公开(公告)号：US20090076113A1

公开(公告)日：2009-03-19

申请号：US12097753

申请日：2006-12-05

Applicant: Ralf Dunkel ,  Hans-Ludwig Elbe ,  Jorg Nico Greul ,  Herbert Gayer ,  Arnd Voerste ,  Ulrike Wachendorff-Neumann ,  Peter Dahmen

Inventor： Ralf Dunkel ,  Hans-Ludwig Elbe ,  Jorg Nico Greul ,  Herbert Gayer ,  Arnd Voerste ,  Ulrike Wachendorff-Neumann ,  Peter Dahmen

IPC: A01N43/56 ,  C07D231/10 ,  C07C229/00 ,  A01N37/44 ,  C07C211/44 ,  A01N33/02 ,  C07D271/00

CPC classification number: C07D231/14 ,  A01N43/56

Abstract: Novel biphenylcarboxamides of the formula (I) There is further provided a plurality of processes for preparing these compounds and their use for controlling unwanted microorganisms, and also novel intermediates and their preparation.

Abstract translation: 式（I）的新型联苯甲酰胺进一步提供了多种制备这些化合物的方法及其用于防治有害微生物的用途，以及新型中间体及其制备方法。

公开(公告)号：US20080058389A1

公开(公告)日：2008-03-06

申请号：US10588491

申请日：2005-01-22

Applicant: Ralf Dunkel ,  Hans-Ludwig Elbe ,  Benoit Hartmann ,  Jorg Nico Greul ,  Stefan Herrmann ,  Ulrike Wachendorff-Neumann ,  Peter Dahmen ,  Karl-Heinz Kuck

Inventor： Ralf Dunkel ,  Hans-Ludwig Elbe ,  Benoit Hartmann ,  Jorg Nico Greul ,  Stefan Herrmann ,  Ulrike Wachendorff-Neumann ,  Peter Dahmen ,  Karl-Heinz Kuck

IPC: A01N37/18 ,  A01N43/08 ,  A01N43/10 ,  A01N43/18 ,  A01N43/32 ,  A01N43/40 ,  A01N43/56 ,  A01N43/78 ,  A01P1/00 ,  C07C233/00 ,  C07D231/02 ,  C07D277/02 ,  C07D307/02 ,  C07D319/12 ,  C07D327/06 ,  C07D333/06 ,  C07D335/02

CPC classification number: A01N43/36 ,  A01N43/10 ,  A01N43/32 ,  A01N43/56 ,  A01N43/78 ,  C07D207/34 ,  C07D231/14 ,  C07D231/16 ,  C07D277/56 ,  C07D327/06 ,  C07D333/38

Abstract: The invention relates to novel carboxamides of formula (I), in which M represents a phenyl ring, pyridine ring or pyrimidine, pyridazine or pyrazine ring, respectively monosubstituted by R8, or represents a thiazole ring substituted by R8-A; R8 represents hydrogen, fluorine, chlorine, methyl, isopropyl, methylthio or trifluoromethyl; R8 can also represent methoxy; R8-A represents hydrogen, methyl, methylthio or trifluoromethyl; L1 represents C1-C10 alkene (alkanediyl); Q represents O, S, SO, SO2 or NR9; L2 represents a direct bond, SiR10R11 or CO; R represents hydrogen, C1-C8 alkyl, C1-C8 alkoxy, C1-C4 alkoxy-C1-C4-alkyl, C1-C4 alkylthio-C1-C4-alkyl, C2-C8 alkenyl, C2-C8 alkynyl, C1-C6 haloalkyl, C2-C6-haloalkenyl, C2-C6 haloalkynyl or C3-C6 cycloalkyl; A represents the group of formula (AI); the remaining substituents are defined in claim 1. The inventive substances have a powerful microbicidal action and can be used to control undesirable micro-organisms such as fungi and bacteria in the phyto-protection and material protection fields.

