公开(公告)号：US4713379A

公开(公告)日：1987-12-15

申请号：US735498

申请日：1985-05-17

申请人： Wolfgang Kramer ,  Joachim Weissmuller ,  Wolf Reiser ,  Dieter Berg ,  Wilhelm Brandes ,  Paul Reinecke

发明人： Wolfgang Kramer ,  Joachim Weissmuller ,  Wolf Reiser ,  Dieter Berg ,  Wilhelm Brandes ,  Paul Reinecke

IPC分类号： A01N43/36 ,  A01N43/40 ,  A01N43/46 ,  A01N43/50 ,  A01N43/54 ,  A01N43/60 ,  A01N43/653 ,  A01N43/84 ,  A01N47/38 ,  A01N47/42 ,  A01N43/64

CPC分类号： A01N43/84 ,  A01N43/36 ,  A01N43/40 ,  A01N43/50 ,  A01N43/54 ,  A01N43/60 ,  A01N43/653 ,  A01N47/38 ,  A01N47/42

摘要： A synergistic fungicidal composition comprising a fungicidally effective amount of at least one amino compound of the formula ##STR1## in which R represents optionally substituted, cycloalkyl or optionally substituted aryl,R.sup.1 represents hydrogen or alkyl,R.sup.2 represents alkyl,R.sup.3 represents alkyl andR.sup.4 represents alkyl, alkenyl or alkinyl, orR.sup.3 and R.sup.4, together with the nitrogen atom to which they are bonded, represent an optionally substituted saturated heterocyclic radical, which can contain further hetero-atoms,X represents oxygen or sulphur,Y represents oxygen, sulphur or the methylene group,m represents 0 or 1 andn represents 0 or 1,or an addition product thereof with an acid, metal salt or quaternizing agent, and at least one member selected from the group consisting of several individually known fungicides.

摘要翻译： 一种协同杀真菌组合物，其包含杀真菌有效量的至少一种式“IMAGE”氨基化合物，其中R表示任选取代的环烷基或任选取代的芳基，R 1表示氢或烷基，R 2表示烷基，R 3表示烷基，R 4表示 烷基，烯基或炔基，或者R 3和R 4与它们所键合的氮原子一起代表任选取代的饱和杂环基，其可含有其它杂原子，X表示氧或硫，Y表示氧，硫或 亚甲基，m表示0或1，n表示0或1，或其与酸，金属盐或季铵化剂的加成产物，以及选自几种单独已知的杀真菌剂中的至少一种。

公开(公告)号：US4755521A

公开(公告)日：1988-07-05

申请号：US55487

申请日：1987-05-28

申请人： Wolfgang Kramer ,  Joachim Weissmuller ,  Wolf Reiser ,  Dieter Berg ,  Wilhelm Brandes ,  Paul Reinecke

发明人： Wolfgang Kramer ,  Joachim Weissmuller ,  Wolf Reiser ,  Dieter Berg ,  Wilhelm Brandes ,  Paul Reinecke

IPC分类号： A01N43/36 ,  A01N43/40 ,  A01N43/46 ,  A01N43/50 ,  A01N43/54 ,  A01N43/60 ,  A01N43/653 ,  A01N43/84 ,  A01N47/38 ,  A01N47/42 ,  A01N43/64

CPC分类号： A01N43/84 ,  A01N43/36 ,  A01N43/40 ,  A01N43/50 ,  A01N43/54 ,  A01N43/60 ,  A01N43/653 ,  A01N47/38 ,  A01N47/42

摘要： A synergistic fungicidal composition comprising a fungicidally effective amount of at least one amino compound of the formula ##STR1## in which R represents optionally substituted cycloalkyl or optionally substituted aryl,R.sup.1 represents hydrogen or alkyl,R.sup.2 represents alkyl,R.sup.3 represents alkyl andR.sup.4 represents alkyl, alkenyl or alkinyl, orR.sup.3 and R.sup.4, together with the nitrogen atom to which they are bonded, represent an optionally substituted saturated heterocyclic radical, which can contain further hetero-atoms,X represents oxygen or sulphur,Y represents oxygen, sulphur or the methylene group,m represents 0 or 1 andn represents 0 or 1,or an addition product thereof with an acid, metal salt or quaternizing agent, and at least one member selected from the group consisting of several individually known fungicides.

