsulphonylamino(thio)carbonyl-triazolin(thi)ones of the formula (I) useful as herbicides.

摘要翻译： 本发明涉及用作除草剂的式（I）的新型取代的芳基磺酰基氨基（硫代）羰基 - 三唑啉（thi）。

公开(公告)号：US06677277B1

公开(公告)日：2004-01-13

申请号：US09194261

申请日：1999-05-13

申请人： Otto Schallner ,  Mark-Wilhelm Drewes ,  Kurt Findeisen ,  Ernst-Rudolf F. Gesing ,  Johannes-Rudolf Jansen ,  Rolf Kirsten ,  Joachim Kluth ,  Klaus-Helmut Müller ,  Klaus König ,  Ulrich Philipp ,  Hans-Jochem Riebel ,  Peter Wolfrum ,  Markus Dollinger

发明人： Otto Schallner ,  Mark-Wilhelm Drewes ,  Kurt Findeisen ,  Ernst-Rudolf F. Gesing ,  Johannes-Rudolf Jansen ,  Rolf Kirsten ,  Joachim Kluth ,  Klaus-Helmut Müller ,  Klaus König ,  Ulrich Philipp ,  Hans-Jochem Riebel ,  Peter Wolfrum ,  Markus Dollinger

IPC分类号： A01N4738

CPC分类号： C07D271/06 ,  A01N47/38 ,  C07C311/65 ,  C07C317/14 ,  C07C323/67 ,  C07D249/12

摘要： The invention relates to novel sulfonylamino(thio)carbonyl compounds of the formula (I), in which n represents the numbers 0, 1 or 2, A represents a single bond, or oxygen or sulfur, or the grouping N—R, in which R represents hydrogen, alkyl, alkenyl, alkinyl or cycloalkyl, Q represents oxygen or sulfur, R1 represents hydrogen or formyl, or represents respectively optionally substituted alkyl, alkoxy, alkylamino, alkoxyamino, dialkylamino, N-alkoxy-N-alkyl-amino, alkylcarbonyl, alkoxycarbonyl, alkylsulfonyl, alkenyl, alkinyl, cycloalkyl, cycloalkylcarbonyl or cycloalkylsulfonyl, R2 represents cyano or halogen, or represents respectively optionally substituted alkyl, alkoxy, alkylthio, alkylsulfinyl, alkylsulfonyl, dialkylaminosulfonyl, alkenyl, alkinyl, alkenyloxy or alkinyloxy, and R3 represents respectively optionally substituted heterocyclyl having 5 ring members of which at least one is oxygen, sulfur or nitrogen and from one to three further ring members can be nitrogen, and salts of compounds of the formula (I), a plurality of processes and novel intermediates for preparing them and their use as herbicides.

摘要翻译： 本发明涉及式（I）的新型磺酰基氨基（硫代）羰基化合物，其中n代表数字0,1或2，A代表单键，或氧或硫，或分组NR，其中R表示氢 烷基，烯基，炔基或环烷基，Q表示氧或硫，R 1表示氢或甲酰基，或分别表示任选取代的烷基，烷氧基，烷基氨基，烷氧基氨基，二烷基氨基，N-烷氧基-N-烷基 - 氨基， 烷氧基羰基，烷基磺酰基，烯基，炔基，环烷基，环烷基羰基或环烷基磺酰基，R 2表示氰基或卤素，或分别表示任选取代的烷基，烷氧基，烷硫基，烷基亚磺酰基，烷基磺酰基，二烷基氨基磺酰基，烯基，炔基，烯氧基或烷氧基， 3分别表示具有5个环成员的任选取代的杂环基，其中至少一个是氧，硫或氮，并且一个至三个另外的环成员可以是氮，并且盐 f式（I）化合物，多种方法和用于制备它们的新型中间体及其作为除草剂的用途。

公开(公告)号：USRE39607E1

公开(公告)日：2007-05-01

申请号：US10603997

申请日：2003-06-25

申请人： Klaus-Helmut Müller ,  Rolf Kirsten ,  Ernst Rudolf F. Gesing ,  Joachim Kluth ,  Mark Wilhelm Drewes ,  Kurt Findeisen ,  Johannes Rudolf Jansen ,  Klaus König ,  Hans-Jochem Riebel ,  Otto Schallner ,  Markus Dollinger ,  Hans-Joachim Santel

