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公开(公告)号:US10100059B2
公开(公告)日:2018-10-16
申请号:US15374386
申请日:2016-12-09
Applicant: Research Triangle Institute
Inventor: Scott P. Runyon , Rangan Maitra , Sanju Narayanan , James Barnwell Thomas , Kenneth S. Rehder , Srinivas Olepu
IPC: C07D491/107 , C07D231/14 , C07D401/12 , C07D401/14 , C07D487/08 , C07D405/12 , C07D417/12 , C07D413/12 , C07D409/04 , C07D403/04 , C07D413/04 , C07D417/04 , C07D403/14 , C07D403/12 , C07D471/08 , A61K45/06 , A61K31/454 , A61K31/415 , A61K31/5377 , A61K31/497 , A61K31/4439 , A61K31/55 , A61K31/427 , A61K31/422 , C07D417/14 , A61K31/4196 , A61K31/4245 , A61K31/439
Abstract: This disclosure is directed to agonists of the apelin receptor (APJ) and uses of such agonists.
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公开(公告)号:US10954247B2
公开(公告)日:2021-03-23
申请号:US15983519
申请日:2018-05-18
Applicant: Research Triangle Institute
Inventor: Scott P. Runyon , Rangan Maitra , Sanju Narayanan , James Barnwell Thomas , Kenneth S. Rehder , Srinivas Olepu
IPC: C07D491/107 , C07D403/04 , A61K31/5377 , C07D401/12 , C07D403/14 , C07D405/12 , C07D417/04 , C07D409/04 , C07D403/12 , C07D417/12 , C07D403/06 , C07D231/14 , C07D471/08 , C07D413/12 , C07D401/14 , C07D417/14 , A61K45/06 , C07D487/08 , C07D407/12 , A61K31/55 , A61K31/427 , A61K31/422 , A61K31/415 , A61K31/4245 , A61K31/4196 , A61K31/454 , A61K31/497 , A61K31/4439 , A61K31/439 , C07D413/04
Abstract: This disclosure is directed to agonists of the apelin receptor (APJ) and uses of such agonists.
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公开(公告)号:US11535630B2
公开(公告)日:2022-12-27
申请号:US17082650
申请日:2020-10-28
Applicant: Research Triangle Institute
Inventor: Scott P. Runyon , Rangan Maitra , Sanju Narayanan , James Barnwell Thomas , Kenneth S. Rehder , Srinivas Olepu
IPC: C07D491/107 , C07D403/12 , C07D231/14 , C07D403/06 , C07D407/12 , C07D413/12 , A61K31/415 , A61K31/4196 , A61K31/422 , A61K31/4245 , A61K31/427 , A61K31/439 , A61K31/4439 , A61K31/454 , A61K31/497 , A61K31/5377 , A61K31/55 , A61K45/06 , C07D401/12 , C07D401/14 , C07D405/12 , C07D409/04 , C07D413/04 , C07D417/04 , C07D417/12 , C07D417/14 , C07D471/08 , C07D487/08 , C07D403/04 , C07D403/14
Abstract: This disclosure is directed to agonists of the apelin receptor (APJ) and uses of such agonists.
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公开(公告)号:US20160207889A1
公开(公告)日:2016-07-21
申请号:US15023510
申请日:2015-06-05
Applicant: Scott P. RUNYON , Rangan MAITRA , Sanju NARAYANAN , James Barnwell THOMAS , RESEARCH TRIANGLE INSTITUTE
Inventor: Scott P. Runyon , Rangan Maitra , Sanju Narayanan , James Barnwell Thomas
IPC: C07D231/14 , A61K45/06 , A61K31/415 , C07D405/12 , A61K31/422 , A61K31/454 , A61K31/4155 , A61K31/496 , C07D413/12
CPC classification number: C07D231/14 , A61K31/415 , A61K31/4155 , A61K31/422 , A61K31/454 , A61K31/496 , A61K45/06 , C07D403/06 , C07D403/12 , C07D405/12 , C07D407/12 , C07D413/12
Abstract: This disclosure is directed to agonists of the apelin receptor (APJ) and uses of such agonists.
