公开(公告)号：US06350748B1

公开(公告)日：2002-02-26

申请号：US09529817

申请日：2000-06-02

申请人： Toshiaki Takeyama ,  Toshimasa Hamada ,  Hiroaki Takahashi ,  Junichi Watanabe ,  Kazuhiro Yamagishi ,  Masanori Nishioka ,  Hiroyuki Suzuki

发明人： Toshiaki Takeyama ,  Toshimasa Hamada ,  Hiroaki Takahashi ,  Junichi Watanabe ,  Kazuhiro Yamagishi ,  Masanori Nishioka ,  Hiroyuki Suzuki

IPC分类号： C07D40306

CPC分类号： C07D249/08 ,  A01N43/653 ,  A01N43/84 ,  A01N43/90 ,  C07D249/12 ,  C07D403/12 ,  C07D471/04

摘要： A sulfamoyl compound of the general formulae (1): wherein R1 and R2 are each independently C1-4 alkyl, or R1 and R2 together are C4-6 alkylene or C4-6 alkyleneoxy, Y is H, halogen, C1-8 alkyl, C1-8 alkoxy, C1-8 alkylthio, C1-8 haloalkyl, C1-8 haloalkoxy or C1-8 haloalkylthio, A is a predetermined heterocyclic group, B is a predetermined heterocyclic group which is identical with or different from A, W is a chemical bond or O, V is O or S, D, E, F and G are each independently N, CR7, CR8, CR9 or CR10, and R3, R4, R5, R6, R7, R8, R9, R10 and R11 are each independently predetermined group such as H, or an unsubstituted or substituted aliphatic, aromatic or heterocyclic group. The sulfamoyl compound is useful as an agricultural and horticultural fungicide.

摘要翻译： 通式（1）的氨磺酰基化合物：其中R 1和R 2各自独立地为C 1-4烷基，或者R 1和R 2一起为C 4-6亚烷基或C 4-6亚烷氧基，Y为H，卤素，C 1-8烷基，C 1 烷氧基，C 1-8烷硫基，C 1-8卤代烷基，C 1-8卤代烷氧基或C 1-8卤代烷硫基，A是预定的杂环基，B是与A相同或不同的预定杂环基，W是化学 键或O，V为O或S，D，E，F和G各自独立地为N，CR7，CR8，CR9或CR10，R3，R4，R5，R6，R7，R8，R9，R10和R11各自独立地为 预定基团如H，或未取代或取代的脂族，芳族或杂环基团。 氨磺酰化合物可用作农业和园艺杀真菌剂。

公开(公告)号：US07067656B2

公开(公告)日：2006-06-27

申请号：US10614871

申请日：2003-07-09

申请人： Toshiaki Takeyama ,  Toshimasa Hamada ,  Hiroaki Takahashi ,  Junichi Watanabe ,  Kazuhiro Yamagishi ,  Masanori Nishioka ,  Hiroyuki Suzuki

发明人： Toshiaki Takeyama ,  Toshimasa Hamada ,  Hiroaki Takahashi ,  Junichi Watanabe ,  Kazuhiro Yamagishi ,  Masanori Nishioka ,  Hiroyuki Suzuki

IPC分类号： C07D413/00 ,  C07D211/06 ,  C07D401/00 ,  C07D405/00 ,  C07D409/00

CPC分类号： C07D249/08 ,  A01N43/653 ,  A01N43/84 ,  A01N43/90 ,  C07D249/12 ,  C07D403/12 ,  C07D471/04

摘要： A sulfamoyl compound of the general formulae (1): wherein R1 and R2 are each independently C1-4 alkyl, or R1 and R2 together are C4-6 alkylene or C4-6 alkyleneoxy, Y is H, halogen, C1-8 alkyl, C1-8 alkoxy, C1-8 alkylthio, C1-8 haloalkyl, C1-8 haloalkoxy or C1-8 haloalkylthio, A is a predetermined heterocyclic group, B is a predetermined heterocyclic group which is identical with or different from A, W is a chemical bond or O, V is O or S, D, E, F and G are each independently N, CR7, CR8, CR9 or CR10, and R3, R4, R5, R6, R7, R8, R9, R10 and R11 are each independently predetermined group such as H, or an unsubstituted or substituted aliphatic, aromatic or heterocyclic group. The sulfamoyl compound is useful as an agricultural and horticultural fungicide.

