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    Tricyclic indole compounds having an affinity against serotonin receptors
    1.
    发明申请
    Tricyclic indole compounds having an affinity against serotonin receptors 审中-公开
    对5-羟色胺受体具有亲和力的三环吲哚化合物

    公开(公告)号：US20050043387A1

    公开(公告)日：2005-02-24

    申请号：US10947172

    申请日：2004-09-23

    申请人： Yoshikazu Fukui ,  Makoto Adachi ,  Takashi Sasatani

    发明人： Yoshikazu Fukui ,  Makoto Adachi ,  Takashi Sasatani

    IPC分类号： A61P5/28 ,  A61P25/00 ,  A61P25/04 ,  A61P25/06 ,  A61P25/16 ,  A61P25/18 ,  A61P25/22 ,  A61P25/24 ,  A61P43/00 ,  C07D491/06 ,  A61K31/55 ,  A61K31/407 ,  A61K31/454 ,  C07D491/02

    CPC分类号： C07D491/06

    摘要： Having an affinity against serotonine receptors, compound (I) shown below is useful as a therapeutic agent against various kinds of diseases of central nervous systems. (wherein R1 is hydrogen; R2 is hydrogen or lower alkyl; R3 is hydrogen, —COOR12 and so on; R4 is hydrogen, lower alkyl and so on, or R3 and R4 taken together may form ═O or ═S; R5 is hydrogen, or R3 and R5 taken together may form a bond; R6 is hydrogen, —COOR24 and so on; R7 is hydrogen, halogen, lower alkyl and so on; R8 is hydrogen, lower alkyl, cycloalkyl and so on; R9, R10 and R11 are each independently hydrogen, halogen, lower alkyl and so on)

    摘要翻译： 对于5-羟色胺受体具有亲和性，下文所示的化合物（I）可用作抗各种中枢神经系统疾病的治疗剂。 （其中R 1为氢; R 2为氢或低级烷基; R 3为氢，-COOR 12等; R 4为氢，低级烷基等，或R R 3和R 4一起可以形成= O或= S; R 5是氢，或者R 3和R 5一起可以形成键; R 6是氢， COOR 24等; R 7是氢，卤素，低级烷基等; R 8是氢，低级烷基，环烷基等; R 9，R 10和R 10， 11>各自独立地为氢，卤素，低级烷基等）

    Tricyclic indole compounds having affinity for serotonin receptor
    2.
    发明授权
    Tricyclic indole compounds having affinity for serotonin receptor 失效
    对5-羟色胺受体具有亲和力的三环吲哚化合物

    公开(公告)号：US06858640B2

    公开(公告)日：2005-02-22

    申请号：US10312818

    申请日：2001-09-17

    申请人： Yoshikazu Fukui ,  Makoto Adachi ,  Takashi Sasatani

    发明人： Yoshikazu Fukui ,  Makoto Adachi ,  Takashi Sasatani

    IPC分类号： A61P5/28 ,  A61P25/00 ,  A61P25/04 ,  A61P25/06 ,  A61P25/16 ,  A61P25/18 ,  A61P25/22 ,  A61P25/24 ,  A61P43/00 ,  C07D491/06 ,  A61K31/40 ,  C07D491/044

    CPC分类号： C07D491/06

    摘要： Having an affinity against serotonine receptors, compound (I) shown below is useful as a therapeutic agent against various kinds of diseases of central nervous systems; (wherein R1 is hydrogen; R2 is hydrogen or lower alkyl; R3 is hydrogen, —COOR12 and so on; R4 is hydrogen, lower alkyl and so on, or R3 and R4 taken together may form ═O or ═S; R5 is hydrogen, or R3 and R5 taken together may form a bond; R6 is hydrogen, —COOR24 and so on; R7 is hydrogen, halogen, lower alkyl and so on; R8 is hydrogen, lower alkyl, cycloalkyl and so on; R9, R10 and R11 are each independently hydrogen, halogen, lower alkyl and so on).

    摘要翻译： 对于5-羟色胺受体具有亲和力，下文所示的化合物（I）可用作抗各种中枢神经系统疾病的治疗剂;（其中R 1是氢; R 2是氢或低级烷基; 3>是氢，-COOR 12等; R 4是氢，低级烷基等，或者R 3和R 4一起可以形成= O或= S; R 5 >是氢，或R 3和R 5一起形成键; R 6是氢，-COOR 24等; R 7是氢，卤素，低级烷基等 R 8是氢，低级烷基，环烷基等; R 9，R 10和R 11各自独立地是氢，卤素，低级烷基等）。

    Pyrrolo[1,2-b] pyridazine derivatives having sPLA2 inhibitory effect
    5.
    发明授权
    Pyrrolo[1,2-b] pyridazine derivatives having sPLA2 inhibitory effect 失效
    具有sPLA2抑制作用的吡咯并[1,2-b]哒嗪衍生物