Abstract translation: 本发明涉及式（I）的新型甲酰胺，其中M表示分别被R 8单取代的苯环，吡啶环或嘧啶，哒嗪或吡嗪环，或代表被R 8取代的噻唑环 8-A; R 8表示氢，氟，氯，甲基，异丙基，甲硫基或三氟甲基; R 8也可以表示甲氧基; R 8 A表示氢，甲基，甲硫基或三氟甲基; L 1表示C 1 -C 10烷基（烷二基）; Q表示O，S，SO，SO 2或NR 9; L 2表示直接键合，SiR 10 R 11或CO; R代表氢，C 1 -C 8烷基，C 1 -C 8烷氧基，C 1 -C 8烷基，C 1 -C 8烷基， C 1 -C 4烷氧基-C 1 -C 4 - 亚烷基，C 1 -C C 1 -C 4烷基硫代C 1 -C 4 - 烷基，C 2 -C 8亚烷基 烯基，C 2 -C 8炔基，C 1 -C 6卤代烷基，C 2 C 1 -C 6 - 卤代烯基，C 2 -C 6卤代炔基或C 3 -C 3 - C 6环烷基; A代表式（AI）的基团; 其余的取代基如权利要求1中所定义。本发明的物质具有强大的杀微生物作用，可用于防止植物保护和材料保护领域中的不期望的微生物如真菌和细菌。

公开(公告)号：US20120178116A1

公开(公告)日：2012-07-12

申请号：US13330873

申请日：2011-12-20

Applicant: Christoph Andreas Braun ,  Peter Schreier ,  Klaus-Gunther Tietjen ,  Michael Edmund Beck ,  Amos Mattes ,  Jorg Nico Greul ,  Oliver Gutbrod ,  Sandra Tuckmantel ,  Daniel Raun

Inventor： Christoph Andreas Braun ,  Peter Schreier ,  Klaus-Gunther Tietjen ,  Michael Edmund Beck ,  Amos Mattes ,  Jorg Nico Greul ,  Oliver Gutbrod ,  Sandra Tuckmantel ,  Daniel Raun

IPC: C12Q1/48 ,  C12N15/63 ,  C12N9/12 ,  C12N1/19 ,  C12N1/21 ,  C12N1/15 ,  C12N5/10 ,  C12N15/54 ,  C07K16/40

CPC classification number: C07K14/37 ,  C12N9/1205 ,  C12Q1/18 ,  C12Q1/485

Abstract: The invention relates to a combination of polypeptides from phytopathogenic fungi having the biological activity of an aurora kinase and the function of an aurora kinase activator, to nucleic acids coding therefore, to the use of the polypeptides and nucleic acids for identifying modulators of an aurora kinase, to processes for identifying such modulators and to the use of these modulators as fungicides.

Abstract translation: 本发明涉及具有极光激酶的生物活性和极光激酶激活剂的功能的植物病原性真菌的多肽与所述多肽和核酸用于鉴定极光激酶调节剂的核酸的组合 ，用于鉴定这种调节剂的方法以及将这些调节剂用作杀真菌剂的方法。

公开(公告)号：US20080064874A1

公开(公告)日：2008-03-13

申请号：US10588293

申请日：2005-01-22

Applicant: Ralf Dunkel ,  Hans-Ludwig Elbe ,  Jorg Nico Greul ,  Benoit Hartmann ,  Peter Dahmen ,  Karl-Heinz Kuck ,  Ulrike Wachendorff-Neumann

Inventor： Ralf Dunkel ,  Hans-Ludwig Elbe ,  Jorg Nico Greul ,  Benoit Hartmann ,  Peter Dahmen ,  Karl-Heinz Kuck ,  Ulrike Wachendorff-Neumann

IPC: C07D401/00 ,  C07D277/00 ,  C07D307/00 ,  C07D409/00 ,  C07D333/02

CPC classification number: C07D307/68 ,  A01N43/08 ,  A01N43/10 ,  A01N43/40 ,  C07D333/38 ,  C07D495/12

Abstract: Novel 2-halofuryl/thienyl-3-carboxamides of the formula (I) in which A, Hal, R, M and Z are as defined in the description, a plurality of processes for preparing these compounds and their use for controlling unwanted microorganisms, and also novel intermediates and their preparation.