摘要翻译： 一种协同杀真菌组合物，其包含杀真菌有效量的至少一种下式的氨基化合物，其中R表示任选取代的环烷基或任选取代的芳基，R 1表示氢或烷基，R 2表示烷基，R 3表示烷基，R 4表示烷基 ，链烯基或炔基，或者R 3和R 4与它们所键合的氮原子一起代表任选取代的饱和杂环基，其可含有其它杂原子，X表示氧或硫，Y表示氧，硫或 亚甲基，m表示0或1，n表示0或1，或其与酸，金属盐或季铵化剂的加成产物，以及选自几种单独已知的杀真菌剂中的至少一种。

公开(公告)号：US4826857A

公开(公告)日：1989-05-02

申请号：US176479

申请日：1988-04-01

申请人： Wolfgang Kramer ,  Joachim Weissmuller ,  Wolf Reiser ,  Dieter Berg ,  Wilhelm Brandes ,  Paul Reinecke

发明人： Wolfgang Kramer ,  Joachim Weissmuller ,  Wolf Reiser ,  Dieter Berg ,  Wilhelm Brandes ,  Paul Reinecke

IPC分类号： A01N43/36 ,  A01N43/40 ,  A01N43/46 ,  A01N43/50 ,  A01N43/54 ,  A01N43/60 ,  A01N43/653 ,  A01N43/84 ,  A01N47/38 ,  A01N47/42 ,  A01N43/64

CPC分类号： A01N43/84 ,  A01N43/36 ,  A01N43/40 ,  A01N43/50 ,  A01N43/54 ,  A01N43/60 ,  A01N43/653 ,  A01N47/38 ,  A01N47/42

摘要： A synergistic fungicidal composition comprising a fungicidally effective amount of at least one amino compound of the formula ##STR1## in which R represents optionally substituted cycloalkyl or optionally substituted aryl,R.sup.1 represents hydrogen or alkyl,R.sup.2 represents alkyl,R.sup.3 represents alkyl andR.sup.4 represents alkyl, alkenyl or alkinyl, orR.sup.3 and R.sup.4, together with the nitrogen atom to which they are bonded, represent an optionally substituted saturated heterocyclic radical, which can contain further hetero-atoms,X represents oxygen or sulphur,Y represents oxygen, sulphur or the methylene group,m represents 0 or 1 andn represents 0 or 1,or an addition product thereof with an acid, metal salt or quaternizing agent, and at least one member selected from the group consisting of several individually known fungicides.

摘要翻译： 一种协同杀真菌组合物，其包含杀真菌有效量的至少一种下式的氨基化合物，其中R表示任选取代的环烷基或任选取代的芳基，R 1表示氢或烷基，R 2表示烷基，R 3表示烷基，R 4表示烷基 ，链烯基或炔基，或者R 3和R 4与它们所键合的氮原子一起代表任选取代的饱和杂环基，其可含有其它杂原子，X表示氧或硫，Y表示氧，硫或 亚甲基，m表示0或1，n表示0或1，或其与酸，金属盐或季铵化剂的加成产物，以及选自几种单独已知的杀真菌剂中的至少一种。

公开(公告)号：US4988729A

公开(公告)日：1991-01-29

申请号：US423607

申请日：1989-10-17

申请人： Wolfgang Kramer ,  Joachim Weissmuller ,  Graham Holmwood ,  Dieter Berg ,  Stefan Dutzmann ,  Wilhelm Brandes ,  Gerd Hanssler ,  Paul Reinecke

发明人： Wolfgang Kramer ,  Joachim Weissmuller ,  Graham Holmwood ,  Dieter Berg ,  Stefan Dutzmann ,  Wilhelm Brandes ,  Gerd Hanssler ,  Paul Reinecke

