公开(公告)号：US08729083B2

公开(公告)日：2014-05-20

申请号：US13120052

申请日：2009-09-23

申请人： Steffen Groβ ,  Karsten Körber ,  Wolfgang von Deyn ,  Florian Kaiser ,  Prashant Deshmukh ,  Joachim Dickhaut ,  Ronan Le Vezouet ,  Sebastian Sörgel ,  Matthias Pohlman ,  Douglas D. Anspaugh ,  Deborah L. Culbertson ,  Faraneh Oloumi

发明人： Steffen Groβ ,  Karsten Körber ,  Wolfgang von Deyn ,  Florian Kaiser ,  Prashant Deshmukh ,  Joachim Dickhaut ,  Ronan Le Vezouet ,  Sebastian Sörgel ,  Matthias Pohlman ,  Douglas D. Anspaugh ,  Deborah L. Culbertson ,  Hassan Oloumi-Sadeghi

IPC分类号： C07D403/12 ,  C07D403/14 ,  A01M1/24

CPC分类号： A01N43/58 ,  A01N43/56 ,  A01N43/60 ,  A01N43/647 ,  A01N43/653 ,  A01N43/82 ,  C07D401/14 ,  C07D403/12 ,  C07D403/14 ,  C07D409/14 ,  C07D413/14 ,  C07D417/14

摘要： The present invention relates to pyrazole compounds of formulae I or II and the salts and N-oxides thereof, wherein A is a pyrazole radical of formulae A1, A2 or A3, wherein # denotes the binding site; R41, R42, R43, R51 are H, halogen, CN, NO2, C1-C10-alkyl and the like; R52, R53 are H, halogen, CN, NO2, C1-C10-alkyl, and the like; R61, R62, R63 are H, CN, NO2, C1-C10-alkyl, and the like; T is C(Rt) or N; U is C(Ru) or N; V is C(Rv) or N; W is C(Rw) or N; with the proviso that at least one of the groups T, U, V and W is N; Rt, Ru, Rv, Rw are H, halogen, C1-C4-alkyl and the like; X1 is S, O or NR1a, wherein R1a is selected H, C1-C10-alkyl and the like; X2 is OR2a, NR2bR2c, S(O)mR2d, wherein m is 0, 1 or 2, R2a is C1-C4-alkyl, C1-C4-haloalkyl and the like, R2b, R2c are H, C1-C4-alkyl, C1-C4-haloalkyl and the like, or R2b and R2c together with the nitrogen atom to which they are bound form a heterocycle, and R2d is C1-C4-alkyl, C1-C4-haloalkyl, C3-C6-cycloalkyl and the like; and R1 is H, CN, C1-C10-alkyl and the like. The present invention further relates to a method for controlling invertebrate pests, to a method for protecting plant propagation material and/or the plants which grow therefrom, to plan propagation material, comprising at least one compound according to the present invention, to a method for treating or protecting an animal from infestation or infection by parasites and to an agricultural composition containing at least one compound according to the present invention.

摘要翻译： 本发明涉及式I或II的吡唑化合物及其盐和N-氧化物，其中A是式A1，A2和A3的吡唑基，其中＃表示结合位点; R 41，R 42，R 43，R 51为H，卤素，CN，NO 2，C 1 -C 10 - 烷基等; R 52，R 53为H，卤素，CN，NO 2，C 1 -C 10 - 烷基等; R61，R62，R63是H，CN，NO2，C1-C10-烷基等; T为C（Rt）或N; U是C（Ru）或N; V是C（Rv）或N; W是C（Rw）或N; 条件是组T，U，V和W中的至少一个为N; R 1，R u，R v，R w为H，卤素，C 1 -C 4 - 烷基等; X1是S，O或NR1a，其中R1a选自H，C1-C10-烷基等; X2是OR2a，NR2bR2c，S（O）mR2d，其中m是0,1或2，R2a是C1-C4-烷基，C1-C4-卤代烷基等，R2b，R2c是H，C1-C4-烷基， C1-C4卤代烷基等，或R2b和R2c与它们所结合的氮原子一起形成杂环，R2d是C1-C4-烷基，C1-C4卤代烷基，C3-C6-环烷基等 ; R1为H，CN，C1-C10-烷基等。 本发明还涉及一种控制无脊椎害虫的方法，一种用于保护植物繁殖材料和/或从其生长的植物的方法，以将包含至少一种本发明化合物的繁殖材料计划到一种方法 治疗或保护动物免受寄生虫侵袭或感染，以及含有至少一种本发明化合物的农药组合物。

