摘要:
The invention relates to spirohydantoins of the formula I ##STR1## where R.sub.1 and R.sub.2 are defined hereinbelow. Also disclosed are methods of preparation, pharmaceutical compositions containing at least one of these compounds, and methods of using said compounds for treatment and prevention of complications of diabetes and galactosemia.
摘要:
The new amino-alcohol derivatives according to the invention have the formula: ##STR1## wherein: (a) R.sub.1 is hydrogen, an alkylthio C.sub.1 -C.sub.5 radical, a cycloalkylthio C.sub.5 -C.sub.6 radical, an alkoxy C.sub.1 -C.sub.5 radical, a cycloalkyloxy C.sub.5 -C.sub.6 radical, an alkyl C.sub.1 -C.sub.5 radical, a cycloalkyl C.sub.5 -C.sub.6 radical or a halogen atom;(b) R.sub.2 is a lower alkyl C.sub.1 -C.sub.3 radical;(c) R.sub.3 is an alkyl C.sub.1 -C.sub.18 radical, substituted or not, an alkenyl C.sub.6 -C.sub.18 radical substituted or not, a cycloalkyl C.sub.5 -C.sub.9 radical;(d) R.sub.4 is an acyl group having the formula: ##STR2## in which R.sub.5 represents an alkyl C.sub.1 -C.sub.10 substituted or not, an alkenyl C.sub.2 -C.sub.4, a cycloalkyl C.sub.3 -C.sub.8, a phenyl substituted or not or a cinnamyl radical, R.sub.4 being hydrogen if R.sub.1 is hydrogen, an alkyl, alkoxy, cycloalkoxy or cycloalkyl radical or a halogen atom.
摘要:
The circuit disclosed can be used to process synchronous video signals, especially those coming from two standard CCD sensors. It comprises two channels connected at the output to the two inputs, respectively, of an adder circuit which gives the mixed video signal. The first channel comprises a subtractor circuit which receives the two video signals, a high-frequency filter circuit to eliminate the low-frequency spectrum ranging between 0 and a determined limit frequency, an amplifier circuit to balance the gain of the two channels and a fast change-over/sampler circuit connected to the first input of the adder during half of each dot cycle, while the second input of the adder continually receives one of the video signals. The mixed signal thus comprises an unchanged low-frequency component which eliminates faults in the sensors related to non-homogeneity. The high-frequency component recovered corresponds to the first signal during the first half of the dot cycle and to the second signal during the second half of the dot cycle.
摘要:
A bispectral pick-up and false color display system which comprises a bispectral camera for analyzing a picture in the visible range and a picture in the infrared range, and outputting two respective video signals, one for the visible range and one for the infrared range. A mixer then mixes these two video signals and derives, therefrom, three color control signals, each color control signal being a linear combination of the two video signals given by the bispectral camera. A manual setting device then sets or adjusts the coefficients of each of the combinations. A standard color television monitor then can display a picture as a function of the three color control signals. The disclosed device can be applied to target-sighting and target-tracking devices for land vehicles.
摘要:
The new amino-alcohols according to the invention are represented by the formula ##SPC1##Wherein: R.sub.1 represents a RS, RSO or RSO.sub.2 group in which R is a linear or branched alkyl group (C.sub.1 -C.sub.10), an acetyl radical or hydrogen; R.sub.2 and R.sub.3, which may be identical or different, represent a halogen atom or an alkyl (C.sub.1 -C.sub.3), amino, alkylamino (C.sub.1 -C.sub.4), acylamino, nitro, carboxy, carbalkoxy, trifluoromethyl, alkoxy (C.sub.1 -C.sub.4) or alkylthio (C.sub.1 -C.sub.4) radical; R.sub.4 represents hydrogen or a linear or branched alkyl radical containing 1 - 4 carbon atoms; R.sub.5 and R.sub.6, which may be identical or different, represent hydrogen, a substituted or not, linear or branched alkyl (C.sub.1 -C.sub.16) radical, a cycloalkyl (C.sub.5 -C.sub.6) radical, an alkynyl (C.sub.3 -C.sub.4) radical, an alkenyl (C.sub.3 -C.sub.4) radical or a heterocycle of the kind piperidine, morpholine, pyridine or pyridimine, R.sub.5 and R.sub.6 can also form with adjacent nitrogen atom a heterocyclic radical, substituted or not; one of said R.sub.2 and R.sub.3 can be a hydrogen atom or can be both a hydrogen atom provided that simultaneously R is a lower alkyl (C.sub.1 -C.sub.3) radical in the group RS, R.sub.4 and R.sub.5 are hydrogen atoms and R.sub.6 is an isopropyl or t-butyl radical or if simultaneously R is a methyl radical in the group RSO.sub.2, R.sub.4 and R.sub.5 are hydrogen atoms and R.sub.6 is an isopropyl radical.When R.sub.5 and R.sub.6 represent an alkyl, the latter can be substituted by amino, alkylamino, hydroxy, alkoxy, phenoxy, substituted phenoxy, phenyl, substituted phenyl radical or a heterocycle such as piperidino or morpholino.
摘要:
The invention relates to a self-propelled machine with flexible caterpillar treads maintained in position by guide wheels (5-8). The two guide wheels of each end are mounted on a rocker (15-24) whose of oscillation (17,25) is different from the axes of rotation of the wheels carried by it, and at least one of these rockers is equipped with a device (18-23) able to oppose its oscillation movement.