摘要翻译： 通式（1）的氨磺酰基化合物：其中R 1和R 2各自独立地为C 1-4烷基，或R 1， SUP 1和R 2一起为C 4-6亚烷基或C 4-6亚烷基氧基，Y为H，卤素 C 1-8烷基，C 1-8烷氧基，C 1-8烷硫基，C 1-8烷基 卤代烷基，C 1-8卤代烷氧基或C 1-8卤代烷硫基，A为预定的杂环基，B为与A相同或不同的预定杂环基 W是化学键或O，V是O或S，D，E，F和G各自独立地为N，CR 7，CR 8，CR 0 > 9或CR 10，R 3，R 4，R 5，R 5， R 6，R 7，R 8，R 9，R 10和R 10， SUP> 11个各自独立地是预定的基团，例如H，或未取代或取代的脂族，芳族或杂环基团。 氨磺酰化合物可用作农业和园艺杀真菌剂。

公开(公告)号：US06620812B2

公开(公告)日：2003-09-16

申请号：US09964357

申请日：2001-09-28

申请人： Toshiaki Takeyama ,  Toshimasa Hamada ,  Hiroaki Takahashi ,  Junichi Watanabe ,  Kazuhiro Yamagishi ,  Masanori Nishioka ,  Hiroyuki Suzuki

发明人： Toshiaki Takeyama ,  Toshimasa Hamada ,  Hiroaki Takahashi ,  Junichi Watanabe ,  Kazuhiro Yamagishi ,  Masanori Nishioka ,  Hiroyuki Suzuki

IPC分类号： C07D40306

CPC分类号： C07D249/08 ,  A01N43/653 ,  A01N43/84 ,  A01N43/90 ,  C07D249/12 ,  C07D403/12 ,  C07D471/04

摘要： A sulfamoyl compound of the general formulae (1): wherein R1 and R2 are each independently C1-4 alkyl, or R1 and R2 together are C4-6 alkylene or C4-6 alkyleneoxy, Y is H, halogen, C1-8 alkyl, C1-8 alkoxy, C1-8 alkylthio, C1-8 haloalkyl, C1-8 haloalkoxy or C1-8 haloalkylthio, A is a predetermined heterocyclic group, B is a predetermined heterocyclic group which is identical with or different from A, W is a chemical bond or O, V is O or S, D, E, F and G are each independently N, CR7, CR8, CR9 or CR10, and R3, R4, R5, R6, R7, R8, R9, R10 and R11 are each independently predetermined group such as H, or an unsubstituted or substituted aliphatic, aromatic or heterocyclic group. The sulfamoyl compound is useful as an agricultural and horticultural fungicide.

公开(公告)号：US5039694A

公开(公告)日：1991-08-13

申请号：US344895

申请日：1989-04-28

申请人： Hideo Suzuki ,  Takeshi Mita ,  Toshiaki Takeyama ,  Yoshinori Ochiai ,  Masami Hanaue ,  Masao Nishikubo ,  Kazuhiro Yamagishi

发明人： Hideo Suzuki ,  Takeshi Mita ,  Toshiaki Takeyama ,  Yoshinori Ochiai ,  Masami Hanaue ,  Masao Nishikubo ,  Kazuhiro Yamagishi

IPC分类号： A01N43/50 ,  A01N43/56 ,  A01N43/653 ,  A01N43/74 ,  A01N43/80 ,  C07D231/14 ,  C07D233/90 ,  C07D261/18 ,  C07D263/34 ,  C07D275/02 ,  C07D275/03 ,  C07D277/56 ,  C07D405/12 ,  C07D409/12 ,  C07D413/12 ,  C07D417/12 ,  C07D521/00

CPC分类号： C07D263/34 ,  A01N43/50 ,  A01N43/56 ,  A01N43/653 ,  A01N43/74 ,  A01N43/80 ,  C07D231/12 ,  C07D231/14 ,  C07D233/56 ,  C07D233/90 ,  C07D249/08 ,  C07D261/18 ,  C07D275/03 ,  C07D277/56 ,  C07D405/12 ,  C07D409/12 ,  C07D413/12 ,  C07D417/12

摘要： Disclosed are substituted-amido derivatives of a general formula (I): ##STR1## in which R.sub.1 represents a group as specifically defined herein; R.sub.2 represents a hydrogen atom, a methyl group, a methoxy group or a halogne atom; B represents a 5-membered hetero-aromatic group as specifically defined herein, as well as a method for preparation of the said derivatives and a fungicide containing the said derivative as an active ingredient.