IPC分类号： A01N43/08 ,  A01N43/28 ,  C07D307/14 ,  C07D307/22 ,  C07D317/28 ,  C07D327/04 ,  C07D407/12 ,  C07D417/12

CPC分类号： C07D407/12 ,  A01N43/08 ,  A01N43/28 ,  C07D307/14 ,  C07D317/28 ,  C07D327/04

摘要： Combattting fungi and bacteria with aminomethylheterocyclic compounds of the formula ##STR1## in which R.sup.1 represents hydrogen, alkyl, alkenyl, in each case optionally substituted tetrahydronaphthyl, decahydronaphthyl, cycloalkyl or cycloalkenyl, furthermore alkyl which is substituted by cycloalkyl, cycloalkenyl, cycloalkyloxy or cycloalkylthio, where the cyclic radicals may optionally be substituted, furthermore optionally substituted aryl, in addition alkyl which is substituted by aryl, aryloxy, arylthio, arylsulphinyl or arylsulphonyl, or alkenyl which is substituted by aryl, where the aryl radicals may in each case optionally be substituted;R.sup.2 represents hydrogen or methyl,R.sup.3 represents alkyl, alkenyl, alkinyl, alkoxyalkyl, hydroxyalkyl, hydroxyalkoxyalkyl, dialkoxyalkyl, or in each case optionally substituted cycloalkyl, cycloalkylalkyl, aryl, aralkyl, aralkenyl, furanylalkyl, tetrahydrofuranylalkyl, tetrahydropyranylalkyl, dioxolanylalkyl or dioxanylalkyl, andX represents oxygen, sulphur or a CH.sub.2 group,or acid additon salts thereof. Many of the compounds wherein R.sup.1 has a narrower meaning are new.

摘要翻译： 用下式（Ⅰ）的氨基甲基杂环化合物与R1代表氢，烷基，烯基，各取代四氢萘基，十氢萘基，环烷基或环烯基，以及被环烷基，环烯基，环烷氧基 或环烷硫基，其中环状基团可任选被取代，此外任选取代的芳基，另外被芳基，芳氧基，芳硫基，芳基亚磺酰基或芳基磺酰基取代的烷基或被芳基取代的烯基，其中芳基可以在每种情况下 任选被取代; R 2表示氢或甲基，R 3表示烷基，烯基，炔基，烷氧基烷基，羟基烷基，羟基烷氧基烷基，二烷氧基烷基，或在每种情况下任选取代的环烷基，环烷基烷基，芳基，芳烷基，芳烯基，呋喃基烷基，四氢呋喃基烷基，四氢吡喃基烷基，二氧戊环烷基或二烷基烷基，X 代表氧，硫或CH2基，或其酸加成盐。 其中R1具有较窄含义的许多化合物是新的。

公开(公告)号：US4615725A

公开(公告)日：1986-10-07

申请号：US720827

申请日：1985-04-08

申请人： Joachim Weissmuller ,  Wolfgang Kramer ,  Dieter Berg ,  Paul Reinecke ,  Wilhelm Brandes ,  Gerd Hanssler ,  Klaus Lurssen

发明人： Joachim Weissmuller ,  Wolfgang Kramer ,  Dieter Berg ,  Paul Reinecke ,  Wilhelm Brandes ,  Gerd Hanssler ,  Klaus Lurssen

IPC分类号： C07D317/28 ,  A01N43/08 ,  C07C17/26 ,  C07C33/48 ,  C07C43/23 ,  C07D303/22 ,  C07D307/10 ,  C07D307/12 ,  C07D307/14 ,  C07D405/06 ,  C07D413/06 ,  A01N43/40

CPC分类号： C07D303/22 ,  A01N43/08 ,  C07C17/2632 ,  C07C33/483 ,  C07C43/23 ,  C07D307/10 ,  C07D307/12 ,  C07D307/14 ,  C07D405/06 ,  C07D413/06

摘要： Tetrahydrofuran-2-ylmethylamines of the formula ##STR1## in which R.sup.1 represents optionally substituted naphthyl, optionally substituted cycloalkyl or cycloalkenyl, optionally substituted phenyl, or alkyl which is substituted by in each case optionally substituted phenyl, phenoxy or phenylthio,R.sup.2 represents hydrogen or methyl,R.sup.3 represents alkyl andR.sup.4 represents alkyl, alkenyl, alkinyl or optionally substituted aralkyl, orR.sup.3 and R.sup.4, together with the nitrogen atom to which they are bonded, represent an optionally substituted heterocyclic radical, which can contain further hetero-atoms,excluding the compounds in which R.sup.3 and R.sup.4 both represent methyl, R.sup.1 represents unsubstituted phenyl and R.sup.2 at the same time represents hydrogen, or plant-tolerated addition products thereof with acids or metal salts, which possess fungicidal and plant growth regulating activities.

