公开(公告)号：US09006266B2

公开(公告)日：2015-04-14

申请号：US13993262

申请日：2011-08-24

申请人： Tomoki Tsuchiya ,  Pierre Wasnaire ,  Sebastian Hoffmann ,  Pierre Cristau ,  Thomas Seitz ,  Joachim Kluth ,  Stefan Hillebrand ,  Juergen Benting ,  Daniela Portz ,  Ulrike Wachendorff-Neumann

发明人： Tomoki Tsuchiya ,  Pierre Wasnaire ,  Sebastian Hoffmann ,  Pierre Cristau ,  Thomas Seitz ,  Joachim Kluth ,  Stefan Hillebrand ,  Juergen Benting ,  Daniela Portz ,  Ulrike Wachendorff-Neumann

IPC分类号： A61K31/445 ,  C07D405/00 ,  A01N43/78 ,  A01N43/80 ,  A01N47/38 ,  A01N55/00 ,  C07D417/14

CPC分类号： A01N43/80 ,  A01N43/78 ,  A01N47/22 ,  A01N47/38 ,  A01N55/00 ,  C07D417/14 ,  C07F7/0812

摘要： Heteroarylpiperidine and -piperazine derivatives of the formula (I) in which the symbols A, X, Y, L1, L2, G, Q, p, R1, R2 and R10 are each as defined in the description, and salts, metal complexes and N-oxides of the compounds of the formula (I), and the use thereof for controlling phytopathogenic harmful fungi and processes for preparing compounds of the formula (I).

摘要翻译： 符号A，X，Y，L1，L2，G，Q，p，R1，R2和R10各自如说明书中所定义的式（I）的杂芳基哌啶和哌嗪衍生物，以及盐，金属络合物和 式（I）化合物的N-氧化物及其用于控制​​植物病原性有害真菌的用途及其制备式（I）化合物的方法。

公开(公告)号：US20130296272A1

公开(公告)日：2013-11-07

申请号：US13993262

申请日：2011-08-24

申请人： Tomoki Tsuchiya ,  Pierre Wasnaire ,  Sebastian Hoffmann ,  Pierre Cristau ,  Thomas Seitz ,  Joachim Kluth ,  Stefan Hillebrand ,  Juergen Benting ,  Daniela Portz ,  Ulrike Wachendorff-Neumann

发明人： Tomoki Tsuchiya ,  Pierre Wasnaire ,  Sebastian Hoffmann ,  Pierre Cristau ,  Thomas Seitz ,  Joachim Kluth ,  Stefan Hillebrand ,  Juergen Benting ,  Daniela Portz ,  Ulrike Wachendorff-Neumann

IPC分类号： A01N55/00 ,  A01N43/80

CPC分类号： A01N43/80 ,  A01N43/78 ,  A01N47/22 ,  A01N47/38 ,  A01N55/00 ,  C07D417/14 ,  C07F7/0812

摘要： Heteroarylpiperidine and -piperazine derivatives of the formula (I) in which the symbols A, X, Y, L1, L2, G, Q, p, R1, R2 and R10 are each as defined in the description, and salts, metal complexes and N-oxides of the compounds of the formula (I), and the use thereof for controlling phytopathogenic harmful fungi and processes for preparing compounds of the formula (I).

公开(公告)号：US08759527B2

公开(公告)日：2014-06-24

申请号：US13216033

申请日：2011-08-23

申请人： Tomoki Tsuchiya ,  Pierre Wasnaire ,  Sebastian Hoffmann ,  Pierre Cristau ,  Thomas Seitz ,  Joachim Kluth ,  Stefan Hillebrand ,  Jürgen Benting ,  Daniela Portz ,  Ulrike Wachendorff-Neumann

发明人： Tomoki Tsuchiya ,  Pierre Wasnaire ,  Sebastian Hoffmann ,  Pierre Cristau ,  Thomas Seitz ,  Joachim Kluth ,  Stefan Hillebrand ,  Jürgen Benting ,  Daniela Portz ,  Ulrike Wachendorff-Neumann

IPC分类号： C07D417/14 ,  A61K31/4535

CPC分类号： A01N43/80 ,  A01N43/78 ,  A01N47/22 ,  A01N47/38 ,  A01N55/00 ,  C07D417/14 ,  C07F7/0812

摘要： Heteroarylpiperidine and -piperazine derivatives of the formula (I) in which the symbols A, X, Y, L1, L2, G, Q, p, R1, R2 and R10 are each as defined in the description, and salts, metal complexes and N-oxides of the compounds of the formula (I), and the use thereof for controlling phytopathogenic harmful fungi and processes for preparing compounds of the formula (I).

