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公开(公告)号:US5021442A
公开(公告)日:1991-06-04
申请号:US267317
申请日:1988-11-04
IPC分类号: A01N43/653 , A01N43/50 , A01P3/00 , C07C323/52 , C07D233/60 , C07D233/61 , C07D249/08 , C07D521/00
CPC分类号: C07D231/12 , A01N43/653 , C07C323/52 , C07D233/56 , C07D249/08
摘要: There are described compounds having general formula: ##STR1## wherein: R.sup.1 is selected from the group comprising F, Cl, Br, CF.sub.3, a phenyl, a C.sub.1 -C.sub.2 alkoxy, a C.sub.1 -C.sub.2 haloalkoxy, an alkylthio, a haloalkylthio radical, in which the halogen is F, Cl, Br;R.sup.2 is selected from the group comprising H, F, Cl, Br, CF.sub.3 ;R.sup.3, R.sup.4 and R.sup.5, which may be the same or different, are H, a C.sub.1 -C.sub.4 alkyl or a C.sub.3 -C.sub.6 cycloalkyl radical, on condition that R.sup.5 is different from R.sup.3, when R.sup.4 is H;Y is selected from the group comprising H, CH.sub.3, OH, CN, F;n is 1,2;m is 0,1;X is O or S;Rf is selected from the group consisting of C.sub.1 -C.sub.5 polyfluoroalkyl, C.sub.2 -C.sub.4 polyfluoroalkenyl, polyfluoroalkoxyalkyl and polyfluoroalkoxyalkenyl radicals, everyone of them containing at least two fluorine atoms and, optionally, other halogen atoms selected from Cl and Br;Z is CH or N.
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公开(公告)号:US5036094A
公开(公告)日:1991-07-30
申请号:US408945
申请日:1989-09-18
申请人: Roberto Colle , Giovanni Camaggi , Franco Gozzo , Giuseppina Ratti , Luigi Mirenna , Carlo Garavaglia
发明人: Roberto Colle , Giovanni Camaggi , Franco Gozzo , Giuseppina Ratti , Luigi Mirenna , Carlo Garavaglia
IPC分类号: C07D317/00 , A01N43/50 , A01N43/653 , A01P3/00 , A61K20060101 , C07D20060101 , C07D249/08 , C07D317/22 , C07D405/06 , C07D409/06 , C07D521/00
CPC分类号: C07D231/12 , A01N43/50 , A01N43/653 , C07D233/56 , C07D249/08 , C07D317/22
摘要: Disclosed are compounds, having the general formula: ##STR1## wherein: m=0, 1, 2; n=0, 1 with the condition that when m=0, also n=0;p=0, 1; q=1, 2;X is either oxygen or sulphur;A=N, CH;R is H, CH.sub.3, F;R.sub.1 is selected from chlorine, bromine, fluorine, CF.sub.3, phe=nyl, C.sub.1 -C.sub.2 -alkoxy, C.sub.1 -C.sub.2 -haloalkoxy, alkylthio, haloalkyl=thio, wherein the halogen is Cl, Br, F;R.sub.2 is selected from H, chlorine, bromine, fluorine;R.sub.f is selected from the group formed by alkyls containing from 2 to 4 carbon atoms, and containing at least 4 atoms of halogen selected from F, Cl and Br, of which at least 3 are F atoms; alkenyls and alkynyls containing up to 4 carbon atoms, containing at least 2 F atoms and, optionally, other halogens selected between Cl and Br.The present invention relates to azolyl-derivatives, more particularly to substituted azolyldioxanes and azolyldioxolanes, endowed with high fungicidal activity, to the process for their preparation, and to their related use in the agrarian field.