    公开(公告)号：US06472389B1

    公开(公告)日：2002-10-29

    申请号：US09673413

    申请日：2000-10-18

    申请人： Mitsuaki Ohtani ,  Masahiro Fuji ,  Yoshikazu Fukui ,  Makoto Adachi

    发明人： Mitsuaki Ohtani ,  Masahiro Fuji ,  Yoshikazu Fukui ,  Makoto Adachi

    IPC分类号： A61K315025

    CPC分类号： C07D487/04

    摘要： The present invention provides a compound having sPLA2 inhibiting activity. The compound represented by the formula (I): wherein R1 is —(L1)—R6 wherein L1 is a divalent linking group of 1 to 18 atoms or the like, and R6 is a carbocyclic ring substituted by at least one non-interfering substituent or the like; R2 is C1 to C3 alkyl or the like; R3 is —(L2)-(acidic group); R4 and R5 are hydrogen atoms, non-interfering substituents, carbocyclic groups or the like; X is independently oxygen atom of sulfur atom; and RA is —C(═X)—C(═X)—NH2 or the like; the prodrugs thereof, their pharmaceutically acceptable salts, or their solvates, and a composition for inhibiting sPLA2 containing them as effective ingredients.

    摘要翻译： 本发明提供具有sPLA2抑制活性的化合物。式（I）表示的化合物：其中R1为 - （L1）-R6，其中L1为1至18个原子的二价连接基团等，R6为 被至少一个非干扰取代基等取代的碳环; R2是C1-C3烷基等; R3是 - （L2） - （酸性基团）; R4和R5是氢原子，非干扰取代基，碳环基团等; X独立地是硫原子的氧原子; RA为-C（= X）-C（= X）-NH 2等; 其前体药物，其药学上可接受的盐或其溶剂合物，以及用于抑制含有它们作为有效成分的sPLA2的组合物。

    Method and apparatus for two-channel recording of video signals
    6.
    发明授权
    Method and apparatus for two-channel recording of video signals 失效
    用于视频信号双通道录像的方法和装置

    公开(公告)号：US5394276A

    公开(公告)日：1995-02-28

    申请号：US49589

    申请日：1993-04-20

    申请人： Makoto Adachi

    发明人： Makoto Adachi

    IPC分类号： H04N5/92 ,  H04N7/015 ,  H04N9/797 ,  H04N9/81 ,  H04N5/78

    CPC分类号： H04N9/7973 ,  Y10S348/91

    摘要： A video signal recording apparatus is provided with first and second channels for transmitting an input video signal. The first channel has a line memory for conducting a 1H delay on data and a time-base-extension line memory for conducting time base extension on the data with the 1H delay. The data subjected to the time base extension undergoes D/A conversion to be an output of the first channel. On the other hand, the second channel does not have a line memory for a 1H delay, and the video signal without delay is subjected to time base extension and undergoes D/A conversion to be an output of the second channel. In the arrangement, odd lines and even lines respectively contained in adjoining two frames in each channel are reversed such that in a certain frame, odd lines of the input video signal are transmitted through the first channel with even lines through the second channel. In the next frame, even lines are transmitted through the first channel with odd lines through the second channel. Thus, influences on the reproduced picture due to the difference of circuit characteristics is averaged and the perception to unevenness of color or brightness is avoided.

    摘要翻译： 视频信号记录装置具有用于发送输入视频信号的第一和第二信道。 第一通道具有用于在数据上进行1H延迟的行存储器和用于对1H延迟的数据进行时基扩展的时基扩展线存储器。 经过时基扩展的数据经历D / A转换为第一通道的输出。 另一方面，第二通道不具有用于1H延迟的行存储器，并且没有延迟的视频信号经受时基扩展，并且经历D / A转换为第二通道的输出。 在这种布置中，分别包含在每个通道中的相邻两个帧中的奇数行和偶数行被反转，使得在某个帧中，输入视频信号的奇数行通过第二通道的偶数行通过第一通道传输。 在下一帧中，偶数行通过第二通道以奇数行通过第一通道传输。 因此，由于电路特性的差异对对再现图像的影响被平均，并且避免了对颜色或亮度的不均匀性的感知。

    Solar heat powered plant
    7.
    发明授权
    Solar heat powered plant 失效
    太阳能热力发电厂

    公开(公告)号：US4569331A

    公开(公告)日：1986-02-11

    申请号：US559248

    申请日：1983-12-08

    申请人： Tatsuo Tani ,  Sinji Sawata ,  Tadayoshi Tanaka ,  Koichi Sakuta ,  Yuuji Nagata ,  Yasushi Eto ,  Makoto Adachi ,  Yasunori Matsurra