公开(公告)号：US10004232B2

公开(公告)日：2018-06-26

申请号：US14342606

申请日：2012-09-11

申请人： Stefan Hillebrand ,  Tomoki Tsuchiya ,  Sebastian Hoffmann ,  Pierre Cristau ,  Pierre Wasnaire ,  Thomas Seitz ,  Juergen Benting ,  Ulrike Wachendorff-Neumann ,  Peter Jan Schmidt

发明人： Stefan Hillebrand ,  Tomoki Tsuchiya ,  Sebastian Hoffmann ,  Pierre Cristau ,  Pierre Wasnaire ,  Thomas Seitz ,  Juergen Benting ,  Ulrike Wachendorff-Neumann ,  Peter Jan Schmidt

IPC分类号： C07D417/14 ,  A01N43/80

CPC分类号： A01N43/80 ,  C07D417/14

摘要： The invention relates to heteroarylpiperidine and -piperazine derivatives of formula (I) to agrochemically active salts thereof, to their use and also to methods and compositions for controlling phytopathogenic harmful fungi in and/or on plants or in and/or on seed of plants, to methods for producing such compositions and to treated seed, and also to the use thereof for controlling phytopathogenic harmful plants in agriculture, horticulture and forestry, in animal health, in materials protection and also in the household and hygiene sector. The present invention further relates to a method for producing heteroarylpiperidine and -piperazine derivatives.

公开(公告)号：US20140005224A1

公开(公告)日：2014-01-02

申请号：US13879876

申请日：2011-10-25

申请人： Stefan Hillebrand ,  Pierre Cristau ,  Sebastian Hoffmann ,  Joachim Kluth ,  Pierre Wasnaire ,  Tomoki Tsuchiya ,  Jürgen Benting ,  Ulrike Wachendorff-Neumann ,  Thomas SEITZ

发明人： Stefan Hillebrand ,  Pierre Cristau ,  Sebastian Hoffmann ,  Joachim Kluth ,  Pierre Wasnaire ,  Tomoki Tsuchiya ,  Jürgen Benting ,  Ulrike Wachendorff-Neumann ,  Thomas SEITZ

IPC分类号： A01N43/80 ,  C07D417/14

CPC分类号： C07D417/14 ,  A01N43/80

摘要： Heteroarylpiperidine and -piperazine derivatives of the formula (I) in which the symbols A, X, Y, L1, L2, G, Q, p, R1, R2 and R10 are each as defined in the description, and salts, metal complexes and N-oxides of the compounds of the formula (I), and the use thereof for controlling phytopathogenic harmful fungi and processes for preparing compounds of the formula (I).

摘要翻译： 符号A，X，Y，L1，L2，G，Q，p，R1，R2和R10各自如说明书中所定义的式（I）的杂芳基哌啶和哌嗪衍生物，以及盐，金属络合物和 式（I）化合物的N-氧化物及其用于控制​​植物病原性有害真菌的用途及其制备式（I）化合物的方法。

公开(公告)号：US20110237612A1

公开(公告)日：2011-09-29

申请号：US13061930

申请日：2009-08-22

申请人： Jörg Nico Greul ,  Hendrik Helmke ,  Stefan Hillebrand ,  Amos Mattes ,  Carl Friedrich Nising ,  Pierre Wasnaire ,  Ulrike Wachendorff-Neumann ,  Peter Dahmen ,  Arnd Voerste ,  Ruth Meissner ,  Christoph Andreas Braun ,  Martin Kaussmann ,  Hiroyuki Hadano

发明人： Jörg Nico Greul ,  Hendrik Helmke ,  Stefan Hillebrand ,  Amos Mattes ,  Carl Friedrich Nising ,  Pierre Wasnaire ,  Ulrike Wachendorff-Neumann ,  Peter Dahmen ,  Arnd Voerste ,  Ruth Meissner ,  Christoph Andreas Braun ,  Martin Kaussmann ,  Hiroyuki Hadano

IPC分类号： A01N43/54 ,  C07D409/12 ,  C07D239/48 ,  A01P3/00

CPC分类号： C07D409/12 ,  A01N43/54

摘要： Thienylaminopyrimidines of the formula (I) in which to R1 to R10 and X1 and X2 have the meanings given in the description, and agrochemically active salts thereof, their use and also methods and compositions for controlling phytopathogenic harmful fungi in and/or on plants or in and/or on seed of plants, processes for preparing such compositions and treated seed and also their use for controlling phytopathogenic harmful fungi in agriculture, horticulture and forestry, in the protection of materials and in the domestic and hygiene field. The present invention furthermore relates to a process for preparing thienylaminopyrimidines of the formula (I).