摘要翻译： 式“IMAGE”的四氢呋喃-2-基甲胺，其中R 1表示任选取代的萘基，任选取代的环烷基或环烯基，任选取代的苯基或被各种情况下被任意取代的苯基，苯氧基或苯硫基取代的烷基，R 2表示氢或 甲基，R 3表示烷基，R 4表示烷基，烯基，炔基或任选取代的芳烷基，或者R 3和R 4与它们所键合的氮原子一起代表任选取代的杂环基，其可含有其它杂原子，不包括 其中R3和R4都表示甲基，R1代表未取代的苯基和R2同时表示具有杀真菌和植物生长调节活性的氢或其与酸或金属盐的植物耐受加成产物。

公开(公告)号：US4542130A

公开(公告)日：1985-09-17

申请号：US624889

申请日：1984-06-27

申请人： Joachim Weissmuller ,  Wolfgang Kramer ,  Dieter Berg ,  Paul Reinecke ,  Wilhelm Brandes ,  Gerd Hanssler

发明人： Joachim Weissmuller ,  Wolfgang Kramer ,  Dieter Berg ,  Paul Reinecke ,  Wilhelm Brandes ,  Gerd Hanssler

IPC分类号： A01N43/28 ,  A01N43/46 ,  A01N43/60 ,  A01N43/84 ,  C07D327/00 ,  C07D327/04 ,  C07D411/06 ,  C07D413/06

CPC分类号： C07D411/06 ,  A01N43/28 ,  C07D327/04

摘要： MIcrobicidally active 5-aminomethyl-1,3-oxathiolanes of the formula ##STR1## in which R.sup.1 is tetrahydronaphthyl, decahydronaphthyl or optionally substituted naphthyl, optionally substituted cycloalkyl or cycloalkenyl, optionally substituted phenyl, or alkyl which is substituted by phenyl, phenoxy, phenylthio, cyclohexyl, cyclohexyloxy or cyclohexylthio, each of which is optionally substituted,R.sup.2 is hydrogen or methyl,R.sup.3 is alkyl, andR.sup.4 is alkyl, alkenyl or optionally substituted aralkyl, orR.sup.3 and R.sup.4, together with the nitrogen atom to which they are bonded, form an optionally substituted saturated heterocyclic structure which can contain further heteroatoms,or a plant-tolerated addition product thereof with an acid or metal salt.

摘要翻译： 其中R 1为四氢萘基，十氢萘基或任选取代的萘基，任选取代的环烷基或环烯基，任选取代的苯基，或被苯基，苯氧基，苯硫基取代的烷基的除草活性的5-氨基甲基-1,3-氧硫杂环戊烷 环己基，环己氧基或环己基硫基，其各自任选被取代，R 2是氢或甲基，R 3是烷基，R 4是烷基，烯基或任选被取代的芳烷基，或者R 3和R 4与它们所键合的氮原子一起 形成可以含有其它杂原子的任选取代的饱和杂环结构，或其含有酸或金属盐的植物耐受的加成产物。

公开(公告)号：US5128368A

公开(公告)日：1992-07-07

申请号：US595143

申请日：1990-10-10

申请人： Wolfgang Kramer ,  Joachim Weissmuller ,  Graham Holmwood ,  Dieter Berg ,  Stefan Dutzmann ,  Wilhelm Brandes ,  Gerd Hanssler ,  Paul Reinecke

发明人： Wolfgang Kramer ,  Joachim Weissmuller ,  Graham Holmwood ,  Dieter Berg ,  Stefan Dutzmann ,  Wilhelm Brandes ,  Gerd Hanssler ,  Paul Reinecke

