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公开(公告)号:US4818762A
公开(公告)日:1989-04-04
申请号:US815692
申请日:1986-01-02
IPC分类号: A01N43/50 , A01N43/653 , C07D233/56 , C07D233/64 , C07D249/08 , C07D405/06 , C07D521/00
CPC分类号: C07D231/12 , A01N43/50 , A01N43/653 , C07D233/56 , C07D249/08
摘要: Hydroxyalkynyl-azolyl derivatives of the formula ##STR1## in which Az is 1,2,4-triazolyl or imidazolyl,X is optionally substituted phenyl or alkyl,R is ##STR2## R.sup.1 is hydrogen or halogen, R.sup.2 is halogen,R.sup.3 is alkylthio, halogenoalkoxy, halogenoalkylthio, alkenyl, alkoxycarbonyl or cyano, or in each case optionally substituted phenyl, phenoxy, phenylthio, phenylalkoxy or phenylalkylthio,n is 0, 1 or 2,m is 0 or 1, andHet is optionally substituted dioxolanyl or dioxanyl,or an addition product thereof with acids or metal salts, which exhibit fungicidal activity.
摘要翻译: 其中Az是1,2,4-三唑基或咪唑基,X是任选取代的苯基或烷基,R是R 1是氢或卤素,R 2是卤素,R 3是烷硫基 ,卤代烷氧基,卤代烷硫基,烯基,烷氧基羰基或氰基,或在每种情况下任选取代的苯基,苯氧基,苯硫基,苯基烷氧基或苯基烷硫基,n为0,1或2,m为0或1,Het为任选取代的二氧戊环基或二恶烷基, 或其与酸或金属盐的加成产物,其具有杀真菌活性。
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公开(公告)号:US4622333A
公开(公告)日:1986-11-11
申请号:US547806
申请日:1983-11-01
IPC分类号: A01N43/50 , A01N43/653 , C07D233/56 , C07D233/64 , C07D249/08 , C07D405/06 , C07D521/00
CPC分类号: C07D231/12 , A01N43/50 , A01N43/653 , C07D233/56 , C07D249/08
摘要: Hydroxyalkynyl-azolyl derivatives of the formula ##STR1## in which Az is 1,2,4-triazolyl or imidazolyl,X is optionally substituted phenyl or alkyl,R is ##STR2## R.sup.1 is hydrogen or halogen, R.sup.2 is halogen,R.sup.3 is alkylthio, halogenoalkoxy, halogenoalkylthio, alkenyl, alkoxycarbonyl or cyano, or in each case optionally substituted phenyl, phenoxy, phenylthio, phenylalkoxy or phenylalkylthio,n is 0, 1 or 2,m is 0 or 1, andHet is optionally substituted dioxolanyl or dioxanyl,or an addition product thereof with acids or metal salts, which exhibit fungicidal activity.
摘要翻译: 其中Az是1,2,4-三唑基或咪唑基,X是任选取代的苯基或烷基,R是R 1是氢或卤素,R 2是卤素,R 3是烷硫基 ,卤代烷氧基,卤代烷硫基,烯基,烷氧基羰基或氰基,或在每种情况下任选取代的苯基,苯氧基,苯硫基,苯基烷氧基或苯基烷硫基,n为0,1或2,m为0或1,Het为任选取代的二氧戊环基或二恶烷基, 或其与酸或金属盐的加成产物,其具有杀真菌活性。
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公开(公告)号:US5025030A
公开(公告)日:1991-06-18
申请号:US376721
申请日:1989-07-07
申请人: Reinhard Lantzsch , Ernst Kysela , Karl H. Buchel , Stefan Dutzmann , Wilhelm Brandes , Gerd Hanssler
发明人: Reinhard Lantzsch , Ernst Kysela , Karl H. Buchel , Stefan Dutzmann , Wilhelm Brandes , Gerd Hanssler
IPC分类号: A01N43/653 , C07C45/45 , C07C49/567 , C07D249/08 , C07D303/08 , C07D521/00
CPC分类号: C07D249/08 , A01N43/653 , C07C45/455 , C07C49/567 , C07D231/12 , C07D233/56 , C07D303/08
摘要: Novel hydroxyalkinyl-azolyl derivatives of the formula ##STR1## in which Ar represents optionally substituted aryl,R represents alkyl, optionally substituted aryl or optionally substituted aralkyl,X.sup.1 represents halogen,X.sup.2 represents hydrogen or halogen,X.sup.3 represents hydrogen or halogen,X.sup.4 represents hydrogen or halogen andn represents 0 or 1,and acid addition salts and metal salt complexes thereof, are outstandingly effective as fungicides.
