PROCESS FOR PREPARING 3-[(4S)-8-BROMO-1-METHYL-6-(2-PYRIDINYL)-4H-IMIDAZO[1,2-A][1,4]BENZODIAZEPINE-4-YL]PROPIONIC ACID METHYL ESTER OR THE BENZENE SULFONATE SALT THEREOF, AND COMPOUNDS USEFUL IN THAT PROCESS
    6.
    发明申请
    PROCESS FOR PREPARING 3-[(4S)-8-BROMO-1-METHYL-6-(2-PYRIDINYL)-4H-IMIDAZO[1,2-A][1,4]BENZODIAZEPINE-4-YL]PROPIONIC ACID METHYL ESTER OR THE BENZENE SULFONATE SALT THEREOF, AND COMPOUNDS USEFUL IN THAT PROCESS 有权
    制备3 - [(4S)-8-溴-1-甲基-6-(2-吡啶基)-4H-咪唑并[1,2-A] [1,4]苯并噻吩并[4-y]]丙酸甲酯的方法 ESTER或其中的苯甲磺酸盐及其用途的化合物

    公开(公告)号:US20150368199A1

    公开(公告)日:2015-12-24

    申请号:US14841899

    申请日:2015-09-01

    IPC分类号: C07D213/50

    摘要: The invention concerns a new process for preparing 3-[(4S)-8-bromo-1-methyl-6-(2-pyridinyl)-4H-imidazo[1,2-a][1,4]benzodiazepine-4-yl]-propionic acid methyl ester or 3-[(4S)-8-bromo-1-methyl-6-(2-pyridinyl)-4H-imidazo[1,2-a][1,4]benzodiazepine-4-yl]propionic acid methyl ester benzene sulfonate (P) which comprises reacting 3-[(S)-7-bromo-2-((R and/or S)-2-hydroxy-propylamino)-5-pyridin-2-yl-3H-benzo[e][1,4]diazepin-3-yl]-propionic acid methyl ester of formula (EM) with an oxidizing agent and optionally treating the reaction product under acidic conditions, such as to produce the compound of formula (F) or the compound (P), and new compounds useful as starting material or as intermediate for performing that process.

    摘要翻译: 本发明涉及一种制备3 - [(4S)-8-溴-1-甲基-6-(2-吡啶基)-4H-咪唑并[1,2-a] [1,4]苯并二氮杂- 吡啶-3-基] - 丙酸甲酯或3 - [(4S)-8-溴-1-甲基-6-(2-吡啶基)-4H-咪唑并〔1,2-a〕〔1,4〕苯并二氮杂-4- 吡啶-2-基]丙酸甲酯苯磺酸盐(P),其包括使3 - [(S)-7-溴-2 - ((R和/或S)-2-羟基 - 丙基氨基) -3H-苯并[e] [1,4]二氮杂-3-基] - 丙酸甲酯与氧化剂反应,并在酸性条件下任选地处理反应产物,例如制备式 (F)或化合物(P),以及可用作原料的新化合物或用于进行该方法的中间体。

    POWER SWITCH FOR PREVENTING ACCIDENTAL ARCS
    8.
    发明申请
    POWER SWITCH FOR PREVENTING ACCIDENTAL ARCS 有权
    用于防止意外ARCS的电源开关

    公开(公告)号:US20100214724A1

    公开(公告)日:2010-08-26

    申请号:US12599224

    申请日:2008-05-09

    IPC分类号: H02B1/00

    CPC分类号: H02H1/0023 H02H3/023 H02H3/08

    摘要: A power switch disposed in a housing includes a contact breaker configured to connect and disconnect a low-voltage switchgear from a power source supplying the low-voltage switchgear, a triggering device configured to disconnect the low-voltage switchgear in an overload event, a current detection device, a control device, a first evaluation device configured to evaluate an accidental arc overcurrent, and a second evaluation device configured to evaluate the accidental arc overcurrent. The power switch is configured to be activated via an overcurrent signal generated by an arc monitoring system in response to the accidental arc overcurrent. The overcurrent signal is linked to the at least one triggering signal. The second evaluation has a threshold above a threshold of the first evaluation device. The triggering device is configured to be activated via a turn-off pulse when a signal from the current detection device is above the threshold of the second evaluation device.