公开(公告)号：US08853125B2

公开(公告)日：2014-10-07

申请号：US13120208

申请日：2009-09-23

申请人： Steffen Groβ ,  Karsten Körber ,  Wolfgang von Deyn ,  Florian Kaiser ,  Ronan Le Vezouet ,  Sebastian Sörgel ,  Matthias Pohlman ,  Prashant Deshmukh ,  Joachim Dickhaut ,  Douglas D. Anspaugh ,  Deborah L. Culbertson ,  Faraneh Oloumi

发明人： Steffen Groβ ,  Karsten Körber ,  Wolfgang von Deyn ,  Florian Kaiser ,  Ronan Le Vezouet ,  Sebastian Sörgel ,  Matthias Pohlman ,  Prashant Deshmukh ,  Joachim Dickhaut ,  Douglas D. Anspaugh ,  Deborah L. Culbertson ,  Hassan Oloumi-Sadeghi

IPC分类号： A01N43/54 ,  A01N43/56 ,  A01N43/58 ,  A01N43/90 ,  A01P5/00 ,  A01P7/02 ,  A01P7/04 ,  C07D498/04 ,  C07D471/04 ,  C07D487/04

CPC分类号： A01N43/90 ,  C07D471/04 ,  C07D487/04 ,  C07D498/04

摘要： The present invention relates to a method for controlling invertebrate pests which method comprises treating the pests, their food supply, their habitat or their breeding ground or a plant, seed, soil, area, material or environment in which the pests are growing or may grow, or the materials, plants, seeds, soils, surfaces or spaces to be protected from pest attack or infestation with a pesticidally effective amount of a pyrazole compound of formulae I or II or a salt or an N-oxide thereof, wherein A is a pyrazole radical of the formulae A1 or A2, wherein # denotes the binding; D is a 5- or 6-membered heterocyclic radical fused to the pyrazole moiety; Rp1, Rp2 and Rpx are H, halogen, CN, NO2, C1-C10-alkyl, C2-C10-alkenyl, C2-C10-alkynyl, etc.; n is 0 to 4; or two radicals Rpx bound to the same ring-member may form an oxo substituent, or two radicals Rpx bound to adjacent ring-members may form a 3- to 7-membered fused cyclic radical; B is N or CR4, wherein R4 is H, halogen, CN, NO2, C1-C4-alkyl, C1-C4-haloalkyl, C1-C4-alkoxy, etc.; X1 is S, O or NR1a, wherein R1a is H, C1-C10-alkyl, etc.; X2 is O2a, NR2bR2c or S(O)mR2d, wherein m is 0, 1 or 2; R2a is C1-C4-alkyl, C1-C4-haloalkyl, C3-C6-cycloalkyl, etc.; R2b, R2c are H, C1-C4-alkyl, C1-C4-haloalkyl, C3-C6-cycloalkyl, etc.; R2d is C1-C4-alkyl, C1-C4-haloalkyl, C3-C6-cycloalkyl, etc.; R1 is H, CN, C1-C10-alkyl, C1-C10-haloalkyl, C3-C10-cycloalkyl, etc.; R2, R3 and R5 are H, halogen, CN, NO2, C1-C4-alkyl, C1-C4-haloalkyl, C1-C4-alkoxy, etc., to a method for protecting plant propagation material and/or the plants which grow threfrom, to plant propagation material comprising at least one compound of formulae I or II, to a method for treating or protecting an animal from infestation or infection by parasites, to novel pyrazole compounds of formulae I or II and agricultural composition containing those compounds.

