-
1.发明授权Anti-ulcer agent comprising chalcone derivative as effective ingredient and novel chalcone derivative 失效将包含CHALCONE衍生物的抗真菌剂作为有效成分和新型氯胺酮衍生物
公开(公告)号：US5106871A
公开(公告)日：1992-04-21
申请号：US733003
申请日：1991-07-19
IPC分类号： C07C45/62 , C07C45/67 , C07C45/68 , C07C45/71 , C07C45/74 , C07C49/83 , C07C49/835 , C07C49/84 , C07C59/90
CPC分类号： C07C59/90 , C07C45/62 , C07C45/673 , C07C45/68 , C07C45/71 , C07C45/74 , C07C49/83 , C07C49/835 , C07C49/84
摘要： The present invention relates to an anti-ulcer agent comprising a compound represented by the following general formula I as the effective ingredient, and a novel chalcone derivative included in the compound represented by this general formula I: ##STR1## wherein X and Y independently stand for a hydrogen atom or together form a single bond, R.sub.1 stands for a hydroxyl group, an acetoxy group, a carboxymethoxy group or a methoxycarbonylmethoxy group, R.sub.2 stands for a hydrogen atom, an isoprenyl group, isopentyl group or a propyl group, R.sub.3 stands for hydroxyl group or a methoxy group, R.sub.4 stands for a hydrogen atom, a hydroxyl group or a methoxy group, R.sub.5 stands for a hydrogen atom, a hydroxyl group, a methoxy group or an isopentyl group, R.sub.6 stands for a hydroxyl group, a methoxy group or a carboxymethoxy group, and R.sub.7 stands for a hydrogen atom or a methoxy group.
-
公开(公告)号：US5234951A
公开(公告)日：1993-08-10
申请号：US797063
申请日：1991-11-25
IPC分类号： C07C45/62 , C07C45/67 , C07C45/68 , C07C45/71 , C07C45/74 , C07C49/83 , C07C49/835 , C07C49/84 , C07C59/90
CPC分类号： C07C59/90 , C07C45/62 , C07C45/673 , C07C45/68 , C07C45/71 , C07C45/74 , C07C49/83 , C07C49/835 , C07C49/84 , Y10S514/925
摘要： The present invention relates to an anti-ulcer agent comprising a compound represented by the following general formula I as the effective ingredient, and a novel chalcone derivative included in the compound represented by this general formula I: ##STR1## wherein X and Y independently stand for a hydrogen atom or together form a single bond, R.sub.1 stands for a hydroxyl group, an acetoxy group, a carboxymethoxy group or a methoxycarbonylmethoxy group, R.sub.2 stands for a hydrogen atom, an isoprenyl group, isopentyl group or a propyl group, R.sub.3 stands for a hydroxyl group or a methoxy group, R.sub.4 stands for a hydrogen atom, a hydroxyl group or a methoxy group, R.sub.5 stands for a hydrogen atom, a hydroxyl group, a methoxy group or an isopentyl group, R.sub.6 stands for a hydroxyl group, a methoxy group or a carboxymethoxy group, and R.sub.7 stands for a hydrogen atom or a methoxy group.
摘要翻译： 本发明涉及包含以下通式I表示的化合物作为有效成分的抗溃疡剂，以及由通式I表示的化合物中包含的新型查耳酮衍生物：其中X和Y独立地为 代表氢原子或一起形成单键，R1代表羟基，乙酰氧基，羧甲氧基或甲氧基羰基甲氧基，R2代表氢原子，异戊二烯基，异戊基或丙基，R3 代表羟基或甲氧基，R4代表氢原子，羟基或甲氧基，R5代表氢原子，羟基，甲氧基或异戊基，R6代表羟基 ，甲氧基或羧甲氧基，R7表示氢原子或甲氧基。
-
公开(公告)号：US4962211A
公开(公告)日：1990-10-09
申请号：US445977
申请日：1989-11-21
IPC分类号： C07D317/68 , A61K31/357 , A61K31/36 , A61P1/16
CPC分类号： C07D317/68
摘要： The present invention relates to a novel biphenyl derivative having a liver ailment-moderating action, which is effective for the remedy of liver diseases such as acute hepatitis and chronic hepatitis, a process for the preparation of this derivative and a liver ailment-moderating agent comprising this derivative as an active ingredient. Moreover, the present invention relates to a compound valuable as the intermediate compound for the synthesis of this derivative and a process for efficiently preparing this intermediate compound.
