-
1.Method of blocking nerve conduction by treatment with branched-chain esters of 2-�4-(2-piperidine-ethoxy)-benzoyl!-benzoic acid and pharmaceutically acceptable salts thereof 失效
标题翻译: 通过用2- [4-(2-哌啶 - 乙氧基) - 苯甲酰基] - 苯甲酸的支链酯处理阻断神经传导的方法及其药学上可接受的盐公开(公告)号:US5821252A
公开(公告)日:1998-10-13
申请号:US474550
申请日:1995-06-07
申请人: Swati Bal-Tembe , Jurgen Blumbach , Alihussein Nomanbhai Dohadwalla, deceased , Bansi Lal , Narayan Sudhindra Punekar , Ramanujam Rajgopalan , Richard Helmut Rupp , Martin Bickel
发明人: Swati Bal-Tembe , Jurgen Blumbach , Alihussein Nomanbhai Dohadwalla, deceased , Bansi Lal , Narayan Sudhindra Punekar , Ramanujam Rajgopalan , Richard Helmut Rupp , Martin Bickel
IPC分类号: A61K31/445 , C07D211/34
CPC分类号: A61K31/445
摘要: Compounds of the formula III ##STR1## in which R.sub.4 and R.sub.5 are CH.sub.3 amd R.sub.6 is hydrogen, have prolonged spasmolytic and anaesthetic activity.
摘要翻译: 其中R4和R5是CH3的R6的化合物III是氢,具有延长的解痉和麻醉活性。
-
2.Labdane derivatives, a process for their preparation, and their use as medicaments 失效
标题翻译: LABDANE衍生物,其制备方法及其作为药物使用公开(公告)号:US5093331A
公开(公告)日:1992-03-03
申请号:US595751
申请日:1990-10-09
申请人: Bansi Lal , Ashok K. Gangopadbya , Alihussein N. Dohadwalla , Ramanujam Rajgopalan , Richard H. Rupp
发明人: Bansi Lal , Ashok K. Gangopadbya , Alihussein N. Dohadwalla , Ramanujam Rajgopalan , Richard H. Rupp
IPC分类号: A61K31/35 , A61K31/352 , A61K31/443 , A61K31/445 , A61K31/495 , A61K31/535 , A61K31/55 , A61P9/12 , A61P27/02 , C07D311/92 , C07D405/12 , C07D413/12
CPC分类号: C07D405/12 , C07D311/92 , C07D413/12
摘要: The present invention relates to polyoxygenated labdane-derivatives of the formula ##STR1## a process for their preparation and the use of these substances as medicaments, preferably as medicaments having a positive inotropic effect, an effect of lowering intraocular pressure and lowering blood pressure.
摘要翻译: 本发明涉及下式的聚氧化实体丹丹衍生物:其制备方法和这些物质作为药物的使用,优选作为具有正性肌力作用的药物,降低眼内压和降低血压的作用。
-