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公开(公告)号：US5493034A
公开(公告)日：1996-02-20
申请号：US443522
申请日：1995-05-18
IPC分类号： A01N43/28 , A01N43/30 , C07D317/72 , C07D327/04 , C07D411/12
CPC分类号： C07D317/72 , A01N43/28 , A01N43/30 , C07D327/04 , C07D411/12
摘要： Fungicidally active compounds of the formula ##STR1## in which X represents oxygen or sulphur,R represents cycloalkyl, or represents optionally substituted aryl, or represents the radical ##STR2## R.sup.1 and R.sup.2 each independently is hydrogen or an organic radical, or together with the nitrogen atom form a heterocyclic radical,R.sup.3 represents hydrogen, alkyl or optionally substituted aryl, andR.sup.4 represents alkyl or cycloalkyl, or represents optionally substituted aryl,but wherein R.sup.3 and R.sup.4 may not simultaneously represent methyl,and acid addition salts thereof, as well as intermediates therefor.
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公开(公告)号：US4988729A
公开(公告)日：1991-01-29
申请号：US423607
申请日：1989-10-17
申请人： Wolfgang Kramer , Joachim Weissmuller , Graham Holmwood , Dieter Berg , Stefan Dutzmann , Wilhelm Brandes , Gerd Hanssler , Paul Reinecke
发明人： Wolfgang Kramer , Joachim Weissmuller , Graham Holmwood , Dieter Berg , Stefan Dutzmann , Wilhelm Brandes , Gerd Hanssler , Paul Reinecke
IPC分类号： A01N43/08 , A01N43/28 , C07D307/14 , C07D307/22 , C07D317/28 , C07D327/04 , C07D407/12 , C07D417/12
CPC分类号： C07D407/12 , A01N43/08 , A01N43/28 , C07D307/14 , C07D317/28 , C07D327/04
摘要： Combattting fungi and bacteria with aminomethylheterocyclic compounds of the formula ##STR1## in which R.sup.1 represents hydrogen, alkyl, alkenyl, in each case optionally substituted tetrahydronaphthyl, decahydronaphthyl, cycloalkyl or cycloalkenyl, furthermore alkyl which is substituted by cycloalkyl, cycloalkenyl, cycloalkyloxy or cycloalkylthio, where the cyclic radicals may optionally be substituted, furthermore optionally substituted aryl, in addition alkyl which is substituted by aryl, aryloxy, arylthio, arylsulphinyl or arylsulphonyl, or alkenyl which is substituted by aryl, where the aryl radicals may in each case optionally be substituted;R.sup.2 represents hydrogen or methyl,R.sup.3 represents alkyl, alkenyl, alkinyl, alkoxyalkyl, hydroxyalkyl, hydroxyalkoxyalkyl, dialkoxyalkyl, or in each case optionally substituted cycloalkyl, cycloalkylalkyl, aryl, aralkyl, aralkenyl, furanylalkyl, tetrahydrofuranylalkyl, tetrahydropyranylalkyl, dioxolanylalkyl or dioxanylalkyl, andX represents oxygen, sulphur or a CH.sub.2 group,or acid additon salts thereof. Many of the compounds wherein R.sup.1 has a narrower meaning are new.