摘要翻译: 公开了具有以下通式的化合物:其中:m = 0,1,2; n = 0,1,条件是当m = 0时,n = 0; p = 0,1, q = 1,2; X是氧或硫; A = N,CH; R为H,CH 3,F; R 1选自氯,溴,氟,CF 3,phe = nyl,C 1 -C 2 - 烷氧基,C 1 -C 2卤代烷氧基,烷硫基,卤代烷基=硫代,其中卤素是Cl,Br,F; R2选自H,氯,溴,氟; Rf选自由含有2至4个碳原子的烷基形成的基团,并且含有至少4个选自F,Cl和Br的卤素,其中至少3个是F原子; 含有至多4个碳原子的烯基和炔基,其含有至少2个F原子,以及任选的选自Cl和Br之间的其它卤素。 本发明涉及唑类衍生物,更具体地涉及具有高杀真菌活性的取代的azolyldioxanes和azolyldioxolanes,其制备方法及其在土地领域的相关用途。
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公开(公告)号:US4929631A
公开(公告)日:1990-05-29
申请号:US133602
申请日:1987-12-16
申请人: Roberto Colle , Giovanni Camaggi , Franco Gozzo , Giuseppina Ratti , Carlo Garavaglia , Luigi Mirenna
发明人: Roberto Colle , Giovanni Camaggi , Franco Gozzo , Giuseppina Ratti , Carlo Garavaglia , Luigi Mirenna
IPC分类号: A01N43/50 , A01N43/653 , C07D233/60 , C07D233/61 , C07D249/08 , C07D521/00
CPC分类号: C07D231/12 , A01N43/50 , A01N43/653 , C07D233/56 , C07D249/08
摘要: Fungicidal compounds having the formula: ##STR1## wherein: R.sup.1 is selected from the group consisting of F, Cl, Br, CF.sub.3, a phenyl, a C.sub.1 -C.sub.2 alkoxy, a C.sub.1 -C.sub.2 haloalkoxy, an alkylthio, and a haloalkylthio radical, in which the halogen is F, Cl, or Br;R.sup.2 is selected from the group consisting of H, F, Cl, Br, and CF.sub.3 ;R.sup.3 is H, a C.sub.1 -C.sub.4 alkyl or a C.sub.3 -C.sub.6 cycloalkyl radical;Y is selected from the group consisting of H, CH.sub.3, OH, CN, and F;n is 1, 2, 3, 4 with the proviso that Y is OH when n is 1;m is 0 or 1;X is O or S;Rf is selected from the group consisting of C.sub.1 -C.sub.5 polyfluoroalkyl, C.sub.2 -C.sub.4 polyfluoroalkenyl, polyfluoroalkoxyalkyl and polyfluoroalkoxyalkenyl radicals, each one of them containing at least two fluorine atoms and, optionally, other halogen atoms selected from the group consisting of Cl and Br; andZ is CH or N.
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公开(公告)号:US4940724A
公开(公告)日:1990-07-10
申请号:US310338
申请日:1989-02-14
IPC分类号: A01N43/50 , A01N43/653 , A01N47/02 , C07D317/22 , C07D405/06 , C07D413/06 , C07D417/06 , C07D521/00
CPC分类号: C07D249/08 , A01N43/653 , A01N47/02 , C07D231/12 , C07D233/56 , C07D317/22
摘要: Compounds having the formula: ##STR1## wherein: m=1 or 2;q=1 or 2;Y=a haloethylene or haloethenyl group;X is oxygen or sulfur;A=N or CH;R is H, CH.sub.3 or F;R.sub.1 is selected from the group comprising chlorine, bromine, fluorine, CF.sub.3, phenyl, C.sub.1 -C.sub.2 alkoxy, C.sub.1 -C.sub.2 haloalkoxy, alkylthio, haloalkylthio radical, wherein the halogen is Cl, Br or F;R.sub.2 is selected from the group comprising H, chlorine, bromine or fluorine; andR.sub.f is a C.sub.1 -C.sub.5 polyfluoroalkyl or a C.sub.2 -C.sub.4 polyfluoroalkenyl radical containing at least 3 fluorine aotms and, optionally, other halogen atoms selected from the group comprising Cl and Br. These compounds have good fungicidal activity.