摘要翻译： 其中R 1至R 10和X 1和X 2具有其描述中给出的含义的式（I）的噻吩基氨基嘧啶及其农业化学活性盐，其用途以及用于控制植物中和/或植物上的植物病原性有害真菌的方法和组合物， 在植物的种子和/或种子中，用于制备这种组合物和处理的种子的方法，以及它们用于控制农业，园艺和林业中的植物病原性有害真菌，在材料的保护和家庭和卫生领域中的用途。 本发明还涉及制备式（I）的噻吩基氨基嘧啶的方法。

公开(公告)号：US20110245284A1

公开(公告)日：2011-10-06

申请号：US13061896

申请日：2009-08-21

申请人： Jörg Nico Greul ,  Hendrik Helmke ,  Stefan Hillebrand ,  Amos Mattes ,  Pierre Wasnaire ,  Carl Friedrich Nising ,  Ulrike Wachendorff-Neumann ,  Peter Dahmen ,  Arnd Voerste ,  Ruth Meissner ,  Chirstoph Andreas Braun ,  Martin Kaubmann ,  Hiroyuki Hadano ,  Ulrich Heinemann

发明人： Jörg Nico Greul ,  Hendrik Helmke ,  Stefan Hillebrand ,  Amos Mattes ,  Pierre Wasnaire ,  Carl Friedrich Nising ,  Ulrike Wachendorff-Neumann ,  Peter Dahmen ,  Arnd Voerste ,  Ruth Meissner ,  Chirstoph Andreas Braun ,  Martin Kaubmann ,  Hiroyuki Hadano ,  Ulrich Heinemann

IPC分类号： A01N43/54 ,  C07D239/48 ,  C07D239/42 ,  C07C205/11 ,  C07C321/20 ,  A01P3/00

CPC分类号： C07D239/48

摘要： Alkoxy- and alkylthio-substituted anilinopyrimidines of the formula (I) in which R1 to R14 and E1, E2, E3, X and Y have the meanings given in the description, and agrochemically active salts thereof, their use, and methods and compositions for controlling phytopathogenic harmful fungi in and/or on plants or in and/or on seeds of plants, processes for preparing such compositions and treated seeds and also their use for controlling phytopathogenic hal inful fungi in agriculture, horticulture and forestry, in the protection of materials and in the domestic and hygiene field. The present invention furthermore relates to a process for the preparation of alkoxy- and alkylthio-substituted anilinopyrimidines of the formula (I).

摘要翻译： 其中R1至R14和E1，E2，E3，X和Y具有本说明书中给出的含义的式（I）的烷氧基​​ - 和烷硫基取代的苯胺基嘧啶，及其农业化学活性盐，其用途和方法和组合物 控制植物内部和/或植物中或植物种子和/或种子上的植物病原性有害真菌，以及用于制备这些组合物和处理过的种子的方法，以及它们用于控制农业，园艺和林业中植物病原性真菌的用途，以保护材料 并在国内和卫生领域。 本发明还涉及制备式（I）的烷氧基​​ - 和烷硫基取代的苯胺基嘧啶亚胺的方法。

公开(公告)号：US20110245249A1

公开(公告)日：2011-10-06

申请号：US13061932

申请日：2009-08-22

申请人： Pierre Wasnaire ,  Jorg Nico Greul ,  Oliver Gaertzen ,  Hendrik Helmke ,  Stefan Hillebrand ,  Amos Mattes ,  Carl Friedrich Nising ,  Ulrike Wachendorff-Neumann ,  Peter Dahmen ,  Arnd Voerste ,  Ruth Meissner ,  Christoph Andreas Braun ,  Martin Kaussmann ,  Hiroyuki Hadano

发明人： Pierre Wasnaire ,  Jorg Nico Greul ,  Oliver Gaertzen ,  Hendrik Helmke ,  Stefan Hillebrand ,  Amos Mattes ,  Carl Friedrich Nising ,  Ulrike Wachendorff-Neumann ,  Peter Dahmen ,  Arnd Voerste ,  Ruth Meissner ,  Christoph Andreas Braun ,  Martin Kaussmann ,  Hiroyuki Hadano

IPC分类号： A01N43/54 ,  C07D405/12 ,  C07D239/48 ,  C07D409/12 ,  C07D413/14 ,  A01N43/84 ,  C07D493/04 ,  A01N43/90 ,  A01P3/00

CPC分类号： C07D405/12 ,  C07D239/48 ,  C07D409/12 ,  C07D411/12

摘要： Heterocyclically substituted anilinopyrimidines of the formula (I) in which R1 to R12 and E1, E2, E3, L1, Y, Z and L2 have the meanings given in the description, and agrochemically active salts thereof, their use and also methods and compositions for controlling phytopathogenic harmful fungi in and/or on plants or in and/or on seed of plants, processes for preparing such compositions and treated seed and also their use for controlling phytopathogenic harmful fungi in agriculture, horticulture and forestry, in the protection of materials and in the domestic and hygiene field. The present invention furthermore relates to a process for preparing heterocyclically substituted anilinopyrimidinenes of the formula (I).