发明人： Klaus-Helmut Müller ,  Rolf Kirsten ,  Ernst Rudolf F. Gesing ,  Joachim Kluth ,  Mark Wilhelm Drewes ,  Kurt Findeisen ,  Johannes Rudolf Jansen ,  Klaus König ,  Hans-Jochem Riebel ,  Otto Schallner ,  Markus Dollinger ,  Hans-Joachim Santel

IPC分类号： A01N43/653 ,  C07D249/12

CPC分类号： C07D263/34 ,  A01N43/76 ,  A01N43/82 ,  A01N47/38 ,  C07C249/12 ,  C07C309/87 ,  C07C311/29 ,  C07C311/65 ,  C07C331/32 ,  C07D249/12 ,  C07D249/14 ,  C07D263/42 ,  C07D271/06 ,  C07D271/10 ,  C07D487/04

摘要： The invention relates to novel sulphonylamino(thio) carbonyl compounds of the formula (I), in which A represents a single bond, oxygen, sulphur or the group N—R, in which R represents hydrogen, alkyl, alkenyl, alkinyl or cycloalkyl, Q represents oxygen or sulphur, R1 represents hydrogen or formyl or represents in each case optionally substituted alkyl, alkenyl, alkinyl, alkylcarbonyl, alkoxycarbonyl, alkylsulphonyl, cycloalkyl, cycloalkylcarbonyl or cycloalkylsulphonyl, R2 represents cyano or halogen or represents in each case optionally substituted alkyl, alkenyl, alkinyl, alkoxy, alkenyloxy or alkinyloxy, and R3 represents in each case optionally substituted heterocyclyl having 5 ring members of which at least one is oxygen, sulphur or nitrogen and from one to three further ring members can be nitrogen, and salts of compounds of the formula (I), the previously known compounds 4,5-dimethoxy-2-(2,5-dimethoxy-phenylsulphonylaminocarbonyl)-2,4-dihydro-3H-1,2,4-triazol-3-one, 4,5-diethoxy-2-(2,5-dimethoxy-phenylsulphonylaminocarbonyl)-2,4-dihydro-3H-1,2,4-triazol-3-one and N-(2,5-dimethoxy-phenylsulphonyl)-1,5-dimethyl-1H-pyrazole-3-carboxamide being excluded by disclaimer; and also to processes and novel intermediates for the preparation of the novel substances and to their use as herbicides.

摘要翻译： 本发明涉及式（I）的新型磺酰基氨基（硫代）羰基化合物，其中A表示单键，氧，硫或基团NR，其中R表示氢，烷基，烯基，炔基或环烷基，Q表示 氧或硫，R 1表示氢或甲酰基，或在各种情况下表示任选取代的烷基，烯基，炔基，烷基羰基，烷氧基羰基，烷基磺酰基，环烷基，环烷基羰基或环烷基磺酰基，R 2 >表示氰基或卤素，或表示在各种情况下任选取代的烷基，烯基，炔基，烷氧基，烯氧基或烷氧基，R 3表示在每种情况下任选取代的具有5个环成员的杂环基，其中至少一个 是氧，硫或氮，并且一至三个其它的环成员可以是氮，并且式（I）化合物的盐，先前已知的化合物4,5-二甲氧基-2-（2,5-二甲氧基 - 苯基磺酰基氨基羰基） -2,4-二氢-3H- 1,2,4-三唑-3-酮，4,5-二乙氧基-2-（2,5-二甲氧基 - 苯基磺酰基氨基羰基）-2,4-二氢-3H-1,2,4-三唑-3-酮和 通过免责声明排除N-（2,5-二甲氧基 - 苯基磺酰基）-1,5-二甲基-1H-吡唑-3-甲酰胺; 以及用于制备新物质及其作为除草剂的用途的方法和新型中间体。