摘要翻译: 式(I)的新型羟基烯基 - 唑基衍生物,其中Ar表示任选取代的芳基,R表示烷基,任选取代的芳基或任选取代的芳烷基,X 1表示卤素,X 2表示氢或卤素,X 3表示氢或卤素, X 4表示氢或卤素,n表示0或1,并且其酸加成盐和金属盐络合物作为杀真菌剂显着有效。
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公开(公告)号:US4999440A
公开(公告)日:1991-03-12
申请号:US395233
申请日:1989-08-17
申请人: Graham Holmwood , Udo Kraatz , Karl H. Buchel , Wilhelm Brandes , Stefan Dutzmann , Paul Reinecke
发明人: Graham Holmwood , Udo Kraatz , Karl H. Buchel , Wilhelm Brandes , Stefan Dutzmann , Paul Reinecke
IPC分类号: A01N43/653 , C07C15/44 , C07C25/24 , C07D249/08 , C07D303/06 , C07D303/08 , C07D303/22 , C07D303/34 , C07D303/36 , C07D521/00
CPC分类号: C07D249/08 , A01N43/653 , C07C15/44 , C07C25/24 , C07D231/12 , C07D233/56 , C07D303/08
摘要: Fungicidal hydroxyalkyl-triazdyl derivatives of the formula ##STR1## in which R represents a radical of the formula --CH.sub.2 --CH(CH.sub.3).sub.2, --(CH.sub.2).sub.4 --CH.sub.3, --(CH.sub.2).sub.5 --CH.sub.3, --(CH.sub.2).sub.6 --CH.sub.3, ##STR2## Z represents halogen, alkyl with 1 to 4 carbon atoms, halogenoalkyl with 1 or 2 carbon atoms and 1 to 5 halogen atoms, halogenoalkoxy with 1 or 2 carbon atoms and 1 to 5 halogen atoms, halogenoalkylthio with 1 or 2 carbon atoms and 1 to 5 halogen atoms, phenyl or alkoximinimethyl with 1 to 4 carbon atoms in the alkoxy group andm represents the numbers 0, 1, 2 or 3,and addition products thereof with acids and metal salts. Intermediates of the formulas ##STR3## are also new.
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5.
公开(公告)号:US4878939A
公开(公告)日:1989-11-07
申请号:US258108
申请日:1988-10-13
申请人: Gerhard Jager , Manfred Jautelat , Wolfgang Kramer , Karl H. Buchel , Paul Reinecke , Wilhelm Brandes , Gerd Hanssler , Klaus Lurssen
发明人: Gerhard Jager , Manfred Jautelat , Wolfgang Kramer , Karl H. Buchel , Paul Reinecke , Wilhelm Brandes , Gerd Hanssler , Klaus Lurssen
IPC分类号: C07C43/225 , A01N43/50 , A01N43/653 , C07C41/00 , C07C45/00 , C07C49/167 , C07C49/175 , C07C67/00 , C07D233/60 , C07D249/08 , C07D521/00
CPC分类号: C07D231/12 , A01N43/50 , A01N43/653 , C07D233/56 , C07D249/08
摘要: Azolyl ether ketones and alcohols of the formula ##STR1## in which R.sup.1 and R.sup.2 each independently represents alkyl with more than one carbon atom, orR.sup.1 represents dichloromethyl, trichloromethyl, chlorovinyl or dichlorovinyl, andR.sup.2 represents alkyl,R.sup.3 represents alkyl,A represents the keto group or a CH(OH) grouping,Z represents a nitrogen atom or the CH group,X represents oxygen or sulphur andAr represents optionally substituted phenyl,or addition products thereof with acids and metal salts, are active against fungi and in regulating the growth of plants. New intermediates therefor are also shown.
摘要翻译: 其中R 1和R 2各自独立地表示具有多于一个碳原子的烷基,或者R 1表示二氯甲基,三氯甲基,氯乙烯基或二氯乙烯基,并且R 2表示烷基,R 3表示烷基, 酮基或CH(OH)基,Z表示氮原子或CH基,X表示氧或硫,Ar表示任选取代的苯基,或其与酸和金属盐的加成产物对真菌有活性, 植物生长。 还显示了其新的中间体。
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6.