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公开(公告)号:US4810718A
公开(公告)日:1989-03-07
申请号:US74352
申请日:1987-07-16
IPC分类号: A01N43/50 , A01N43/653 , A01N47/02 , C07D317/22 , C07D405/06 , C07D413/06 , C07D417/06 , C07D521/00 , C07D249/12
CPC分类号: C07D249/08 , A01N43/653 , A01N47/02 , C07D231/12 , C07D233/56 , C07D317/22
摘要: Compounds having the formula: ##STR1## wherein: m=1 or 2;q=1 or 2;Y=a haloethylene or haloethenyl group;X is oxygen or sulfur;A=N or CH;R is H, CH.sub.3 or F;R.sub.1 is selected from the group comprising chlorine, bromine, fluorine CF.sub.3, phenyl, C.sub.1 -C.sub.2 alkoxy, C.sub.1 -C.sub.2 haloalkoxy, alkylthio, haloalkylthio radical, wherein the halogen is Cl, Br or F;R.sub.2 is selected from the group comprising H, chlorine, bromine or fluorine; andR.sub.f is a C.sub.1 -C.sub.5 polyfluoroalkyl or a C.sub.2 -C.sub.4 polyfluoroalkenyl radical containing at least 3 fluorine atoms and, optionally, other halogen atoms selected from the group comprising Cl and Br. These compounds have good fungicidal activity.
摘要翻译: 具有下式的化合物:其中:m = 1或2; q = 1或2; Y =卤代乙烯基或卤代乙烯基; X是氧或硫; A = N或CH; R为H,CH 3或F; R 1选自氯,溴,氟CF 3,苯基,C 1 -C 2烷氧基,C 1 -C 2卤代烷氧基,烷硫基,卤代烷硫基,其中卤素是Cl,Br或F; R2选自H,氯,溴或氟; 并且Rf是含有至少3个氟原子的C1-C5多氟烷基或C2-C4多氟烯基,以及任选的选自Cl和Br的其它卤素原子。 这些化合物具有良好的杀真菌活性。
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公开(公告)号:US5081141A
公开(公告)日:1992-01-14
申请号:US549648
申请日:1990-07-06
申请人: Roberto Colle , Francesco Corda , Giovanni Camaggi , Franco Gozzo , Luigi Mirenna , Carlo Garavaglia
发明人: Roberto Colle , Francesco Corda , Giovanni Camaggi , Franco Gozzo , Luigi Mirenna , Carlo Garavaglia
IPC分类号: C07D249/12 , A01N43/50 , A01N43/653 , A01P3/00 , C07C67/343 , C07C253/00 , C07D233/56 , C07D233/60 , C07D233/61 , C07D249/08 , C07D521/00
CPC分类号: C07D231/12 , A01N43/50 , A01N43/653 , C07C255/00 , C07D233/56 , C07D249/08
摘要: Disclosed are compounds having the formula: ##STR1## wherein: m=0, 1;n=0, 1;Z=CH, N;R.sub.1 is selected from chlorine, bromine, fluorine, CF.sub.3, phenyl, C.sub.1 -C.sub.2 -alkoxy, C.sub.1 -C.sub.2 -haloalkoxy, alkylthio, and haloalkylthio, wherein the halogen is Cl, Br, F;R.sub.2 is H, fluorine, chlorine, or bromine;R.sub.3 represents H, CH.sub.3, CN, or also F when m=1 or when n=1 and R.sub.4, R.sub.5 are H;R.sub.4, R.sub.5 are independently H or F;R.sub.3 and R.sub.4, furthermore, when m=0, may represent, taken together, a second bond between the two carbon atoms to which they are linked in formula (I); andR.sub.f is selected from the group consisting of polyfluoroalkyls, polyfluoroalkenyls and polyfluoroalkynyls containing up to 4 carbon atoms, containing at least 2 F atoms and, optionally, other halogens selected from Cl and Br.Anti-fungal compositions containing these new compounds.