摘要翻译： 公开了通式（I）的取代的酰氨基衍生物：其中R 1表示本文具体定义的基团; R2表示氢原子，甲基，甲氧基或卤代原子; B表示本文具体定义的5元杂芳族基团，以及制备所述衍生物的方法和含有所述衍生物作为活性成分的杀真菌剂。

公开(公告)号：US5126362A

公开(公告)日：1992-06-30

申请号：US412220

申请日：1989-09-25

申请人： Hideo Suzuki ,  Takeshi Mita ,  Toshiaki Takeyama ,  Masami Hanaue ,  Masao Nishikubo ,  Kazuhiro Yamagishi

发明人： Hideo Suzuki ,  Takeshi Mita ,  Toshiaki Takeyama ,  Masami Hanaue ,  Masao Nishikubo ,  Kazuhiro Yamagishi

IPC分类号： A01N43/08 ,  A01N43/10 ,  A01N43/40 ,  A01N43/56 ,  A01N47/06 ,  A01N47/24 ,  C07D231/12 ,  C07D231/14 ,  C07D333/24 ,  C07D405/12 ,  C07D409/12

CPC分类号： C07D405/12 ,  A01N43/08 ,  A01N43/10 ,  A01N43/40 ,  A01N43/56 ,  A01N47/06 ,  A01N47/24 ,  C07D231/14 ,  C07D333/24 ,  C07D409/12

摘要： An oxime derivative represented by the general formula [1]: ##STR1## wherein A, B, Y and W represent each a specified group, and an optically active isomer thereof and a fungicide for agricultural and horticultural use for containing said derivative or an optically active isomer thereof as an active ingredient are disclosed.

公开(公告)号：US6043262A

公开(公告)日：2000-03-28

申请号：US125988

申请日：1998-11-24

申请人： Norihito Hayakawa ,  Masatoshi Baba ,  Norihiro Suwa ,  Kazuhiro Yamagishi

发明人： Norihito Hayakawa ,  Masatoshi Baba ,  Norihiro Suwa ,  Kazuhiro Yamagishi

IPC分类号： A01N43/78 ,  C07D277/54 ,  C07D277/56

CPC分类号： C07D277/56 ,  A01N43/78

摘要： The present invention provides thifluzamide which has changed its crystalline form, its preparation method, and a pesticide composition containing thifluzamide as its effective ingredient. The rate of dissolution of the thifluzamide obtained is high and the pesticide compounds containing it has improved efficacy.

摘要翻译： PCT No.PCT / JP97 / 00613 Sec。 371日期：1998年11月24日 102（e）1998年11月24日PCT PCT 1997年2月28日提交PCT公布。 公开号WO97 / 31908 日期1997年9月4日本发明提供了改变其结晶形式的噻泊胺，其制备方法和含有thifluzamide作为其有效成分的农药组合物。 获得的thifluzamide的溶出速度高，含有的杀虫剂化合物具有改善的疗效。

公开(公告)号：US5837721A

公开(公告)日：1998-11-17

申请号：US804160

申请日：1997-02-20

申请人： Norihito Hayakawa ,  Masatoshi Baba ,  Norihiro Suwa ,  Kazuhiro Yamagishi

发明人： Norihito Hayakawa ,  Masatoshi Baba ,  Norihiro Suwa ,  Kazuhiro Yamagishi

IPC分类号： C07D277/20 ,  A01N43/78 ,  C07D277/56

CPC分类号： A01N43/78 ,  C07D277/56

摘要： The disclosed invention is thifluzamide with an altered crystalline form, prepared by heat-melting and then cooling, and agricultural chemical compositions comprising such a thifluzamide as its effective ingredient.

摘要翻译： 所公开的发明是通过加热熔化然后冷却制备的具有改变的结晶形式的thifluzamide以及包含这种thifluzamide作为其有效成分的农业化学组合物。