公开(公告)号：US06200931B1

公开(公告)日：2001-03-13

申请号：US09242253

申请日：1999-05-13

申请人： Klaus-Helmut Müller ,  Mark Wilhelm Drewes ,  Kurt Findeisen ,  Ernst Rudolf F. Gesing ,  Johannes Rudolf Jansen ,  Rolf Kirsten ,  Joachim Kluth ,  Ulrich Philipp ,  Hans-Jochem Riebel ,  Klaus König ,  Markus Dollinger ,  Hans-Joachim Santel

发明人： Klaus-Helmut Müller ,  Mark Wilhelm Drewes ,  Kurt Findeisen ,  Ernst Rudolf F. Gesing ,  Johannes Rudolf Jansen ,  Rolf Kirsten ,  Joachim Kluth ,  Ulrich Philipp ,  Hans-Jochem Riebel ,  Klaus König ,  Markus Dollinger ,  Hans-Joachim Santel

IPC分类号： A01N4388

CPC分类号： C07D413/12 ,  A01N47/38 ,  C07D413/14

摘要： The invention relates to novel substituted sulphonylamino(thio)carbonyl compounds of the formula (I) in which A represents a single bond, represents oxygen, imino (NH), alkanediyl (alkylene) or alkylimino (N-alkyl), J represents a (hetero)aryl grouping selected from the series phenyl, pyridyl, pyrazolyl, thienyl which is substituted by a 5,6-dihydro-[1,4,2]-dioxazin-3-yl group (which may for its part be substituted by halogen, alkyl or halogenoalkyl) and optionally by one or two further radicals selected from the series cyano, halogeno, alkyl, halogenoalkyl, phenyl, pyridyl, Q represents oxygen or sulphur and, R represents optionally substituted heterocyclyl having 5 ring members of which at least one is oxygen, sulphur or nitrogen and one to three more may be nitrogen, and salts of compounds of the formula (I), processes and specific novel intermediates for their preparation and their use as herbicides.

摘要翻译： 本发明涉及式（I）的新型取代磺酰基氨基（硫代）羰基化合物，其中A代表单键，代表氧，亚氨基（NH），烷二基（亚烷基）或烷基亚氨基（N-烷基），J代表 ）芳基，其选自苯并吡啶基，吡唑基，噻吩基，其被5,6-二氢 - [1,4,2] - 二恶嗪-3-基（其可以被卤素取代）取代， 烷基或卤代烷基）和任选地一个或两个选自氰基，卤代，烷基，卤代烷基，苯基，吡啶基，Q代表氧或硫的其它基团，R代表任选取代的具有5个环成员的杂环基，其中至少一个是 氧，硫或氮，一至三个可以是氮，以及式（I）化合物的盐，其制备方法和具体的新型中间体及其作为除草剂的用途。

公开(公告)号：US06838414B2

公开(公告)日：2005-01-04

申请号：US10195979

申请日：2002-07-16

申请人： Ernst Rudolf F. Gesing ,  Rolf Kirsten ,  Joachim Kluth ,  Klaus-Helmut Müller ,  Mark Wilhelm Drewes ,  Johannes Rudolf Jansen ,  Ulrich Philipp ,  Hans-Jochem Riebel ,  Otto Schallner ,  Markus Dollinger ,  Hans-Joachim Santel

发明人： Ernst Rudolf F. Gesing ,  Rolf Kirsten ,  Joachim Kluth ,  Klaus-Helmut Müller ,  Mark Wilhelm Drewes ,  Johannes Rudolf Jansen ,  Ulrich Philipp ,  Hans-Jochem Riebel ,  Otto Schallner ,  Markus Dollinger ,  Hans-Joachim Santel

IPC分类号： A01N47/36 ,  C07D239/42 ,  C07D239/46 ,  C07D239/52 ,  C07D251/16 ,  C07D251/46 ,  C07D521/00 ,  A01N43/54 ,  C07D239/697

