Azolyl derivatives of carbocyclic and heterocyclic ketones having
fungicidal activity
    1.
    发明授权
    Azolyl derivatives of carbocyclic and heterocyclic ketones having fungicidal activity 失效
    具有杀真菌活性的碳环和杂环酮的唑基衍生物

    公开(公告)号:US4725614A

    公开(公告)日:1988-02-16

    申请号:US802001

    申请日:1985-12-03

    摘要: There are disclosed compounds having general formula (I): ##STR1## wherein: X is H, a phenyl, phenylalkyl, phenylcarbonyl, phenyloxy group, optionally substituted with a halogen; Y is N or CH; R.sup.1 is H or a phenyl group; R.sup.2 and R.sup.3, equal or different, are H, an alkyl, alkoxy group or together they are an atom of ketonic oxygen; R.sup.4 and R.sup.5, equal or different, are H or an alkyl group; R.sup.6 and R.sup.7, equal or different, are H, an alkyl group or one of them forms with R.sup.2 or R.sup.3 an alkylidenic or etheric bridge; or they form a dioxyalkylidenic or alkylidenic ring; m=0, 1; n=0, 1, 2, 3. The compounds are endowed with fungicide and systemic properties.

    摘要翻译: 公开了具有通式(I)的化合物:其中:X为H,苯基,苯基烷基,苯基羰基,苯氧基,任选被卤素取代; Y为N或CH; R1是H或苯基; R2和R3相同或不同,是H,烷基,烷氧基或它们一起是酮氧原子; R4和R5相同或不同,为H或烷基; R6和R7相同或不同,为H,烷基或其中一个与R2或R3形成亚烷基或醚桥; 或它们形成二环烯基或亚烷基环; m = 0,1, 这些化合物具有杀真菌剂和系统性质。

    Azolyl-derivatives endowed with antifungal activity
    2.
    发明授权
    Azolyl-derivatives endowed with antifungal activity 失效
    具有抗真菌活性的唑基衍生物

    公开(公告)号:US5036094A

    公开(公告)日:1991-07-30

    申请号:US408945

    申请日:1989-09-18

    摘要: Disclosed are compounds, having the general formula: ##STR1## wherein: m=0, 1, 2; n=0, 1 with the condition that when m=0, also n=0;p=0, 1; q=1, 2;X is either oxygen or sulphur;A=N, CH;R is H, CH.sub.3, F;R.sub.1 is selected from chlorine, bromine, fluorine, CF.sub.3, phe=nyl, C.sub.1 -C.sub.2 -alkoxy, C.sub.1 -C.sub.2 -haloalkoxy, alkylthio, haloalkyl=thio, wherein the halogen is Cl, Br, F;R.sub.2 is selected from H, chlorine, bromine, fluorine;R.sub.f is selected from the group formed by alkyls containing from 2 to 4 carbon atoms, and containing at least 4 atoms of halogen selected from F, Cl and Br, of which at least 3 are F atoms; alkenyls and alkynyls containing up to 4 carbon atoms, containing at least 2 F atoms and, optionally, other halogens selected between Cl and Br.The present invention relates to azolyl-derivatives, more particularly to substituted azolyldioxanes and azolyldioxolanes, endowed with high fungicidal activity, to the process for their preparation, and to their related use in the agrarian field.

    摘要翻译: 公开了具有以下通式的化合物:其中:m = 0,1,2; n = 0,1,条件是当m = 0时,n = 0; p = 0,1, q = 1,2; X是氧或硫; A = N,CH; R为H,CH 3,F; R 1选自氯,溴,氟,CF 3,phe = nyl,C 1 -C 2 - 烷氧基,C 1 -C 2卤代烷氧基,烷硫基,卤代烷基=硫代,其中卤素是Cl,Br,F; R2选自H,氯,溴,氟; Rf选自由含有2至4个碳原子的烷基形成的基团,并且含有至少4个选自F,Cl和Br的卤素,其中至少3个是F原子; 含有至多4个碳原子的烯基和炔基,其含有至少2个F原子,以及任选的选自Cl和Br之间的其它卤素。 本发明涉及唑类衍生物,更具体地涉及具有高杀真菌活性的取代的azolyldioxanes和azolyldioxolanes,其制备方法及其在土地领域的相关用途。