公开(公告)号：US20110269770A1

公开(公告)日：2011-11-03

申请号：US13120052

申请日：2009-09-23

申请人： Steffen Gross ,  Karsten Körber ,  Wolfgang von Deyn ,  Florian Kaiser ,  Prashant Deshmukh ,  Joachim Dickhaut ,  Ronan Le Vezouet ,  Sebastian Sörgel ,  Matthias Pohlman ,  Douglas D. Anspaugh ,  Deborah L. Culbertson ,  Hassan Oloumi-Sadeghi ,  Faraneh Oloumi

发明人： Steffen Gross ,  Karsten Körber ,  Wolfgang von Deyn ,  Florian Kaiser ,  Prashant Deshmukh ,  Joachim Dickhaut ,  Ronan Le Vezouet ,  Sebastian Sörgel ,  Matthias Pohlman ,  Douglas D. Anspaugh ,  Deborah L. Culbertson ,  Hassan Oloumi-Sadeghi ,  Faraneh Oloumi

IPC分类号： A01N43/58 ,  A01P7/04 ,  A61P33/00 ,  A01P7/00 ,  C07D403/12 ,  A61K31/501

CPC分类号： A01N43/58 ,  A01N43/56 ,  A01N43/60 ,  A01N43/647 ,  A01N43/653 ,  A01N43/82 ,  C07D401/14 ,  C07D403/12 ,  C07D403/14 ,  C07D409/14 ,  C07D413/14 ,  C07D417/14

摘要： The present invention relates to pyrazole compounds of formulae I or II and the salts and N-oxides thereof, wherein A is a pyrazole radical of formulae A1, A2 or A3, wherein # denotes the binding site; R41, R42, R43, R51 are H, halogen, CN, NO2, C1-C10-alkyl and the like; R52, R53 are H, halogen, CN, NO2, C1-C10-alkyl, and the like; R61, R62, R63 are H, CN, NO2, C1-C10-alkyl, and the like; T is C(Rt) or N; U is C(Ru) or N; V is C(Rv) or N; W is C(Rw) or N; with the proviso that at least one of the groups T, U, V and W is N; Rt, Ru, Rv, Rw are H, halogen, C1-C4-alkyl and the like; X1 is S, O or NR1a, wherein R1a is selected H, C1-C10-alkyl and the like; X2 is OR2a, NR2bR2c, S(O)mR2d, wherein m is 0, 1 or 2, R2a is C1-C4-alkyl, C1-C4-haloalkyl and the like, R2b, R2c are H, C1-C4-alkyl, C1-C4-haloalkyl and the like, or R2b and R2c together with the nitrogen atom to which they are bound form a heterocycle, and R2d is C1-C4-alkyl, C1-C4-haloalkyl, C3-C6-cycloalkyl and the like; and R1 is H, CN, C1-C10-alkyl and the like.The present invention further relates to a method for controlling invertebrate pests, to a method for protecting plant propagation material and/or the plants which grow therefrom, to plant propagation material, comprising at least one compound according to the present invention, to a method for treating or protecting an animal from infestation or infection by parasites and to an agricultural composition containing at least one compound according to the present invention.

摘要翻译： 本发明涉及式I或II的吡唑化合物及其盐和N-氧化物，其中A是式A1，A2和A3的吡唑基，其中＃表示结合位点; R 41，R 42，R 43，R 51为H，卤素，CN，NO 2，C 1 -C 10 - 烷基等; R 52，R 53为H，卤素，CN，NO 2，C 1 -C 10 - 烷基等; R61，R62，R63是H，CN，NO2，C1-C10-烷基等; T为C（Rt）或N; U是C（Ru）或N; V是C（Rv）或N; W是C（Rw）或N; 条件是组T，U，V和W中的至少一个为N; R 1，R u，R v，R w为H，卤素，C 1 -C 4 - 烷基等; X1是S，O或NR1a，其中R1a选自H，C1-C10-烷基等; X2是OR2a，NR2bR2c，S（O）mR2d，其中m是0,1或2，R2a是C1-C4-烷基，C1-C4-卤代烷基等，R2b，R2c是H，C1-C4-烷基， C1-C4卤代烷基等，或R2b和R2c与它们所结合的氮原子一起形成杂环，R2d是C1-C4-烷基，C1-C4卤代烷基，C3-C6-环烷基等 ; R1为H，CN，C1-C10-烷基等。 本发明还涉及一种控制无脊椎害虫的方法，一种用于保护植物繁殖材料和/或从其生长的植物的方法，包括至少一种根据本发明的化合物的植物繁殖材料的方法， 治疗或保护动物免受寄生虫侵袭或感染，以及含有至少一种本发明化合物的农药组合物。