CPC分类号： C07D239/42 ,  A01N47/36 ,  C07D239/47 ,  C07D239/52 ,  C07D251/16 ,  C07D251/46 ,  C07D521/00

摘要： The invention relates to novel substituted arylsulphonyl(thio)ureas in which A represents nitrogen or a CH grouping, Q represents oxygen or sulphur, R1 represents hydrogen, halogen or respectively optionally substituted alkyl, alkoxy, alkylthio, alkylamino, dialkylamino, cycloalkyl, cycloalkyloxy or heterocyclyloxy, R2 represents hydrogen, halogen or respectively optionally substituted alkyl, alkoxy, alkylthio, alkylamino, dialkylamino, cycloalkyl, cycloalkyloxy or heterocyclyloxy, R3 represents hydrogen or optionally substituted alkyl, R4 represents respectively optionally substituted alkyl, alkoxy, alkenyl, alkinyl, alkenyloxy, alkinyloxy, cycloalkyl, cycloalkyloxy or cycloalkylalkyl, and R5 represents hydrogen, formyl or respectively optionally substituted alkyl, alkylcarbonyl, alkoxycarbonyl, alkylsulphonyl, alkenyl, alkinyl, cycloalkyl, cycloalkylcarbonyl, cycloalkylsulphonyl or heterocyclyl, and to salts of compounds of the formula (I), except for the compound N-(4,6-dimethyl-pyrimidin-2-yl)-N′-[2-(1,1,2,2-tetrafluoro-ethoxy)-6-methyl-phenylsulphonyl]-urea, to processes for preparing the novel compounds and to their use as herbicides.

摘要翻译： 本发明涉及A代表氮或CH基的新型取代芳基磺酰基（硫代）脲脲，Q表示氧或硫，R 1表示氢，卤素或分别任意取代的烷基，烷氧基，烷硫基，烷基氨基，二烷基氨基，环烷基，环烷氧基 或杂环氧基，R 2表示氢，卤素或分别任选取代的烷基，烷氧基，烷硫基，烷基氨基，二烷基氨基，环烷基，环烷氧基或杂环氧基，R 3表示氢或任选取代的烷基， 烷基，烷氧基，烯基，炔基，烯氧基，烷氧基，环烷基，环烷基氧基或环烷基烷基，R 5表示氢，甲酰基或分别任选取代的烷基，烷基羰基，烷氧基羰基，烷基磺酰基，烯基，炔基，环烷基，环烷基羰基，环烷基磺酰基或杂环基， 和式（I）化合物的盐，除了化合物N-（4,6-二甲基 - 吡啶-2-基） 亚氨基-2-基）-N' - [2-（1,1,2,2-四氟 - 乙氧基）-6-甲基 - 苯基磺酰基] - 脲，用于制备新化合物及其作为除草剂的用途。

公开(公告)号：US06451737B1

公开(公告)日：2002-09-17

申请号：US09125997

申请日：1998-08-28

申请人： Ernst Rudolf F. Gesing ,  Rolf Kirsten ,  Joachim Kluth ,  Klaus-Helmut Müller ,  Mark Wilhelm Drewes ,  Johannes Rudolf Jansen ,  Ulrich Philipp ,  Hans-Jochem Riebel ,  Otto Schallner ,  Markus Dollinger ,  Hans-Joachim Santel

发明人： Ernst Rudolf F. Gesing ,  Rolf Kirsten ,  Joachim Kluth ,  Klaus-Helmut Müller ,  Mark Wilhelm Drewes ,  Johannes Rudolf Jansen ,  Ulrich Philipp ,  Hans-Jochem Riebel ,  Otto Schallner ,  Markus Dollinger ,  Hans-Joachim Santel

IPC分类号： A01N4370

CPC分类号： C07D239/42 ,  A01N47/36 ,  C07D239/47 ,  C07D239/52 ,  C07D251/16 ,  C07D251/46 ,  C07D521/00

摘要： The invention related to novel substituted arylsulphonyl(thio)ureas wherein: A is nitrogen or a CH grouping, Q is oxygen or sulphur, R1 is hydrogen, halogen or optionally substituted alkyl, alkoxy, alkylthio, alkylamino, dialkylamino, cycloalkyl, cycloalkyloxy or heterocyclyloxy, R2 is hydrogen, halogen or optionally substituted alkyl, alkoxy, alkylthio, alkylamino, dialkylamino, cycloalkyl, cycloalkyloxy or heterocyclyloxy, R3 is hydrogen or optionally substituted alkyl, R4 is optionally substituted alkyl, alkoxy, alkenyl, alkinyl, alkenyloxy, alkinyloxy, cycloalkyl, cycloalkyloxy or cycloalkylalkyl, and R5 is hydrogen, formyl or optionally substituted alkyl, alkylcarbonyl, alkoxycarbonyl, alkylsulphonyl, alkenyl, alkinyl, cycloalkyl, cycloalkylcarbonyl, cycloalkylsulphonyl or heterocyclyl, and salts of compounds of the formula (I), except for the compound N-(4,6-dimethyl-pyrimidin-2-yl)-N′-[2-(1,1,2,2-tetrafluoro-ethoxy)-6-methyl-phenylsulphonyl]-urea.