摘要翻译: 公开了具有下式的化合物:其中:m = 0,1; n = 0,1; Z = CH,N; R1选自氯,溴,氟,CF3,苯基,C1-C2-烷氧基,C1-C2-卤代烷氧基,烷硫基和卤代烷硫基,其中卤素为Cl,Br,F; R2是H,氟,氯或溴; 当m = 1或当n = 1且R 4,R 5为H时,R 3表示H,CH 3,CN或F。 R4,R5独立地为H或F; 此外,当m = 0时,R 3和R 4可以一起表示在式(I)中它们连接的两个碳原子之间的第二键; 并且Rf选自包含至少2个F原子的含有至多4个碳原子的多氟烷基,多氟烯基和多氟炔基,以及任选的选自Cl和Br的其它卤素。 含有这些新化合物的抗真菌组合物。
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公开(公告)号:US5334605A
公开(公告)日:1994-08-02
申请号:US14131
申请日:1993-02-05
申请人: Giovanni Camaggi , Lucio Filippini , Marilena Gusmeroli , Raul Riva , Carlo Garavaglia , Luigi Mirenna , Luigi Mirenna
发明人: Giovanni Camaggi , Lucio Filippini , Marilena Gusmeroli , Raul Riva , Carlo Garavaglia , Luigi Mirenna , Luigi Mirenna
IPC分类号: A01N43/78 , C07D417/04 , C07D277/22
CPC分类号: C07D417/04 , A01N43/78
摘要: Compounds based on 2-thiazole-2-ylpyrrole, with a fungicidal activity, having the general formula (I): ##STR1##
摘要翻译: 具有通式(I)的具有杀真菌活性的2-噻唑-2-基吡咯的化合物:(I)
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公开(公告)号:US5378707A
公开(公告)日:1995-01-03
申请号:US155545
申请日:1993-11-22
IPC分类号: A01N43/84 , A01N33/10 , A01N43/40 , A01N43/54 , A01N55/00 , A01N55/10 , A01P3/00 , C07D213/64 , C07D213/643 , C07D239/34 , C07D265/30 , C07D295/096 , C07D413/06 , C07F7/08 , C07F7/10 , C07F7/18
CPC分类号: C07D213/643 , A01N33/10 , A01N43/40 , A01N43/54 , A01N55/00 , C07D239/34 , C07D295/096 , C07F7/0812 , C07F7/1856 , C07C2101/02 , C07C2101/08
摘要: Aryl-propyl-aminic compounds having the following formula ##STR1## have high activity and are useful in the agricultural field as fungicides.
摘要翻译: 具有下式(I)的芳基 - 丙基 - 氨基化合物具有高活性,并且在农田中用作杀真菌剂。
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公开(公告)号:US5464836A
公开(公告)日:1995-11-07
申请号:US131880
申请日:1993-10-05
申请人: Giovanni Camaggi , Lucio Filippini , Marilena Gusmeroli , Raul Riva , Carlo Garavaglia , Luigi Mirenna
发明人: Giovanni Camaggi , Lucio Filippini , Marilena Gusmeroli , Raul Riva , Carlo Garavaglia , Luigi Mirenna
IPC分类号: A01N37/44 , A01N35/04 , A01N43/84 , C07C45/51 , C07C49/86 , C07C217/22 , C07C225/06 , C07C225/16 , C07C233/69 , C07D265/30 , C07D279/12 , C07D295/092 , C07D295/112 , A61K31/535 , C07C211/27
CPC分类号: C07D295/088 , A01N35/04 , C07C217/22 , C07C225/16 , C07C45/512 , C07C49/86 , C07D295/112
摘要: A description follows of benzophenones having an antifungal activity and responding to the general formula (I): ##STR1## wherein: R.sub.1 and R.sub.2, the same or different, represent C.sub.1 -C.sub.6 alkyl groups, C.sub.7 -C.sub.10 arylalkyl groups; or R.sub.1 and R.sub.2, considered jointly with N, represent a C.sub.3 -C.sub.8 heterocyclic group or a C.sub.2 -C.sub.7 heterocyclic group containing a second hetero-atom selected from O and S, said heterocyclic groups being optionally subsituted with one or more C.sub.1 -C.sub.4 alkyl groups;R.sub.3 and R.sub.4, the same or different, represent H atoms, C.sub.1 -C.sub.3 alkyl groups;K represents an oxygen atom or methylene;A represents a benzene group, optionally sustituted with one or more halogen atoms, C.sub.1 -C.sub.4 alkyl or haloalkyl groups, C.sub.1 -C.sub.4 alkoxylics, C.sub.1 -C.sub.4 haloalkoxylics;Y represents a C.sub.6 -C.sub.10 aryl group; said group may be optionally substituted with one or more halogen atomos, C.sub.1 -C.sub.4 alkyl or haloalkyl groups, C.sub.1 -C.sub.4 alkoxylics, C.sub.1 -C.sub.4 haloalkoxylics.