IPC分类号： A01N43/08 ,  A01N43/28 ,  C07D307/14 ,  C07D307/22 ,  C07D317/28 ,  C07D327/04 ,  C07D407/12 ,  C07D417/12

CPC分类号： C07D407/12 ,  A01N43/08 ,  A01N43/28 ,  C07D307/14 ,  C07D317/28 ,  C07D327/04

摘要： Combatting fungi and bacteria with aminomethylheterocyclic compounds of the formula ##STR1## in which R.sup.1 represents hydrogen, alkyl, alkenyl, in each case optionally substituted tetrahydronaphthyl, decahydronaphthyl, cycloalkyl or cycloalkenyl, furthermore alkyl which is substituted by cycloalkyl, cycloalkenyl, cycloalkyloxy or cycloalkylthio, where the cyclic radicals may optionally be substituted, furthermore optionally substituted aryl, in addition alkyl which is substituted by aryl, aryloxy, arylthio, arylsulphinyl or arylsulphonyl, or alkenyl which is substituted by aryl, where the aryl radicals may in each case optionally be substituted;R.sup.2 represents hydrogen or methyl,R.sup.3 represents alkyl, alkenyl, alkinyl, alkoxyalkyl, hydroxyalkyl, hydroxyalkoxyalkyl, dialkoxyalkyl, or in each case optionally substituted cycloalkyl, cycloalkylalkyl, aryl, aralkyl, aralkenyl, furanylalkyl, tetrahydrofuranylalkyl, tetrahydropyranylalkyl, dioxolanylalkyl or dioxanylalkyl, andX represents oxygen, sulphur or a CH.sub.2 group,or acid addition salts thereof.Many of the compounds wherein R.sup.1 has a narrower meaning are new.

摘要翻译： 用下式（Ⅰ）的氨基甲基杂环化合物与R1代表氢，烷基，烯基，各取代四氢萘基，十氢萘基，环烷基或环烯基，以及被环烷基，环烯基，环烷基 或环烷硫基，其中环状基团可任选被取代，此外任选取代的芳基，另外被芳基，芳氧基，芳硫基，芳基亚磺酰基或芳基磺酰基取代的烷基或被芳基取代的烯基，其中芳基可以在每种情况下 任选被取代; R 2表示氢或甲基，R 3表示烷基，烯基，炔基，烷氧基烷基，羟基烷基，羟基烷氧基烷基，二烷氧基烷基，或在每种情况下任选取代的环烷基，环烷基烷基，芳基，芳烷基，芳烯基，呋喃基烷基，四氢呋喃基烷基，四氢吡喃基烷基，二氧戊环烷基或二烷基烷基，X 代表氧，硫或CH2基，或其酸加成盐。 其中R1具有较窄含义的许多化合物是新的。

公开(公告)号：US4563447A

公开(公告)日：1986-01-07

申请号：US630487

申请日：1984-07-13

申请人： Wolfgang Kramer ,  Joachim Weissmuller ,  Dieter Berg ,  Paul Reinecke ,  Gerd Hanssler ,  Wilhelm Brandes

发明人： Wolfgang Kramer ,  Joachim Weissmuller ,  Dieter Berg ,  Paul Reinecke ,  Gerd Hanssler ,  Wilhelm Brandes

IPC分类号： A01N43/40 ,  C07D317/00 ,  C07D317/16 ,  C07D317/28 ,  C07D405/06 ,  C07D405/14

CPC分类号： C07D405/06 ,  A01N43/40 ,  C07D317/16 ,  C07D317/28 ,  C07D405/14

摘要： Substituted 4-piperidinomethyl-1,3-dioxolanes of the formula ##STR1## in which R.sup.1 is tetrahydronaphthyl, decahydronaphthyl, optionally substituted naphthyl, optionally substituted cycloalkyl or cycloalkenyl, optionally substituted phenyl, or alkyl which is substituted by in each case optionally substituted phenyl, phenoxy, phenylthio, cyclohexyl, cyclohexyloxy or cyclohexylthio,R.sup.2 is hydrogen or methyl,R.sup.3 is hydrogen or an acyl radicalor plant-tolerated addition products thereof with acids or metal salts, which possess fungicidal activity.