公开(公告)号:US4875928A
公开(公告)日:1989-10-24
申请号:US792089
申请日:1985-10-28
申请人: Erik Regel , Klaus Bockmann , Karl H. Buchel , Klaus Lurssen , Wilhelm Brandes , Jorg Konze , Paul Reinecke
发明人: Erik Regel , Klaus Bockmann , Karl H. Buchel , Klaus Lurssen , Wilhelm Brandes , Jorg Konze , Paul Reinecke
IPC分类号: A01N43/50 , A01N43/653 , C07D233/60 , C07D249/08 , C07D333/00 , C07D403/06 , C07D405/06 , C07D409/06 , C07D521/00
CPC分类号: C07D231/12 , A01N43/50 , A01N43/653 , C07D233/56 , C07D249/08 , Y02P60/246
摘要: Substituted azolylcyclopropyl-azolylmethyl-carbinol derivatives of the formula ##STR1## in which Ar is optionally substituted aryl or optionally substituted heteroaryl,R is hydrogen, alkyl, alkenyl, alkinyl, trialkylsilyl, optionally substituted phenylalkyl or an acyl radical, andX and Y each independently is a nitrogen atom or a CH group,and addition products thereof with acids and metal salts are effective in regulating plant growth and combating fungi. New intermediates are described, some of which are themselves active.
摘要翻译: 其中Ar是任选取代的芳基或任选取代的杂芳基,R是氢,烷基,烯基,炔基,三烷基甲硅烷基,任选取代的苯基烷基或酰基,以及X和Y各自独立地取代的具有式“IMAGE”的唑基环丙基 - 甲基 - 甲醇衍生物 独立地是氮原子或CH基团,其与酸和金属盐的加成产物在调节植物生长和对抗真菌中是有效的。 描述了新的中间体,其中一些本身是活性的。
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公开(公告)号:US4622335A
公开(公告)日:1986-11-11
申请号:US645464
申请日:1984-09-11
IPC分类号: C07D249/08 , A01N43/50 , A01N43/56 , A01N43/653 , C07C45/43 , C07C45/51 , C07C45/63 , C07C49/255 , C07D20060101 , C07D233/60 , C07D233/61 , C07D521/00
CPC分类号: C07D231/12 , A01N43/50 , A01N43/653 , C07C45/43 , C07C45/515 , C07C45/63 , C07C49/255 , C07D233/56 , C07D249/08
摘要: Fungicidally active novel hydroxyethylazolyl-oxime derivatives of the formula ##STR1## in which Ar is optionally substituted aryl,R.sup.1 is hydrogen or alkyl,R.sup.2 is hydrogen, alkyl, alkenyl, alkinyl, optionally substituted aralkyl or optionally substituted cycloalkylalkyl, andX is a nitrogen atom or the CH group,and addition products thereof with acids and metal salts.
摘要翻译: 其中Ar为任选取代的芳基,R 1为氢或烷基,R 2为氢,烷基,链烯基,炔基,任选取代的芳烷基或任选取代的环烷基烷基,X为氮原子的杀真菌活性的新型羟乙唑基肟衍生物 原子或CH基团,以及其与酸和金属盐的加成产物。
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公开(公告)号:US4618619A
公开(公告)日:1986-10-21
申请号:US589613
申请日:1984-03-14
申请人: Erik Regel , Karl H. Buchel , Paul Reinecke , Wilhelm Brandes
发明人: Erik Regel , Karl H. Buchel , Paul Reinecke , Wilhelm Brandes
IPC分类号: A01N31/14 , A01N31/00 , A01N31/02 , A01N33/04 , A01N33/08 , A01N43/48 , A01N43/50 , A01N43/56 , A01N43/64 , A01N43/653 , C07D249/08 , C07D303/22 , C07D303/24 , C07D303/34 , C07D303/36 , C07D521/00
CPC分类号: C07D303/22 , A01N43/50 , A01N43/56 , A01N43/653 , C07C323/00 , C07D231/12 , C07D233/56 , C07D249/08 , C07D303/24 , C07D303/34 , C07D303/36
摘要: A method of combating plant pathogenic fungi which comprises administering to such fungi or to a habitat thereof a plant pathogenic fungicidally effective amount of a substituted tert.-butanol derivative of the formula ##STR1## in which R.sup.1, R.sup.2 and R.sup.3 are identical or different and represent azolyl, optionally substituted phenoxy, optionally substituted phenylthio, alkylthio, alkenyl, alkinyl, optionally substituted phenylacetylenyl, alkylamino, dialkylamino, optionally substituted phenylamino, optionally substituted phenyl-N-alkyl-amino, optionally substituted cycloalkylamino, optionally substituted cycloalkyl-N-alkyl-amino, aminoethoxy, alkylaminoethoxy or dialkylaminoethyoxy,or an acid addition salt or metal salt complex thereof.