摘要翻译： 用下式（Ⅰ）的氨基甲基杂环化合物与R1代表氢，烷基，烯基，各取代四氢萘基，十氢萘基，环烷基或环烯基，以及被环烷基，环烯基，环烷氧基 或环烷硫基，其中环状基团可任选被取代，此外任选取代的芳基，另外被芳基，芳氧基，芳硫基，芳基亚磺酰基或芳基磺酰基取代的烷基或被芳基取代的烯基，其中芳基可以在每种情况下 任选被取代; R 2表示氢或甲基，R 3表示烷基，烯基，炔基，烷氧基烷基，羟基烷基，羟基烷氧基烷基，二烷氧基烷基，或在每种情况下任选取代的环烷基，环烷基烷基，芳基，芳烷基，芳烯基，呋喃基烷基，四氢呋喃基烷基，四氢吡喃基烷基，二氧戊环烷基或二烷基烷基，X 代表氧，硫或CH2基，或其酸加成盐。 其中R1具有较窄含义的许多化合物是新的。
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公开(公告)号：US4985421A
公开(公告)日：1991-01-15
申请号：US395231
申请日：1989-08-17
IPC分类号： A01N43/30 , C07D317/72 , C07D405/06 , C07D407/06 , C07D407/12 , C07D413/06
CPC分类号： C07D317/72 , C07D407/12
摘要： Fungicidal substituted dioxolanylethylamine of the formula ##STR1## in which R represents alkyl, or represents in each case optionally substituted cycloalkylalkyl, aralkyl, cycloalkyl or aryl, andR.sup.1 and R.sup.2 independently of one another each represents hydrogen, alkyl, alkenyl, alkinyl, alkoxyalkyl, dialkoxyalkyl, hydroxyalkyl, hydroxyalkoxyalkyl, alkoxycarbonylalkyl, dioxolanylalkyl, dioxanylalkyl or oxolanylalkyl, or represents in each case optionally substituted cycloalkylalkyl, cycloalkyl, aralkyl, aralkenyl or aryl, orR.sup.1 and R.sup.2, together with the nitrogen atom to which they are bonded, represent an optionally substituted saturated heterocyclic radical, which can optionally contain further hetero atoms,and acid addition salts thereof.Intermediates wherein the amino group is an electron-withdrawing leaving group are also new.
摘要翻译： 式（I）的杀真菌取代的二氧戊环二乙胺其中R代表烷基，或在每种情况下表示任选取代的环烷基烷基，芳烷基，环烷基或芳基，R 1和R 2彼此独立地表示氢，烷基，链烯基，炔基 烷氧基烷基，二烷氧基烷基，羟烷基，羟基烷氧基烷基，烷氧基羰基烷基，二氧戊环烷基，二烷基烷基或氧代烷基烷基，或在各种情况下表示任选取代的环烷基烷基，环烷基，芳烷基，芳烯基或芳基，或者R1和R2与它们所键合的氮原子一起， 代表任选取代的饱和杂环基团，其可任选地含有其它杂原子，及其酸加成盐。 其中氨基是吸电子离去基团的中间体也是新的。
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公开(公告)号：US5177103A
公开(公告)日：1993-01-05
申请号：US616155
申请日：1990-11-20
IPC分类号： A01N43/28 , A01N43/30 , C07D317/72 , C07D327/04 , C07D411/12
CPC分类号： C07D317/72 , A01N43/28 , A01N43/30 , C07D327/04 , C07D411/12
摘要： Fungicidally active compounds of the formula ##STR1## in which X represents oxygen or sulphur,R represents cycloalkyl, or represents optionally substituted aryl, or represents the radical ##STR2## R.sup.1 and R.sup.2 each independently is hydrogen or an organic radical, or together with the nitrogen atom form a heterocyclic radical,R.sup.3 represents hydrogen, alkyl or optionally substituted aryl, andR.sup.4 represents alkyl or cycloalkyl, or represents optionally substituted aryl,but wherein R.sup.3 and R.sup.4 may not simultaneously represent methyl,and acid addition salts thereof, as well as intermediates therefor.