公开(公告)号：US20110173726A1

公开(公告)日：2011-07-14

申请号：US13120208

申请日：2009-09-23

申请人： Steffen Groß ,  Karsten Körber ,  Wolfgang Von Deyn ,  Florian Kaiser ,  Ronan Le Vezouet ,  Sebastian Sörgel ,  Matthias Pohlman ,  Prashant Deshmukh ,  Joachim Dickhaut ,  Douglas D. Anspaugh ,  Deborah L. Culbertson ,  Hassan Oloumi-Sadeghi

发明人： Steffen Groß ,  Karsten Körber ,  Wolfgang Von Deyn ,  Florian Kaiser ,  Ronan Le Vezouet ,  Sebastian Sörgel ,  Matthias Pohlman ,  Prashant Deshmukh ,  Joachim Dickhaut ,  Douglas D. Anspaugh ,  Deborah L. Culbertson ,  Hassan Oloumi-Sadeghi

IPC分类号： A01H5/00 ,  A01N43/40 ,  C07D471/04 ,  A01N43/54 ,  C07D487/04 ,  C07D401/14 ,  A01N43/60 ,  A01N43/58 ,  A01N43/84 ,  C07D498/04 ,  A01N43/42 ,  A01P7/00

CPC分类号： A01N43/90 ,  C07D471/04 ,  C07D487/04 ,  C07D498/04

摘要： The present invention relates to a method for controlling invertebrate pests which method comprises treating the pests, their food supply, their habitat or their breeding ground or a plant, seed, soil, area, material or environment in which the pests are growing or may grow, or the materials, plants, seeds, soils, surfaces or spaces to be protected from pest attack or infestation with a pesticidally effective amount of a pyrazole compound of formulae I or II or a salt or an N-oxide thereof, wherein A is a pyrazole radical of the formulae A1 or A2, wherein # denotes the binding; D is a 5- or 6-membered heterocyclic radical fused to the pyrazole moiety; Rp1, Rp2 and Rpx are H, halogen, CN, NO2, C1-C10-alkyl, C2-C10-alkenyl, C2-C10-alkynyl, etc.; n is 0 to 4; or two radicals Rpx bound to the same ring-member may form an oxo substituent, or two radicals Rpx bound to adjacent ring-members may form a 3- to 7-membered fused cyclic radical; B is N or CR4, wherein R4 is H, halogen, CN, NO2, C1-C4-alkyl, C1-C4-haloalkyl, C1-C4-alkoxy, etc.; X1 is S, O or NR1a, wherein R1a is H, C1-C10-alkyl, etc.; X2 is O2a, NR2bR2c or S(O)mR2d, wherein m is 0, 1 or 2; R2a is C1-C4-alkyl, C1-C4-haloalkyl, C3-C6-cycloalkyl, etc.; R2b, R2c are H, C1-C4-alkyl, C1-C4-haloalkyl, C3-C6-cycloalkyl, etc.; R2d is C1-C4-alkyl, C1-C4-haloalkyl, C3-C6-cycloalkyl, etc.; R1 is H, CN, C1-C10-alkyl, C1-C10-haloalkyl, C3-C10-cycloalkyl, etc.; R2, R3 and R5 are H, halogen, CN, NO2, C1-C4-alkyl, C1-C4-haloalkyl, C1-C4-alkoxy, etc., to a method for protecting plant propagation material and/or the plants which grow threfrom, to plant propagation material comprising at least one compound of formulae I or II, to a method for treating or protecting and animal from infestation or infection by parasites, to novel pyrazole compounds of formulae I or II and agricultural composition containing those compounds.

公开(公告)号：US08765774B2

公开(公告)日：2014-07-01

申请号：US13254182

申请日：2010-03-03

申请人： Steffen Groβ ,  Karsten Körber ,  Wolfgang von Deyn ,  Florian Kaiser ,  Prashant Deshmukh ,  Joachim Dickhaut ,  Nina Gertrud Bandur ,  Arun Narine ,  Matthias Pohlman ,  Michael Puhl ,  Sarah Thompson ,  Cecille Ebuenga ,  Douglas D. Anspaugh ,  Deborah L. Culbertson ,  Faraneh Oloumi

发明人： Steffen Groβ ,  Karsten Körber ,  Wolfgang von Deyn ,  Florian Kaiser ,  Prashant Deshmukh ,  Joachim Dickhaut ,  Nina Gertrud Bandur ,  Arun Narine ,  Matthias Pohlman ,  Michael Puhl ,  Sarah Thompson ,  Cecille Ebuenga ,  Douglas D. Anspaugh ,  Deborah L. Culbertson ,  Hassan Oloumi-Sadeghi