    摘要翻译: 设置在壳体中的电源开关包括接触断路器,其被配置为将低压开关设备与供应低压开关设备的电源连接和断开;触发装置,其被配置为在过载事件中断开低压开关设备,电流 检测装置,控制装置,被配置为评估意外的过电流的第一评估装置,以及被配置为评估意外的电弧过电流的第二评估装置。 电源开关被配置为通过由电弧监视系统响应于意外的电弧过电流而产生的过电流信号而被激活。 过电流信号与至少一个触发信号相连。 第二评估具有高于第一评估装置的阈值的阈值。 触发装置被配置为当来自当前检测装置的信号高于第二评估装置的阈值时通过关断脉冲被激活。

    CIRCUIT BREAKER AND SHORT CIRCUITER COMBINATION
    9.
    发明申请
    CIRCUIT BREAKER AND SHORT CIRCUITER COMBINATION 失效
    断路器和短路电路组合

    公开(公告)号:US20080007881A1

    公开(公告)日:2008-01-10

    申请号:US11773575

    申请日:2007-07-05

    IPC分类号: H02H9/00

    摘要: A circuit breaker for multi-phase power includes an opening-closing apparatus configured to open and close each phase of the multiphase power, a detection unit configured to detect a fault current in at least one phase of an electrical installation being protected by the circuit breaker, a plurality of connecting bars disposed on a load side of the circuit breaker, and a short circuiter disposed on the connecting bars and configured to produce a short circuit between the connecting bars if a fault current is detected by the fault-current detection unit. When a fault current occurs, a tripping signal can be transmitted by the detection system to the short circuiter. The circuit breaker is also fully operational, even without a function-activated short circuiter.

    摘要翻译: 一种用于多相电力的断路器包括:开闭装置,其被配置为打开和关闭所述多相电力的每个相;检测单元,被配置为检测由所述断路器保护的电气设备的至少一相中的故障电流; 设置在所述断路器的负载侧的多个连接杆,以及设置在所述连接杆上的短路器,其被配置为如果所述故障电流检测单元检测到故障电流,则在所述连接条之间产生短路。 当发生故障电流时,检测系统可以向短路器发送跳闸信号。 断路器也是完全可操作的,即使没有功能激活的短路器。

    Method for producing an optical arrangement
    10.
    发明申请
    Method for producing an optical arrangement 有权
    光学装置的制造方法

    公开(公告)号:US20050053327A1

    公开(公告)日:2005-03-10

    申请号:US10686982

    申请日:2003-10-16

    IPC分类号: G02B6/42 G02B6/26

    CPC分类号: G02B6/4226 G02B6/4212

    摘要: The invention relates to a method for producing an optical arrangement (10, 300), in which an optical component (355, 20) is optically connected to at least one waveguide (90, 320, 330) provided on or in a carrier substrate (100, 310). In order to enable an optical component to be connected to an optical waveguide of a carrier substrate in a particularly simple and thus cost-effective manner, the invention provides for there to be arranged between the optical component (20, 355) and the waveguide (90, 320, 330) an adjustment device (40, 350) with at least one auxiliary waveguide (60, 410, 440), the waveguide ends (50, 70, 400, 420, 430, 450) of which are in each case movable and an optical adjustment between the optical component (20, 355) and the waveguide (90, 320, 330) of the carrier substrate (100, 310) is effected by a mechanical adjustment of the movable waveguide ends (50, 70, 400, 420, 430, 450).

    摘要翻译: 本发明涉及一种用于制造光学装置(10,300)的方法,其中光学部件(355,20)光学地连接到设置在载体衬底上或载体衬底上的至少一个波导(90,320,330) 100,310)。 为了使光学部件能够以特别简单且因此成本有效的方式连接到载体基板的光波导,本发明提供了一种布置在光学部件(20,355)和波导( 90,320,330)具有至少一个辅助波导(60,410,440)的调节装置(40,350),其波导端部(50,70,400,420,430,450)在每种情况下 通过对可移动波导端部(50,70,400)的机械调节来实现光学部件(20,355)和载体基板(100,310)的波导(90,320,330)之间的可移动和光学调节 ,420,430,450)。