摘要翻译： 式（I）的杀真菌活性化合物，其中X表示氧或硫，R表示环烷基，或表示任选取代的芳基，或表示基团R 1和R 2各自独立地为氢或有机基团，或 与氮原子一起形成杂环基，R 3表示氢，烷基或任选取代的芳基，R 4表示烷基或环烷基，或表示任选取代的芳基，但其中R 3和R 4可不同时表示甲基，及其酸加成盐， 以及其中间体。
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公开(公告)号：US5376660A
公开(公告)日：1994-12-27
申请号：US924764
申请日：1992-08-03
IPC分类号： A01N43/28 , A01N43/30 , C07D317/72 , C07D327/04 , C07D411/12 , C07D413/06 , C07D417/06
CPC分类号： C07D317/72 , A01N43/28 , A01N43/30 , C07D327/04 , C07D411/12
摘要： Fungicidally active compounds of the formula ##STR1## in which X represents oxygen or sulphur,R represents cycloalkyl, or represents optionally substituted aryl, or represents the radical ##STR2## R.sup.1 and R.sup.2 each independently is hydrogen or an organic radical, or together with the nitrogen atom form a heterocyclic radical,R.sup.3 represents hydrogen, alkyl or optionally substituted aryl, andR.sup.4 represents alkyl or cycloalkyl, or represents optionally substituted aryl,but wherein and R.sup.3 and R.sup.4 may not simultaneously represent methyl,and acid addition salts thereof, as well as intermediates therefore.
摘要翻译： 式（I）的杀真菌活性化合物，其中X表示氧或硫，R表示环烷基，或表示任选取代的芳基，或表示基团R 1和R 2各自独立地为氢或有机基团，或 与氮原子一起形成杂环基，R 3表示氢，烷基或任选取代的芳基，R 4表示烷基或环烷基，或表示任选取代的芳基，但其中R 3和R 4可不同时表示甲基，及其酸加成盐 ，以及中间体。
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公开(公告)号：US5128368A
公开(公告)日：1992-07-07
申请号：US595143
申请日：1990-10-10
申请人： Wolfgang Kramer , Joachim Weissmuller , Graham Holmwood , Dieter Berg , Stefan Dutzmann , Wilhelm Brandes , Gerd Hanssler , Paul Reinecke
发明人： Wolfgang Kramer , Joachim Weissmuller , Graham Holmwood , Dieter Berg , Stefan Dutzmann , Wilhelm Brandes , Gerd Hanssler , Paul Reinecke
IPC分类号： A01N43/08 , A01N43/28 , C07D307/14 , C07D307/22 , C07D317/28 , C07D327/04 , C07D407/12 , C07D417/12
CPC分类号： C07D407/12 , A01N43/08 , A01N43/28 , C07D307/14 , C07D317/28 , C07D327/04
摘要： Combatting fungi and bacteria with aminomethylheterocyclic compounds of the formula ##STR1## in which R.sup.1 represents hydrogen, alkyl, alkenyl, in each case optionally substituted tetrahydronaphthyl, decahydronaphthyl, cycloalkyl or cycloalkenyl, furthermore alkyl which is substituted by cycloalkyl, cycloalkenyl, cycloalkyloxy or cycloalkylthio, where the cyclic radicals may optionally be substituted, furthermore optionally substituted aryl, in addition alkyl which is substituted by aryl, aryloxy, arylthio, arylsulphinyl or arylsulphonyl, or alkenyl which is substituted by aryl, where the aryl radicals may in each case optionally be substituted;R.sup.2 represents hydrogen or methyl,R.sup.3 represents alkyl, alkenyl, alkinyl, alkoxyalkyl, hydroxyalkyl, hydroxyalkoxyalkyl, dialkoxyalkyl, or in each case optionally substituted cycloalkyl, cycloalkylalkyl, aryl, aralkyl, aralkenyl, furanylalkyl, tetrahydrofuranylalkyl, tetrahydropyranylalkyl, dioxolanylalkyl or dioxanylalkyl, andX represents oxygen, sulphur or a CH.sub.2 group,or acid addition salts thereof.Many of the compounds wherein R.sup.1 has a narrower meaning are new.