    Fungicidal azolyl-derivatives
    4.
    发明授权
    Fungicidal azolyl-derivatives 失效
    真菌化合物衍生物

    公开(公告)号:US5081141A

    公开(公告)日:1992-01-14

    申请号:US549648

    申请日:1990-07-06

    摘要: Disclosed are compounds having the formula: ##STR1## wherein: m=0, 1;n=0, 1;Z=CH, N;R.sub.1 is selected from chlorine, bromine, fluorine, CF.sub.3, phenyl, C.sub.1 -C.sub.2 -alkoxy, C.sub.1 -C.sub.2 -haloalkoxy, alkylthio, and haloalkylthio, wherein the halogen is Cl, Br, F;R.sub.2 is H, fluorine, chlorine, or bromine;R.sub.3 represents H, CH.sub.3, CN, or also F when m=1 or when n=1 and R.sub.4, R.sub.5 are H;R.sub.4, R.sub.5 are independently H or F;R.sub.3 and R.sub.4, furthermore, when m=0, may represent, taken together, a second bond between the two carbon atoms to which they are linked in formula (I); andR.sub.f is selected from the group consisting of polyfluoroalkyls, polyfluoroalkenyls and polyfluoroalkynyls containing up to 4 carbon atoms, containing at least 2 F atoms and, optionally, other halogens selected from Cl and Br.Anti-fungal compositions containing these new compounds.

    摘要翻译: 公开了具有下式的化合物:其中:m = 0,1; n = 0,1; Z = CH,N; R1选自氯,溴,氟,CF3,苯基,C1-C2-烷氧基,C1-C2-卤代烷氧基,烷硫基和卤代烷硫基,其中卤素为Cl,Br,F; R2是H,氟,氯或溴; 当m = 1或当n = 1且R 4,R 5为H时,R 3表示H,CH 3,CN或F。 R4,R5独立地为H或F; 此外,当m = 0时,R 3和R 4可以一起表示在式(I)中它们连接的两个碳原子之间的第二键; 并且Rf选自包含至少2个F原子的含有至多4个碳原子的多氟烷基,多氟烯基和多氟炔基,以及任选的选自Cl和Br的其它卤素。 含有这些新化合物的抗真菌组合物。

    Triazolyl-keto-derivatives endowed with a fungicidal activity
    6.
    发明授权
    Triazolyl-keto-derivatives endowed with a fungicidal activity 失效
    具有杀真菌活性的三唑基 - 酮衍生物

    公开(公告)号:US4704398A

    公开(公告)日:1987-11-03

    申请号:US687282

    申请日:1984-12-28

    摘要: Described herein are .alpha.-(1-triazolyl)-keto-derivatives of general formula: ##STR1## wherein R is phenyl or heteroaryl, optionally substituted, alkyl; R.sup.1 is alkoxyl, optionally substituted aryloxy, alkyl, alkenyl, alkynyl, alkoxyalkyl, alkoxycarbonyl, cyano, optionally substituted phenyl, or, along with R.sup.2, an alkylidene; R.sup.2 is H or, along with R.sup.1, an alkylidene; R.sup.3 is alkylcarbonyl, alkoxycarbonyl, arylcarbonyl, cyano or alkoxyalkylcarbonyl; such compounds being endowed with a high fungicidal activity.

    摘要翻译: 本文描述的是以下通式的α-(1-三唑基) - 酮衍生物:其中R是苯基或杂芳基,任选取代的烷基; R 1为烷氧基,任选取代的芳氧基,烷基,烯基,炔基,烷氧基烷基,烷氧基羰基,氰基,任选取代的苯基,或与R 2一起为亚烷基; R2是H或与R1一起是亚烷基; R3是烷基羰基,烷氧基羰基,芳基羰基,氰基或烷氧基烷基羰基; 这种化合物被赋予高杀真菌活性。