IPC分类号： A01N43/54 ,  A61K31/517 ,  C07D401/00 ,  C07D403/00 ,  C07D413/00 ,  C07D417/00 ,  C07D419/00

CPC分类号： C07D239/88 ,  C07D401/04 ,  C07D403/04

摘要： The present invention relates to the 3-arylquinazolin-4-one compounds of the formula I and the salts thereof, wherein n is 0, 1 or 2; X is O, S or N—R4; Y1 is N or CH; Y2 is N or C—R5; R1 is C1-C10-alkyl, C1-C10-haloalkyl, C2-C10-alkenyl, C2-C10-haloalkenyl, C2-C10-alkynyl, C2-C10-haloalkynyl, C3-C12-cycloalkyl, C5-C12-cycloalkenyl, C3-C12-cycloalkyl-C1-C4-alkyl, C5-C12-cycloalkenyl-C1-C4-alkyl, where the cycloalkyl radical and the cycloalkenyl radical in the last four mentioned radicals are unsubstituted, partially or fully halogenated and/or carry 1, 2, 3, 4, or 5 C1-C4-alkyl radicals; R2 is hydrogen, halogen, CN, C(Z)NH2, C1-C4-alkyl or C1-C4-haloalkyl, wherein Z is O, S or NR6; and the variables k, R, R3, R4, R5 and R6 are as defined in the claims. The invention also relates to the use of novel compounds of formula I for combating invertebrate pests and to a method for controlling invertebrate pests. The invention also relates to a plant propagation material and to an agricultural composition comprising a 3-arylquinazolin-4-one compound of formula I.

摘要翻译： 本发明涉及式I的3-芳基喹唑啉-4-酮化合物及其盐，其中n为0,1或2; X为O，S或N-R4; Y1是N或CH; Y2是N或C-R5; R 1是C 1 -C 10 - 烷基，C 1 -C 10 - 卤代烷基，C 2 -C 10 - 烯基，C 2 -C 10 - 卤代烯基，C 2 -C 10 - 炔基，C 2 -C 10 - 卤代炔基，C 3 -C 12 - 环烷基，C 5 -C 12 - 环烯基， C 3 -C 12 - 环烷基-C 1 -C 4 - 烷基，C 5 -C 12 - 环烯基-C 1 -C 4烷基，其中最后四个所述基团中的环烷基和环烯基是未取代的，部分或完全卤化和/或携带1 ，2,3,4或5个C 1 -C 4 - 烷基; R 2是氢，卤素，CN，C（Z）NH 2，C 1 -C 4烷基或C 1 -C 4卤代烷基，其中Z是O，S或NR 6; 变量k，R，R3，R4，R5和R6如权利要求中所定义。 本发明还涉及新颖的式I化合物用于防治无脊椎动物害虫以及控制无脊椎害虫的方法。 本发明还涉及植物繁殖材料和农业组合物，其包含式I的3-芳基喹唑啉-4-酮化合物。

公开(公告)号：US20120053052A1

公开(公告)日：2012-03-01

申请号：US13254182

申请日：2010-03-03

申请人： Steffen Gross ,  Karsten Körber ,  Wolfgang von Deyn ,  Florian Kaiser ,  Prashant Deshmukh ,  Joachim Dickhaut ,  Nina Gertrud Bandur ,  Arun Narine ,  Matthias Pohlman ,  Michael Puhl ,  Sarah Thompson ,  Cecille Ebuenga ,  Douglas D. Anspaugh ,  Deborah L. Culbertson ,  Hassan Oloumi-Sadeghi ,  Faraneh Oloumi

发明人： Steffen Gross ,  Karsten Körber ,  Wolfgang von Deyn ,  Florian Kaiser ,  Prashant Deshmukh ,  Joachim Dickhaut ,  Nina Gertrud Bandur ,  Arun Narine ,  Matthias Pohlman ,  Michael Puhl ,  Sarah Thompson ,  Cecille Ebuenga ,  Douglas D. Anspaugh ,  Deborah L. Culbertson ,  Hassan Oloumi-Sadeghi ,  Faraneh Oloumi