Abstract translation: 其中A，Hal，R，M和Z如说明书中所定义的式（I）的新型2-卤呋喃基/噻吩基-3-甲酰胺，制备这些化合物的多种方法及其控制不想要的微生物的用途， 还有新型中间体及其制备方法。

公开(公告)号：US20080021045A1

公开(公告)日：2008-01-24

申请号：US10581891

申请日：2004-12-08

Applicant: Olaf Gebauer ,  Ulrich Heinemann ,  Stefan Herrmann ,  Herbert Gayer ,  Jorg Nico Greul ,  Stefan Hillebrand ,  Hans-Ludwig Elbe ,  Ronald Ebbert ,  Ulrike Wachendorff-Neumann ,  Peter Dahmen ,  Karl-Heinz Kuck

Inventor： Olaf Gebauer ,  Ulrich Heinemann ,  Stefan Herrmann ,  Herbert Gayer ,  Jorg Nico Greul ,  Stefan Hillebrand ,  Hans-Ludwig Elbe ,  Ronald Ebbert ,  Ulrike Wachendorff-Neumann ,  Peter Dahmen ,  Karl-Heinz Kuck

IPC: C07D487/04 ,  A01N43/54 ,  A01P1/00 ,  A01P3/00

CPC classification number: C07D487/04

Abstract: Novel pyrazolopyrimidines of the formula in which R1, R2, R3, R4, R5 and Hal are as defined in the description, a plurality of processes for preparing these compounds and their use for controlling unwanted microorganisms.

Abstract translation: 下式的新的吡唑并嘧啶其中R 1，R 2，R 3，R 4，R 4， > 5和Hal如说明书中所定义，多种制备这些化合物的方法及其用于防治有害微生物的用途。

公开(公告)号：US20090105311A1

公开(公告)日：2009-04-23

申请号：US11916436

申请日：2006-05-26

Applicant: Ralf Dunkel ,  Hans-Ludwig Elbe ,  Herbert Gayer ,  Jorg Nico Greul ,  Ulrike Wachendorff-Neumann ,  Peter Dahmen ,  Ingo Wetcholowsky ,  Haruko Sawada ,  Hiroyuki Hadano

Inventor： Ralf Dunkel ,  Hans-Ludwig Elbe ,  Herbert Gayer ,  Jorg Nico Greul ,  Ulrike Wachendorff-Neumann ,  Peter Dahmen ,  Ingo Wetcholowsky ,  Haruko Sawada ,  Hiroyuki Hadano

IPC: A01N43/40 ,  A01N43/56 ,  A01N43/78 ,  A01N43/828 ,  A01N37/18

CPC classification number: A01N43/56 ,  A01N43/78

Abstract: Use of carboxamides of the formula (I) in which A, R1, M, Q and R are as defined in the description for controlling certain rust fungi, such as soya bean rust and coffee rust, in crop protection.

Abstract translation: 使用式（I）的甲酰胺，其中A，R 1，M，Q和R如描述中所定义，用于在作物保护中控制某些锈病真菌，例如大豆锈病和咖啡锈。

公开(公告)号：US20110245249A1

公开(公告)日：2011-10-06

申请号：US13061932

申请日：2009-08-22

Applicant: Pierre Wasnaire ,  Jorg Nico Greul ,  Oliver Gaertzen ,  Hendrik Helmke ,  Stefan Hillebrand ,  Amos Mattes ,  Carl Friedrich Nising ,  Ulrike Wachendorff-Neumann ,  Peter Dahmen ,  Arnd Voerste ,  Ruth Meissner ,  Christoph Andreas Braun ,  Martin Kaussmann ,  Hiroyuki Hadano

Inventor： Pierre Wasnaire ,  Jorg Nico Greul ,  Oliver Gaertzen ,  Hendrik Helmke ,  Stefan Hillebrand ,  Amos Mattes ,  Carl Friedrich Nising ,  Ulrike Wachendorff-Neumann ,  Peter Dahmen ,  Arnd Voerste ,  Ruth Meissner ,  Christoph Andreas Braun ,  Martin Kaussmann ,  Hiroyuki Hadano