    发明人： Tatsuo Tani ,  Sinji Sawata ,  Tadayoshi Tanaka ,  Koichi Sakuta ,  Yuuji Nagata ,  Yasushi Eto ,  Makoto Adachi ,  Yasunori Matsurra

    IPC分类号： F24S90/00 ,  F24D11/00 ,  F24D17/00

    CPC分类号： F24D11/003 ,  Y02B10/20

    摘要： In a solar heat powered plant according to the present invention, hot water is normally circulated through a hot-water tank, a low-temperature-side heat load unit, a return tank, a low-temperature-side heat exchanger, and again through the hot-water tank, in the order named, under the condition in which first and second valves are opened and closed, respectively. On the other hand, in warming up the hot-water tank, the first and second valves are closed and opened, respectively, so that the hot water is circulated between the hot-after tank and the low-temperature-side heat exchanger, through a by-pass pipe. Thus, the warming up of the hot-water tank can be achieved in a short time.

    摘要翻译： 在本发明的太阳能热力发电设备中，热水通常循环通过热水箱，低温侧热负荷单元，回流箱，低温侧热交换器，再次通过 分别在第一和第二阀门打开和关闭的条件下按照命名的顺序排列热水箱。 另一方面，在对热水箱进行预热时，第一和第二阀分别关闭并打开，使得热水在热水箱和低温侧热交换器之间循环，通过 旁路管。 因此，可以在短时间内实现热水箱的升温。

    Opening/closing body control device, opening/closing body control system, power window device, and power window system
    9.
    发明授权
    Opening/closing body control device, opening/closing body control system, power window device, and power window system 有权

    公开(公告)号：US11480005B2

    公开(公告)日：2022-10-25

    申请号：US16659212

    申请日：2019-10-21

    申请人： Takashi Aragai ,  Makoto Adachi ,  Tomohiro Murase

    发明人： Takashi Aragai ,  Makoto Adachi ,  Tomohiro Murase

    IPC分类号： E05F15/695 ,  E05F15/40 ,  E05F15/70

    摘要： An opening/closing body control device continues an as-needed operation where the opening/closing body is controlled in response to the operation instruction signal even when an abnormality in an opening/closing position of the opening/closing body is detected, continues opening and closing the opening/closing body until it is determined that the abnormal state in the opening/closing instruction signal is confirmed even when an abnormality in the opening/closing instruction signal is detected during the as-needed opening/closing operation, and stops opening and closing the opening/closing body the abnormal state in the opening/closing instruction signal is confirmed. The confirmation time at the presence of the opening/closing position abnormality is shorter than that at the absence of opening/closing position abnormality.

    Image decoding apparatus and image decoding method
    10.
    发明授权
    Image decoding apparatus and image decoding method 有权
    图像解码装置和图像解码方法

    公开(公告)号：US08885707B2

    公开(公告)日：2014-11-11

    申请号：US11887441

    申请日：2006-03-31

    申请人： Makoto Adachi ,  Hiroaki Toida ,  Kiyofumi Abe

    发明人： Makoto Adachi ,  Hiroaki Toida ,  Kiyofumi Abe

    IPC分类号： H04N7/12 ,  H04N19/593 ,  H04N19/61 ,  H04N19/89 ,  H04N19/44 ,  H04N19/11 ,  H04N19/176 ,  H04N19/46

    CPC分类号： H04N19/159 ,  H04N19/11 ,  H04N19/136 ,  H04N19/176 ,  H04N19/423 ,  H04N19/44 ,  H04N19/46 ,  H04N19/593 ,  H04N19/61 ,  H04N19/89

    摘要： An image decoding apparatus and an image decoding method capable of generating a decoded image even in the case where a pixel in a block is necessary as a reference pixel, the block where an intra prediction mode specified in a stream is unavailable according to a standard, due to a transmission error, a coding-method error, or the like. An image decoding apparatus determines whether or not a reference block necessary for a specified intra prediction mode is available, based on intra-prediction mode information extracted by an intra-prediction mode extraction unit and peripheral block pixel information stored in a line memory. The image decoding apparatus includes a reference pixel determination unit which controls a switch unit; and a substitute intra-prediction image generation unit which generates a substitute intra-prediction image in the case where a reference block necessary for a specified intra prediction mode is unavailable.

    摘要翻译： 即使在需要块中的像素作为参考像素的情况下也能够生成解码图像的图像解码装置和图像解码方法，流中指定的帧内预测模式的块根据标准不可用， 由于传输错误，编码方法错误等。 图像解码装置基于由帧内预测模式提取单元提取的帧内预测模式信息和存储在行存储器中的周边块像素信息来确定指定帧内预测模式所需的参考块是否可用。 图像解码装置包括控制开关单元的参考像素确定单元; 以及在指定的帧内预测模式所需的基准块不可用的情况下，生成替代帧内预测图像的替代帧内预测图像生成单元。