摘要翻译: 一种防治植物致病真菌的方法,其包括向所述真菌或其栖息地施用植物病原真菌有效量的式(I)的取代的叔丁醇衍生物,其中R 1,R 2和R 3相同 任选取代的苯基乙酰基,烷基氨基,二烷基氨基,任选取代的苯基氨基,任选取代的苯基-N-烷基 - 氨基,任选取代的环烷基氨基,任选取代的环烷基 - N-烷基 - 氨基,氨基乙氧基,烷基氨基乙氧基或二烷基氨基乙氧基,或其酸加成盐或金属盐络合物。
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公开(公告)号:US4472416A
公开(公告)日:1984-09-18
申请号:US403988
申请日:1982-08-02
IPC分类号: A01N43/50 , A01N43/653 , C07D233/60 , C07D249/08 , C07D521/00 , A01N43/64 , C07D233/61
CPC分类号: C07D231/12 , C07D233/56 , C07D249/08
摘要: A substituted azolyl-phenoxy derivative of the formula ##STR1## in which A is a nitrogen atom or a CH group,B is a keto group or a CH(OH) grouping,R.sup.1 is an alkyl or halogenoalkyl group of an optionally substituted aryl group,R.sup.2 is a hydrogen atom, an alkyl group or an optionally substituted phenyl group,R.sup.3 is a hydrogen atom, an alkyl, alkenyl or alkinyl group,m is 1 or 2,X is a halogen atom, or an alkyl, alkoxy, alkylthio, halogenoalkyl, halogenoalkoxy or halogenoalkylthio group, andn is 0, 1 or 2,or an addition product thereof with an acid or metal salt, which possesses fungicidal activity particularly for combating cereal diseases as well as rust and scab diseases.
摘要翻译: A为氮原子或CH基团的取代的吡唑基 - 苯氧基衍生物,其中A为氮原子或CH基团,B为酮基或CH(OH)基团,R 1为任选取代的芳基的烷基或卤代烷基 R2是氢原子,烷基或可以具有取代基的苯基,R3是氢原子,烷基,烯基或炔基,m是1或2,X是卤素原子或烷基,烷氧基,烷硫基 ,卤代烷基,卤代烷氧基或卤代烷硫基,n为0,1或2,或其与酸或金属盐的加成产物,其具有特别用于防治谷物疾病以及防锈和痂病的杀真菌活性。
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10.
公开(公告)号:US4917720A
公开(公告)日:1990-04-17
申请号:US256808
申请日:1988-10-12
申请人: Gerhard Jager , Manfred Jautelat , Wolfgang Kramer , Karl H. Buchel , Paul Reinecke , Wilhelm Brandes , Gerd Hanssler , Klaus Lurssen
发明人: Gerhard Jager , Manfred Jautelat , Wolfgang Kramer , Karl H. Buchel , Paul Reinecke , Wilhelm Brandes , Gerd Hanssler , Klaus Lurssen
IPC分类号: C07C43/225 , A01N43/50 , A01N43/653 , C07C41/00 , C07C45/00 , C07C49/167 , C07C49/175 , C07C67/00 , C07D233/60 , C07D249/08 , C07D521/00
CPC分类号: C07D231/12 , A01N43/50 , A01N43/653 , C07D233/56 , C07D249/08
摘要: Azolyl ether ketones and alcohols of the formula ##STR1## in which R.sup.1 and R.sup.2 each independently represents alkyl with more than one carbon atom, orR.sup.1 represents dichloromethyl, trichloromethyl, chlorovinyl or dichlorovinyl, andR.sup.2 represents alkyl,R.sup.3 represents alkyl,A represents the keto group or a CH(OH) grouping,Z represents a nitrogen atom or the CH group,X represents oxygen or sulfur andAr represents optionally substituted phenyl,or addition products thereof with acids and metal salts, are active against fungi and in regulating the growth of plants. New intermediates therefor are also shown.
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