IPC: A01N43/54 ,  C07D405/12 ,  C07D239/48 ,  C07D409/12 ,  C07D413/14 ,  A01N43/84 ,  C07D493/04 ,  A01N43/90 ,  A01P3/00

CPC classification number: C07D405/12 ,  C07D239/48 ,  C07D409/12 ,  C07D411/12

Abstract: Heterocyclically substituted anilinopyrimidines of the formula (I) in which R1 to R12 and E1, E2, E3, L1, Y, Z and L2 have the meanings given in the description, and agrochemically active salts thereof, their use and also methods and compositions for controlling phytopathogenic harmful fungi in and/or on plants or in and/or on seed of plants, processes for preparing such compositions and treated seed and also their use for controlling phytopathogenic harmful fungi in agriculture, horticulture and forestry, in the protection of materials and in the domestic and hygiene field. The present invention furthermore relates to a process for preparing heterocyclically substituted anilinopyrimidinenes of the formula (I).

Abstract translation: R 1至R 12和E 1，E 2，E 3，L 1，Y，Z和L 2具有本说明书中给出的含义的式（I）的杂环取代的苯胺基嘧啶及其农业化学活性盐，其用途和方法和组合物 控制植物内部和/或植物中或植物种子和/或种子上的植物病原性有害真菌，以及用于制备这些组合物和处理过的种子的方法，以及它们用于控制农业，园艺和林业中植物病原性有害真菌，保护材料和 在国内和卫生领域。 本发明还涉及制备式（I）的杂环取代的苯胺基嘧啶并苯的方法。

公开(公告)号：US20100167926A1

公开(公告)日：2010-07-01

申请号：US12530767

申请日：2008-03-04

Applicant: Klaus Kunz ,  Ralf Dunkel ,  Jorg Nico Greul ,  Kerstin Ilg ,  Birgit Kuhn ,  Wahed Ahmed Moradi ,  Thomas Seitz ,  Darren James Mansfield ,  Oliver Guth ,  Peter Dahmen ,  Ulrike Wachendorff-Neumann ,  Arnd Voerste ,  Robert Dale Mitchell ,  Tom Hough

Inventor： Klaus Kunz ,  Ralf Dunkel ,  Jorg Nico Greul ,  Kerstin Ilg ,  Birgit Kuhn ,  Wahed Ahmed Moradi ,  Thomas Seitz ,  Darren James Mansfield ,  Oliver Guth ,  Peter Dahmen ,  Ulrike Wachendorff-Neumann ,  Arnd Voerste ,  Robert Dale Mitchell ,  Tom Hough

IPC: A01C1/06 ,  C07C257/18 ,  A01N37/52 ,  C07C43/20 ,  A01N31/14 ,  C07C211/45 ,  A01N33/02 ,  C07C217/04 ,  A01N33/08 ,  A01N37/18 ,  C07C233/03 ,  C07C233/04

CPC classification number: C07C205/38 ,  A01N37/52 ,  C07C217/90 ,  C07C257/12 ,  C07C2601/02 ,  C07D211/14 ,  C07D265/30 ,  C07D295/125 ,  C07F7/1804

Abstract: The present invention relates to 3-substituted phenylamidines of the general formula (I), to a process for their preparation, to the use of the amidines according to the invention for controlling unwanted microorganisms and also to a composition for this purpose, comprising the phenoxyamidines according to the invention. Furthermore, the invention relates to a method for controlling unwanted microorganisms by applying the compounds according to the invention to the microorganisms and/or their habitat.