-
公开(公告)号：US5032685A
公开(公告)日：1991-07-16
申请号：US439840
申请日：1989-11-21
IPC分类号： C07D317/68 , A61K31/357 , A61K31/36 , A61P1/16
CPC分类号： C07D317/68
摘要： The present invention relates to a novel biphenyl derivative having a liver ailment-moderating action, which is effective for the remedy of liver diseases such as acute hepatitis and chronic hepatitis, a process for the preparation of this derivative and a liver ailment-moderating agent comprising this derivative as an active ingredient. Moreover, the present invention relates to a compound valuable as the intermediate compound for the synthesis of this derivative and a process for efficiently preparing this intermediate compound.
-
公开(公告)号：US4987240A
公开(公告)日：1991-01-22
申请号：US450211
申请日：1989-11-21
IPC分类号： C07D317/68 , A61K31/357 , A61K31/36 , A61P1/16
CPC分类号： C07D317/68
摘要： The present invention relates to a novel biphenyl derivative having a liver ailment-moderating action, which is effective for the remedy of liver diseases such as acute hepatitis and chronic hepatitis, a process for the preparation of this derivative and a liver ailment-moderating agent comprising this derivative as an active ingredient. Moreover, the present invention relates to a compound valuable as the intermediate compound for the synthesis of this derivative and a process for efficiently preparing this intermediate compound.
-
公开(公告)号：US4904694A
公开(公告)日：1990-02-27
申请号：US180107
申请日：1988-02-10
IPC分类号： C07D317/68 , A61K31/357 , A61K31/36 , A61P1/16
CPC分类号： C07D317/68
摘要： The present invention relates to a novel biphenyl derivative having a liver ailment-moderating action, which is effective for the remedy of liver diseases such as acute hepatitis and chronic hepatitis, a process for the preparation of this derivative and a liver ailment-moderating agent comprising this derivative as an active ingredient. Moreover, the present invention relates to a compound valuable as the intermediate compound for the synthesis of this derivative and a process for efficiently preparing this intermediate compound.
-
7.发明授权
公开(公告)号：US5227398A
公开(公告)日：1993-07-13
申请号：US798202
申请日：1991-11-26
IPC分类号： C07D317/60 , C07D317/66 , C07D409/06 , C07D409/12
CPC分类号： C07D409/06 , C07D317/60 , C07D317/66 , C07D409/12
摘要： Hepatopathy improvers contain as an effective ingredient one or more of benzodioxole derivatives represented by the following formula: ##STR1## wherein A means a particular N- or S-containing group. Most of these benzodioxole derivatives are novel.
-
公开(公告)号：US4925872A
公开(公告)日：1990-05-15
申请号：US341803
申请日：1989-04-24
IPC分类号： C07D317/68
CPC分类号： C07D317/68
摘要： The present invention relates to a novel biphenyl derivative having a liver ailment-moderating action and effective as a remedy for acute hepatitis and chronic hepatitis, a process for the preparation of this biphenyl derivative and a liver ailment-moderating agent comprising this diphenyl derivative as an effective ingredient. This diphenyl derivative is represented by the following formula: ##STR1## wherein R.sub.0 and R.sub.1 independently stand for a lower alkyl group or R.sub.0 and R.sub.1 together represent a group O.dbd.C
-
9.发明授权Certain 1,3,4-thiadiazole derivatives and anti-ulcer agent comprising said derivatives as active ingredient 失效某些1,3,4-噻二唑衍生物和包含作为活性成分的所述衍生物的抗真菌剂
公开(公告)号：US5106859A
公开(公告)日：1992-04-21
申请号：US613693
申请日：1990-07-30
IPC分类号： A61K31/44 , A61P1/04 , C07D417/14
CPC分类号： C07D417/14
摘要： A novel thiadiazole derivative represented by the following formula I: ##STR1## wherein when n is 0, m is 0, and when n is 1, m is 0 or 1, and the preparation of this derivative and the use of this derivative as an anti-ulcer agent.
-
公开(公告)号：US4996331A
公开(公告)日：1991-02-26
申请号：US341813
申请日：1989-04-24
IPC分类号： C07D317/68
CPC分类号： C07D317/68
摘要： The present invention relates to a novel biphenyl derivative having a liver ailment-moderating action and effective as a remedy for acute hepatitis and chronic hepatitis, a process for the preparation of this biphenyl derivative and a liver ailment-moderating agent comprising this diphenyl derivative as an effective ingredient. This diphenyl derivative is represented by the following formula: ##STR1## wherein R.sub.0 and R.sub.1 independently stand for a lower alkyl group or R.sub.0 and R.sub.1 together represent a group O.dbd.C
-
-
-
-
-
-
-
-
-
搜索结果
16 条记录 (耗时 0.024 秒)