摘要翻译： 用下式（Ⅰ）的氨基甲基杂环化合物与R1代表氢，烷基，烯基，各取代四氢萘基，十氢萘基，环烷基或环烯基，以及被环烷基，环烯基，环烷基 或环烷硫基，其中环状基团可任选被取代，此外任选取代的芳基，另外被芳基，芳氧基，芳硫基，芳基亚磺酰基或芳基磺酰基取代的烷基或被芳基取代的烯基，其中芳基可以在每种情况下 任选被取代; R 2表示氢或甲基，R 3表示烷基，烯基，炔基，烷氧基烷基，羟基烷基，羟基烷氧基烷基，二烷氧基烷基，或在每种情况下任选取代的环烷基，环烷基烷基，芳基，芳烷基，芳烯基，呋喃基烷基，四氢呋喃基烷基，四氢吡喃基烷基，二氧戊环烷基或二烷基烷基，X 代表氧，硫或CH2基，或其酸加成盐。 其中R1具有较窄含义的许多化合物是新的。
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公开(公告)号：US5010101A
公开(公告)日：1991-04-23
申请号：US395391
申请日：1989-08-17
IPC分类号： A01N43/28 , A01N43/30 , A01N43/36 , A01N43/40 , A01N43/46 , A01N43/84 , C07D317/72 , C07D327/04 , C07D411/12
CPC分类号： C07D317/72 , A01N43/28 , A01N43/30 , C07D327/04 , C07D411/12
摘要： Fungicidally active compounds of the formula ##STR1## in which X represents oxygen or sulphur,R represents cycloalkyl, or represents optionally substituted aryl, or represents the radical ##STR2## R.sup.1 and R.sup.2 each independently is hydrogen or an organic radical, or together with the nitrogen atom form a heterocyclic radical,R.sup.3 represents hydrogen, alkyl or optionally substituted aryl, andR.sup.4 represents alkyl or cycloalkyl, or represents optionally substituted aryl,but wherein R.sup.3 and R.sup.4 may not simultaneously represent methyl,and acid addition salts thereof, as well as intermediates therefor.
摘要翻译： 式（I）的杀真菌活性化合物，其中X表示氧或硫，R表示环烷基，或表示任选取代的芳基，或表示基团R 1和R 2各自独立地为氢或有机基团，或 与氮原子一起形成杂环基，R 3表示氢，烷基或任选取代的芳基，R 4表示烷基或环烷基，或表示任选取代的芳基，但其中R 3和R 4可不同时表示甲基，及其酸加成盐， 以及其中间体。
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公开(公告)号：US5447927A
公开(公告)日：1995-09-05
申请号：US279933
申请日：1994-07-25
IPC分类号： A01N43/28 , A01N43/30 , C07D317/72 , C07D327/04 , C07D411/12 , A01N43/84 , A01N43/46 , C07D411/06 , C07D413/06
CPC分类号： C07D317/72 , A01N43/28 , A01N43/30 , C07D327/04 , C07D411/12
摘要： Fungicidally active compounds of the formula ##STR1## in which X represents oxygen or sulphur,R represents cycloalkyl, or represents optionally substituted aryl, or represents the radical ##STR2## R.sup.1 and R.sup.2 each independently is hydrogen or an organic radical, or together with the nitrogen atom form a heterocyclic radical,R.sup.3 represents hydrogen, alkyl or optionally substituted aryl, andR.sup.4 represents alkyl or cycloalkyl, or represents optionally substituted aryl,but wherein R.sup.3 and R.sup.4 may not simultaneously represent methyl,and acid addition salts thereof, as well as intermediates therefor.
摘要翻译： 式（I）的杀真菌活性化合物，其中X表示氧或硫，R表示环烷基，或表示任选取代的芳基，或表示基团R 1和R 2各自独立地为氢或有机基团，或 与氮原子一起形成杂环基，R 3表示氢，烷基或任选取代的芳基，R 4表示烷基或环烷基，或表示任选取代的芳基，但其中R 3和R 4可不同时表示甲基，及其酸加成盐， 以及其中间体。
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公开(公告)号：US4851405A
公开(公告)日：1989-07-25
申请号：US161830
申请日：1988-02-29
IPC分类号： A01N43/28 , A01N43/30 , C07D317/72 , C07D327/04 , C07D405/06 , C07D407/12 , C07D411/06 , C07D411/12 , C07D413/06
CPC分类号： C07D317/72 , A01N43/28 , A01N43/30 , C07D327/04 , C07D407/12 , C07D411/12
摘要： Fungicidally effective aminomethyl heterocyclic compounds of the formula ##STR1## in which X represents oxygen or sulphur,R represents hydrogen or alkyl, or represents in each case optionally substituted cyclohexyl or phenyl andR.sup.1 and R.sup.2 independently of one another each represent hydrogen, alkyl, alkenyl, alkinyl, alkoxyalkyl, dialkoxyalkyl, hydroalkyl, hydroxyalkoxyalkyl, alkoxycarbonylalkyl, dioxolanylalkyl, dioxanylalkyl or oxolanylalkyl, or represent in each case optionally substituted cycloalkylalkyl, cycloalkyl, aralkyl, aralkenyl or aryl, orR.sup.1 and R.sup.2, together with the nitrogen atom to which they are bonded, represent an optionally substituted saturated heterocyclic radical, which can optionally contain further hetero atoms,or acid addition salts thereof.