IPC分类号： A01N43/54 ,  C07D401/04 ,  A61K31/517 ,  A01P7/02 ,  A01P5/00 ,  A01C1/06 ,  C07D239/91 ,  A01P7/04

CPC分类号： C07D239/88 ,  C07D401/04 ,  C07D403/04

摘要： The present invention relates to the 3-arylquinazolin-4-one compounds of the formula I and the salts thereof, wherein n is 0, 1 or 2; X is O, S or N—R4; Y1 is N or CH; Y2 is N or C—R5; R1 is C1-C10-alkyl, C1-C10-haloalkyl, C2-C10-alkenyl, C2-C10-haloalkenyl, C2-C10-alkynyl, C2-C10-haloalkynyl, C3-C12-cycloalkyl, C5-C12-cycloalkenyl, C3-C12-cycloalkyl-C1-C4-alkyl, C5-C12-cycloalkenyl-C1-C4-alkyl, where the cycloalkyl radical and the cycloalkenyl radical in the last four mentioned radicals are unsubstituted, partially or fully halogenated and/or carry 1, 2, 3, 4, or 5 C1-C4-alkyl radicals; R2 is hydrogen, halogen, CN, C(Z)NH2, C1-C4-alkyl or C1-C4-haloalkyl, wherein Z is O, S or NR6; and the variables k, R, R3, R4, R5 and R6 are as defined in the claims. The invention also relates to the use of novel compounds of formula I for combating invertebrate pests and to a method for controlling invertebrate pests. The invention also relates to a plant propagation material and to an agricultural composition comprising a 3-arylquinazolin-4-one compound of formula I.

摘要翻译： 本发明涉及式I的3-芳基喹唑啉-4-酮化合物及其盐，其中n为0,1或2; X为O，S或N-R4; Y1是N或CH; Y2是N或C-R5; R 1是C 1 -C 10 - 烷基，C 1 -C 10 - 卤代烷基，C 2 -C 10 - 烯基，C 2 -C 10 - 卤代烯基，C 2 -C 10 - 炔基，C 2 -C 10 - 卤代炔基，C 3 -C 12 - 环烷基，C 5 -C 12 - 环烯基， C 3 -C 12 - 环烷基-C 1 -C 4 - 烷基，C 5 -C 12 - 环烯基-C 1 -C 4烷基，其中最后四个所述基团中的环烷基和环烯基是未取代的，部分或完全卤化和/或携带1 ，2,3,4或5个C 1 -C 4 - 烷基; R 2是氢，卤素，CN，C（Z）NH 2，C 1 -C 4烷基或C 1 -C 4卤代烷基，其中Z是O，S或NR 6; 变量k，R，R3，R4，R5和R6如权利要求中所定义。 本发明还涉及新颖的式I化合物用于防治无脊椎动物害虫以及控制无脊椎害虫的方法。 本发明还涉及植物繁殖材料和农业组合物，其包含式I的3-芳基喹唑啉-4-酮化合物。

公开(公告)号：US20120030841A1

公开(公告)日：2012-02-02

申请号：US13260788

申请日：2010-03-31

申请人： Karsten Koerber ,  Florian Kaiser ,  Wolfgang von Deyn ,  Matthias Pohlman ,  Steffen Gross ,  Prashant Deshmukh ,  Joachim Dickhaut ,  Nina Gertrud Bandur ,  Deborah L. Culbertson ,  Douglas D. Anspaugh ,  Franz-Josef Braun ,  Cecille Ebuenga ,  Nancy B. Rankl

发明人： Karsten Koerber ,  Florian Kaiser ,  Wolfgang von Deyn ,  Matthias Pohlman ,  Steffen Gross ,  Prashant Deshmukh ,  Joachim Dickhaut ,  Nina Gertrud Bandur ,  Deborah L. Culbertson ,  Douglas D. Anspaugh ,  Franz-Josef Braun ,  Cecille Ebuenga ,  Nancy B. Rankl

IPC分类号： A01N43/80 ,  A61K31/4709 ,  A01P7/04 ,  A01P7/00 ,  A61P33/14 ,  A01P7/02 ,  C07D413/04 ,  A01H5/00

CPC分类号： C07D413/04

摘要： The present invention relates to isoxazoline compounds which are useful for combating or controlling invertebrate pests, in particular arthropod pests and nematodes. The invention also relates to a method for controlling invertebrate pests by using these compounds and to plant propagation material and to an agricultural and a veterinary composition comprising said compounds.