摘要翻译： R 1至R 12和E 1，E 2，E 3，L 1，Y，Z和L 2具有本说明书中给出的含义的式（I）的杂环取代的苯胺基嘧啶及其农业化学活性盐，其用途和方法和组合物 控制植物内部和/或植物中或植物种子和/或种子上的植物病原性有害真菌，以及用于制备这些组合物和处理过的种子的方法，以及它们用于控制农业，园艺和林业中植物病原性有害真菌，保护材料和 在国内和卫生领域。 本发明还涉及制备式（I）的杂环取代的苯胺基嘧啶并苯的方法。

公开(公告)号：US07999137B2

公开(公告)日：2011-08-16

申请号：US12063659

申请日：2006-09-12

申请人： Klaus Kunz ,  Jörg Greul ,  Oliver Guth ,  Benoît Hartmann ,  Kerstin Ilg ,  Wahed Ahmed Moradi ,  Thomas Seitz ,  Peter Dahmen ,  Arnd Voerste ,  Ulrike Wachendorff-Neumann ,  Mark Drewes ,  Ralf Dunkel ,  Ronald Ebbert ,  Herbert Gayer ,  Stefan Hillebrand ,  Eva-Maria Franken ,  Olga Malsam ,  Ulrich Ebbinghaus-Kintscher

发明人： Klaus Kunz ,  Jörg Greul ,  Oliver Guth ,  Benoît Hartmann ,  Kerstin Ilg ,  Wahed Ahmed Moradi ,  Thomas Seitz ,  Peter Dahmen ,  Arnd Voerste ,  Ulrike Wachendorff-Neumann ,  Mark Drewes ,  Ralf Dunkel ,  Ronald Ebbert ,  Herbert Gayer ,  Stefan Hillebrand ,  Eva-Maria Franken ,  Olga Malsam ,  Ulrich Ebbinghaus-Kintscher

IPC分类号： C07C257/00 ,  A01N25/26

CPC分类号： C07D295/195 ,  A01N37/52 ,  A01N41/06 ,  A01N41/10 ,  A01N43/36 ,  A01N43/40 ,  A01N43/56 ,  A01N43/58 ,  A01N55/00 ,  C07C257/12 ,  C07C335/30 ,  C07C2601/08 ,  C07C2601/14 ,  C07F7/081

摘要： The present invention relates to bi-phenyl-amidine derivatives of formula (I) in which the substituents are as in the description, their process of preparation, their use as fungicide or insecticide active agents, particularly in the form of fungicide or insecticide compositions, and methods for the control of phytopathogenic fungi or damaging insects, notably of plants, using these compounds or compositions:

摘要翻译： 本发明涉及式（I）的双苯基 - 脒衍生物，其中取代基如说明书，其制备方法，其作为杀真菌剂或杀虫剂活性剂的用途，特别是杀真菌剂或杀虫剂组合物的形式， 以及使用这些化合物或组合物来控制植物病原真菌或损害昆虫，特别是植物的昆虫的方法：

公开(公告)号：US07781439B2

公开(公告)日：2010-08-24

申请号：US11816253

申请日：2006-02-07

申请人： Stefan Herrmann ,  Olaf Gebauer ,  Herbert Gayer ,  Stefan Hillebrand ,  Ulrich Heinemann ,  Oliver Guth ,  Kerstin Ilg ,  Thomas Seitz ,  Ronald Ebbert ,  Ulrike Wachendorff-Neumann ,  Peter Dahmen ,  Karl-Heinz Kuck ,  Horst-Peter Antonicek

发明人： Stefan Herrmann ,  Olaf Gebauer ,  Herbert Gayer ,  Stefan Hillebrand ,  Ulrich Heinemann ,  Oliver Guth ,  Kerstin Ilg ,  Thomas Seitz ,  Ronald Ebbert ,  Ulrike Wachendorff-Neumann ,  Peter Dahmen ,  Karl-Heinz Kuck ,  Horst-Peter Antonicek

IPC分类号： A01N43/90 ,  A61K31/519 ,  C07D487/00

CPC分类号： C07D487/04 ,  A01N43/90

摘要： Pyrazolopyrimidines of the formula in which R1, R2, R3, R4, R5 and X are as defined in the description, processes for preparing these compounds and their use for controlling unwanted microorganisms.

摘要翻译： 其中R 1，R 2，R 3，R 4，R 5和X如说明书中所定义的式的吡唑并嘧啶用于制备这些化合物及其用于防治有害微生物的方法。