Azolyl-derivatives endowed with antifungal activity
    2.
    发明授权
    Azolyl-derivatives endowed with antifungal activity 失效
    具有抗真菌活性的唑基衍生物

    公开(公告)号:US5036094A

    公开(公告)日:1991-07-30

    申请号:US408945

    申请日:1989-09-18

    摘要: Disclosed are compounds, having the general formula: ##STR1## wherein: m=0, 1, 2; n=0, 1 with the condition that when m=0, also n=0;p=0, 1; q=1, 2;X is either oxygen or sulphur;A=N, CH;R is H, CH.sub.3, F;R.sub.1 is selected from chlorine, bromine, fluorine, CF.sub.3, phe=nyl, C.sub.1 -C.sub.2 -alkoxy, C.sub.1 -C.sub.2 -haloalkoxy, alkylthio, haloalkyl=thio, wherein the halogen is Cl, Br, F;R.sub.2 is selected from H, chlorine, bromine, fluorine;R.sub.f is selected from the group formed by alkyls containing from 2 to 4 carbon atoms, and containing at least 4 atoms of halogen selected from F, Cl and Br, of which at least 3 are F atoms; alkenyls and alkynyls containing up to 4 carbon atoms, containing at least 2 F atoms and, optionally, other halogens selected between Cl and Br.The present invention relates to azolyl-derivatives, more particularly to substituted azolyldioxanes and azolyldioxolanes, endowed with high fungicidal activity, to the process for their preparation, and to their related use in the agrarian field.

    摘要翻译: 公开了具有以下通式的化合物:其中:m = 0,1,2; n = 0,1,条件是当m = 0时,n = 0; p = 0,1, q = 1,2; X是氧或硫; A = N,CH; R为H,CH 3,F; R 1选自氯,溴,氟,CF 3,phe = nyl,C 1 -C 2 - 烷氧基,C 1 -C 2卤代烷氧基,烷硫基,卤代烷基=硫代,其中卤素是Cl,Br,F; R2选自H,氯,溴,氟; Rf选自由含有2至4个碳原子的烷基形成的基团,并且含有至少4个选自F,Cl和Br的卤素,其中至少3个是F原子; 含有至多4个碳原子的烯基和炔基,其含有至少2个F原子,以及任选的选自Cl和Br之间的其它卤素。 本发明涉及唑类衍生物,更具体地涉及具有高杀真菌活性的取代的azolyldioxanes和azolyldioxolanes,其制备方法及其在土地领域的相关用途。

    Azolyl-derivatives having fungicidal activity
    5.
    发明授权
    Azolyl-derivatives having fungicidal activity 失效
    具有杀真菌活性的唑基衍生物

    公开(公告)号:US4810718A

    公开(公告)日:1989-03-07

    申请号:US74352

    申请日:1987-07-16

    摘要: Compounds having the formula: ##STR1## wherein: m=1 or 2;q=1 or 2;Y=a haloethylene or haloethenyl group;X is oxygen or sulfur;A=N or CH;R is H, CH.sub.3 or F;R.sub.1 is selected from the group comprising chlorine, bromine, fluorine CF.sub.3, phenyl, C.sub.1 -C.sub.2 alkoxy, C.sub.1 -C.sub.2 haloalkoxy, alkylthio, haloalkylthio radical, wherein the halogen is Cl, Br or F;R.sub.2 is selected from the group comprising H, chlorine, bromine or fluorine; andR.sub.f is a C.sub.1 -C.sub.5 polyfluoroalkyl or a C.sub.2 -C.sub.4 polyfluoroalkenyl radical containing at least 3 fluorine atoms and, optionally, other halogen atoms selected from the group comprising Cl and Br. These compounds have good fungicidal activity.

    摘要翻译: 具有下式的化合物:其中:m = 1或2; q = 1或2; Y =卤代乙烯基或卤代乙烯基; X是氧或硫; A = N或CH; R为H,CH 3或F; R 1选自氯,溴,氟CF 3,苯基,C 1 -C 2烷氧基,C 1 -C 2卤代烷氧基,烷硫基,卤代烷硫基,其中卤素是Cl,Br或F; R2选自H,氯,溴或氟; 并且Rf是含有至少3个氟原子的C1-C5多氟烷基或C2-C4多氟烯基,以及任选的选自Cl和Br的其它卤素原子。 这些化合物具有良好的杀真菌活性。

    Fungicidal azolyl-derivatives
    6.
    发明授权
    Fungicidal azolyl-derivatives 失效
    真菌化合物衍生物

