公开(公告)号：US08288416B2

公开(公告)日：2012-10-16

申请号：US12311243

申请日：2007-09-22

申请人： Vijaykumar Jadgishwar Patil ,  Mahesh Vithalbhai Patel ,  Bharat Kalidas Trivedi ,  Deepak Vijaykumar Dekhane ,  Mohammad Usman Shaikh ,  Yati Chugh ,  Rajesh Prabhakar Chavan ,  Mohammad Alam Jafri

发明人： Vijaykumar Jadgishwar Patil ,  Mahesh Vithalbhai Patel ,  Bharat Kalidas Trivedi ,  Deepak Vijaykumar Dekhane ,  Mohammad Usman Shaikh ,  Yati Chugh ,  Rajesh Prabhakar Chavan ,  Mohammad Alam Jafri

IPC分类号： A61K31/445 ,  C07D413/14

CPC分类号： C07D413/10 ,  C07F9/65583

摘要： The present invention relates to oxazolidinones of Formula I and pharmaceutically acceptable salts, pharmaceutically acceptable solvates or polymorphs thereof. The invention also relates to processes for the preparation of the compound of Formula I and pharmaceutically acceptable salts, pharmaceutically acceptable solvates or polymorphs thereof, and to pharmaceutical compositions containing the compounds of Formula I and pharmaceutically acceptable salts, pharmaceutically acceptable solvates or polymorphs thereof and to methods for treating or preventing microbial infections using the compounds of Formula I and pharmaceutically acceptable salts, pharmaceutically acceptable solvates or polymorphs thereof.

摘要翻译： 本发明涉及式I的恶唑烷酮及其药学上可接受的盐，药学上可接受的溶剂化物或其多晶型物。 本发明还涉及制备式I化合物及其药学上可接受的盐，药学上可接受的溶剂合物或多晶型物的方法，以及含有式I化合物及其药学上可接受的盐，药学上可接受的溶剂化物或多晶型物的药物组合物，以及 使用式I化合物及其药学上可接受的盐，药学上可接受的溶剂合物或多晶型物治疗或预防微生物感染的方法。

公开(公告)号：US20100120721A1

公开(公告)日：2010-05-13

申请号：US12311243

申请日：2007-09-22

申请人： Vijaykumar Jadgishwar Patil ,  Mahesh Vithalbhai Patel ,  Bharat Kalidas Trivedi ,  Deepak Vijaykumar Dekhane ,  Mohammad Usman Shaikh ,  Yati Chugh ,  Rajesh Prabhakar Chavan ,  Mohammad Alam Jafri

发明人： Vijaykumar Jadgishwar Patil ,  Mahesh Vithalbhai Patel ,  Bharat Kalidas Trivedi ,  Deepak Vijaykumar Dekhane ,  Mohammad Usman Shaikh ,  Yati Chugh ,  Rajesh Prabhakar Chavan ,  Mohammad Alam Jafri

IPC分类号： A61K31/454 ,  C07F9/117 ,  C07D413/14 ,  C07D413/10 ,  A61K31/661 ,  A61P31/04 ,  A61P31/00

CPC分类号： C07D413/10 ,  C07F9/65583

摘要： The present invention relates to oxazolidinones of Formula I and pharmaceutically acceptable salts, pharmaceutically acceptable solvates or polymorphs thereof. The invention also relates to processes for the preparation of the compound of Formula I and pharmaceutically acceptable salts, pharmaceutically acceptable solvates or polymorphs thereof, and to pharmaceutical compositions containing the compounds of Formula I and pharmaceutically acceptable salts, pharmaceutically acceptable solvates or polymorphs thereof and to methods for treating or preventing microbial infections using the compounds of Formula I and pharmaceutically acceptable salts, pharmaceutically acceptable solvates or polymorphs thereof.

摘要翻译： 本发明涉及式I的恶唑烷酮及其药学上可接受的盐，药学上可接受的溶剂化物或其多晶型物。 本发明还涉及制备式I化合物及其药学上可接受的盐，药学上可接受的溶剂合物或多晶型物的方法，以及含有式I化合物及其药学上可接受的盐，药学上可接受的溶剂化物或多晶型物的药物组合物，以及 使用式I化合物及其药学上可接受的盐，药学上可接受的溶剂合物或多晶型物治疗或预防微生物感染的方法。