摘要翻译： 取代的式“IMAGE”的4-哌啶甲基-1,3-二氧戊烷，其中R 1是四氢萘基，十氢萘基，任选取代的萘基，任选取代的环烷基或环烯基，任选取代的苯基或被各种情况下被取代的任选取代的苯基 ，苯氧基，苯硫基，环己基，环己氧基或环己基硫基，R2是氢或甲基，R3是氢或具有杀真菌活性的酸或其盐的酰基或植物耐受的加成产物。

公开(公告)号：US5493034A

公开(公告)日：1996-02-20

申请号：US443522

申请日：1995-05-18

申请人： Wolfgang Kramer ,  Joachim Weissmuller ,  Dieter Berg ,  Wilhelm Brandes ,  Stefan Dutzmann

发明人： Wolfgang Kramer ,  Joachim Weissmuller ,  Dieter Berg ,  Wilhelm Brandes ,  Stefan Dutzmann

IPC分类号： A01N43/28 ,  A01N43/30 ,  C07D317/72 ,  C07D327/04 ,  C07D411/12

CPC分类号： C07D317/72 ,  A01N43/28 ,  A01N43/30 ,  C07D327/04 ,  C07D411/12

摘要： Fungicidally active compounds of the formula ##STR1## in which X represents oxygen or sulphur,R represents cycloalkyl, or represents optionally substituted aryl, or represents the radical ##STR2## R.sup.1 and R.sup.2 each independently is hydrogen or an organic radical, or together with the nitrogen atom form a heterocyclic radical,R.sup.3 represents hydrogen, alkyl or optionally substituted aryl, andR.sup.4 represents alkyl or cycloalkyl, or represents optionally substituted aryl,but wherein R.sup.3 and R.sup.4 may not simultaneously represent methyl,and acid addition salts thereof, as well as intermediates therefor.

公开(公告)号：US4740515A

公开(公告)日：1988-04-26

申请号：US632138

申请日：1984-07-18

申请人： Joachim Weissmuller ,  Wolfgang Kramer ,  Karl H. Buchel ,  Wilhelm Brandes ,  Paul Reinecke

发明人： Joachim Weissmuller ,  Wolfgang Kramer ,  Karl H. Buchel ,  Wilhelm Brandes ,  Paul Reinecke

IPC分类号： A01N43/653 ,  C07C17/14 ,  C07D249/08 ,  C07D521/00

CPC分类号： C07D231/12 ,  A01N43/653 ,  C07C17/14 ,  C07D233/56 ,  C07D249/08

摘要： 3-(1,2,4-Triazol-1-yl)-prop-1-enes of the general formula (I) ##STR1## in which X.sup.1 and X.sup.2 independently of one another represent hydrogen or methyl,R.sup.1 represents alkyl, alkenyl, in each case optionally substituted cycloalkyl or cycloalkenyl or in each case optionally substituted phenyl or benzyl andR.sup.2 represents alkyl, alkenyl, in each case optionally substituted cycloalkyl or cycloalkenyl, halogenoalkyl, in each case optionally substituted phenyl or phenylalkyl, phenoxyalkyl or phenylthioalkyl, in each case optionally substituted in the phenyl part,but whereinR.sup.1 and R.sup.2 may not simultaneously represent optionally substituted phenyl if X.sup.1 and/or X.sup.2 represent hydrogen,and acid addition salts and metal salt complexes thereof which are tolerated by plants, exhibit fungicidal activity.

摘要翻译： 其中X 1和X 2彼此独立地表示氢或甲基的通式（I）的（I）的3-（1,2,4-三唑-1-基） - 丙-1-烯，R 1表示 烷基，烯基，在每种情况下均为任选取代的环烷基或环烯基，或在每种情况下为任选取代的苯基或苄基，并且R 2表示烷基，烯基，在每种情况下为任选取代的环烷基或环烯基，卤代烷基，在每种情况下为任选取代的苯基或苯基烷基，苯氧基烷基或 苯硫基烷基，在每种情况下都可以在苯基部分被取代，但如果X1和/或X2代表氢，其中R1和R2不能同时代表任选取代的苯基，并且其被植物耐受的酸加成盐和金属盐络合物显示为杀真菌剂 活动。