摘要翻译： 化学式为“IMAGE”的杀真菌有效的氨基甲基杂环化合物，其中X表示氧或硫，R表示氢或烷基，或在各种情况下表示任选取代的环己基或苯基，R 1和R 2彼此独立地表示氢，烷基，烯基 ，烷氧基烷基，烷氧基烷基，烷氧基烷基，二烷氧基烷基，氢烷基，羟基烷氧基烷基，烷氧基羰基烷基，二氧戊环烷基，二烷基烷基或氧代烷基烷基，或在每种情况下表示任选取代的环烷基烷基，环烷基，芳烷基，芳烯基或芳基，或R 1和R 2与它们所在的氮原子一起 代表任选取代的饱和杂环基，其可以任选地含有另外的杂原子，或其酸加成盐。
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公开(公告)号：US4713379A
公开(公告)日：1987-12-15
申请号：US735498
申请日：1985-05-17
申请人： Wolfgang Kramer , Joachim Weissmuller , Wolf Reiser , Dieter Berg , Wilhelm Brandes , Paul Reinecke
发明人： Wolfgang Kramer , Joachim Weissmuller , Wolf Reiser , Dieter Berg , Wilhelm Brandes , Paul Reinecke
IPC分类号： A01N43/36 , A01N43/40 , A01N43/46 , A01N43/50 , A01N43/54 , A01N43/60 , A01N43/653 , A01N43/84 , A01N47/38 , A01N47/42 , A01N43/64
CPC分类号： A01N43/84 , A01N43/36 , A01N43/40 , A01N43/50 , A01N43/54 , A01N43/60 , A01N43/653 , A01N47/38 , A01N47/42
摘要： A synergistic fungicidal composition comprising a fungicidally effective amount of at least one amino compound of the formula ##STR1## in which R represents optionally substituted, cycloalkyl or optionally substituted aryl,R.sup.1 represents hydrogen or alkyl,R.sup.2 represents alkyl,R.sup.3 represents alkyl andR.sup.4 represents alkyl, alkenyl or alkinyl, orR.sup.3 and R.sup.4, together with the nitrogen atom to which they are bonded, represent an optionally substituted saturated heterocyclic radical, which can contain further hetero-atoms,X represents oxygen or sulphur,Y represents oxygen, sulphur or the methylene group,m represents 0 or 1 andn represents 0 or 1,or an addition product thereof with an acid, metal salt or quaternizing agent, and at least one member selected from the group consisting of several individually known fungicides.
摘要翻译： 一种协同杀真菌组合物，其包含杀真菌有效量的至少一种式“IMAGE”氨基化合物，其中R表示任选取代的环烷基或任选取代的芳基，R 1表示氢或烷基，R 2表示烷基，R 3表示烷基，R 4表示 烷基，烯基或炔基，或者R 3和R 4与它们所键合的氮原子一起代表任选取代的饱和杂环基，其可含有其它杂原子，X表示氧或硫，Y表示氧，硫或 亚甲基，m表示0或1，n表示0或1，或其与酸，金属盐或季铵化剂的加成产物，以及选自几种单独已知的杀真菌剂中的至少一种。
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