摘要翻译： 本发明涉及新型取代的芳基磺酰基（硫代）脲：其中A为氮或CH基团，Q为氧或硫，R1为氢，卤素或任选取代的烷基，烷氧基，烷硫基，烷基氨基，二烷基氨基，环烷基，环烷氧基或杂环氧基， R2是氢，卤素或任选取代的烷基，烷氧基，烷硫基，烷基氨基，二烷基氨基，环烷基，环烷氧基或杂环氧基，R 3是氢或任选取代的烷基，R 4是任选取代的烷基，烷氧基，烯基，炔基，烯氧基， 环烷基氧基或环烷基烷基，R 5为氢，甲酰基或任选取代的烷基，烷基羰基，烷氧基羰基，烷基磺酰基，烯基，炔基，环烷基，环烷基羰基，环烷基磺酰基或杂环基，以及式（I）化合物的盐， （4,6-二甲基 - 嘧啶-2-基）-N' - [2-（1,1,2,2-四氟 - 乙氧基）-6-甲基 - 苯基磺酰基] - 脲。

公开(公告)号：US07723266B2

公开(公告)日：2010-05-25

申请号：US10901780

申请日：2004-07-29

申请人： Ernst Rudolf F. Gesing ,  Rolf Kirsten ,  Joachim Kluth ,  Klaus-Helmut Müller ,  Mark Wilhelm Drewes ,  Johannes Rudolf Jansen ,  Ulrich Philipp ,  Hans-Jochem Riebel ,  Otto Schallner ,  Markus Dollinger ,  Hans-Joachim Santel

发明人： Ernst Rudolf F. Gesing ,  Rolf Kirsten ,  Joachim Kluth ,  Klaus-Helmut Müller ,  Mark Wilhelm Drewes ,  Johannes Rudolf Jansen ,  Ulrich Philipp ,  Hans-Jochem Riebel ,  Otto Schallner ,  Markus Dollinger ,  Hans-Joachim Santel

IPC分类号： A01N43/54 ,  C07D239/02

CPC分类号： C07D239/42 ,  A01N47/36 ,  C07D239/47 ,  C07D239/52 ,  C07D251/16 ,  C07D251/46 ,  C07D521/00

摘要： The invention relates to novel substituted arylsulphonyl(thio)ureas in which A represents nitrogen or a CH grouping, Q represents oxygen or sulphur, R1 represents hydrogen, halogen or respectively optionally substituted alkyl, alkoxy, alkylthio, alkylamino, dialkylamino, cycloalkyl, cycloalkyloxy or heterocyclyloxy, R2 represents hydrogen, halogen or respectively optionally substituted alkyl, alkoxy, alkylthio, alkylamino, dialkylamino, cycloalkyl, cycloalkyloxy or heterocyclyloxy, R3 represents hydrogen or optionally substituted alkyl, R4 represents respectively optionally substituted alkyl, alkoxy, alkenyl, alkinyl, alkenyloxy, alkinyloxy, cycloalkyl, cycloalkyloxy or cycloalkylalkyl, and R5 represents hydrogen, formyl or respectively optionally substituted alkyl, alkylcarbonyl, alkoxycarbonyl, alkylsulphonyl, alkenyl, alkinyl, cycloalkyl, cycloalkylcarbonyl, cycloalkylsulphonyl or heterocyclyl, and to salts of compounds of the formula (I), except for the compound N-(4,6-dimethyl-primidin-2-yl)-N′-[2-1,1,2,2-tetrafluoro-ethoxy-6-methyl-phenylsulphonyl]-urea, to process for preparing the novel compounds and to their use as herbicides.