Abstract translation: 本发明涉及通式（I）的3-取代苯基脒，其制备方法，使用根据本发明的脒控制不需要的微生物，还涉及用于该目的的组合物，其包含苯氧基脒基 根据本发明。 此外，本发明涉及通过将根据本发明的化合物施用于微生物和/或其栖息地来控制不想要的微生物的方法。

公开(公告)号：US20090030024A1

公开(公告)日：2009-01-29

申请号：US12067634

申请日：2006-09-12

Applicant: Jorg Nico Greul ,  Oliver Gaertzen ,  Ralf Dunkel ,  Oliver Guth ,  Stefan Hillebrand ,  Kerstin Ilg ,  Peter Schreier ,  Ulrike Wachendorff-Neumann ,  Peter Dahmen ,  Arnd Voerste ,  Hiroyuki Hadano ,  Samir Bennabi

Inventor： Jorg Nico Greul ,  Oliver Gaertzen ,  Ralf Dunkel ,  Oliver Guth ,  Stefan Hillebrand ,  Kerstin Ilg ,  Peter Schreier ,  Ulrike Wachendorff-Neumann ,  Peter Dahmen ,  Arnd Voerste ,  Hiroyuki Hadano ,  Samir Bennabi

IPC: A01N43/54 ,  C07D417/04 ,  A01P3/00 ,  C07D417/14

CPC classification number: C07D417/04 ,  A01N43/78 ,  C07D417/14

Abstract: Use of compounds of the formula (I), in which R1, R2, R3, R4, R5, R6, R7, R8 and X, Y, Z are as defined in the description as fungicides. Compounds of the formula (Ia), R1, R2, R3, R4, R5, R6, R7, R8, R14, A, X, Y and Z are as defined in the description, process for preparing these compounds and their use for controlling unwanted microorganisms.

Abstract translation: 使用式（I）化合物，其中R 1，R 2，R 3，R 4，R 5，R 6，R 7，R 8和X，Y，Z如描述中所定义，作为杀真菌剂。 式（Ia），R 1，R 2，R 3，R 4，R 5，R 6，R 7，R 8，R 14，A，X，Y和Z的化合物如说明书中所定义，制备这些化合物的方法及其用于控制 不想要的微生物。

公开(公告)号：US20080085924A1

公开(公告)日：2008-04-10

申请号：US10538242

申请日：2003-12-01

Applicant: Ralf Dunkel ,  Hans-Ludwig Elbe ,  Heiko Rieck ,  Ulrike Wachendorff-Neumann ,  Peter Dahmen ,  Peter Losel ,  Karl-Heinz Kuck ,  Astrid Mauler-Machnik ,  Jorg Nico Greul

Inventor： Ralf Dunkel ,  Hans-Ludwig Elbe ,  Heiko Rieck ,  Ulrike Wachendorff-Neumann ,  Peter Dahmen ,  Peter Losel ,  Karl-Heinz Kuck ,  Astrid Mauler-Machnik ,  Jorg Nico Greul

IPC: A01N37/18 ,  A01N43/08 ,  A01N43/10 ,  A01N43/32 ,  A01N43/36 ,  A01N43/40 ,  A01N43/56 ,  A01N43/86 ,  A01P5/00 ,  A01P7/00 ,  C07C233/75 ,  C07D207/34 ,  C07D213/82 ,  C07D277/56 ,  C07D307/68 ,  C07D327/06 ,  C07D333/38

CPC classification number: C07D213/82 ,  A01N37/22 ,  A01N43/08 ,  A01N43/10 ,  A01N43/32 ,  A01N43/40 ,  A01N43/56 ,  A01N43/78 ,  C07C225/22 ,  C07C251/48 ,  C07D207/34 ,  C07D231/14 ,  C07D231/16 ,  C07D277/56 ,  C07D307/68 ,  C07D327/06 ,  C07D333/38

Abstract: This invention relates to novel biphenylcarboxamides of the formula (I) in which R, Z, X, Y, m, n and A are as defined in the disclosure, to a plurality of processes for preparing these compounds and their use for controlling unwanted microorganisms, and to novel intermediates and their preparation.

Abstract translation: 本发明涉及式（I）的新型联苯甲酰胺，其中R，Z，X，Y，m，n和A如本公开所定义，涉及多种制备这些化合物的方法及其用于防治有害微生物 ，以及新型中间体及其制备方法。