摘要翻译： 本发明涉及可用于对抗或控制无脊椎害虫，特别是节肢动物害虫和线虫的异恶唑啉化合物。 本发明还涉及通过使用这些化合物和植物繁殖材料以及包含所述化合物的农业和兽用组合物来控制无脊椎害虫的方法。

公开(公告)号：US08633134B2

公开(公告)日：2014-01-21

申请号：US13141264

申请日：2009-12-14

申请人： Florian Kaiser ,  Karsten Koerber ,  Matthias Pohlman ,  Steffen Gross ,  Prashant Deshmukh ,  Joachim Dickhaut ,  Nina Gertrud Bandur ,  Wolfgang von Deyn ,  Deborah L. Culbertson ,  Douglas D. Anspaugh ,  Franz-Josef Braun ,  Cecille Ebuenga

发明人： Florian Kaiser ,  Karsten Koerber ,  Matthias Pohlman ,  Steffen Gross ,  Prashant Deshmukh ,  Joachim Dickhaut ,  Nina Gertrud Bandur ,  Wolfgang von Deyn ,  Deborah L. Culbertson ,  Douglas D. Anspaugh ,  Franz-Josef Braun ,  Cecille Ebuenga

IPC分类号： A01N43/836 ,  A01N43/40 ,  A01N43/80 ,  A61P33/00 ,  A61K31/4245 ,  A61K31/4439 ,  A61K31/42 ,  A61K31/444 ,  C07D261/04 ,  C07D413/04 ,  C07D413/10 ,  C07D413/14

CPC分类号： C07D261/04 ,  A01N43/80 ,  A01N43/82 ,  C07C257/18 ,  C07C257/22 ,  C07C259/18 ,  C07C2601/02 ,  C07D413/04 ,  C07D413/10 ,  C07D413/12 ,  C07D413/14

摘要： The invention relates to substituted amidine compounds of formula (I), to the enantiomers, diastereomers and salts thereof and to compositions comprising such compounds. The invention also relates to the use of the substituted amidine compounds, of their salts or of compositions comprising them for combating animal pests. Furthermore the invention relates also to methods of applying such substituted amidine compounds.The substituted amidine compounds of the present invention are defined by the following formula I: wherein A1 to A4, B1 to B3, R1 to R3, (R4)p, (R5)q, X and Y are defined as in the description.

摘要翻译： 本发明涉及式（I）的取代的脒化合物，其涉及其对映体，非对映异构体和盐以及包含这些化合物的组合物。 本发明还涉及取代的脒化合物，其盐或包含它们的组合物用于对抗动物害虫的用途。 此外，本发明还涉及应用这种取代的脒化合物的方法。 本发明的取代的脒化合物由下式I定义：其中A1至A4，B1至B3，R1至R3，（R4）p，（R5）q，X和Y如说明书所定义。

公开(公告)号：US20110257011A1

公开(公告)日：2011-10-20

申请号：US13141264

申请日：2009-12-14

申请人： Florian Kaiser ,  Karsten Koerber ,  Matthias Pohlman ,  Steffen Gross ,  Prashant Deshmukh ,  Joachim Dickhaut ,  Nina Gertrud Bandur ,  Wolfgang Von Deyn ,  Deborah L. Culbertson ,  Douglas D. Anspaugh ,  Franz-Josef Braun ,  Cecille Ebuenga

发明人： Florian Kaiser ,  Karsten Koerber ,  Matthias Pohlman ,  Steffen Gross ,  Prashant Deshmukh ,  Joachim Dickhaut ,  Nina Gertrud Bandur ,  Wolfgang Von Deyn ,  Deborah L. Culbertson ,  Douglas D. Anspaugh ,  Franz-Josef Braun ,  Cecille Ebuenga

IPC分类号： A01C1/06 ,  A01N43/836 ,  A61K31/4245 ,  C07D413/14 ,  A01N43/40 ,  A01P7/00 ,  C07D413/04 ,  A61K31/4439 ,  C07D261/04 ,  A01N43/80 ,  A61K31/42 ,  A61P33/00 ,  C07D413/10 ,  A61K31/444

CPC分类号： C07D261/04 ,  A01N43/80 ,  A01N43/82 ,  C07C257/18 ,  C07C257/22 ,  C07C259/18 ,  C07C2601/02 ,  C07D413/04 ,  C07D413/10 ,  C07D413/12 ,  C07D413/14

摘要： The invention relates to substituted amidine compounds of formula (I), to the enantiomers, diastereomers and salts thereof and to compositions comprising such compounds. The invention also relates to the use of the substituted amidine compounds, of their salts or of compositions comprising them for combating animal pests. Furthermore the invention relates also to methods of applying such substituted amidine compounds.The substituted amidine compounds of the present invention are defined by the following formula I: wherein A1 to A4, B1 to B3, R1 to R3, (R4)p, (R5)q, X and Y are defined as in the description.