摘要翻译： 本发明涉及新的取代芳基磺酰基（硫代）脲，其中A代表氮或CH基团，Q代表氧或硫，R1代表氢，卤素或分别任意取代的烷基，烷氧基，烷硫基，烷基氨基，二烷基氨基，环烷基，环烷氧基或 烷氧基，烷硫基，烷基氨基，二烷基氨基，环烷基，环烷氧基或杂环氧基，R 3表示氢或任选取代的烷基，R 4表示分别为任选取代的烷基，烷氧基，烯基，炔基，烯氧基， 烷氧基羰基，烷基磺酰基，烯基，炔基，环烷基，环烷基羰基，环烷基磺酰基或杂环基，以及式（I）化合物的盐， 除了化合物N-（4,6-二甲基 - 咪唑-2-基）-N' - [2-1,1,2,2-四氟 - 乙氧基-6-甲基 - 苯基磺酰基] - 脲，用于制备新化合物及其作为除草剂的用途。

公开(公告)号：US06297195B1

公开(公告)日：2001-10-02

申请号：US09214773

申请日：1999-05-10

申请人： Ernst Rudolf F. Gesing ,  Mark Wilhelm Drewes ,  Johannes R. Jansen ,  Rolf Kirsten ,  Joachim Kluth ,  Klaus-Helmut Müller ,  Ulrich Philipp ,  Hans-Jochem Riebel ,  Otto Schallner ,  Detlef Wollweber ,  Markus Dollinger ,  Klaus Stenzel ,  Christoph Erdelen

发明人： Ernst Rudolf F. Gesing ,  Mark Wilhelm Drewes ,  Johannes R. Jansen ,  Rolf Kirsten ,  Joachim Kluth ,  Klaus-Helmut Müller ,  Ulrich Philipp ,  Hans-Jochem Riebel ,  Otto Schallner ,  Detlef Wollweber ,  Markus Dollinger ,  Klaus Stenzel ,  Christoph Erdelen

IPC分类号： A01N4388

CPC分类号： C07D487/04 ,  A01N43/90

摘要： The invention concerns novel substituted triazoloazine sulphonamides of formula (I) in which Q1 stands for nitrogen or a CH group: Q2 stands for nitrogen or a CH group; R1 stands for hydrogen or halogen, or for C1-C4 alkyl, C1-C4 alkoxy, C1-C4 alkylthio, C1-C4 alkylamino or di(C1-C4 alkyl)amino, in each case optionally substituted by hydroxy, halogen or C1-C4 alkoxy; R2 stands for hydrogen or halogen, or for C1-C4 alkyl, C1-C4 alkoxy, C1-C4 alkylthio, C1-C4 alkylamino or di(C1-C4 alkyl)amino, in each case optionally substituted by halogen; and Ar stands for 4-cyano-2,5-difluoro-phenyl, 2,6-dimethoxy-phenyl, 2-bromo-3-trifluoro-methyl-phenyl, 2-bromo-5-trifluoromethyl-phenyl, 6-chloro-pyridine-3-yl-methyl or one of the 5- or 6-member (hetero)cyclic groups mentioned in the description. The invention also concerns salts of these substances, a process for preparing the novel compounds, and their use as plant-treatment agents.

摘要翻译： 本发明涉及式（I）的新型取代的三唑并乙酰胺，其中Q 1代表氮或CH基：Q 2代表氮或CH基; R1代表氢或卤素，或C1-C4烷基，C1-C4烷氧基，C1-C4烷硫基，C1-C4烷基氨基或二（C1-C4烷基）氨基，各自任选被羟基，卤素或C1- C4烷氧基; R2代表氢或卤素，或C1-C4烷基，C1-C4烷氧基，C1-C4烷硫基，C1-C4烷基氨基或二（C1-C4烷基）氨基，各自任选被卤素取代; Ar代表4-氰基-2,5-二氟 - 苯基，2,6-二甲氧基 - 苯基，2-溴-3-三氟 - 甲基 - 苯基，2-溴-5-三氟甲基 - 苯基，6-氯 - 吡啶-3-基 - 甲基或说明书中提到的5-或6-元（杂）环基之一。 本发明还涉及这些物质的盐，一种制备新化合物的方法及其作为植物处理剂的用途。