Substituted 1-aryl-3-tert.-butyl-pyrazoles
    3.
    发明授权
    Substituted 1-aryl-3-tert.-butyl-pyrazoles 失效
    取代的1-芳基-3-叔丁基 - 吡唑

    公开(公告)号:US4826867A

    公开(公告)日:1989-05-02

    申请号:US89474

    申请日:1987-08-25

    摘要: Insecticidally and acaricidally active novel 1-aryl-3-tert.-butyl-pyrazoles of the formula ##STR1## in which R.sup.1 represents nitro or halogen,R.sup.2 represents halogen or the --NR.sup.3 R.sup.4 group, and also may represent hydrogen when R.sup.1 denotes halogen,whereR.sup.3 represents hydrogen, in each case optionally substituted alkyl, alkenyl or alkinyl, and in each case optionally substituted cycloalkyl or cycloalkylalkyl andR.sup.4, independently of R.sup.3, represents the same radicals as R.sup.3l , and, in addition, a ##STR2## radical, where X represents oxygen or sulphur andR.sup.5 represents hydrogen, alkyl, alkenyl, alkinyl, halogenoalkyl, alkoxyalkyl, alkylthioalkyl, optionally substituted cycloalkyl, optionally substituted aryl, alkoxy, alkylthio, optionally substituted aryloxy, optionally substituted arylthio, alkylamino, dialkylamino or optionally substituted arylamino; andAr represents optionally substituted phenyl, apart from dinitrophenyl, or optionally substituted pyridyl. Intermediates where R.sup.1 is replaced by hydrogen are also new and are also pesticidally active.

    摘要翻译: 杀虫剂和杀螨剂活性的式“IMAGE”的1-芳基-3-叔丁基 - 吡唑,其中R 1表示硝基或卤素,R 2表示卤素或-NR 3 R 4基团,当R1表示卤素时也可以表示氢, 其中R 3表示氢,在各种情况下均为任选取代的烷基,烯基或炔基,并且在每种情况下为任选取代的环烷基或环烷基烷基,R 4独立于R 3,表示与R 3相同的基团,另外, 其中X表示氧或硫,R5表示氢,烷基,烯基,炔基,卤代烷基,烷氧基烷基,烷硫基烷基,任选取代的环烷基,任选取代的芳基,烷氧基,烷硫基,任选取代的芳氧基,任选取代的芳硫基,烷基氨基,二烷基氨基或任选取代的芳基氨基 ; Ar表示除二硝基苯基以外的任意取代的苯基,或任意取代的吡啶基。 R1被氢取代的中间体也是新的,也是杀虫活性的。

    4-haloalkylthio-5-amino-1-arylpyrazoles, composition containing them,
and insecticidal and acaricidal method of using them
    6.
    发明授权
    4-haloalkylthio-5-amino-1-arylpyrazoles, composition containing them, and insecticidal and acaricidal method of using them 失效
    4-卤代烷硫基-5-氨基-1-芳基吡唑,含有它们的组合物,以及使用它们的杀虫和杀螨方法

    公开(公告)号:US4771066A

    公开(公告)日:1988-09-13

    申请号:US13741

    申请日:1987-02-12

    摘要: Insecticidally and acarididally active 1-arylpyrazoles of the formula ##STR1## in which R.sup.1 represents hydrogen, alkyl or halogen alkyl,R.sup.2 represents alkyl, alkenyl, alkinyl, cycloalkyl, halogenoalkyl, halogenoalkenyl, alkoxyalkyl, alkylthioalkyl, alkylsulphinylalkyl, alkylsulphonylalkyl, optionally substituted aralkyl or optionally substituted aryl,R.sup.3 represents alkyl, alkenyl, alkinyl, halogenoalkyl, halogenoalkenyl, alkoxyalkyl, alkylthioalkyl, cycloalkyl or optionally substituted aralkyl,R.sup.4 represents alkyl, alkenyl, alkinyl, halogenoalkyl, halogenoalkenyl, alkoxyalkyl, alkylthioalkyl, cycloalkyl or optionally substituted aralkyl, and, in addition, also represents hydrogen in the case where R.sup.3 does not simultaneously represent unsubstituted alkyl, orR.sup.3 and R.sup.4, together with the nitrogen atom to which they are bound, represent a saturated heterocycle, which can optionally contain further heteroatoms,Ar represents in each case optionally substituted phenyl or pyridyl, andn represents a number 0, 1 or 2.

    摘要翻译: 具有式“IMAGE”的杀虫和杀螨活性1-芳基吡唑其中R1代表氢,烷基或卤素烷基,R2代表烷基,烯基,炔基,环烷基,卤代烷基,卤代烯基,烷氧基烷基,烷硫基烷基,烷基亚磺酰基烷基,烷基磺酰基烷基,任选取代的芳烷基或 任选取代的芳基,R 3表示烷基,烯基,炔基,卤代烷基,卤代烯基,烷氧基烷基,烷硫基烷基,环烷基或任选取代的芳烷基,R 4表示烷基,烯基,炔基,卤代烷基,卤代烯基,烷氧基烷基,烷硫基烷基,环烷基或任选取代的芳烷基, 此外,在R3不同时表示未取代的烷基的情况下也表示氢,或者R 3和R 4与它们所连接的氮原子一起代表饱和的杂环,其可以任选地含有另外的杂原子,Ar表示每个 任选取代的苯基或吡啶基,n表示 数字0,1或2。