摘要翻译： 本发明涉及式（I）的取代的脒化合物，其涉及其对映体，非对映异构体和盐以及包含这些化合物的组合物。 本发明还涉及取代的脒化合物，其盐或包含它们的组合物用于对抗动物害虫的用途。 此外，本发明还涉及应用这种取代的脒化合物的方法。 本发明的取代的脒化合物由下式I定义：其中A1至A4，B1至B3，R1至R3，（R4）p，（R5）q，X和Y如说明书所定义。

公开(公告)号：US08119568B2

公开(公告)日：2012-02-21

申请号：US12523802

申请日：2008-01-14

申请人： Wolfgang von Deyn ,  Matthias Pohlman ,  Florian Kaiser ,  Joachim Dickhaut ,  Douglas D. Anspaugh ,  Deborah L. Culbertson ,  Hassan Oloumi-Sadeghi

发明人： Wolfgang von Deyn ,  Matthias Pohlman ,  Florian Kaiser ,  Joachim Dickhaut ,  Douglas D. Anspaugh ,  Deborah L. Culbertson ,  Hassan Oloumi-Sadeghi

IPC分类号： A01N43/80 ,  C07D275/06

CPC分类号： C07D417/14 ,  A01N43/80 ,  A01N43/90 ,  C07D275/04 ,  C07D275/06 ,  C07D417/12

摘要： The invention provides 3-amino-1,2-benzisothiazole compounds of formula (I) wherein n, R1, R2, R3, R4 and A are defined as in the description. The invention provides further agricultural compositions comprising an amount of at least one compound of the formula (I) or an enantiomer, diastereomer or salt thereof; the use of a compound of formula (I) or an enantiomer, diastereomer or salt thereof for combating animal pests; a method of combating animal pests which comprises contacting the animal pests, their habit, breeding ground, food supply, plant, seed, soil, area, material or environment in which the animal pests are growing or may grow, or the materials, plants, seeds, soils, surfaces or spaces to be protected from animal attack or infestation with a pesticidally effective amount of at least one compound of the formula (I) or an enantiomer, diastereomer or salt thereof; a method for protecting crops from attack or infestation by animal pests, which comprises contacting a crop with a pesticidally effective amount of at least one compound of the formula (I) or an enantiomer, diastereomer or salt thereof; a method for the protection of seeds from soil insects and of the seedlings' roots and shoots from soil and foliar insects comprising contacting the seeds before sowing and/or after pregermination with at least one compound of the formula (I), or the enantiomers, diastereomers or salts thereof; and seeds comprising a compound of the formula I or an enantiomer, diastereomer or salt thereof.

摘要翻译： 本发明提供式（I）的3-氨基-1,2-苯并异噻唑化合物，其中n，R 1，R 2，R 3，R 4和A如描述中所定义。 本发明提供了包含一定量的至少一种式（I）化合物或其对映异构体，非对映体或其盐的进一步农业组合物; 使用式（I）化合物或其对映异构体，非对映体或其盐来防治动物害虫; 一种防治动物害虫的方法，包括使动物有害生物，其习惯，繁殖地，食物供应，植物，种子，土壤，区域，动物害虫生长或可能生长的区域，物质或环境，或材料，植物， 种子，土壤，表面或空间，以防止动物攻击或侵袭与杀虫有效量的至少一种式（I）化合物或其对映体，非对映体或其盐; 包括使作物与杀虫有效量的至少一种式（I）化合物或其对映异构体，非对映异构体或其盐接触的方法，用于保护作物不被动物害虫侵袭或侵染。 包括防止种子从土壤昆虫和幼苗根和土壤和叶面昆虫的芽中保护种子的方法，包括在种子播种前和/或之后与种子接种后与至少一种式（I）的化合物或对映异构体接触， 非对映体或其盐; 和包含式I化合物或其对映体，非对映体或其盐的种子。