    公开(公告)号:US5081141A

    公开(公告)日:1992-01-14

    申请号:US549648

    申请日:1990-07-06

    摘要: Disclosed are compounds having the formula: ##STR1## wherein: m=0, 1;n=0, 1;Z=CH, N;R.sub.1 is selected from chlorine, bromine, fluorine, CF.sub.3, phenyl, C.sub.1 -C.sub.2 -alkoxy, C.sub.1 -C.sub.2 -haloalkoxy, alkylthio, and haloalkylthio, wherein the halogen is Cl, Br, F;R.sub.2 is H, fluorine, chlorine, or bromine;R.sub.3 represents H, CH.sub.3, CN, or also F when m=1 or when n=1 and R.sub.4, R.sub.5 are H;R.sub.4, R.sub.5 are independently H or F;R.sub.3 and R.sub.4, furthermore, when m=0, may represent, taken together, a second bond between the two carbon atoms to which they are linked in formula (I); andR.sub.f is selected from the group consisting of polyfluoroalkyls, polyfluoroalkenyls and polyfluoroalkynyls containing up to 4 carbon atoms, containing at least 2 F atoms and, optionally, other halogens selected from Cl and Br.Anti-fungal compositions containing these new compounds.

    摘要翻译: 公开了具有下式的化合物:其中:m = 0,1; n = 0,1; Z = CH,N; R1选自氯,溴,氟,CF3,苯基,C1-C2-烷氧基,C1-C2-卤代烷氧基,烷硫基和卤代烷硫基,其中卤素为Cl,Br,F; R2是H,氟,氯或溴; 当m = 1或当n = 1且R 4,R 5为H时,R 3表示H,CH 3,CN或F。 R4,R5独立地为H或F; 此外,当m = 0时,R 3和R 4可以一起表示在式(I)中它们连接的两个碳原子之间的第二键; 并且Rf选自包含至少2个F原子的含有至多4个碳原子的多氟烷基,多氟烯基和多氟炔基,以及任选的选自Cl和Br的其它卤素。 含有这些新化合物的抗真菌组合物。

    Benzophenones having an antifungal activity
    9.
    发明授权
    Benzophenones having an antifungal activity 失效
    具有抗真菌活性的二苯甲酮

    公开(公告)号:US5464836A

    公开(公告)日:1995-11-07

    申请号:US131880

    申请日:1993-10-05

    摘要: A description follows of benzophenones having an antifungal activity and responding to the general formula (I): ##STR1## wherein: R.sub.1 and R.sub.2, the same or different, represent C.sub.1 -C.sub.6 alkyl groups, C.sub.7 -C.sub.10 arylalkyl groups; or R.sub.1 and R.sub.2, considered jointly with N, represent a C.sub.3 -C.sub.8 heterocyclic group or a C.sub.2 -C.sub.7 heterocyclic group containing a second hetero-atom selected from O and S, said heterocyclic groups being optionally subsituted with one or more C.sub.1 -C.sub.4 alkyl groups;R.sub.3 and R.sub.4, the same or different, represent H atoms, C.sub.1 -C.sub.3 alkyl groups;K represents an oxygen atom or methylene;A represents a benzene group, optionally sustituted with one or more halogen atoms, C.sub.1 -C.sub.4 alkyl or haloalkyl groups, C.sub.1 -C.sub.4 alkoxylics, C.sub.1 -C.sub.4 haloalkoxylics;Y represents a C.sub.6 -C.sub.10 aryl group; said group may be optionally substituted with one or more halogen atomos, C.sub.1 -C.sub.4 alkyl or haloalkyl groups, C.sub.1 -C.sub.4 alkoxylics, C.sub.1 -C.sub.4 haloalkoxylics.

    摘要翻译: 以下描述具有抗真菌活性并对应于通式(I)的二苯甲酮:其中:R1和R2相同或不同,表示C1-C6烷基,C7-C10芳基烷基; 或与N一起考虑的R 1和R 2表示含有选自O和S的第二杂原子的C 3 -C 8杂环基或C 2 -C 7杂环基,所述杂环基任选被一个或多个C 1 -C 4烷基取代 团体 R3和R4相同或不同,表示H原子,C1-C3烷基; K表示氧原子或亚甲基; A表示任选被一个或多个卤素原子取代的苯基,C 1 -C 4烷基或卤代烷基,C 1 -C 4烷氧基,C 1 -C 4卤代烷氧基; Y表示C6-C10芳基; 所述基团可以任选地被一个或多个卤素原子,C 1 -C 4烷基或卤代烷基,C 1 -C 4烷氧基,C 1 -C 4卤代烷氧基取代。