摘要翻译: 以下描述具有抗真菌活性并对应于通式(I)的二苯甲酮:其中:R1和R2相同或不同,表示C1-C6烷基,C7-C10芳基烷基; 或与N一起考虑的R 1和R 2表示含有选自O和S的第二杂原子的C 3 -C 8杂环基或C 2 -C 7杂环基,所述杂环基任选被一个或多个C 1 -C 4烷基取代 团体 R3和R4相同或不同,表示H原子,C1-C3烷基; K表示氧原子或亚甲基; A表示任选被一个或多个卤素原子取代的苯基,C 1 -C 4烷基或卤代烷基,C 1 -C 4烷氧基,C 1 -C 4卤代烷氧基; Y表示C6-C10芳基; 所述基团可以任选地被一个或多个卤素原子,C 1 -C 4烷基或卤代烷基,C 1 -C 4烷氧基,C 1 -C 4卤代烷氧基取代。
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公开(公告)号:US5470863A
公开(公告)日:1995-11-28
申请号:US943333
申请日:1992-09-10
申请人: Giovanni Camaggi , Lucio Filippini , Marilena Gusmeroli , Giovanni Meazza , Giampaolo Zanardi , Carlo Garavaglia , Luigi Mirenna
发明人: Giovanni Camaggi , Lucio Filippini , Marilena Gusmeroli , Giovanni Meazza , Giampaolo Zanardi , Carlo Garavaglia , Luigi Mirenna
IPC分类号: A01N43/36 , A01N43/40 , A01N43/78 , A01P3/00 , C07D207/32 , C07D207/335 , C07D207/337 , C07D401/12 , C07D417/12
CPC分类号: C07D207/335 , A01N43/36 , A01N43/78 , C07D417/12
摘要: A description follows of oximic derivatives with a fungicide activity, for agricultural use, having the formula (I): ##STR1## wherein: A, B, D, are N, or .dbd.C--G;G is H, halogen, NO.sub.2, CN, --COOR.sub.4, C.sub.1 -C.sub.6 (halo)alkylR.sub.1, R.sub.2, R.sub.4 and R.sub.5, are C.sub.1 -C.sub.6 (halo)alkyl;R.sub.3 is H, C.sub.1 -C.sub.6 (halo)alkyl or --COOR.sub.5 ;W is C.sub.2 -C.sub.10 alkylene;L represents O or S;Y represents phenyl, naphthyl, heterocycle, substituted alkyl.
摘要翻译: 以下描述具有式(I)的农业用杀真菌活性的肟化衍生物:其中:A,B,D为N或= C-G; G是H,卤素,NO 2,CN,-COOR 4,C 1 -C 6(卤代)烷基,R 1,R 2和R 4是C 1 -C 6(卤代) R3是H,C1-C6(卤代)烷基或-COOR5; W是C 2 -C 10亚烷基; L表示O或S; Y表示苯基,萘基,杂环,取代的烷基。
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