Abstract translation: 本公开涉及apelin受体(APJ)的激动剂和这种激动剂的用途。
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公开(公告)号:USRE49594E1
公开(公告)日:2023-08-01
申请号:US16974363
申请日:2020-05-04
Applicant: Research Triangle Institute
Inventor: Scott P. Runyon , Rangan Maitra , Sanju Narayanan , James Barnwell Thomas , Kenneth S. Rehder , Srinivas Olepu
IPC: C07D491/107 , C07D403/12 , C07D231/14 , C07D403/06 , C07D407/12 , C07D413/12 , A61K31/415 , A61K31/4196 , A61K31/422 , A61K31/4245 , A61K31/427 , A61K31/439 , A61K31/4439 , A61K31/454 , A61K31/497 , A61K31/5377 , A61K31/55 , A61K45/06 , C07D401/12 , C07D401/14 , C07D403/04 , C07D403/14 , C07D405/12 , C07D409/04 , C07D413/04 , C07D417/04 , C07D417/12 , C07D417/14 , C07D471/08 , C07D487/08
CPC classification number: C07D491/107 , A61K31/415 , A61K31/4196 , A61K31/422 , A61K31/427 , A61K31/4245 , A61K31/439 , A61K31/4439 , A61K31/454 , A61K31/497 , A61K31/5377 , A61K31/55 , A61K45/06 , C07D231/14 , C07D401/12 , C07D401/14 , C07D403/04 , C07D403/06 , C07D403/12 , C07D403/14 , C07D405/12 , C07D407/12 , C07D409/04 , C07D413/04 , C07D413/12 , C07D417/04 , C07D417/12 , C07D417/14 , C07D471/08 , C07D487/08
Abstract: This disclosure is directed to agonists of the apelin receptor (APJ) and uses of such agonists.
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公开(公告)号:US11267789B2
公开(公告)日:2022-03-08
申请号:US16448976
申请日:2019-06-21
Applicant: Research Triangle Institute
Inventor: Scott P. Runyon , Rangan Maitra , Sanju Narayanan , James Barnwell Thomas
IPC: C07D231/14 , C07D405/12 , A61K45/06 , A61K31/415 , A61K31/4155 , A61K31/422 , C07D403/12 , A61K31/496 , C07D413/12 , C07D407/12 , C07D403/06 , A61K31/454
Abstract: This disclosure is directed to agonists of the apelin receptor (APJ) and uses of such agonists.
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公开(公告)号:US10377718B2
公开(公告)日:2019-08-13
申请号:US15023510
申请日:2015-06-05
Applicant: Research Triangle Institute , Scott P. Runyon , Rangan Maitra , Sanju Narayanan , James Barnwell Thomas
Inventor: Scott P. Runyon , Rangan Maitra , Sanju Narayanan , James Barnwell Thomas
IPC: C07D231/14 , A61K45/06 , A61K31/415 , C07D405/12 , A61K31/422 , A61K31/454 , A61K31/4155 , A61K31/496 , C07D413/12 , C07D403/12 , C07D403/06 , C07D407/12
Abstract: This disclosure is directed to agonists of the apelin receptor (APJ) and uses of such agonists.
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公开(公告)号:US20170166577A1
公开(公告)日:2017-06-15
申请号:US15374386
申请日:2016-12-09
Applicant: Research Triangle Institute
Inventor: Scott P. Runyon , Rangan Maitra , Sanju Narayanan , James Barnwell Thomas , Kenneth S. Rehder , Srinivas Olepu
IPC: C07D491/107 , A61K31/454 , C07D231/14 , A61K31/415 , A61K31/5377 , A61K31/497 , A61K31/4439 , C07D401/12 , C07D401/14 , A61K31/55 , C07D487/08 , C07D405/12 , A61K31/427 , C07D417/12 , A61K31/422 , C07D413/12 , C07D409/04 , C07D403/04 , C07D413/04 , C07D417/04 , C07D417/14 , A61K31/4196 , A61K31/4245 , C07D403/14 , C07D403/12 , A61K31/439 , C07D471/08 , A61K45/06
CPC classification number: C07D491/107 , A61K31/415 , A61K31/4196 , A61K31/422 , A61K31/4245 , A61K31/427 , A61K31/439 , A61K31/4439 , A61K31/454 , A61K31/497 , A61K31/5377 , A61K31/55 , A61K45/06 , C07D231/14 , C07D401/12 , C07D401/14 , C07D403/04 , C07D403/06 , C07D403/12 , C07D403/14 , C07D405/12 , C07D407/12 , C07D409/04 , C07D413/04 , C07D413/12 , C07D417/04 , C07D417/12 , C07D417/14 , C07D471/08 , C07D487/08
Abstract: This disclosure is directed to agonists of the apelin receptor (APJ) and uses of such agonists.
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